naltrexone and diprenorphine

naltrexone has been researched along with diprenorphine in 66 studies

Research

Studies (66)

Timeframe	Studies, this research(%)	All Research%
pre-1990	30 (45.45)	18.7374
1990's	21 (31.82)	18.2507
2000's	11 (16.67)	29.6817
2010's	3 (4.55)	24.3611
2020's	1 (1.52)	2.80

Authors

Authors	Studies
Klein, P; Nelson, WL	1
Portoghese, PS; Takemori, AE	1
Bell, GI; Chen, Y; Kong, H; Raynor, K; Reisine, T; Yasuda, K; Yu, L	1
Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A	1
Strassburg, CP; Tukey, RH	1
Briddon, SJ; Canals, M; Graham, B; Kellam, B; Scammells, PJ; Schembri, LS; Stoddart, LA	1
Herz, A; Höllt, V	1
Colombel, MC; Jacob, J; Tremblay, E	1
Gray, AP; Guardina, WJ	2
Riley, AL; Smurthwaite, ST	2
Caudle, RM; Chavkin, C; Wagner, JJ	1
Geter, B; Kautz, MA; Riley, AL; Smurthwaite, ST	1
Barg, J; Belcheva, MM; Chuang, DM; Coscia, CJ; Gao, XM; McHale, RJ	1
Lawrence, AJ; Traynor, JR	1
Barbas, DP; Portoghese, PS; Song, ZH; Takemori, AE	1
Barg, J; Levy, R; Simantov, R	1
France, CP; Morse, WH	1
Cooper, SJ; Kirkham, TC	1
Kotlińska, J; Langwiński, R	1
Gallagher, M	2
Cho, TM; Nozaki, M	1
Mantegazza, P; Panerai, AE; Sacerdote, P	1
Corbett, AD; Kosterlitz, HW; Traynor, JR	1
Bruzzone, ME; Marusic, ET	1
France, CP; Woods, JH	2
Baskin, DS; Grevel, JC; Hosobuchi, Y	1
Dykstra, LA	1
Bostock, E; Gallagher, M; King, R	1
Freye, E; Hartung, E; Schenk, GK	1
Billington, CJ; Gosnell, BA; Levine, AS; Morley, JE	1
Cheng, RS; Pomeranz, BH	1
Brown, DR; Holtzman, SG; Locke, KW	1
Grevel, J; Sadée, W	1
Herman, BH; Holtzman, SG	1
Gioannini, TL; Hiller, JM; Howard, A; Simon, EJ	1
Katz, RJ; Manik, CP	1
Cooper, SJ; Holtzman, SG	1
Brown, DR; Holtzman, SG	1
Gates, CC; Haigh, JC	1
Chen, C; Chen, YW; Kim de Riel, J; Kunapuli, S; Liu-Chen, LY; Xue, JC; Yu, L; Zhu, J	1
Elliott, J; Lambert, DG; Smart, D; Traynor, JR	1
Chen, C; DeRiel, JK; Kunapuli, S; Liu-Chen, LY; Xue, JC; Yu, L; Zhu, J	1
Lipinsky, D; Oron, Y; Sarne, Y	1
Butour, JL; Meunier, JC; Moisand, C; Mollereau, C; Parmentier, M	1
Kübler, W; Mura, RA; Niroomand, F; Piacentini, L	1
Cheung, P; Li, JG; Liu-Chen, LY; Raffa, RB; Tzeng, TB	1
Clark, MJ; Emmerson, PJ; Medzihradsky, F; Remmers, AE	1
Baamonde, A; Gutiérrez, M; Hidalgo, A; Menéndez, L; SanMartín, S	1
Newman, LC; Stevens, CW; Wallace, DR	1
Cho, KP; Kim, KW; Shin, BS; Son, Y	1
Bahia, DS; Cavalli, A; Hoffmann, M; Massotte, D; Milligan, G; Moon, HE	1
Brillet, K; Bucher, B; Lecat, S; Pattus, F; Perret, BG; Rabut, G; Wagner, R	1
Brown, DR; Townsend, DW	1
Emmerson, PJ; McKinzie, JH; Mitch, CH; Statnick, MA; Surface, PL; Suter, TM	1
Claude-Geppert, PA; Erickson-Herbrandson, LJ; Law, PY; Liu, J; Loh, HH; Solberg, J	1
Holtzman, SG; White, DA	1
Sterious, SN; Walker, EA	1
Luger, P; Messerschmidt, M; Morgenroth, W; Paulmann, C; Scheins, S	1
Howells, RD; Wannemacher, KM; Yadav, PN	1
Diatchenko, L; Ding, F; Dokholyan, NV; Gauthier, J; Gibson, DG; Maixner, W; Serohijos, AW; Yin, S	1
Ingram, SL; Lamberts, JT; Li, MH; Neubig, RR; Smith, CE; Traynor, JR	1
Beytell, P; du Preez, JH; du Preez, P; Felippe, J; Gleed, RD; Jago, M; Kotting, B; Manuel, B; Miller, MA; Morkel, E; Morkel, PV; Parry, SA; Radcliffe, RW	1

