naltrexone and dronabinol

naltrexone has been researched along with dronabinol in 39 studies

Research

Studies (39)

TimeframeStudies, this research(%)All Research%
pre-19904 (10.26)18.7374
1990's8 (20.51)18.2507
2000's17 (43.59)29.6817
2010's9 (23.08)24.3611
2020's1 (2.56)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Järbe, TU; Ohlin, GC1
Cheney, DL; Costa, E; Revuelta, AV; Wood, PL1
Coscia, CJ; Devane, WA; Howlett, AC; Spain, JW1
Ayhan, IH; Portoghese, PS; Takemori, AE; Tulunay, FC1
Compton, DR; Martin, BR; Mechoulam, R; Razdan, RK; Smith, PB; Welch, SP1
Foltz, RL; Fraser, MD; Nelson, CC; Wilfahrt, JK1
Martin, BR; Smith, PB; Welch, SP1
Welch, SP2
Fuentes, JA; Reche, I; Ruiz-Gayo, M2
Lowe, J; Mason, DJ; Welch, SP1
de Wit, H; Wachtel, SR1
Greenwald, MK; Stitzer, ML1
Berrendero, F; Maldonado, R1
Delatte, MS; Moerschbaecher, JM; Winsauer, PJ1
Gardell, LR; Lai, J; Ossipov, MH; Porreca, F; Vanderah, TW1
Bisaga, A; Foltin, RW; Haney, M1
Goldberg, SR; Justinova, Z; Munzar, P; Tanda, G1
Cox, ML; Welch, SP1
Goldberg, SR; Solinas, M1
Acquas, E; Di Chiara, G; Fenu, S; Pisanu, A1
Flau, K; Kathmann, M; Redmer, A; Schlicker, E; Tränkle, C1
Haney, M1
Becker, GL; France, CP; Gerak, LR; Li, JX; McMahon, LR1
Cooper, ZD; Haney, M1
Kurose, M; Meng, ID; Okada-Ogawa, A1
Craft, RM; Wakley, AA1
Braley, G; Carbuto, M; D'Souza, DC; Elander, J; Perry, E; Pittman, B; Radhakrishnan, R; Ranganathan, M; Sewell, RA1
Cheng, K; Flax, SM; Rice, KC; Riley, AL; Wakeford, AG1
Bisaga, A; Carpenter, KM; Glass, A; Haney, M; Levin, FR; Mariani, JJ; Mishlen, K; Nunes, EV; Pavlicova, M; Raby, WN; Sullivan, MA1
Ding, H; Kiguchi, N; Kishioka, S; Ko, MC; Mabry, KM1

Reviews

1 review(s) available for naltrexone and dronabinol

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

6 trial(s) available for naltrexone and dronabinol

ArticleYear
Naltrexone does not block the subjective effects of oral Delta(9)-tetrahydrocannabinol in humans.
    Drug and alcohol dependence, 2000, Jun-01, Volume: 59, Issue:3

    Topics: Adolescent; Adult; Affect; Analysis of Variance; Behavior, Addictive; Cross-Over Studies; Double-Blind Method; Dronabinol; Female; Heart Rate; Humans; Male; Marijuana Smoking; Naltrexone; Narcotic Antagonists; Psychomotor Performance; Psychotropic Drugs

2000
Antinociceptive, subjective and behavioral effects of smoked marijuana in humans.
    Drug and alcohol dependence, 2000, Jun-01, Volume: 59, Issue:3

    Topics: Adolescent; Adult; Affect; Analgesics, Non-Narcotic; Double-Blind Method; Dronabinol; Female; Humans; Male; Marijuana Smoking; Middle Aged; Naltrexone; Narcotic Antagonists; Pain Measurement; Psychomotor Performance

2000
Interaction between naltrexone and oral THC in heavy marijuana smokers.
    Psychopharmacology, 2003, Volume: 166, Issue:1

    Topics: Administration, Oral; Adult; Analgesics, Non-Narcotic; Analysis of Variance; Choice Behavior; Dose-Response Relationship, Drug; Double-Blind Method; Dronabinol; Drug Interactions; Female; Heart Rate; Humans; Male; Marijuana Smoking; Methadone; Naltrexone; Narcotic Antagonists; Pain Measurement; Psychomotor Performance; Reaction Time

2003
Opioid antagonism enhances marijuana's effects in heavy marijuana smokers.
    Psychopharmacology, 2010, Volume: 211, Issue:2

