naltrexone and cocaine

naltrexone has been researched along with cocaine in 147 studies

Research

Studies (147)

TimeframeStudies, this research(%)All Research%
pre-199011 (7.48)18.7374
1990's50 (34.01)18.2507
2000's37 (25.17)29.6817
2010's38 (25.85)24.3611
2020's11 (7.48)2.80

Authors

AuthorsStudies
Carroll, FI1
Jolivette, LJ; Ward, KW1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Blumberg, H; Ikeda, C1
Masukawa, Y; Misawa, M; Nagase, H; Shiozaki, Y; Suzuki, T1
Doty, P; Dykstra, LA; Johnson, AB; Picker, MJ1
Bilsky, EJ; Menkens, K; Porreca, F; Portoghese, PS; Reid, LD; Wild, KD1
Byck, R; Compton, M; Fleming, J; Gawin, FH; Jatlow, P; Kosten, T; Kosten, TA; Silverman, DG1
Bilsky, EJ; Delong, CL; Montegut, MJ; Reid, LD1
Goldberg, SR; Grayson, NA; Jaffe, JH; Johnson, RE; Katz, JL; Rice, KC; Witkin, JM1
Bansinath, M; Goldfrank, LR; Shukla, VK; Turndorf, H1
Ramsey, NF; van Ree, JM2
Mello, NK1
Kamien, JB; Lukas, SE; Mello, NK; Mendelson, JH1
Coen, KM; Corrigall, WA1
Bree, MP; Lukas, SE; Mello, NK; Mendelson, JH1
Schuster, CR; Snyder, M1
De Vry, J; Donselaar, I; Van Ree, JM1
Winger, G1
Kleber, HD; Kosten, TR; Morgan, C1
Mello, NK; Mendelson, JH1
Corrigall, WA; Vaccarino, FJ1
Williams, A1
Carroll, ME; Kragh, R; Lac, ST; Newman, T; Walker, MJ1
Bloom, FE; Ettenberg, A; Koob, GF; Pettit, HO1
Dackis, CA; Gold, MS1
Bilsky, EJ; French, ED; Glick, SD; Menkens, KA; Porreca, F; Reid, LD1
Heidbreder, C; Shippenberg, TS1
Archer, S; Glick, SD; Maisonneuve, IM; Raucci, J1
Braida, D; Colombo, M; Gori, E; Groppetti, A; Parenti, M; Sacco, S; Sala, M1
Funada, M; Misawa, M; Mori, T; Nagase, H; Suzuki, T1
Archer, S; Glick, SD; Maisonneuve, IM1
Carroll, ME; Comer, SD; Curtis, LK; Lac, ST1
Misawa, M; Mori, T; Nagase, H; Suzuki, T; Tsuji, M1
Kameyama, T; Mizutani, M; Ukai, M1
Goldberg, SR; Heidbreder, C; Shippenberg, TS1
Drieze, J; Lukas, SE; Mello, NK; Mendelson, JH1
Bowen, WD; Holtzman, SG; Jones, DN; Portoghese, PS1
Acquas, E; Di Chiara, G; Meloni, M1
Bilsky, EJ; Glaccum, MB; Hubbell, CL; Porreca, F; Portoghese, PS; Reid, LD1
Kameyama, T; Mori, E; Ukai, M1
Babovic-Vuksanovic, D; de Vries, TJ; Elmer, G; Shippenberg, TS1
France, CP; Gerak, LR1
Heidbreder, C; LeFevour, A; Shippenberg, TS1
Dworkin, SI; Hemby, SE; Smith, JE1
Heidbreder, C; Shippenberg, TS; Shoaib, M1
Cox, BM; Izenwasser, S; Katz, JL; Newman, AH1
Bigelow, GE; Garner, JE; Preston, KL; Sullivan, JT; Walsh, SL1
Litten, RZ1
Cramer, CM; Hubbell, CL; Pabello, NG; Reid, LD1
Lin, CE; Mello, NK; Negus, SS; Portoghese, PS1
Holtzman, SG; Kimmel, HL1
Gordon, FJ; Holtzman, SG; Patterson, AB1
Boedeker, KL; Cramer, CM; Gardell, LR; Harris, JR; Hubbell, CL; Reid, LD1
Rowlett, JK; Wilcox, KM; Woolverton, WL1
Cramer, CM; Hubbell, CL; Reid, LD1
DeMontis, MG; Dworkin, SI; Kim, SA; Martin, TJ; Sizemore, GM; Smith, JE1
Gerrits, MA; Kuzmin, AV; Van Ree, JM1
Brodkin, ES; Carlezon, WA; Duman, RS; Hiroi, N; Lane-Ladd, SB; Nestler, EJ; Neve, RL; Olson, VG; Thome, J1
Anders, KA; Czapiga, M; Dallman, E; Kruschel, CK; Mitchem, LD; Panos, JJ; Steinpreis, RE1
Hersh, D; Kranzler, HR; Mulgrew, CL; Van Kirk, J1
Gerrits, MA; Ramsey, NF; Van Ree, JM1
Grech, DM; Platt, DM; Rowlett, JK; Spealman, RD1
Platt, DM; Rowlett, JK; Spealman, RD1
Mello, NK; Negus, SS1
Bian, D; Cannon, DG; Kim, SA; Martin, TJ; Porreca, F; Sizemore, GM; Smith, JE1
Justice, JB; Sharpe, LG; Shippenberg, TS; Thompson, AC; Vaughan, RA; Zapata, A1
Collins, SL; D'Addario, C; Gerdes, RM; Izenwasser, S1
France, CP; Sell, SL1
Mackler, SA; O'Brien, CP; Sengpiel, T; Stromberg, MF; Vogel, WH; Volpicelli, JR1
Chavkin, C; Marton-Popovici, M; McLaughlin, JP1
Martin, TJ; Roberts, DC; Ward, SJ1
France, CP; McMahon, LR; Sell, SL1
Izenwasser, S; Platt, DM; Rowlett, JK; Spealman, RD1
Goldberg, SR; Justinova, Z; Munzar, P; Tanda, G1
Butelman, ER; Ho, A; Kreek, MJ; Schlussman, SD; Zhang, Y1
Ansonoff, MA; Hummel, M; Pintar, JE; Unterwald, EM1
Negus, SS1
Alekseyenko, OV; Bondar, NP; Burbach, JP; Gerrits, MA; Hordijk, M; Lesscher, HM; van Ree, JM1
Sable, HJ; Steinpreis, RE; White, SL1
France, CP; Koek, W; McMahon, LR; Sell, SL1
Chavkin, C; Chavkin, TA; Li, S; McLaughlin, JP; Valdez, J1
Fantoma, A; Gerra, G; Zaimovic, A1
Chefer, VI; Shippenberg, TS1
Comer, SD; Dackis, C; Kampman, K; Kleber, HD; O'Brien, CP; Rothenberg, JL; Sullivan, MA; Yu, E1
Le Merrer, J; Stephens, DN1
Jasmin, L; Narasaiah, M; Tien, D1
Kaminski, RM; Shippenberg, TS; Witkin, JM1
Antonilli, L; Cioce, AM; Giudici, FD; Grassi, MC; Nencini, P1
Bienkowski, P; Kostowski, W; Mierzejewski, P; Stefanski, R1
Roberts, DC; Ward, SJ1
Co, C; Coller, M; Martin, TJ; Smith, JE1
Ding, Z; Phillips, AG; Powell, JA; Raffa, RB; Rawls, SM; Ross, G; Stagliano, GW1
Antapasis, J; Bolaños Guzmán, CA; Herrera, CM; Poveromo, LB; Wiley, MD1
Achat-Mendes, C; Platt, DM; Rowlett, JK; Spealman, RD; Valdez, GR1
Cashman, JR; Ghirmai, S; Koob, GF; Orio, L; Wee, S1
Di Paolo, T; Grégoire, L; Lévesque, D; Morissette, M; Ouattara, B; Rouillard, C; Samadi, P; Tamim, MK1
Aita, M; Bruchas, MR; Chavkin, C; Giardino, WJ; Hnasko, TS; Land, BB; Messinger, D; Palmiter, RD; Schattauer, S1
Chavkin, C; Li, S; Schindler, AG1
Chung, NN; Gibula-Bruzda, E; Izdebski, J; Kotlinska, JH; Kunce, D; Pachuta, A; Schiller, PW; Witkowska, E1
Dong, Y; Mu, P; Neumann, PA; Panksepp, J; Schlüter, OM1
Aklin, WM; Bigelow, GE; DeFulio, A; Donlin, WD; Everly, JJ; Fingerhood, M; Koffarnus, MN; Leoutsakos, JM; Silverman, K; Umbricht, A1
Carlezon, WA; Chartoff, E; Pliakas, A; Potter, D; Rachlin, A; Sawyer, A1
Carlezon, WA; Chartoff, EH; Cohen, BM; Damez-Werno, D; Potter, DN1
Chudnovskaya, D; Cowan, A; Huang, P; Liu-Chen, LY; Rasakham, K; Wang, YJ1
Friedman, TC; Hamid, A; Kieffer, B; Lutfy, K; Marquez, P; Nguyen, AT1
Bühler, KM; Echeverry-Alzate, V; Giné, E; Gorriti, MÁ; Huertas, E; López-Moreno, JA; Olmos, P; Rodríguez de Fonseca, F; Santos, Á; Tuda-Arízcun, M1
Koob, GF; Misra, KK; Schlosburg, JE; Vendruscolo, LF; Wee, S1
Allen, CP; Leri, F; Zhou, Y1
Chavkin, C; Chavkin, NW; Gustin, RM; Hagan, CE; Lemos, JC; Messinger, DI; Neumaier, JF; Schattauer, SS; Schindler, AG; Shankar, H; Smith, JS1
Bailey, CP; Cordery, SF; Delgado-Charro, MB; Guy, RH; Husbands, SM; Ridzwan, IE; Taverner, A1
Agovic, MS; Banerjee, SP; Chan, CY; Friedman, E; Jashanmal, I; Ragnauth, A; Sostris, V; Vidal, L1
Askalsky, P; Berkower, EL; Comer, SD; Cooper, ZD; Foltin, RW; Haney, M; Jones, JD; Manubay, JM; Martinez, D; Mogali, S; Pines, A; Roux, P; Rubin, E; Saccone, PA; Sullivan, MA; Vosburg, SK; Walker, EA1
Al-Hasani, R; Bruchas, MR; Foshage, AM; McCall, JG1
Gibula-Bruzda, E; Izdebski, J; Kotlinska, JH; Witkowska, E1
Clark, JK; Hammond, S; Keralapurath, MM; Wagner, JJ1
Chavkin, C; Groblewski, PA; Phillips, PE; Willuhn, I; Zietz, C1
Banks, ML; Cheng, K; Hutsell, BA; Negus, SS; Rice, KC1
Abbott, S; Boyapati, V; Deakin, JF; Elliott, R; Erritzoe, D; Ersche, KD; Faluyi, Y; Faravelli, L; Fernandez-Egea, E; Flechais, RS; Kalk, NJ; Kuchibatla, SS; Lingford-Hughes, AR; McGonigle, J; Metastasio, A; Mick, I; Murphy, A; Nestor, L; Nutt, DJ; Orban, C; Passetti, F; Paterson, LM; Rabiner, EA; Reed, LJ; Robbins, TW; Smith, DG; Suckling, J; Tait, R; Taylor, EM; Waldman, AD1
Eans, SO; Ganno, ML; Hunkele, A; Le Rouzic, V; Majumdar, S; Marrone, GF; McLaughlin, JP; Pasternak, GW; Subrath, JJ; Váradi, A1
de Carvalho, CR; Takahashi, RN1
Bühler, KM; Calleja-Conde, J; Echeverry-Alzate, V; Giné, E; Gual, A; López-Moreno, JA; Maldonado, R; Nadal, R; Rodríguez de Fonseca, F1
Coggiano, M; Hiranita, T; Katz, JL; Mereu, M; Quarterman, JC; Tanda, G1
Bardo, MT; Beckmann, JS; Hofford, RS1
Camirand-Lemyre, F; Desharnais, B; Mireault, P; Skinner, CD1
Bigelow, GE; DeFulio, A; Fingerhood, M; Holtyn, AF; Jarvis, BP; Long, L; Silverman, K; Umbricht, A1
Ciccocioppo, R; de Guglielmo, G; Journigan, VB; Kallupi, M; Shen, Q; Yasuda, D; Zaveri, NT1
Banks, ML; Cheng, K; Moerke, MJ; Negus, SS; Rice, KC1
George, O; Kallupi, M; Martin-Fardon, R; Matzeu, A; Schweitzer, P1
Negus, SS; Sakloth, F1
Kreek, MJ; Reed, B; Windisch, KA1
Giancola, JB; Keighron, JD; Lin, SC; Newman, AH; Scaglione, A; Tanda, G; Zanettini, C1
Bigelow, GE; DeFulio, A; Fingerhood, M; Holtyn, AF; Jarvis, BP; Koffarnus, MN; Leoutsakos, JS; Silverman, K; Umbricht, A1
Carson, RE; Chang, D; Foltin, R; Grassetti, A; Huang, Y; Lin, SF; Martinez, D; Matuskey, D; Nabulsi, N; Ropchan, J; Salling, M; Slifstein, M; Urban, N; Zheng, MQ1
Freeman, KB; Huskinson, SL; Naylor, JE; Prisinzano, TE; Townsend, EA; Zamarripa, CA1
Ayers, C; Chan, B; Freeman, M; Kansagara, D; Kondo, K; Korthuis, PT; Paynter, R1
Azar, MR; Cunningham, JI; Dean, RL; Deaver, DR; Eyerman, DJ; Koob, GF; Todtenkopf, MS1
Kreek, MJ; Morochnik, M; Reed, B; Windisch, KA1
Hallahan, JE; Hillhouse, TM; Husbands, SM; Jutkiewicz, EM; Koppenhaver, PO; Meurice, C; Olson, KM; Ostovar, M; Rysztak, LG; Sears, BF; Traynor, JR; West, JL1
Graham, DP; Hamon, SC; Hillhouse, M; Kosten, TR; Lawson, WB; Ling, W; Nielsen, DA; Nielsen, EM; Rotrosen, J; Saxon, AJ; Settles-Reaves, BD; Shmueli-Blumberg, D; Shores-Wilson, K; Trivedi, MH; Walker, R1
Cami-Kobeci, G; Cippitelli, A; Husbands, SM; Martinez, M; Toll, L; Zribi, G1
Cippitelli, A; Toll, L; Zribi, G1
Alcorn, JL; Bolin, BL; Hays, LR; Lile, JA; Rayapati, AO; Regnier, SD; Reynolds, AR; Rush, CR; Stoops, WW1
Bachtell, RK; Brown, KT; Levis, SC; Levy, C; O'Neill, CE; Rice, KC; Watkins, LR1
Balise, RR; Castillo, F; Feaster, DJ; Hu, MC; Liu, Y; Luo, SX; Nunes, EV; Rotrosen, J; Saxon, AJ; Weiss, RD1