Reviews

3 review(s) available for naltrexone and diprenorphine

Article	Year
Human UDP-glucuronosyltransferases: metabolism, expression, and disease. Annual review of pharmacology and toxicology, 2000, Volume: 40 Topics: Autoimmunity; Chromosome Mapping; Glucuronides; Glucuronosyltransferase; Humans; Hyperbilirubinemia; Neoplasms; Steroids; Terminology as Topic	2000
In vivo receptor occupation by opiates and correlation to the pharmacological effect. Federation proceedings, 1978, Volume: 37, Issue:2 Topics: Animals; Binding Sites; Brain; Cerebellum; Diprenorphine; Dose-Response Relationship, Drug; Etorphine; Mice; Naltrexone; Narcotics; Rats; Receptors, Opioid; Stereoisomerism	1978
Behavioral significance of opioid peptides in relation to hippocampal function. NIDA research monograph, 1988, Volume: 82 Topics: Animals; beta-Endorphin; Diprenorphine; Endorphins; Hippocampus; Learning; Memory; Naloxone; Naltrexone; Neurons, Afferent; Spatial Behavior	1988

Trials

1 trial(s) available for naltrexone and diprenorphine

Article	Year
THE PULMONARY AND METABOLIC EFFECTS OF SUSPENSION BY THE FEET COMPARED WITH LATERAL RECUMBENCY IN IMMOBILIZED BLACK RHINOCEROSES (DICEROS BICORNIS) CAPTURED BY AERIAL DARTING. Journal of wildlife diseases, 2021, 04-01, Volume: 57, Issue:2 Topics: Animals; Animals, Wild; Diprenorphine; Energy Metabolism; Etorphine; Female; Hypnotics and Sedatives; Immobilization; Male; Naltrexone; Narcotic Antagonists; Perissodactyla; Posture; Respiratory Physiological Phenomena	2021

Article

Year

THE PULMONARY AND METABOLIC EFFECTS OF SUSPENSION BY THE FEET COMPARED WITH LATERAL RECUMBENCY IN IMMOBILIZED BLACK RHINOCEROSES (DICEROS BICORNIS) CAPTURED BY AERIAL DARTING.

Journal of wildlife diseases, 2021, 04-01, Volume: 57, Issue:2

Topics: Animals; Animals, Wild; Diprenorphine; Energy Metabolism; Etorphine; Female; Hypnotics and Sedatives; Immobilization; Male; Naltrexone; Narcotic Antagonists; Perissodactyla; Posture; Respiratory Physiological Phenomena