    Topics: Adult; Dose-Response Relationship, Drug; Double-Blind Method; Dronabinol; Drug Interactions; Female; Heart Rate; Humans; Male; Marijuana Abuse; Marijuana Smoking; Naltrexone; Narcotic Antagonists; Psychomotor Performance

2010
Naltrexone does not attenuate the effects of intravenous Δ9-tetrahydrocannabinol in healthy humans.
    The international journal of neuropsychopharmacology, 2012, Volume: 15, Issue:9

    Topics: Adolescent; Adult; Attention; Behavior; Cognition; Cognition Disorders; Double-Blind Method; Dronabinol; Drug Interactions; Euphoria; Female; Hallucinogens; Humans; Inhibition, Psychological; Injections, Intravenous; Male; Marijuana Abuse; Memory; Mental Recall; Middle Aged; Naltrexone; Narcotic Antagonists; Orientation; Perception; Psychoses, Substance-Induced; Recognition, Psychology; Reward; Young Adult

2012
The effects of dronabinol during detoxification and the initiation of treatment with extended release naltrexone.
    Drug and alcohol dependence, 2015, Sep-01, Volume: 154

    Topics: Adult; Cannabinoids; Delayed-Action Preparations; Double-Blind Method; Dronabinol; Drug Administration Schedule; Drug Therapy, Combination; Female; Humans; Male; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Patient Compliance; Substance Withdrawal Syndrome; Young Adult

2015

Other Studies

32 other study(ies) available for naltrexone and dronabinol

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
Stimulus effects of delta(9)-THC and its interaction with naltrexone and catecholamine blockers in rats.
    Psychopharmacology, 1977, Oct-20, Volume: 54, Issue:2

    Topics: Animals; Catecholamines; Columbidae; Dronabinol; Drug Interactions; Injections, Intraperitoneal; Male; Naloxone; Naltrexone; Rats; Receptors, Adrenergic, alpha

1977
GABAergic mediation in the inhibition of hippocampal acetylcholine turnover rate elicited by delta 9-tetrahydrocannabinol.
    Neuropharmacology, 1979, Volume: 18, Issue:6

    Topics: Acetylcholine; Animals; Bicuculline; Dopamine; Dronabinol; gamma-Aminobutyric Acid; Hippocampus; Kinetics; Male; Muscimol; Naltrexone; Norepinephrine; Rats; Substantia Nigra

1979
An assessment of the role of opioid receptors in the response to cannabimimetic drugs.
    Journal of neurochemistry, 1986, Volume: 46, Issue:6

    Topics: Adenylyl Cyclase Inhibitors; Animals; Cannabinoids; Cell Line; Dronabinol; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Etorphine; Morphine; Naltrexone; Neuroblastoma; Neurons; Receptors, Opioid; Receptors, Opioid, delta

1986
Antagonism by chlornaltrexamine of some effects of delta 9-tetrahydrocannabinol in rats.
    European journal of pharmacology, 1981, Mar-12, Volume: 70, Issue:2

    Topics: Analgesia; Animals; Dronabinol; Drug Tolerance; Humans; Hypothermia; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Nitrogen Mustard Compounds; Rats; Receptors, Opioid; Substance-Related Disorders

1981
The pharmacological activity of anandamide, a putative endogenous cannabinoid, in mice.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:1

    Topics: Analgesics; Animals; Arachidonic Acids; Binding, Competitive; Brain; Calcium Channel Blockers; Cyclohexanols; Dronabinol; Drug Administration Routes; Drug Interactions; Endocannabinoids; Male; Membranes; Mice; Mice, Inbred ICR; Naltrexone; Polyunsaturated Alkamides; Receptors, Purinergic P2; Tritium

1994
Gas chromatography/tandem mass spectrometry measurement of delta 9-tetrahydrocannabinol, naltrexone, and their active metabolites in plasma.
    Therapeutic drug monitoring, 1993, Volume: 15, Issue:6

    Topics: Dronabinol; Gas Chromatography-Mass Spectrometry; Humans; Naltrexone; Sensitivity and Specificity

1993
Interactions between delta 9-tetrahydrocannabinol and kappa opioids in mice.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzofurans; Dronabinol; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Mice; Mice, Inbred ICR; Naltrexone; Pyrrolidines; Receptors, Opioid, kappa