Reviews

7 review(s) available for naltrexone and cocaine

ArticleYear
2002 Medicinal Chemistry Division Award address: monoamine transporters and opioid receptors. Targets for addiction therapy.
    Journal of medicinal chemistry, 2003, May-08, Volume: 46, Issue:10

    Topics: Animals; Biogenic Monoamines; Biological Transport; Carrier Proteins; Cocaine; Fluorescent Dyes; Humans; Isoquinolines; Ligands; Morphinans; Narcotic Antagonists; Piperidines; Protein Binding; Radioisotopes; Receptors, Opioid; Structure-Activity Relationship; Substance-Related Disorders

2003
Preclinical evaluation of the effects of buprenorphine, naltrexone and desipramine on cocaine self-administration.
    NIDA research monograph, 1990, Volume: 105

    Topics: Animals; Buprenorphine; Cocaine; Desipramine; Humans; Macaca mulatta; Naltrexone; Self Administration

1990
Pharmacological modifications of cocaine and opioid self-administration.
    NIDA research monograph, 1988, Volume: 88

    Topics: Animals; Chlorpromazine; Cocaine; Naltrexone; Narcotics; Receptors, Dopamine; Receptors, Opioid; Reinforcement, Psychology; Self Administration

1988
Clinical investigations of drug effects in women.
    NIDA research monograph, 1986, Volume: 65

    Topics: Buprenorphine; Cocaine; Desipramine; Female; Heroin Dependence; Humans; Male; Naltrexone; Opioid-Related Disorders; Sex Factors; Substance-Related Disorders

1986
New insights and treatments: opiate withdrawal and cocaine addiction.
    Clinical therapeutics, 1984, Volume: 7, Issue:1

    Topics: Brain Chemistry; Clonidine; Cocaine; Dopamine; Humans; Methadone; Naltrexone; Norepinephrine; Substance Withdrawal Syndrome; Substance-Related Disorders

1984
Interactions between kappa opioid agonists and cocaine. Preclinical studies.
    Annals of the New York Academy of Sciences, 2000, Volume: 909

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Psychological; Discrimination Learning; Humans; Naloxone; Naltrexone; Receptors, Opioid, kappa; Self Administration

2000
A systematic review and meta-analysis of medications for stimulant use disorders in patients with co-occurring opioid use disorders.
    Drug and alcohol dependence, 2020, 11-01, Volume: 216

    Topics: Analgesics, Opioid; Antidepressive Agents; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Female; Humans; Methadone; Naltrexone; Opioid-Related Disorders

2020

Trials

11 trial(s) available for naltrexone and cocaine

ArticleYear
Intravenous cocaine challenges during naltrexone maintenance: a preliminary study.
    Biological psychiatry, 1992, Sep-15, Volume: 32, Issue:6

    Topics: Adult; Blood Pressure; Cocaine; Double-Blind Method; Female; Heart Rate; Humans; Male; Naltrexone; Placebo Effect; Substance Abuse, Intravenous

1992
Effects of naltrexone on response to intravenous cocaine, hydromorphone and their combination in humans.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:2

    Topics: Adult; Buprenorphine; Cocaine; Cross-Over Studies; Double-Blind Method; Drug Interactions; Humans; Hydromorphone; Liver; Male; Naltrexone; Narcotic Antagonists; Narcotics; Respiration; Substance-Related Disorders

1996
The validity of self-reported cocaine use in two groups of cocaine abusers.
    Journal of consulting and clinical psychology, 1999, Volume: 67, Issue:1

    Topics: Adult; Carbamazepine; Cocaine; Cocaine-Related Disorders; Double-Blind Method; Female; Humans; Interview, Psychological; Male; Naltrexone; Predictive Value of Tests; Psychometrics; Reproducibility of Results; Self Disclosure; Substance Abuse Detection