2021

Other Studies

62 other study(ies) available for naltrexone and diprenorphine

Article	Year
O3-(2-carbomethoxyallyl) ethers of opioid ligands derived from oxymorphone, naltrexone, etorphine, diprenorphine, norbinaltorphimine, and naltrindole. Unexpected O3-dealkylation in the opioid radioligand displacement assay. Journal of medicinal chemistry, 1992, Nov-27, Volume: 35, Issue:24 Topics: Alkylation; Animals; Brain; Diprenorphine; Drug Stability; Ethers; Etorphine; Guinea Pigs; Indoles; Methacrylates; Molecular Structure; Morphinans; Naltrexone; Narcotic Antagonists; Narcotics; Oxymorphone; Phenols; Radioligand Assay; Receptors, Opioid; Tritium	1992
Different receptor sites mediate opioid agonism and antagonism. Journal of medicinal chemistry, 1983, Volume: 26, Issue:10 Topics: Animals; Binding Sites; Kinetics; Naltrexone; Narcotic Antagonists; Narcotics; Receptors, Opioid; Structure-Activity Relationship	1983
Pharmacological characterization of the cloned kappa-, delta-, and mu-opioid receptors. Molecular pharmacology, 1994, Volume: 45, Issue:2 Topics: Analgesics; Animals; Binding Sites; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; Ligands; PC12 Cells; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Software	1994
Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications. NIDA research monograph, 1998, Volume: 178 Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders	1998
Synthesis, Biological Evaluation, and Utility of Fluorescent Ligands Targeting the μ-Opioid Receptor. Journal of medicinal chemistry, 2015, Dec-24, Volume: 58, Issue:24 Topics: Animals; Binding, Competitive; Buprenorphine; CHO Cells; Cricetulus; Fluorescent Dyes; HEK293 Cells; Humans; Ligands; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Phosphorylation; Radioligand Assay; Receptors, Opioid, mu; Stereoisomerism; Structure-Activity Relationship	2015
[Precipitation and prevention of abstinence in acutely morphinized rats and mice: comparisons between naloxone, naltrexone, and diprenorphine (author's transl)]. Psychopharmacology, 1976, Aug-26, Volume: 49, Issue:1 Topics: Animals; Diprenorphine; Humans; Male; Mice; Morphinans; Morphine; Morphine Dependence; Naloxone; Naltrexone; Rats; Substance Withdrawal Syndrome; Time Factors	1976
Long-acting narcotic antagonist complexes. National Institute on Drug Abuse research monograph series, 1976, Issue:4 Topics: Animals; Brain; Diprenorphine; Methadone; Mice; Morphine; Naltrexone; Narcotic Antagonists; Reaction Time; Time Factors	1976
Long-acting narcotic antagonist complexes. National Institute on Drug Abuse research monograph series, 1975, Issue:4 Topics: Aluminum; Animals; Brain; Buffers; Chemistry, Pharmaceutical; Delayed-Action Preparations; Diprenorphine; Drug Stability; Methadone; Mice; Morphine; Naltrexone; Narcotic Antagonists; Reaction Time; Zinc	1975
Diprenorphine as a stimulus in drug discrimination learning. Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:3 Topics: Animals; Chlorides; Conditioning, Psychological; Diprenorphine; Discrimination Learning; Dose-Response Relationship, Drug; Female; Generalization, Psychological; Lithium; Lithium Chloride; Morphine; Nalorphine; Naloxone; Naltrexone; Pentobarbital; Rats	1992
Kappa-opioids decrease excitatory transmission in the dentate gyrus of the guinea pig hippocampus. The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:1 Topics: Action Potentials; Animals; Benzeneacetamides; Diprenorphine; Dynorphins; Electrophysiology; Endorphins; Guinea Pigs; Hippocampus; Male; Naloxone; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Synapses	1992
Naloxone as a stimulus in drug discrimination learning: generalization to other opiate antagonists. Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:1 Topics: Animals; Cues; Diprenorphine; Discrimination Learning; Female; Generalization, Psychological; Nalorphine; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Saccharin	1992
Up-regulation of delta opioid receptors in neuroblastoma hybrid cells: evidence for differences in the mechanisms of action of sodium butyrate and naltrexone. The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:1 Topics: Binding Sites; Butyrates; Butyric Acid; Cycloheximide; Diprenorphine; Enkephalin, Leucine-2-Alanine; Hybrid Cells; Naltrexone; Neuroblastoma; Receptors, Opioid; Receptors, Opioid, delta; Tumor Cells, Cultured; Up-Regulation	1991