1994
Blockade of cannabinoid-induced antinociception by norbinaltorphimine, but not N,N-diallyl-tyrosine-Aib-phenylalanine-leucine, ICI 174,864 or naloxone in mice.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dronabinol; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalins; Infusions, Intravenous; Injections, Spinal; Mice; Naloxone; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta

1993
A role for central cannabinoid and opioid systems in peripheral delta 9-tetrahydrocannabinol-induced analgesia in mice.
    European journal of pharmacology, 1996, Apr-22, Volume: 301, Issue:1-3

    Topics: Analgesics; Animals; Central Nervous System; Dose-Response Relationship, Drug; Dronabinol; Dynorphins; Injections, Intravenous; Male; Mice; Naltrexone; Narcotic Antagonists; Pain Measurement; Peripheral Nervous System; Piperidines; Pyrazoles; Reaction Time; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid; Rimonabant

1996
Potentiation of delta 9-tetrahydrocannabinol-induced analgesia by morphine in mice: involvement of mu- and kappa-opioid receptors.
    European journal of pharmacology, 1996, Dec-27, Volume: 318, Issue:1

    Topics: Analgesia; Analgesics, Opioid; Animals; Binding Sites; Dronabinol; Drug Synergism; Male; Mice; Morphine; Naltrexone; Narcotic Antagonists; Pain Measurement; Receptors, Opioid, kappa; Receptors, Opioid, mu

1996
Characterization of anandamide-induced tolerance: comparison to delta 9-THC-induced interactions with dynorphinergic systems.
    Drug and alcohol dependence, 1997, Apr-14, Volume: 45, Issue:1-2

    Topics: Analgesics; Animals; Arachidonic Acids; Cannabinoids; Cyclohexanols; Dose-Response Relationship, Drug; Dronabinol; Drug Tolerance; Dynorphins; Endocannabinoids; Injections, Intraperitoneal; Injections, Spinal; Mice; Naltrexone; Narcotic Antagonists; Pain Measurement; Polyunsaturated Alkamides; Receptors, Cannabinoid; Receptors, Drug

1997
Cannabinoid modulation of dynorphin A: correlation to cannabinoid-induced antinociception.
    European journal of pharmacology, 1999, Aug-13, Volume: 378, Issue:3

    Topics: Analgesics; Animals; Cannabinoids; Cyclohexanols; Dimethyl Sulfoxide; Dronabinol; Dynorphins; Injections, Spinal; Male; Naltrexone; Narcotic Antagonists; Nociceptors; Pain; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant

1999
Involvement of the opioid system in the anxiolytic-like effects induced by Delta(9)-tetrahydrocannabinol.
    Psychopharmacology, 2002, Volume: 163, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Darkness; Dronabinol; Endorphins; Light; Male; Mice; Naltrexone; Narcotic Antagonists; Piperidines; Pyrazoles; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Rimonabant

2002
Tolerance to the disruptive effects of Delta(9)-THC on learning in rats.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 74, Issue:1

    Topics: Animals; Color Perception; Conditioning, Operant; Dose-Response Relationship, Drug; Dronabinol; Drug Tolerance; Hallucinogens; Learning; Male; Naltrexone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rats, Long-Evans; Reinforcement Schedule; Rimonabant

2002
Dynorphin-independent spinal cannabinoid antinociception.
    Pain, 2002, Volume: 100, Issue:3

    Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Benzoxazines; Dose-Response Relationship, Drug; Dronabinol; Dynorphins; Injections, Spinal; Male; Mice; Mice, Knockout; Morpholines; Naltrexone; Naphthalenes; Pain; Pain Measurement; Reference Values; Reproducibility of Results; Sensitivity and Specificity; Single-Blind Method; Species Specificity; Spinal Cord

2002
The opioid antagonist naltrexone reduces the reinforcing effects of Delta 9 tetrahydrocannabinol (THC) in squirrel monkeys.
    Psychopharmacology, 2004, Volume: 173, Issue:1-2

    Topics: Analgesics, Non-Narcotic; Anesthetics, Local; Animals; Behavior, Animal; Cocaine; Conditioning, Operant; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Male; Naltrexone; Narcotic Antagonists; Reinforcement Schedule; Reinforcement, Psychology; Saimiri; Self Administration

2004
The antinociceptive effect of Delta9-tetrahydrocannabinol in the arthritic rat.
    European journal of pharmacology, 2004, Jun-16, Volume: 493, Issue:1-3