1999
Injectable, sustained-release naltrexone for the treatment of opioid dependence: a randomized, placebo-controlled trial.
    Archives of general psychiatry, 2006, Volume: 63, Issue:2

    Topics: Adolescent; Adult; Cocaine; Delayed-Action Preparations; Double-Blind Method; Drug Administration Schedule; Female; Heroin Dependence; Humans; Injections, Subcutaneous; Male; Methadone; Middle Aged; Naltrexone; Narcotics; Placebos; Secondary Prevention; Substance Abuse Detection; Treatment Outcome

2006
Short-term efficacy of Disulfiram or Naltrexone in reducing positive urinalysis for both cocaine and cocaethylene in cocaine abusers: a pilot study.
    Pharmacological research, 2007, Volume: 55, Issue:2

    Topics: Adult; Cocaine; Cocaine-Related Disorders; Cognitive Behavioral Therapy; Combined Modality Therapy; Disulfiram; Humans; Naltrexone; Narcotic Antagonists; Patient Compliance; Pilot Projects; Time Factors; Treatment Outcome

2007
Employment-based reinforcement of adherence to depot naltrexone in unemployed opioid-dependent adults: a randomized controlled trial.
    Addiction (Abingdon, England), 2011, Volume: 106, Issue:7

    Topics: Adolescent; Adult; Aged; Analgesics, Opioid; Cocaine; Delayed-Action Preparations; Dopamine Uptake Inhibitors; Employment; Female; Humans; Injections, Subcutaneous; Male; Medication Adherence; Middle Aged; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Outcome Assessment, Health Care; Reinforcement, Psychology; Salaries and Fringe Benefits; Young Adult

2011
Effects of acute oral naltrexone on the subjective and physiological effects of oral D-amphetamine and smoked cocaine in cocaine abusers.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2013, Volume: 38, Issue:12

    Topics: Administration, Oral; Adult; Cardiovascular System; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Cross-Over Studies; Dextroamphetamine; Dopamine Uptake Inhibitors; Double-Blind Method; Female; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Smoking

2013
The Imperial College Cambridge Manchester (ICCAM) platform study: An experimental medicine platform for evaluating new drugs for relapse prevention in addiction. Part A: Study description.
    Journal of psychopharmacology (Oxford, England), 2015, Volume: 29, Issue:9

    Topics: Adult; Behavior, Addictive; Biomedical Research; Brain; Cocaine; Cross-Over Studies; Drug Discovery; Ethanol; Female; Humans; Impulsive Behavior; Magnetic Resonance Imaging; Male; Middle Aged; Naltrexone; Neurokinin-1 Receptor Antagonists; Pharmaceutical Preparations; Receptors, Dopamine D3; Receptors, Neurokinin-1; Reward; Secondary Prevention; Substance-Related Disorders

2015
The effects of extended-release injectable naltrexone and incentives for opiate abstinence in heroin-dependent adults in a model therapeutic workplace: A randomized trial.
    Drug and alcohol dependence, 2019, 04-01, Volume: 197

    Topics: Adult; Black or African American; Cocaine; Delayed-Action Preparations; Female; Heroin; Humans; Injections; Male; Middle Aged; Motivation; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Substance Abuse Detection; Workplace

2019
Moderation of buprenorphine therapy for cocaine dependence efficacy by variation of the Prodynorphin gene.
    European journal of clinical pharmacology, 2022, Volume: 78, Issue:6

    Topics: Buprenorphine; Buprenorphine, Naloxone Drug Combination; Cocaine; Cocaine-Related Disorders; Delayed-Action Preparations; Enkephalins; Humans; Injections, Intramuscular; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Protein Precursors

2022
Naltrexone-bupropion combinations do not affect cocaine self-administration in humans.
    Pharmacology, biochemistry, and behavior, 2023, Volume: 224

    Topics: Blood Pressure; Bupropion; Cocaine; Drug Combinations; Humans; Naltrexone

2023

Other Studies

129 other study(ies) available for naltrexone and cocaine

ArticleYear
Extrapolation of human pharmacokinetic parameters from rat, dog, and monkey data: Molecular properties associated with extrapolative success or failure.
    Journal of pharmaceutical sciences, 2005, Volume: 94, Issue:7

    Topics: Algorithms; Animals; Dogs; Haplorhini; Humans; Pharmaceutical Preparations; Pharmacokinetics; Rats; Species Specificity; Tissue Distribution

2005
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Naltrexone, morphine and cocaine interactions in mice and rats.
    The Journal of pharmacology and experimental therapeutics, 1978, Volume: 206, Issue:2

    Topics: Animals; Cocaine; Drug Interactions; Lethal Dose 50; Male; Mice; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Reaction Time; Reflex

1978
The role of mu- and kappa-opioid receptors in cocaine-induced conditioned place preference.
    Japanese journal of pharmacology, 1992, Volume: 58, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Buprenorphine; Chlorides; Cocaine; Conditioning, Psychological; Lithium; Lithium Chloride; Male; Naltrexone; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid, kappa; Receptors, Opioid, mu

1992
Discriminative stimulus properties of cocaine, alone and in combination with buprenorphine, morphine and naltrexone.
    Drug and alcohol dependence, 1992, Volume: 30, Issue:3

    Topics: Animals; Buprenorphine; Cocaine; Dextroamphetamine; Discrimination, Psychological; Dose-Response Relationship, Drug; Drug Combinations; Male; Morphine; Naltrexone; Rats; Sodium Chloride

1992
Cocaine place preference is blocked by the delta-opioid receptor antagonist, naltrindole.
    European journal of pharmacology, 1992, Aug-25, Volume: 219, Issue:2

    Topics: Animals; Cocaine; Conditioning, Operant; Indoles; Male; Morphinans; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Lew

1992
Opioidergic modulation of cocaine conditioned place preferences.
    Life sciences, 1992, Volume: 50, Issue:14

    Topics: Analysis of Variance; Animals; Cocaine; Conditioning, Psychological; Male; Methadone; Naltrexone; Rats; Rats, Inbred Strains; Reference Values; Reinforcement, Psychology

1992
The partial opioid agonist, buprenorphine, protects against lethal effects of cocaine.
    Drug and alcohol dependence, 1991, Volume: 27, Issue:2

    Topics: Animals; Brain; Buprenorphine; Cocaine; Dose-Response Relationship, Drug; Methadone; Mice; Mice, Inbred Strains; Morphine; Naltrexone; Receptors, Opioid; Receptors, Opioid, mu; Seizures

1991
Antagonism of acute cocaine toxicity by buprenorphine.
    Life sciences, 1991, Volume: 49, Issue:25

    Topics: Analysis of Variance; Animals; Buprenorphine; Cocaine; Dose-Response Relationship, Drug; L-Lactate Dehydrogenase; Male; Mice; Naloxone; Naltrexone

1991
Intracerebroventricular naltrexone treatment attenuates acquisition of intravenous cocaine self-administration in rats.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 40, Issue:4

    Topics: Animals; Brain; Cocaine; Drug Interactions; Infusions, Intravenous; Injections, Intraventricular; Male; Naltrexone; Rats; Rats, Inbred Strains; Reinforcement, Psychology; Self Administration

1991
Effects of naltrexone on cocaine self-administration by rhesus monkey.
    NIDA research monograph, 1990, Volume: 105

    Topics: Animals; Buprenorphine; Cocaine; Eating; Macaca mulatta; Naltrexone; Self Administration

1990
Opiate antagonists reduce cocaine but not nicotine self-administration.
    Psychopharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Cocaine; Conditioning, Operant; Male; Naloxone; Naltrexone; Narcotic Antagonists; Nicotine; Rats; Reinforcement Schedule; Self Administration

1991
Chronic pretreatment with naltrexone facilitates acquisition of intravenous cocaine self-administration in rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1990, Volume: 1, Issue:1

    Topics: Animals; Cocaine; Conditioning, Operant; Injections, Intravenous; Male; Naltrexone; Rats; Rats, Inbred Strains; Self Administration

1990
Buprenorphine and naltrexone effects on cocaine self-administration by rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:3

    Topics: Animals; Buprenorphine; Cocaine; Conditioning, Operant; Eating; Female; Macaca mulatta; Male; Naltrexone; Self Administration

1990
NIDA's Medication Development Program--1989.
    NIDA research monograph, 1989, Volume: 95

    Topics: Acquired Immunodeficiency Syndrome; Brain; Cocaine; Drug and Narcotic Control; Female; Heroin Dependence; Humans; Infant, Newborn; Methadone; Methadyl Acetate; Naltrexone; Pregnancy; Psychotropic Drugs; Research Support as Topic; Risk Factors; Substance Abuse, Intravenous; Substance-Related Disorders

1989
Food deprivation and acquisition of intravenous cocaine self-administration in rats: effect of naltrexone and haloperidol.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:2

    Topics: Animals; Body Weight; Cocaine; Food Deprivation; Haloperidol; Male; Naltrexone; Rats; Rats, Inbred Strains; Reinforcement, Psychology; Self Administration

1989
Role of opioid antagonists in treating intravenous cocaine abuse.
    Life sciences, 1989, Volume: 44, Issue:13

    Topics: Adult; Buprenorphine; Cocaine; Female; Humans; Injections, Intravenous; Male; Methadone; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Substance-Related Disorders

1989
Antagonist treatment in nucleus accumbens or periaqueductal grey affects heroin self-administration.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:2