Characterisation of opioid binding sites using selective antagonists. Progress in clinical and biological research, 1990, Volume: 328 Topics: Animals; Binding, Competitive; Brain; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guinea Pigs; In Vitro Techniques; Indoles; Morphinans; Naltrexone; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Somatostatin	1990
Isolation of kappa opioid receptor with an aminoethyl-nor-binaltorphimine (AE-norBNI) affinity column. Progress in clinical and biological research, 1990, Volume: 328 Topics: Animals; Binding, Competitive; Brain Chemistry; Chromatography, Affinity; Diprenorphine; Guinea Pigs; Kinetics; Naltrexone; Receptors, Opioid; Receptors, Opioid, kappa	1990
Paradoxical and subtype-specific effects of opiate antagonists on the expression of opioid receptors in rat brain cultures. Journal of neuroscience research, 1989, Volume: 22, Issue:3 Topics: Adenylyl Cyclases; Animals; Brain; Cells, Cultured; Diprenorphine; Naltrexone; Rats; Rats, Inbred Strains; Receptors, Opioid; Time Factors	1989
Pharmacological characterization of supersensitivity to naltrexone in squirrel monkeys. The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3 Topics: Animals; Azocines; Behavior, Animal; Benzomorphans; Diprenorphine; Drug Administration Schedule; Morphine; Naloxone; Naltrexone; Receptors, Opioid; Saimiri	1989
Adrenalectomy and the anorectic effects of benzodiazepine inverse agonists and opiate antagonists in rats fed a palatable diet. Physiology & behavior, 1987, Volume: 40, Issue:4 Topics: Adrenal Glands; Adrenalectomy; Animals; Appetite; Appetite Depressants; Carbolines; Clonazepam; Diprenorphine; Eating; Hunger; Male; Morphinans; Naltrexone; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taste	1987
Does the blockade of opioid receptors influence the development of ethanol dependence? Alcohol and alcoholism (Oxford, Oxfordshire), 1987, Volume: 22, Issue:2 Topics: Alcoholism; Animals; Diprenorphine; Female; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Seizures; Substance Withdrawal Syndrome	1987
Effects of 5,5'-dithiobis-(2-nitrobenzoic acid) on opiate binding to both the membrane-bound receptor and the partially purified opiate receptor. Journal of neurochemistry, 1985, Volume: 45, Issue:2 Topics: Animals; Butorphanol; Cell Membrane; Dihydromorphine; Diprenorphine; Dithionitrobenzoic Acid; Dithiothreitol; Etorphine; Morphine; Nalorphine; Naloxone; Naltrexone; Nitrobenzoates; Oxymorphone; Rats; Receptors, Opioid	1985
Analgesic effects of mu antagonists after naloxone non-reversible stress-induced analgesia. Brain research, 1985, Dec-16, Volume: 359, Issue:1-2 Topics: Analgesics; Animals; Diprenorphine; Electroshock; Male; Nalorphine; Naloxone; Naltrexone; Pain; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Stress, Physiological	1985
Diprenorphine has agonist activity at opioid kappa-receptors in the myenteric plexus of the guinea-pig ileum. European journal of pharmacology, 1987, May-07, Volume: 137, Issue:1 Topics: Animals; Cricetinae; Diprenorphine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphinans; Muscle Contraction; Myenteric Plexus; Naltrexone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens	1987
Effects of opioid peptides on aldosterone production: stimulatory effect of leu-enkephalin. Endocrinology, 1988, Volume: 122, Issue:2 Topics: Adrenal Cortex; Aldosterone; Animals; Cattle; Diprenorphine; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Naloxone; Naltrexone; Perfusion	1988
Acute supersensitivity to the discriminative stimulus effects of naltrexone in pigeons. The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:2 Topics: Animals; Binding Sites; Columbidae; Diprenorphine; Discrimination Learning; Dose-Response Relationship, Drug; Generalization, Stimulus; Morphine; Nalorphine; Naloxone; Naltrexone; Opioid-Related Disorders	1988
Treatment of experimental stroke with opiate antagonists. Effects on neurological function, infarct size, and survival. Journal of neurosurgery, 1986, Volume: 64, Issue:1 Topics: Animals; Brain Ischemia; Cats; Cerebrovascular Disorders; Consciousness; Diprenorphine; Disease Models, Animal; Male; Morphinans; Movement; Naloxone; Naltrexone; Pupil; Sensation	1986