    Topics: Animals; Arthritis, Experimental; Cannabinoid Receptor Antagonists; Dose-Response Relationship, Drug; Dronabinol; Dynorphins; Enkephalin, Leucine; Enkephalin, Methionine; Freund's Adjuvant; Injections, Intradermal; Injections, Intraperitoneal; Male; Morphine; Mycobacterium; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Opioid; Rimonabant

2004
Involvement of mu-, delta- and kappa-opioid receptor subtypes in the discriminative-stimulus effects of delta-9-tetrahydrocannabinol (THC) in rats.
    Psychopharmacology, 2005, Volume: 179, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Benzamides; Conditioning, Operant; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; Food; Hallucinogens; Heroin; Male; Naltrexone; Narcotic Antagonists; Narcotics; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reinforcement, Psychology

2005
Modulation of Delta(9)-THC-induced increase of cortical and hippocampal acetylcholine release by micro opioid and D(1) dopamine receptors.
    Neuropharmacology, 2006, Volume: 50, Issue:6

    Topics: Acetylcholine; Animals; Behavior, Animal; Benzazepines; Dopamine Antagonists; Dronabinol; Drug Interactions; Hippocampus; Male; Microdialysis; Naloxone; Naltrexone; Narcotic Antagonists; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Opioid, mu; Time Factors

2006
Cannabidiol is an allosteric modulator at mu- and delta-opioid receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 372, Issue:5

    Topics: Allosteric Regulation; Analgesics, Opioid; Animals; Cannabidiol; Cerebral Cortex; Dose-Response Relationship, Drug; Dronabinol; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Male; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, mu

2006
Opioid antagonism of cannabinoid effects: differences between marijuana smokers and nonmarijuana smokers.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2007, Volume: 32, Issue:6

    Topics: Adult; Blood Pressure; Cannabinoids; Dronabinol; Female; Hallucinogens; Heart Rate; Humans; Male; Marijuana Smoking; Mental Recall; Methadone; Middle Aged; Naltrexone; Narcotic Antagonists; Narcotics; Psychomotor Performance; Pupil; Recognition, Psychology; Sex Characteristics; Surveys and Questionnaires

2007
Interactions between Delta(9)-tetrahydrocannabinol and mu opioid receptor agonists in rhesus monkeys: discrimination and antinociception.
    Psychopharmacology, 2008, Volume: 199, Issue:2

    Topics: Analgesics; Analgesics, Opioid; Animals; Data Interpretation, Statistical; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Female; Heroin; Hot Temperature; Hypnotics and Sedatives; Macaca mulatta; Male; Midazolam; Morphine; Morphine Dependence; Naltrexone; Narcotic Antagonists; Pain Measurement; Receptors, Opioid, mu; Substance Withdrawal Syndrome

2008
Attenuation of cannabinoid-induced inhibition of medullary dorsal horn neurons by a kappa-opioid receptor antagonist.
    Brain research, 2010, Nov-04, Volume: 1359

    Topics: Animals; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Dronabinol; Male; Medulla Oblongata; Morpholines; Naltrexone; Naphthalenes; Narcotic Antagonists; Patch-Clamp Techniques; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

2010
THC-methadone and THC-naltrexone interactions on discrimination, antinociception, and locomotion in rats.
    Behavioural pharmacology, 2011, Volume: 22, Issue:5-6

    Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Discrimination Learning; Disease Models, Animal; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Locomotion; Male; Methadone; Naltrexone; Narcotic Antagonists; Pain; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

2011
Effect of norbinaltorphimine on ∆⁹-tetrahydrocannabinol (THC)-induced taste avoidance in adolescent and adult Sprague-Dawley rats.
    Psychopharmacology, 2015, Volume: 232, Issue:17

    Topics: Aging; Animals; Appetite Stimulants; Avoidance Learning; Dose-Response Relationship, Drug; Dronabinol; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Taste; Taste Perception

2015
Functional consequences of short-term exposure to opioids versus cannabinoids in nonhuman primates.
    Neuropharmacology, 2023, Feb-01, Volume: 223

    Topics: Analgesics, Opioid; Animals; Cannabinoid Receptor Agonists; Cannabinoids; Dose-Response Relationship, Drug; Dronabinol; Female; Heroin; Male; Morphine; Naltrexone; Rimonabant

2023