    Topics: Animals; Cocaine; Heroin; Male; Microinjections; Naltrexone; Narcotic Antagonists; Nucleus Accumbens; Periaqueductal Gray; Quaternary Ammonium Compounds; Rats; Rats, Inbred Strains; Self Administration

1988
Primary care of parenteral substance abusers.
    The Nurse practitioner, 1986, Volume: 11, Issue:6

    Topics: Acquired Immunodeficiency Syndrome; Administration, Intranasal; Antibodies, Viral; Body Weight; Cocaine; Female; Heart Diseases; Hepatitis; Heroin Dependence; HIV Antibodies; Humans; Injections, Intradermal; Injections, Intravenous; Kidney Diseases; Male; Menstruation Disturbances; Methadone; Naltrexone; Nervous System Diseases; Primary Health Care; Respiratory Tract Diseases; Substance-Related Disorders

1986
Effects of naltrexone on intravenous cocaine self-administration in rats during food satiation and deprivation.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Animals; Cocaine; Diarrhea; Food Deprivation; Male; Naltrexone; Nasal Mucosa; Posture; Rats; Rats, Inbred Strains; Salivation; Self Administration; Time Factors

1986
Heroin and cocaine intravenous self-administration in rats: mediation by separate neural systems.
    Psychopharmacology, 1982, Volume: 78, Issue:3

    Topics: Animals; Cocaine; Conditioning, Operant; Dose-Response Relationship, Drug; Flupenthixol; Heroin; Infusions, Parenteral; Male; Motor Activity; Naltrexone; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Opioid; Self Administration

1982
Cocaine self-administration and naltrindole, a delta-selective opioid antagonist.
    Neuroreport, 1995, Jul-10, Volume: 6, Issue:10

    Topics: Animals; Cocaine; Conditioning, Operant; Drug Implants; Female; Male; Morphine; Morphine Dependence; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Inbred Lew; Rats, Sprague-Dawley; Receptors, Opioid, delta; Self Administration

1995
The delta-opioid receptor antagonist naltrindole prevents sensitization to the conditioned rewarding effects of cocaine.
    European journal of pharmacology, 1995, Jun-23, Volume: 280, Issue:1

    Topics: Animals; Association Learning; Cocaine; Conditioning, Operant; Drug Interactions; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Reward; Sensitivity and Specificity

1995
Kappa opioid inhibition of morphine and cocaine self-administration in rats.
    Brain research, 1995, May-29, Volume: 681, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Cocaine; Dose-Response Relationship, Drug; Extinction, Psychological; Female; Morphine; Naltrexone; Narcotics; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Reinforcement, Psychology; Self Administration

1995
Behavioral and biochemical evidence of opioidergic involvement in cocaine sensitization.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:1

    Topics: Adenylyl Cyclases; Animals; Cocaine; Drug Tolerance; Male; Motor Activity; Naltrexone; Nucleus Accumbens; Opioid Peptides; Rats; Rats, Wistar; Receptors, Dopamine D1; Substance-Related Disorders

1995
Attenuation of the discriminative stimulus properties of cocaine by delta-opioid receptor antagonists.
    European journal of pharmacology, 1994, Sep-22, Volume: 263, Issue:1-2

    Topics: Animals; Benzylidene Compounds; Cocaine; Discrimination Learning; Dose-Response Relationship, Drug; Male; Naltrexone; Rats; Rats, Inbred F344; Receptors, Opioid, delta

1994
U50,488, a kappa opioid receptor agonist, attenuates cocaine-induced increases in extracellular dopamine in the nucleus accumbens of rats.
    Neuroscience letters, 1994, Nov-07, Volume: 181, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cocaine; Dopamine; Extracellular Space; Female; Naltrexone; Nucleus Accumbens; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

1994
Effects of buprenorphine and naltrexone on reinstatement of cocaine-reinforced responding in rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:3

    Topics: Animals; Benzimidazoles; Buprenorphine; Cocaine; Dose-Response Relationship, Drug; Drug Interactions; Male; Naltrexone; Rats; Rats, Wistar; Receptors, Opioid, mu; Reinforcement, Psychology

1993
The role of delta-opioid receptor subtypes in cocaine- and methamphetamine-induced place preferences.
    Life sciences, 1994, Volume: 55, Issue:17

    Topics: Animals; Benzylidene Compounds; Cocaine; Conditioning, Psychological; Male; Methamphetamine; Naltrexone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Reinforcement, Psychology

1994
Opioid peptides selective for receptor types modulate cocaine-induced behavioral responses in mice.
    Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology, 1994, Volume: 14, Issue:3

    Topics: Animals; Behavior, Animal; Cocaine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Naltrexone; Opioid Peptides

1994
Inhibition of cocaine-induced sensitization by the delta-opioid receptor antagonist naltrindole.
    European journal of pharmacology, 1993, Oct-19, Volume: 243, Issue:2

    Topics: Animals; Cocaine; Male; Motor Activity; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta

1993
Naltrexone-buprenorphine interactions: effects on cocaine self-administration.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1993, Volume: 9, Issue:3

    Topics: Animals; Buprenorphine; Cocaine; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Combinations; Eating; Female; Macaca mulatta; Male; Naltrexone; Reinforcement Schedule; Self Administration

1993
Delta-opioid receptor antagonists attenuate motor activity induced by amphetamine but not cocaine.
    European journal of pharmacology, 1993, Nov-09, Volume: 249, Issue:2

    Topics: Amphetamine; Animals; Cocaine; Dose-Response Relationship, Drug; Enkephalin, Leucine-2-Alanine; Male; Motor Activity; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta

1993
Blockade of delta-opioid receptors in the nucleus accumbens prevents ethanol-induced stimulation of dopamine release.
    European journal of pharmacology, 1993, Jan-12, Volume: 230, Issue:2

    Topics: Animals; Cocaine; Dopamine; Ethanol; Indoles; Male; Morphinans; Naltrexone; Narcotic Antagonists; Nucleus Accumbens; Oligopeptides; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta

1993
Naltrindole, an opioid delta receptor antagonist, blocks cocaine-induced facilitation of responding for rewarding brain stimulation.
    Life sciences, 1993, Volume: 52, Issue:9

    Topics: Analysis of Variance; Animals; Brain; Cocaine; Electric Stimulation; Indoles; Male; Morphinans; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Reinforcement, Psychology; Self Stimulation

1993
Cocaine-like discriminative stimulus properties of the delta-selective opioid receptor agonist, [D-Pen2,L-Pen5]enkephalin, in the rat.
    European journal of pharmacology, 1993, Jan-26, Volume: 231, Issue:1

    Topics: Animals; Cocaine; Discrimination Learning; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Generalization, Stimulus; Indoles; Morphinans; Naltrexone; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu

1993
Lack of involvement of delta-opioid receptors in mediating the rewarding effects of cocaine.
    Psychopharmacology, 1995, Volume: 120, Issue:4

    Topics: Animals; Benzazepines; Cocaine; Conditioning, Operant; Dose-Response Relationship, Drug; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Reward; Self Administration; Time Factors

1995
Discriminative stimulus effects of nalbuphine in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:2

    Topics: Analgesics, Opioid; Animals; Cocaine; Dextroamphetamine; Discrimination Learning; Female; Macaca mulatta; Male; Nalbuphine; Naltrexone

1996
kappa-Opioid receptor agonists prevent sensitization to the conditioned rewarding effects of cocaine.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzeneacetamides; Cocaine; Conditioning, Psychological; Dopamine; Male; Naltrexone; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Reward

1996
The effects of eticlopride and naltrexone on responding maintained by food, cocaine, heroin and cocaine/heroin combinations in rats.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 277, Issue:3

    Topics: Analysis of Variance; Animals; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Combinations; Eating; Heroin; Male; Naltrexone; Rats; Rats, Inbred F344; Receptors, Opioid; Salicylamides

1996
Differential role of delta-opioid receptors in the development and expression of behavioral sensitization to cocaine.
    European journal of pharmacology, 1996, Mar-18, Volume: 298, Issue:3

    Topics: Animals; Behavior, Animal; Cocaine; Male; Motor Activity; Naltrexone; Narcotic Antagonists; Narcotics; Nicotine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta

1996
The cocaine-like behavioral effects of meperidine are mediated by activity at the dopamine transporter.
    European journal of pharmacology, 1996, Feb-15, Volume: 297, Issue:1-2

    Topics: Animals; Behavior, Animal; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Meperidine; Models, Molecular; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Saimiri

1996
International update: new findings on promising medications.
    Alcoholism, clinical and experimental research, 1996, Volume: 20, Issue:8 Suppl

    Topics: Acamprosate; Alcohol Deterrents; Alcoholism; Animals; Clinical Trials as Topic; Cocaine; Comorbidity; Europe; Humans; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Taurine; United States

1996
Isradipine in combination with naltrexone as a medicine for treating cocaine abuse.
    Life sciences, 1997, Volume: 60, Issue:8

    Topics: Animals; Calcium Channel Blockers; Cocaine; Drug Therapy, Combination; Electric Stimulation; Isradipine; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Substance-Related Disorders

1997
Effects of kappa opioids on cocaine self-administration by rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Circadian Rhythm; Cocaine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Macaca mulatta; Male; Naloxone; Naltrexone; Pyrrolidines; Receptors, Opioid, kappa; Self Administration; Substance-Related Disorders

1997
Mu opioid agonists potentiate amphetamine- and cocaine-induced rotational behavior in the rat.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:2