Effects of buprenorphine on shock titration in squirrel monkeys. The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:1 Topics: Animals; Buprenorphine; Conditioning, Operant; Diprenorphine; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Male; Morphinans; Morphine; Naloxone; Naltrexone; Saimiri	1985
Antagonistic and rate-suppressing effects of opioid antagonists in the pigeon. The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2 Topics: Animals; Azocines; Benzomorphans; Buprenorphine; Columbidae; Conditioning, Operant; Diprenorphine; Dose-Response Relationship, Drug; Morphine; Naloxone; Naltrexone; Narcotic Antagonists	1985
Effects of opiate antagonists on spatial memory in young and aged rats. Behavioral and neural biology, 1985, Volume: 44, Issue:3 Topics: Age Factors; Aging; Animals; Diprenorphine; Male; Memory; Naloxone; Naltrexone; Rats; Space Perception; Stimulation, Chemical	1985
Effects of three narcotic antagonists (naltrexone, diprenorphine, and S-20682) on blood pressure, heart rate and electrical cortical activity. Pharmacology, 1983, Volume: 26, Issue:2 Topics: Animals; Blood Pressure; Carbon Dioxide; Cerebral Cortex; Diprenorphine; Dogs; Electroencephalography; Electrophysiology; Heart Rate; Morphinans; Naltrexone; Narcotic Antagonists; Respiration	1983
Which opioid receptor mechanism modulates feeding? Appetite, 1984, Volume: 5, Issue:1 Topics: Animals; Azocines; Diprenorphine; Dynorphins; Endorphins; Feeding Behavior; Humans; Mice; Naloxone; Naltrexone; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma	1984
Electroacupuncture analgesia is mediated by stereospecific opiate receptors and is reversed by antagonists of type I receptors. Life sciences, 1980, Feb-25, Volume: 26, Issue:8 Topics: Acupuncture Therapy; Analgesia; Animals; Cyclazocine; Diprenorphine; Electric Stimulation; Female; Mice; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Stereoisomerism; Time Factors	1980
Effects of opiate antagonists and putative mu- and kappa-agonists on milk intake in rat and squirrel monkey. Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:6 Topics: Animals; Buprenorphine; Cyclazocine; Diazepam; Diprenorphine; Drinking; Ethylketocyclazocine; Etorphine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Saimiri; Taste	1982
Naloxone enhancement of memory processes: effects of other opiate antagonists. Behavioral and neural biology, 1982, Volume: 35, Issue:4 Topics: Animals; Avoidance Learning; Diprenorphine; Female; Male; Memory; Mental Recall; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Retention, Psychology	1982
An opiate binding site in the rat brain is highly selective for 4,5-epoxymorphinans. Science (New York, N.Y.), 1983, Sep-16, Volume: 221, Issue:4616 Topics: Animals; Brain Chemistry; Dihydromorphine; Diprenorphine; Morphine; Nalorphine; Naloxone; Naltrexone; Rats; Receptors, Opioid; Sodium; Tissue Distribution	1983
Repeated administration of naltrexone and diprenorphine decreases food intake and body weight in squirrel monkeys. Life sciences, 1984, Jan-02, Volume: 34, Issue:1 Topics: Animals; Body Weight; Diprenorphine; Dose-Response Relationship, Drug; Drinking; Eating; Female; Humans; Male; Morphinans; Naloxone; Naltrexone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Saimiri; Salivation	1984
Affinity chromatography of solubilized opioid binding sites using CH-Sepharose modified with a new naltrexone derivative. Biochemical and biophysical research communications, 1984, Mar-15, Volume: 119, Issue:2 Topics: Animals; Bufo marinus; Cattle; Cell Membrane; Chromatography, Affinity; Corpus Striatum; Diprenorphine; Female; Male; Naloxone; Naltrexone; Rats; Rats, Inbred Strains; Receptors, Opioid; Sepharose	1984
Endogenous opiates and stress. Behavioral activation elicited in the rat and effects of naltrexone, diprenorphine and morphine. Neuropharmacology, 1984, Volume: 23, Issue:12A Topics: Animals; Behavior, Animal; Diprenorphine; Endorphins; Humans; Male; Morphinans; Morphine; Naloxone; Naltrexone; Noise; Rats; Rats, Inbred Strains; Receptors, Drug; Stress, Psychological; Time Factors	1984