    Topics: Amphetamine; Animals; Cocaine; Drug Synergism; Male; Motor Activity; Naltrexone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

1997
Naltrindole, a selective delta-opioid receptor antagonist, potentiates the lethal effects of cocaine by a central mechanism of action.
    European journal of pharmacology, 1997, Aug-20, Volume: 333, Issue:1

    Topics: Animals; Blood Pressure; Central Nervous System; Cisterna Magna; Cocaine; Drug Synergism; Heart Rate; Infusions, Intravenous; Injections; Male; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Seizures

1997
Isradipine combined with naltrexone persistently reduces the reward-relevant effects of cocaine and alcohol.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:2

    Topics: Animals; Body Weight; Calcium Channel Blockers; Central Nervous System Depressants; Cocaine; Conditioning, Operant; Drinking; Drug Interactions; Ethanol; Isradipine; Male; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Sprague-Dawley; Reward

1998
Self-administration of cocaine-heroin combinations by rhesus monkeys: antagonism by naltrexone.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:1

    Topics: Animals; Cocaine; Dose-Response Relationship, Drug; Drug Combinations; Female; Heroin; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Receptors, Opioid, delta; Receptors, Opioid, mu; Self Administration

1998
A combination of isradipine and naltrexone blocks cocaine's enhancement of a cocaine place preference.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:4

    Topics: Animals; Calcium Channel Blockers; Cocaine; Conditioning, Operant; Dose-Response Relationship, Drug; Isradipine; Male; Mental Recall; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Sprague-Dawley; Substance-Related Disorders

1998
Effects of beta-funaltrexamine on dose-effect curves for heroin self-administration in rats: comparison with alteration of [3H]DAMGO binding to rat brain sections.
    Drug and alcohol dependence, 1998, Oct-01, Volume: 52, Issue:2

    Topics: Analgesics, Opioid; Animals; Brain; Caudate Nucleus; Cocaine; Culture Techniques; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Heroin; Heroin Dependence; Motivation; Naltrexone; Narcotic Antagonists; Nucleus Accumbens; Radioligand Assay; Rats; Receptors, Opioid, mu; Self Administration

1998
Kappa-opioid receptor blockade with nor-binaltorphimine modulates cocaine self-administration in drug-naive rats.
    European journal of pharmacology, 1998, Oct-09, Volume: 358, Issue:3

    Topics: Animals; Behavior, Animal; Cocaine; Dose-Response Relationship, Drug; Male; Naltrexone; Narcotics; Nicotinic Antagonists; Rats; Rats, Wistar; Receptors, Opioid, kappa; Self Administration; Time Factors

1998
Regulation of cocaine reward by CREB.
    Science (New York, N.Y.), 1998, Dec-18, Volume: 282, Issue:5397

    Topics: Animals; Cocaine; Conditioning, Psychological; Cyclic AMP Response Element-Binding Protein; Dose-Response Relationship, Drug; Dynorphins; Gene Expression; Gene Expression Regulation; Gene Transfer Techniques; Genetic Vectors; Naltrexone; Narcotic Antagonists; Neurons; Nucleus Accumbens; Point Mutation; Rats; Receptors, Opioid, kappa; Reward; RNA, Messenger; Simplexvirus

1998
The effects of the naltrexone implant on rodent social interactions and cocaine-induced conditioned place preference.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 62, Issue:1

    Topics: Animals; Cocaine; Conditioning, Psychological; Drug Implants; Drug Interactions; Grooming; Male; Motor Activity; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Social Behavior

1999
Naltrexone affects cocaine self-administration in naïve rats through the ventral tegmental area rather than dopaminergic target regions.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1999, Volume: 9, Issue:1-2

    Topics: Animals; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Wistar; Self Administration; Time Factors; Ventral Tegmental Area

1999
Discriminative stimulus effects of morphine in squirrel monkeys: stimulants, opioids, and stimulant-opioid combinations.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Amphetamine; Analgesics, Opioid; Anesthetics, Local; Animals; Anti-Anxiety Agents; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Combinations; Fentanyl; Male; Morphine; Naltrexone; Narcotic Antagonists; Piperazines; Receptors, Opioid; Saimiri; Selective Serotonin Reuptake Inhibitors

1999
Cocaine-like discriminative stimulus effects of heroin in squirrel monkeys: role of active metabolites and opioid receptor mechanisms.
    Psychopharmacology, 2000, Volume: 150, Issue:2

    Topics: Analgesics, Opioid; Animals; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Heroin; Male; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Saimiri

2000
Antagonism of delta(2)-opioid receptors by naltrindole-5'-isothiocyanate attenuates heroin self-administration but not antinociception in rats.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:3

    Topics: Analgesics, Opioid; Animals; Cocaine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Heroin; Injections, Intraventricular; Isothiocyanates; Male; Naltrexone; Narcotic Antagonists; Oligopeptides; Pain Measurement; Rats; Rats, Inbred F344; Receptors, Opioid, delta; Reinforcement, Psychology; Self Administration

2000
Kappa-opioid receptor activation modifies dopamine uptake in the nucleus accumbens and opposes the effects of cocaine.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Dec-15, Volume: 20, Issue:24

    Topics: Analysis of Variance; Animals; Autoradiography; Benzeneacetamides; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Drug Administration Schedule; Drug Antagonism; Extracellular Space; Injections, Intraperitoneal; Injections, Subcutaneous; Iodine Radioisotopes; Linear Models; Male; Membrane Glycoproteins; Membrane Transport Proteins; Microdialysis; Naltrexone; Nerve Tissue Proteins; Nucleus Accumbens; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

2000
Kappa opioid agonists alter dopamine markers and cocaine-stimulated locomotor activity.
    Behavioural pharmacology, 2001, Volume: 12, Issue:4

    Topics: Analgesics; Animals; Benzeneacetamides; Benzomorphans; Caudate Nucleus; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Drug Interactions; Male; Membrane Glycoproteins; Membrane Transport Proteins; Motor Activity; Naltrexone; Nerve Net; Nerve Tissue Proteins; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

2001
Cocaine and amphetamine attenuate the discriminative stimulus effects of naltrexone in opioid-dependent rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 301, Issue:3

    Topics: Amphetamine; Animals; Cocaine; Discrimination, Psychological; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Substance Withdrawal Syndrome

2002
Effect of naltrexone on oral consumption of concurrently available ethanol and cocaine in the rat.
    Alcohol (Fayetteville, N.Y.), 2002, Volume: 28, Issue:3

    Topics: Administration, Oral; Alcohol Drinking; Animals; Behavior, Addictive; Cocaine; Dose-Response Relationship, Drug; Ethanol; Male; Naltrexone; Rats; Rats, Wistar

2002
Kappa opioid receptor antagonism and prodynorphin gene disruption block stress-induced behavioral responses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Jul-02, Volume: 23, Issue:13

    Topics: Analgesia; Animals; Behavior, Animal; Cocaine; Drug Synergism; Enkephalins; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Naltrexone; Narcotic Antagonists; Pain Threshold; Protein Precursors; Reaction Time; Receptors, Opioid, kappa; Reward; Spatial Behavior; Stress, Physiological; Swimming

2003
Beta-funaltrexamine affects cocaine self-administration in rats responding on a progressive ratio schedule of reinforcement.
    Pharmacology, biochemistry, and behavior, 2003, Volume: 75, Issue:2

    Topics: Animals; Cocaine; Conditioning, Operant; Male; Microinjections; Naltrexone; Narcotic Antagonists; Neostriatum; Nucleus Accumbens; Rats; Rats, Inbred F344; Reinforcement Schedule; Self Administration; Ventral Tegmental Area

2003
Cocaine and other indirect-acting monoamine agonists differentially attenuate a naltrexone discriminative stimulus in morphine-treated rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 308, Issue:1

    Topics: Amphetamine; Animals; Biogenic Monoamines; Cocaine; Discrimination Learning; Disease Models, Animal; Dopamine Agents; Dopamine Uptake Inhibitors; Drug Interactions; Imipramine; Macaca mulatta; Morphine; Morphine Dependence; Naltrexone; Narcotics; Substance Withdrawal Syndrome

2004
Opioid partial agonist effects of 3-O-methylnaltrexone in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 308, Issue:3

    Topics: Adenylyl Cyclases; Animals; Cocaine; Discrimination Learning; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Heroin; Heroin Dependence; Macaca mulatta; Male; Morphine; Morphine Derivatives; Naltrexone; Narcotics; Quaternary Ammonium Compounds; Receptors, Opioid, mu; Self Administration

2004
The opioid antagonist naltrexone reduces the reinforcing effects of Delta 9 tetrahydrocannabinol (THC) in squirrel monkeys.
    Psychopharmacology, 2004, Volume: 173, Issue:1-2

    Topics: Analgesics, Non-Narcotic; Anesthetics, Local; Animals; Behavior, Animal; Cocaine; Conditioning, Operant; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Male; Naltrexone; Narcotic Antagonists; Reinforcement Schedule; Reinforcement, Psychology; Saimiri; Self Administration

2004
Effect of the kappa opioid agonist R-84760 on cocaine-induced increases in striatal dopamine levels and cocaine-induced place preference in C57BL/6J mice.
    Psychopharmacology, 2004, Volume: 173, Issue:1-2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Chromatography, High Pressure Liquid; Cocaine; Conditioning, Operant; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Food; Male; Mice; Mice, Inbred C57BL; Microdialysis; Motor Activity; Naltrexone; Narcotic Antagonists; Neostriatum; Pyrrolidines; Receptors, Opioid, kappa; Thiazines

2004
Genetic and pharmacological manipulation of mu opioid receptors in mice reveals a differential effect on behavioral sensitization to cocaine.
    Neuroscience, 2004, Volume: 125, Issue:1

    Topics: Adaptation, Physiological; Animals; Behavior, Animal; Cocaine; Dopamine Uptake Inhibitors; Mice; Mice, Knockout; Motor Activity; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu

2004
Effects of the kappa opioid agonist U50,488 and the kappa opioid antagonist nor-binaltorphimine on choice between cocaine and food in rhesus monkeys.
    Psychopharmacology, 2004, Volume: 176, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Behavior, Addictive; Choice Behavior; Cocaine; Dose-Response Relationship, Drug; Eating; Macaca mulatta; Male; Naltrexone; Receptors, Opioid, kappa

2004
Mu-opioid receptors are not involved in acute cocaine-induced locomotor activity nor in development of cocaine-induced behavioral sensitization in mice.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:2

    Topics: Animals; Behavior, Animal; Cocaine; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Naltrexone; Narcotic Antagonists; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Somatostatin; Stimulation, Chemical

2005
Effects of chronic naltrexone treatment in rats on place preference and locomotor activation after acute administration of cocaethylene or ethanol plus cocaine.
    Alcohol (Fayetteville, N.Y.), 2004, Volume: 33, Issue:1

    Topics: Animals; Cocaine; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Combinations; Ethanol; Male; Motor Activity; Naltrexone; Rats; Rats, Sprague-Dawley

2004
Monoaminergic drugs and directly observable signs of LAAM withdrawal in rhesus monkeys.
    Behavioural pharmacology, 2005, Volume: 16, Issue:1

    Topics: Adrenergic alpha-Agonists; Amphetamine; Analgesics, Opioid; Animals; Antidepressive Agents, Tricyclic; Biogenic Monoamines; Clonidine; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Haloperidol; Imipramine; Macaca mulatta; Male; Methadyl Acetate; Muscle Rigidity; Naltrexone; Narcotic Antagonists; Respiratory Mechanics; Salivation; Substance Withdrawal Syndrome

2005
Social defeat stress-induced behavioral responses are mediated by the endogenous kappa opioid system.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2006, Volume: 31, Issue:6

    Topics: Analysis of Variance; Anesthetics, Local; Animals; Behavior, Animal; Cocaine; Conditioning, Operant; Enkephalins; Immobility Response, Tonic; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Naltrexone; Narcotic Antagonists; Pain Measurement; Protein Precursors; Reaction Time; Receptors, Opioid, kappa; Social Behavior; Stress, Psychological

2006
Naltrexone and buprenorphine combination in the treatment of opioid dependence.
    Journal of psychopharmacology (Oxford, England), 2006, Volume: 20, Issue:6

    Topics: Adult; Affect; Buprenorphine; Cocaine; Cocaine-Related Disorders; Female; Heroin Dependence; Humans; Liver; Male; Naltrexone; Narcotic Antagonists; Opioid-Related Disorders; Psychiatric Status Rating Scales; Substance Abuse Detection; Survival Analysis

2006
Paradoxical effects of prodynorphin gene deletion on basal and cocaine-evoked dopaminergic neurotransmission in the nucleus accumbens.
    The European journal of neuroscience, 2006, Volume: 23, Issue:1

    Topics: Analgesics; Animals; Area Under Curve; Behavior, Animal; Benzeneacetamides; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Dynorphins; Electrochemistry; Mice; Mice, Inbred C57BL; Mice, Knockout; Microdialysis; Motor Activity; Naltrexone; Narcotic Antagonists; Nucleus Accumbens; Pyrrolidines

2006
Food-induced behavioral sensitization, its cross-sensitization to cocaine and morphine, pharmacological blockade, and effect on food intake.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jul-05, Volume: 26, Issue:27

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analgesics, Opioid; Animals; Benzazepines; Benzodiazepines; Cocaine; Conditioning, Psychological; Dopamine Antagonists; Dopamine Uptake Inhibitors; Drug Interactions; Eating; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Feeding Behavior; Male; Mice; Mice, Inbred C57BL; Morphine; Motor Activity; Naltrexone; Narcotic Antagonists; Receptors, Dopamine D1; Sulpiride

2006
Noradrenaline is necessary for the hedonic properties of addictive drugs.
    Vascular pharmacology, 2006, Volume: 45, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Appetitive Behavior; Benzazepines; Biphenyl Compounds; Bupropion; Carbidopa; Cocaine; Dopamine beta-Hydroxylase; Dopamine Uptake Inhibitors; Droxidopa; Female; Genotype; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Morphine; Naltrexone; Narcotic Antagonists; Neurokinin-1 Receptor Antagonists; Norepinephrine; Receptors, Adrenergic, alpha-1; Receptors, Dopamine D1; Reward; Substance-Related Disorders

2006
Pharmacological and genetic manipulation of kappa opioid receptors: effects on cocaine- and pentylenetetrazol-induced convulsions and seizure kindling.
    Neuropharmacology, 2007, Volume: 52, Issue:3

    Topics: Analgesics; Animals; Behavior, Animal; Benzeneacetamides; Cocaine; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Naltrexone; Narcotic Antagonists; Pentylenetetrazole; Pyrrolidines; Receptors, Opioid, kappa; Seizures

2007
History of cocaine self-administration alters morphine reinforcement in the rat.
    European journal of pharmacology, 2007, May-07, Volume: 562, Issue:1-2

    Topics: Analysis of Variance; Animals; Cocaine; Conditioning, Operant; Dose-Response Relationship, Drug; Infusions, Intravenous; Injections, Intraperitoneal; Male; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration

2007
Microinjection of the delta-opioid receptor selective antagonist naltrindole 5'-isothiocyanate site specifically affects cocaine self-administration in rats responding under a progressive ratio schedule of reinforcement.
    Behavioural brain research, 2007, Aug-22, Volume: 182, Issue:1

    Topics: Anesthetics, Local; Animals; Behavior, Animal; Brain; Cocaine; Isothiocyanates; Male; Microinjections; Naltrexone; Rats; Rats, Inbred F344; Receptors, Opioid, delta; Reinforcement Schedule; Self Administration; Time Factors

2007
Micro-opioid receptor alkylation in the ventral pallidum and ventral tegmental area, but not in the nucleus accumbens, attenuates the effects of heroin on cocaine self-administration in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2008, Volume: 33, Issue:5

    Topics: Alkylating Agents; Alkylation; Analysis of Variance; Animals; Behavior, Animal; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Synergism; Globus Pallidus; Heroin; Male; Naltrexone; Narcotics; Nucleus Accumbens; Rats; Rats, Inbred F344; Receptors, Opioid, mu; Self Administration; Ventral Tegmental Area

2008
The kappa-opioid receptor antagonist nor-BNI inhibits cocaine and amphetamine, but not cannabinoid (WIN 52212-2), abstinence-induced withdrawal in planarians: an instance of 'pharmacologic congruence'.
    Brain research, 2008, Feb-08, Volume: 1193

    Topics: Amphetamine; Analgesics; Analysis of Variance; Animals; Behavior, Animal; Benzoxazines; Cocaine; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug Interactions; Morpholines; Naltrexone; Naphthalenes; Narcotic Antagonists; Planarians; Substance Withdrawal Syndrome; Time Factors

2008
Kappa-opioid system regulates the long-lasting behavioral adaptations induced by early-life exposure to methylphenidate.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anxiety; Behavior, Animal; Central Nervous System Stimulants; Cocaine; Conditioning, Psychological; Food Preferences; Male; Methylphenidate; Motor Activity; Naltrexone; Psychotropic Drugs; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Stress, Psychological

2009
Intravenous self-administration of etonitazene alone and combined with cocaine in rhesus monkeys: comparison with heroin and antagonism by naltrexone and naloxonazine.
    Psychopharmacology, 2009, Volume: 204, Issue:3

    Topics: Animals; Benzimidazoles; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Data Interpretation, Statistical; Dose-Response Relationship, Drug; Drug Interactions; Female; Heroin; Injections, Intravenous; Macaca mulatta; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Receptors, Opioid, mu; Reinforcement, Psychology; Self Administration; Substance Abuse, Intravenous

2009
Inhibition of kappa opioid receptors attenuated increased cocaine intake in rats with extended access to cocaine.
    Psychopharmacology, 2009, Volume: 205, Issue:4

    Topics: Animals; CHO Cells; Cocaine; Conditioning, Operant; Cricetinae; Cricetulus; Drug Interactions; Male; Naltrexone; Rats; Rats, Wistar; Receptors, Opioid, kappa; Reinforcement Schedule; Self Administration

2009
Effect of non-dopaminergic drug treatment on Levodopa induced dyskinesias in MPTP monkeys: common implication of striatal neuropeptides.
    Neuropharmacology, 2010, Volume: 58, Issue:1

    Topics: Animals; Antiparkinson Agents; Benzoxazoles; Cocaine; Corpus Striatum; Disease Models, Animal; Docosahexaenoic Acids; Dopamine; Dopamine Uptake Inhibitors; Dynorphins; Dyskinesia, Drug-Induced; Enkephalins; Female; Iodine Isotopes; Levodopa; Macaca fascicularis; Naltrexone; Neuropeptides; Ovariectomy; Parkinsonian Disorders; Piperidines; Protein Precursors; RNA, Messenger; Sulfonamides; Tachykinins; Thiazoles; Time Factors