Patterns of drinking in the rat following the administration of opiate antagonists. Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:3 Topics: Animals; Depression, Chemical; Diprenorphine; Drinking Behavior; Male; Morphinans; Naloxone; Naltrexone; Rats; Rats, Inbred Strains; Water Deprivation	1983
Narcotic antagonists attenuate drinking induced by water deprivation in a primate. Life sciences, 1981, Mar-16, Volume: 28, Issue:11 Topics: Animals; Diprenorphine; Dose-Response Relationship, Drug; Drinking Behavior; Male; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Saimiri; Water Deprivation	1981
Capture of wood bison (Bison bison athabascae) using carfentanil-based mixtures. Journal of wildlife diseases, 1995, Volume: 31, Issue:1 Topics: Analgesics, Opioid; Animals; Bison; Diprenorphine; Drug Combinations; Female; Fentanyl; Hypnotics and Sedatives; Immobilization; Injections, Intramuscular; Injections, Intravenous; Injections, Subcutaneous; Male; Naloxone; Naltrexone; Narcotic Antagonists; Northwest Territories; Piperidines; Tranquilizing Agents; Xylazine	1995
Characterization of irreversible binding of beta-funaltrexamine to the cloned rat mu opioid receptor. The Journal of biological chemistry, 1995, Jul-28, Volume: 270, Issue:30 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Amino Acid Sequence; Animals; Cell Line; Cloning, Molecular; Diprenorphine; Electrophoresis, Polyacrylamide Gel; Enkephalin, Leucine; Glycosylation; Molecular Sequence Data; Naltrexone; Oligopeptides; Protein Binding; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Recombinant Proteins; Sodium; Tritium	1995
Characterisation of mu-opioid receptors on SH-SY5Y cells using naloxonazine and beta-funaltrexamine. European journal of pharmacology, 1994, Aug-16, Volume: 268, Issue:3 Topics: Amino Acid Sequence; Animals; Brain Neoplasms; Cerebral Cortex; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Humans; Ligands; Molecular Sequence Data; Naloxone; Naltrexone; Neuroblastoma; Rats; Receptors, Opioid, mu; Somatostatin; Tumor Cells, Cultured	1994
Nalorphine as a stimulus in drug discrimination learning: assessment of the role of mu- and kappa-receptor subtypes. Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:3 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Diprenorphine; Discrimination Learning; Dose-Response Relationship, Drug; Female; Generalization, Stimulus; Nalorphine; Naloxone; Naltrexone; Pyrrolidines; Rats; Receptors, Opioid, kappa; Receptors, Opioid, mu	1994
Differential binding domains of peptide and non-peptide ligands in the cloned rat kappa opioid receptor. The Journal of biological chemistry, 1994, Dec-02, Volume: 269, Issue:48 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Amino Acid Sequence; Animals; Base Sequence; Benzeneacetamides; Binding Sites; Binding, Competitive; Cell Line; Chlorocebus aethiops; Cloning, Molecular; Diprenorphine; DNA Primers; Dynorphins; Endorphins; Kinetics; Ligands; Molecular Sequence Data; Naltrexone; Polymerase Chain Reaction; Protein Conformation; Protein Structure, Secondary; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Recombinant Fusion Proteins; Transfection	1994
Morphine inhibits calcium influx and the response to acetylcholine in Xenopus oocytes. Journal of neurochemistry, 1993, Volume: 60, Issue:1 Topics: Acetylcholine; Animals; Calcium; Diprenorphine; Electrophysiology; Female; Morphine; Muscarine; Naltrexone; Oocytes; Radioligand Assay; Xenopus laevis	1993
Replacement of Gln280 by His in TM6 of the human ORL1 receptor increases affinity but reduces intrinsic activity of opioids. FEBS letters, 1996, Oct-14, Volume: 395, Issue:1 Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Diprenorphine; Dynorphins; Etorphine; Fentanyl; Glutamine; Histamine; Humans; Kinetics; Ligands; Naltrexone; Narcotic Antagonists; Narcotics; Nociceptin; Nociceptin Receptor; Opioid Peptides; Receptors, Opioid	1996
Opioid receptor agonists activate pertussis toxin-sensitive G proteins and inhibit adenylyl cyclase in canine cardiac sarcolemma. Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:5 Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Analgesics; Analysis of Variance; Animals; Diprenorphine; Dogs; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GTP Phosphohydrolases; GTP-Binding Proteins; Myocardium; Naltrexone; Narcotic Antagonists; Pertussis Toxin; Sarcolemma; Virulence Factors, Bordetella	1996