2010
Activation of the kappa opioid receptor in the dorsal raphe nucleus mediates the aversive effects of stress and reinstates drug seeking.
    Proceedings of the National Academy of Sciences of the United States of America, 2009, Nov-10, Volume: 106, Issue:45

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analysis of Variance; Animals; Cocaine; Enzyme-Linked Immunosorbent Assay; Immunohistochemistry; Lentivirus; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Naltrexone; Raphe Nuclei; Receptors, Opioid, kappa; Stress, Physiological; Ventral Tegmental Area

2009
Behavioral stress may increase the rewarding valence of cocaine-associated cues through a dynorphin/kappa-opioid receptor-mediated mechanism without affecting associative learning or memory retrieval mechanisms.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2010, Volume: 35, Issue:9

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Analysis of Variance; Anesthetics, Local; Animals; Association Learning; Behavior, Animal; Cocaine; Conditioning, Operant; Cues; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Dynorphins; Exploratory Behavior; Male; Mental Recall; Mice; Mice, Inbred C57BL; Naltrexone; Narcotic Antagonists; Receptors, Opioid, kappa; Reward; Stress, Psychological; Swimming

2010
Influence of new deltorphin analogues on reinstatement of cocaine-induced conditioned place preference in rats.
    Behavioural pharmacology, 2010, Volume: 21, Issue:7

    Topics: Animals; Behavior, Addictive; Behavioral Research; Cocaine; Conditioning, Psychological; Infusions, Intraventricular; Maze Learning; Motor Activity; Naltrexone; Narcotic Antagonists; Oligopeptides; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Opioid, delta; Reward

2010
Exposure to cocaine alters dynorphin-mediated regulation of excitatory synaptic transmission in nucleus accumbens neurons.
    Biological psychiatry, 2011, Feb-01, Volume: 69, Issue:3

    Topics: Animals; Cocaine; Drug Interactions; Dynorphins; Excitatory Postsynaptic Potentials; Male; Naltrexone; Neurons; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Synaptic Transmission

2011
Blockade of kappa opioid receptors attenuates the development of depressive-like behaviors induced by cocaine withdrawal in rats.
    Neuropharmacology, 2012, Volume: 62, Issue:1

    Topics: Analysis of Variance; Animals; Cocaine; Conditioning, Operant; Depression; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug Administration Routes; Immobility Response, Tonic; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Opioid, kappa; Reinforcement Schedule; Self Administration; Substance Withdrawal Syndrome; Swimming; Time Factors

2012
Repeated exposure to the κ-opioid receptor agonist salvinorin A modulates extracellular signal-regulated kinase and reward sensitivity.
    Biological psychiatry, 2011, Oct-15, Volume: 70, Issue:8

    Topics: Animals; Cocaine; Cyclic AMP Response Element-Binding Protein; Diterpenes, Clerodane; Drug Interactions; Extracellular Signal-Regulated MAP Kinases; Male; Naltrexone; Nucleus Accumbens; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Reward; Self Stimulation; Signal Transduction; Time Factors

2011
Sex difference in κ-opioid receptor (KOPR)-mediated behaviors, brain region KOPR level and KOPR-mediated guanosine 5'-O-(3-[35S]thiotriphosphate) binding in the guinea pig.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 339, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analgesics, Non-Narcotic; Animals; Brain; Cocaine; Dopamine Uptake Inhibitors; Female; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Male; Mice; Motor Activity; Movement; Naltrexone; Narcotic Antagonists; Posture; Rats; Receptors, Opioid, kappa; Sex Characteristics

2011
The rewarding action of acute cocaine is reduced in β-endorphin deficient but not in μ opioid receptor knockout mice.
    European journal of pharmacology, 2012, Jul-05, Volume: 686, Issue:1-3

    Topics: Animals; Behavior, Animal; beta-Endorphin; Cocaine; Conditioning, Operant; Male; Mice; Mice, Knockout; Morphine; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu; Reward

2012
Cocaine reverses the naltrexone-induced reduction in operant ethanol self-administration: the effects on immediate-early gene expression in the rat prefrontal cortex.
    Neuropharmacology, 2012, Volume: 63, Issue:6

    Topics: Acamprosate; Alcohol Deterrents; Alcohol Drinking; Animals; Carrier Proteins; Cocaine; Conditioning, Operant; Cyclooxygenase 2; Dose-Response Relationship, Drug; Gene Expression; Genes, fos; Genes, Immediate-Early; Homer Scaffolding Proteins; Male; Motor Activity; Naltrexone; Narcotic Antagonists; Prefrontal Cortex; Rats; Rats, Wistar; Real-Time Polymerase Chain Reaction; Self Administration; Taurine

2012
A combination of buprenorphine and naltrexone blocks compulsive cocaine intake in rodents without producing dependence.
    Science translational medicine, 2012, Aug-08, Volume: 4, Issue:146

    Topics: Animals; Buprenorphine; Cocaine; Cocaine-Related Disorders; Male; Naloxone; Naltrexone; Rats; Rats, Wistar; Substance Withdrawal Syndrome

2012
Effect of food restriction on cocaine locomotor sensitization in Sprague-Dawley rats: role of kappa opioid receptors.
    Psychopharmacology, 2013, Volume: 226, Issue:3

    Topics: Animals; Cocaine; Corticosterone; Dose-Response Relationship, Drug; Food Deprivation; Male; Motor Activity; Naltrexone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

2013
Stress produces aversion and potentiates cocaine reward by releasing endogenous dynorphins in the ventral striatum to locally stimulate serotonin reuptake.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Dec-05, Volume: 32, Issue:49

    Topics: Animals; Avoidance Learning; Brain; Cocaine; Corpus Striatum; Dopamine; Dynorphins; G-Protein-Coupled Receptor Kinase 3; Male; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Mice, Transgenic; Microinjections; Naltrexone; Narcotic Antagonists; Nicotine; Nucleus Accumbens; p38 Mitogen-Activated Protein Kinases; Raphe Nuclei; Receptors, Opioid, kappa; Reward; Serotonin; Serotonin Plasma Membrane Transport Proteins; Signal Transduction; Stress, Psychological; Substance Withdrawal Syndrome; Synaptosomes

2012
A non-rewarding, non-aversive buprenorphine/naltrexone combination attenuates drug-primed reinstatement to cocaine and morphine in rats in a conditioned place preference paradigm.
    Addiction biology, 2014, Volume: 19, Issue:4

    Topics: Animals; Behavior, Animal; Buprenorphine; Cocaine; Conditioning, Psychological; Cues; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Therapy, Combination; Male; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Sprague-Dawley; Reward

2014
Neuropsychopharmacological actions of taurine.
    Advances in experimental medicine and biology, 2013, Volume: 775

    Topics: Amino Acids; Animals; Cocaine; Conditioning, Psychological; Extracellular Space; Locomotion; Models, Biological; Naltrexone; Neostriatum; Nervous System; Oligopeptides; Psychotropic Drugs; Rats; Receptors, N-Methyl-D-Aspartate; Taurine

2013
Locus coeruleus kappa-opioid receptors modulate reinstatement of cocaine place preference through a noradrenergic mechanism.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2013, Volume: 38, Issue:12

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-2 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Betaxolol; Clonidine; Cocaine; Conditioning, Psychological; Drug-Seeking Behavior; Locus Coeruleus; Male; Mice; Mice, Inbred C57BL; Naltrexone; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Opioid, kappa

2013
Involvement of delta and mu opioid receptors in the acute and sensitized locomotor action of cocaine in mice.
    Peptides, 2013, Volume: 48

    Topics: Animals; Cocaine; Humans; Mice; Motor Activity; Naltrexone; Oligopeptides; Pain Measurement; Receptors, Opioid, delta; Receptors, Opioid, mu

2013
Cocaine- or stress-induced metaplasticity of LTP in the dorsal and ventral hippocampus.
    Hippocampus, 2014, Volume: 24, Issue:5

    Topics: Animals; Cocaine; Corticosterone; Dopamine Uptake Inhibitors; Drug Administration Schedule; Excitatory Postsynaptic Potentials; Hippocampus; Hormone Antagonists; In Vitro Techniques; Long-Term Potentiation; Male; Mifepristone; Mineralocorticoid Receptor Antagonists; Motor Activity; Naltrexone; Rats; Rats, Sprague-Dawley; Spironolactone; Stress, Psychological

2014
Repeated stress exposure causes strain-dependent shifts in the behavioral economics of cocaine in rats.
    Addiction biology, 2015, Volume: 20, Issue:2

    Topics: Animals; Cocaine; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Economics, Behavioral; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred WKY; Rats, Wistar; Self Administration; Stress, Psychological; Swimming

2015
Effects of the kappa opioid receptor antagonist nor-binaltorphimine (nor-BNI) on cocaine versus food choice and extended-access cocaine intake in rhesus monkeys.
    Addiction biology, 2016, Volume: 21, Issue:2

    Topics: Analysis of Variance; Animals; Cocaine; Conditioning, Operant; Drug-Seeking Behavior; Food Preferences; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Receptors, Opioid, kappa; Self Administration

2016
Synthesis and characterization of a dual kappa-delta opioid receptor agonist analgesic blocking cocaine reward behavior.
    ACS chemical neuroscience, 2015, Nov-18, Volume: 6, Issue:11

    Topics: Analgesics, Opioid; Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Psychological; Dopamine Uptake Inhibitors; Drug Evaluation, Preclinical; Male; Mice, Inbred C57BL; Mice, Knockout; Molecular Structure; Morphinans; Naltrexone; Nociception; Nuclear Receptor Subfamily 1, Group F, Member 1; Random Allocation; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reward; Spatial Behavior

2015
Cannabidiol disrupts the reconsolidation of contextual drug-associated memories in Wistar rats.
    Addiction biology, 2017, Volume: 22, Issue:3

    Topics: Animals; Cannabidiol; Cocaine; Conditioning, Classical; Cues; Disease Models, Animal; Male; Memory; Mental Recall; Morphine; Naltrexone; Rats; Rats, Wistar; Reward

2017
Nalmefene is effective at reducing alcohol seeking, treating alcohol-cocaine interactions and reducing alcohol-induced histone deacetylases gene expression in blood.
    British journal of pharmacology, 2016, Volume: 173, Issue:16

    Topics: Alcohol Drinking; Animals; Cocaine; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Gene Expression Regulation, Enzymologic; Histone Deacetylases; Male; Naltrexone; Rats; Rats, Wistar; Structure-Activity Relationship

2016
Lack of Specific Involvement of (+)-Naloxone and (+)-Naltrexone on the Reinforcing and Neurochemical Effects of Cocaine and Opioids.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2016, Volume: 41, Issue:11

    Topics: Analgesics, Opioid; Anesthetics; Animals; Brain; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dopamine; Extinction, Psychological; Male; Microdialysis; Naloxone; Naltrexone; Narcotic Antagonists; Piperidines; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Remifentanil; Self Administration; Time Factors

2016
Rearing environment differentially modulates cocaine self-administration after opioid pretreatment: A behavioral economic analysis.
    Drug and alcohol dependence, 2016, Oct-01, Volume: 167

    Topics: Analgesics, Opioid; Animals; Behavior, Animal; Cocaine; Economics, Behavioral; Environment; Male; Morphine; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Self Administration; Substance-Related Disorders; Time Factors

2016
Procedure for the Selection and Validation of a Calibration Model I-Description and Application.
    Journal of analytical toxicology, 2017, May-01, Volume: 41, Issue:4

    Topics: Calibration; Chromatography, Liquid; Cocaine; Models, Statistical; Naltrexone; Quality Control; Reference Standards; Tandem Mass Spectrometry

2017
Factors associated with using opiates while under extended-release naltrexone blockade: A descriptive pilot study.
    Journal of substance abuse treatment, 2018, Volume: 85

    Topics: Adult; Behavior, Addictive; Cocaine; Delayed-Action Preparations; Female; Humans; Male; Naltrexone; Narcotic Antagonists; Opiate Alkaloids; Opioid-Related Disorders; Pilot Projects; Randomized Controlled Trials as Topic

2018
Buprenorphine requires concomitant activation of NOP and MOP receptors to reduce cocaine consumption.
    Addiction biology, 2018, Volume: 23, Issue:2

    Topics: Animals; Behavior, Animal; Buprenorphine; Cocaine; Conditioning, Operant; Cycloheptanes; Dopamine Uptake Inhibitors; Naltrexone; Narcotic Antagonists; Nociceptin Receptor; Piperidines; Rats; Receptors, Opioid; Receptors, Opioid, mu; Self Administration

2018
Maintenance on naltrexone+amphetamine decreases cocaine-vs.-food choice in male rhesus monkeys.
    Drug and alcohol dependence, 2017, 12-01, Volume: 181

    Topics: Administration, Intravenous; Animals; Choice Behavior; Cocaine; Dextroamphetamine; Dose-Response Relationship, Drug; Drug Interactions; Food; Macaca mulatta; Male; Morphine; Naltrexone; Receptors, Opioid, mu; Reinforcement, Psychology; Self Administration

2017
Dynorphin Counteracts Orexin in the Paraventricular Nucleus of the Thalamus: Cellular and Behavioral Evidence.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2018, Volume: 43, Issue:5

    Topics: Animals; Behavior, Addictive; Cocaine; Cocaine-Related Disorders; Drug Interactions; Dynorphins; Excitatory Postsynaptic Potentials; Extinction, Psychological; Male; Microinjections; Miniature Postsynaptic Potentials; Naltrexone; Orexins; Paraventricular Hypothalamic Nucleus; Rats; Reward; Self Administration

2018
Naltrexone maintenance fails to alter amphetamine effects on intracranial self-stimulation in rats.
    Experimental and clinical psychopharmacology, 2018, Volume: 26, Issue:2

    Topics: Amphetamine; Animals; Central Nervous System Stimulants; Cocaine; Deep Brain Stimulation; Dose-Response Relationship, Drug; Male; Medial Forebrain Bundle; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Sprague-Dawley; Self Stimulation; Substance-Related Disorders

2018
Naltrexone and nalmefene attenuate cocaine place preference in male mice.
    Neuropharmacology, 2018, 09-15, Volume: 140

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Analgesics, Opioid; Animals; Cocaine; Conditioning, Psychological; Dose-Response Relationship, Drug; Locomotion; Male; Mice; Morphine; Naltrexone; Narcotic Antagonists

2018
Pharmacological classification of centrally acting drugs using EEG in freely moving rats: an old tool to identify new atypical dopamine uptake inhibitors.
    Neuropharmacology, 2019, 12-15, Volume: 161

    Topics: Animals; Central Nervous System Agents; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Discovery; Electroencephalography; Heroin; Ketamine; Male; Methylphenidate; Modafinil; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

2019
Kappa-opioid receptors, dynorphin, and cocaine addiction: a positron emission tomography study.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2019, Volume: 44, Issue:10

    Topics: Adult; Brain; Carbon Radioisotopes; Case-Control Studies; Choice Behavior; Cocaine; Cocaine Smoking; Cocaine-Related Disorders; Dynorphins; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Neostriatum; Piperazines; Positron-Emission Tomography; Pyrrolidines; Receptors, Opioid, kappa; Stress, Psychological

2019
Kappa opioid agonists reduce oxycodone self-administration in male rhesus monkeys.
    Psychopharmacology, 2020, Volume: 237, Issue:5

    Topics: Analgesics, Opioid; Animals; Behavior, Addictive; Cocaine; Diterpenes, Clerodane; Dose-Response Relationship, Drug; Macaca mulatta; Male; Morphinans; Naltrexone; Narcotic Antagonists; Oxycodone; Receptors, Opioid, kappa; Reinforcement, Psychology; Self Administration; Spiro Compounds

2020
Samidorphan, an opioid receptor antagonist, attenuates drug-induced increases in extracellular dopamine concentrations and drug self-administration in male Wistar rats.
    Pharmacology, biochemistry, and behavior, 2021, Volume: 204

    Topics: Amphetamine; Animals; Cocaine; Dopamine; Ethanol; Humans; Male; Microdialysis; Naltrexone; Narcotic Antagonists; Nucleus Accumbens; Oxycodone; Rats; Rats, Wistar; Receptors, Opioid; Receptors, Opioid, mu; Self Administration; Substance-Related Disorders

2021
Nalmefene, a mu opioid receptor antagonist/kappa opioid receptor partial agonist, potentiates cocaine motivation but not intake with extended access self-administration in adult male mice.
    Neuropharmacology, 2021, 07-01, Volume: 192

    Topics: Analgesics, Opioid; Animals; Cocaine; Male; Mice; Mice, Inbred C57BL; Motivation; Naltrexone; Narcotic Antagonists; Receptors, Opioid, kappa; Receptors, Opioid, mu; Self Administration

2021
The Buprenorphine Analogue BU10119 Attenuates Drug-Primed and Stress-Induced Cocaine Reinstatement in Mice.
    The Journal of pharmacology and experimental therapeutics, 2021, Volume: 378, Issue:3

    Topics: Buprenorphine; Cocaine; Naltrexone; Receptors, Opioid, mu

2021
PPL-138 (BU10038): A bifunctional NOP/mu partial agonist that reduces cocaine self-administration in rats.
    Neuropharmacology, 2022, 06-15, Volume: 211

    Topics: Animals; Cocaine; Dose-Response Relationship, Drug; Female; Isoquinolines; Male; Naltrexone; Nociceptin; Opioid Peptides; Phenylpropionates; Rats; Receptors, Opioid; Receptors, Opioid, mu; Self Administration

2022
PPL-103: A mixed opioid partial agonist with desirable anti-cocaine properties.
    Progress in neuro-psychopharmacology & biological psychiatry, 2022, 12-20, Volume: 119

    Topics: Analgesics, Opioid; Animals; Cocaine; Cocaine-Related Disorders; Humans; Naltrexone; Rats; Receptors, Opioid, kappa; Receptors, Opioid, mu; Self Administration

2022
Toll-like receptor 4 antagonists reduce cocaine-primed reinstatement of drug seeking.
    Psychopharmacology, 2023, Volume: 240, Issue:7

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Extinction, Psychological; Lipopolysaccharides; Naltrexone; Rats; Rats, Sprague-Dawley; Self Administration; Toll-Like Receptor 4

2023
Risks of returning to opioid use at treatment entry and early in opioid use disorder treatment: Role of non-opioid substances.
    Drug and alcohol dependence, 2023, Oct-01, Volume: 251

    Topics: Analgesics, Opioid; Buprenorphine; Cocaine; Humans; Methadone; Naltrexone; Opiate Substitution Treatment; Opioid-Related Disorders

2023