Apparent thermodynamic parameters of ligand binding to the cloned rat mu-opioid receptor. European journal of pharmacology, 1998, Aug-07, Volume: 354, Issue:2-3 Topics: Analgesics; Animals; Binding, Competitive; CHO Cells; Cricetinae; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; Ligands; Methadone; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Peptide Fragments; Peptides; Radioligand Assay; Rats; Receptors, Opioid, mu; Somatostatin; Sufentanil; Thermodynamics; Time Factors	1998
Membrane microviscosity modulates mu-opioid receptor conformational transitions and agonist efficacy. Journal of neurochemistry, 1999, Volume: 73, Issue:1 Topics: Animals; Cell Line; Cell Membrane; Cholesterol Esters; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Glioma; Guanosine 5'-O-(3-Thiotriphosphate); Membrane Fluidity; Nalbuphine; Naltrexone; Narcotic Antagonists; Narcotics; Neuroblastoma; Protein Conformation; Rats; Receptors, Opioid, mu; Sodium Chloride; Sufentanil; Tumor Cells, Cultured; Viscosity	1999
Effects of diethylstilbestrol on mouse hippocampal evoked potentials in vitro. Cellular and molecular neurobiology, 1999, Volume: 19, Issue:6 Topics: Animals; Binding, Competitive; Dactinomycin; Diethylstilbestrol; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estrogens; Excitatory Postsynaptic Potentials; Hippocampus; Male; Mice; Naloxone; Naltrexone; Narcotic Antagonists; Nerve Tissue Proteins; Pyramidal Cells; Receptors, Opioid; Receptors, Opioid, mu	1999
Characterization of [3H]-diprenorphine binding in Rana pipiens: observations of filter binding enhanced by naltrexone. Journal of pharmacological and toxicological methods, 1999, Volume: 41, Issue:1 Topics: Animals; Binding, Competitive; Brain; Diprenorphine; Dose-Response Relationship, Drug; Drug Interactions; Filtration; Naltrexone; Narcotic Antagonists; Rana pipiens	1999
Pharmacological effects of naltriben as a ligand for opioid mu and kappa receptors in rat cerebral cortex. Life sciences, 2001, Feb-02, Volume: 68, Issue:11 Topics: Animals; Cerebral Cortex; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Ligands; Male; Naloxone; Naltrexone; Narcotic Antagonists; Norepinephrine; Peptide Fragments; Peptides; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Somatostatin; Tritium	2001
The human delta opioid receptor activates G(i1)alpha more efficiently than G(o1)alpha. Journal of neurochemistry, 2001, Volume: 76, Issue:6 Topics: Adenylyl Cyclases; Cell Line; Colforsin; Diprenorphine; Enkephalin, Leucine-2-Alanine; GTP Phosphohydrolases; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine Triphosphate; Heterotrimeric GTP-Binding Proteins; Humans; Kinetics; Naltrexone; Polymerase Chain Reaction; Receptors, Opioid, delta; Recombinant Fusion Proteins; Recombinant Proteins; Transfection	2001
Expression of EGFP-amino-tagged human mu opioid receptor in Drosophila Schneider 2 cells: a potential expression system for large-scale production of G-protein coupled receptors. Protein expression and purification, 2003, Volume: 31, Issue:1 Topics: Animals; Binding, Competitive; Blotting, Western; Cell Line; Cloning, Molecular; Colforsin; Copper Sulfate; Cyclic AMP; Diprenorphine; DNA, Complementary; Drosophila; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Gene Expression; Genetic Vectors; Green Fluorescent Proteins; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Luminescent Proteins; Metallothionein; Microscopy, Confocal; Morphine; Naloxone; Naltrexone; Oligopeptides; Opioid Peptides; Pertussis Toxin; Polymerase Chain Reaction; Protein Binding; Receptors, G-Protein-Coupled; Receptors, Opioid, mu; Recombinant Fusion Proteins; Spectrometry, Fluorescence; Thermodynamics	2003
Pharmacological characterization of a 7-benzylidenenaltrexone-preferring opioid receptor in porcine ileal submucosa. British journal of pharmacology, 2003, Volume: 140, Issue:4 Topics: Amphibian Proteins; Animals; Anions; Benzamides; Benzylidene Compounds; Biological Transport, Active; Carrier Proteins; Diprenorphine; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Female; Gastrointestinal Motility; Ileum; Intestinal Mucosa; Male; Naltrexone; Neurons, Afferent; Oligopeptides; Piperazines; Quinolines; Receptors, Opioid, delta; Receptors, Opioid, mu; Swine; Tritium	2003
Na+ modulation, inverse agonism, and anorectic potency of 4-phenylpiperidine opioid antagonists. European journal of pharmacology, 2004, Jun-28, Volume: 494, Issue:2-3 Topics: Animals; Appetite Depressants; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Cyclohexanes; Diprenorphine; Dose-Response Relationship, Drug; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Guanosine 5'-O-(3-Thiotriphosphate); Ligands; Naltrexone; Narcotic Antagonists; Piperidines; Radioligand Assay; Rats; Rats, Zucker; Receptors, Opioid; Receptors, Opioid, delta; Sodium	2004
Antagonist efficacy in MORS196L mutant is affected by the interaction between transmembrane domains of the opioid receptor. The Journal of pharmacology and experimental therapeutics, 2005, Volume: 313, Issue:1 Topics: Animals; Cyclic AMP; Diprenorphine; Electrophysiology; Mutagenesis, Site-Directed; Mutation; Naloxone; Naltrexone; Narcotic Antagonists; Oocytes; Patch-Clamp Techniques; Radioligand Assay; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Recombinant Fusion Proteins; RNA, Complementary; Xenopus	2005
Discriminative stimulus effects of acute morphine followed by naltrexone in the squirrel monkey: a further characterization. The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:1 Topics: Analgesics, Opioid; Animals; Buprenorphine; Diprenorphine; Discrimination, Psychological; Dose-Response Relationship, Drug; Drinking; Drug Interactions; Generalization, Stimulus; Male; Meperidine; Mice; Morphine; Nalbuphine; Nalorphine; Naltrexone; Narcotic Antagonists; Saimiri; Water Deprivation	2005
Opioid antagonists differ according to negative intrinsic efficacy in a mouse model of acute dependence. British journal of pharmacology, 2005, Volume: 145, Issue:7 Topics: Animals; Behavior, Animal; Body Weight; Brain; Diprenorphine; Dose-Response Relationship, Drug; Male; Mice; Morphine; Morphine Dependence; Naloxone; Naltrexone; Narcotic Antagonists; Substance Withdrawal Syndrome; Tremor	2005
Electron density analyses of opioids: a comparative study. The journal of physical chemistry. A, 2007, Jun-28, Volume: 111, Issue:25 Topics: Analgesics, Opioid; Codeine; Cold Temperature; Dextromethorphan; Diprenorphine; Electrons; Models, Molecular; Morphine; Naltrexone; X-Ray Diffraction	2007
A select set of opioid ligands induce up-regulation by promoting the maturation and stability of the rat kappa-opioid receptor in human embryonic kidney 293 cells. The Journal of pharmacology and experimental therapeutics, 2007, Volume: 323, Issue:2 Topics: Animals; Benzeneacetamides; Brefeldin A; Cells, Cultured; Cycloheximide; Diprenorphine; Humans; Ligands; Naloxone; Naltrexone; Pyrrolidines; Rats; Receptors, Opioid, kappa; RNA, Messenger; Transfection; Up-Regulation	2007
Structural basis for μ-opioid receptor binding and activation. Structure (London, England : 1993), 2011, Nov-09, Volume: 19, Issue:11 Topics: Amino Acid Substitution; Animals; Binding Sites; Binding, Competitive; Cattle; Cyclic AMP; Databases, Factual; Decapodiformes; Diprenorphine; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Molecular Dynamics Simulation; Morphine; Mutagenesis, Site-Directed; Naltrexone; Protein Binding; Radioligand Assay; Receptors, Opioid, mu; Small Molecule Libraries	2011
Differential control of opioid antinociception to thermal stimuli in a knock-in mouse expressing regulator of G-protein signaling-insensitive Gαo protein. The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Mar-06, Volume: 33, Issue:10 Topics: Analgesics, Opioid; Animals; Brain; Diprenorphine; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine 5'-O-(3-Thiotriphosphate); Hot Temperature; Humans; Hyperalgesia; Inhibitory Postsynaptic Potentials; Isotopes; Male; Methadone; Mice; Mice, Transgenic; Morphine; Mutation; Naloxone; Naltrexone; Narcotic Antagonists; Neurons; Oligopeptides; Pain Measurement; Patch-Clamp Techniques; Pertussis Toxin; Protein Binding; Reaction Time; RGS Proteins; Signal Transduction; Spinal Cord	2013