naftopidil and prazosin

naftopidil has been researched along with prazosin in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (22.22)18.2507
2000's7 (38.89)29.6817
2010's6 (33.33)24.3611
2020's1 (5.56)2.80

Authors

AuthorsStudies
Ang, KK; Arkin, MR; Chen, S; Doyle, PS; Engel, JC; McKerrow, JH1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Kigoshi, S; Muramatsu, I; Yamanaka, K1
Borbe, HO; Peter, G1
Asano, M; Honda, K; Inagaki, O; Kawabe, K; Kimura, R; Mori, R; Suzuki, M; Takenaka, T; Tanaka, C; Yamada, S1
Asano, T; Awaji, T; Hirasawa, A; Ikegaki, I; Shibata, K; Takada, T; Take, H; Tsujimoto, G1
Ikegaki, I1
Miyata, K; Ohtake, A; Saitoh, C; Sasamata, M; Sato, S; Yuyama, H1
Kobayashi, K; Kobayashi, M; Maruyama, I; Shibata, N; Tatemichi, S; Yamazaki, Y1
Jin, J; Kong, CZ; Li, NC; Na, YQ; Qiu, SP; Song, YS; Sun, G; Sun, YC; Sun, YH; Wang, XF; Wu, SL; Ye, ZQ1
Noguchi, Y; Ohtake, A; Sasamata, M; Suzuki, M1
Imanishi, A; Latifpour, J; Ueda, S; Yamamoto, Y; Yono, M; Yoshida, M1
Aizawa, N; Andersson, KE; Chen, Z; Igawa, Y; Imamura, T; Ishizuka, O; Nishizawa, O1
Ashitomi, K; Kadekawa, K; Nishijima, S; Sugaya, K; Yamamoto, H1
Gotoh, A; Kanno, T; Nagaya, H; Nishizaki, T1
Araki, M; Araki, T; Monden, K1
Creta, M; Ficarra, V; Fusco, F; Giannarini, G; Longo, N; Mirone, V; Novara, G; Palmieri, A; Verze, P1
Hattori, T; Uta, D; Yoshimura, M1

Reviews

2 review(s) available for naftopidil and prazosin

ArticleYear
[Pharmacological properties of naftopidil, a drug for treatment of the bladder outlet obstruction for patients with benign prostatic hyperplasia].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2000, Volume: 116, Issue:2

    Topics: Adrenergic alpha-Antagonists; Aged; Animals; Binding, Competitive; Dogs; Humans; Male; Naphthalenes; Piperazines; Prazosin; Pressure; Prostate; Prostatic Hyperplasia; Rabbits; Receptors, Adrenergic, alpha-1; Urinary Bladder Neck Obstruction; Urination Disorders

2000
α1-Blockers Improve Benign Prostatic Obstruction in Men with Lower Urinary Tract Symptoms: A Systematic Review and Meta-analysis of Urodynamic Studies.
    European urology, 2016, Volume: 69, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Clinical Trials as Topic; Doxazosin; Humans; Indoles; Male; Naphthalenes; Piperazines; Prazosin; Prostatism; Quinazolines; Severity of Illness Index; Sulfonamides; Tamsulosin; Urodynamics

2016

Trials

2 trial(s) available for naftopidil and prazosin

ArticleYear
[Comparison of different drugs on the treatment of benign prostate hyperplasia].
    Zhonghua wai ke za zhi [Chinese journal of surgery], 2007, Jul-15, Volume: 45, Issue:14

    Topics: 5-alpha Reductase Inhibitors; Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Androstadienes; Double-Blind Method; Doxazosin; Enzyme Inhibitors; Finasteride; Follow-Up Studies; Humans; Male; Middle Aged; Naphthalenes; Piperazines; Plant Extracts; Prazosin; Prostate; Prostatic Hyperplasia; Quality of Life; Secale; Sulfonamides; Tamsulosin; Treatment Outcome

2007
Comparison of 7 α(1)-adrenoceptor antagonists in patients with lower urinary tract symptoms associated with benign prostatic hyperplasia:a short-term crossover study.
    Acta medica Okayama, 2013, Volume: 67, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adult; Aged; Aged, 80 and over; Cross-Over Studies; Doxazosin; Humans; Indoles; Lower Urinary Tract Symptoms; Male; Middle Aged; Naphthalenes; Piperazines; Prazosin; Prostatic Hyperplasia; Sulfonamides; Tamsulosin; Treatment Outcome

2013

Other Studies

14 other study(ies) available for naftopidil and prazosin

ArticleYear
Image-based high-throughput drug screening targeting the intracellular stage of Trypanosoma cruzi, the agent of Chagas' disease.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:8

    Topics: Animals; Cattle; Cell Line; Cell Line, Tumor; Chagas Disease; Drug Evaluation, Preclinical; Hepatocytes; High-Throughput Screening Assays; Humans; Image Processing, Computer-Assisted; Muscle, Skeletal; Parasitic Sensitivity Tests; Trypanocidal Agents; Trypanosoma cruzi

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Pharmacological profile of the novel alpha-adrenoceptor antagonist KT-611 (naftopidil).
    Japanese journal of pharmacology, 1991, Volume: 55, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Dogs; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Naphthalenes; Piperazines; Prazosin; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Sympathetic Nervous System

1991
Radioreceptor assay for the determination of alpha 1-adrenoceptor-binding material in rat plasma following single oral administration of naftopidil.
    Arzneimittel-Forschung, 1990, Volume: 40, Issue:3

    Topics: Administration, Oral; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Carrier Proteins; Half-Life; Male; Naphthalenes; Piperazines; Prazosin; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1990
Comparative study on alpha 1-adrenoceptor antagonist binding in human prostate and aorta.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:5

    Topics: Adrenergic alpha-Antagonists; Aged; Aorta; Binding Sites; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Humans; Kinetics; Male; Middle Aged; Naphthalenes; Piperazines; Prazosin; Prostate; Sulfonamides; Tamsulosin

1994
Vascular alpha1-adrenoceptor subtype selectivity and alpha1-blocker-induced orthostatic hypotension.
    Japanese journal of pharmacology, 1998, Volume: 77, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Base Sequence; CHO Cells; Cricetinae; DNA Primers; Hypotension, Orthostatic; Iodine Radioisotopes; Male; Naphthalenes; Phenethylamines; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Recombinant Proteins; RNA, Messenger; Tetralones

1998
Effects of tamsulosin on hypogastric nerve stimulation-induced intraurethral pressure elevation in male and female dogs under anesthesia.
    European journal of pharmacology, 2004, Aug-30, Volume: 497, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Dogs; Female; Hypogastric Plexus; Male; Naphthalenes; Piperazines; Prazosin; Pressure; Sex Factors; Sulfonamides; Tamsulosin; Urethra

2004
[Effects of silodosin (KMD-3213) on phenylephrine-induced increase in intraurethral pressure and blood pressure in rats--study of the selectivity for lower urinary tract].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 2006, Volume: 126 Spec no.

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Indoles; Male; Naphthalenes; Phenylephrine; Piperazines; Prazosin; Pressure; Rats; Sulfonamides; Tamsulosin; Urethra

2006
In vivo study on the effects of alpha1-adrenoceptor antagonists on intraurethral pressure in the prostatic urethra and intraluminal pressure in the vas deferens in male dogs.
    European journal of pharmacology, 2008, Feb-02, Volume: 580, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Dogs; Dose-Response Relationship, Drug; Ejaculation; Indoles; Male; Naphthalenes; Phenylephrine; Piperazines; Prazosin; Pressure; Prostate; Quinazolines; Sulfonamides; Tamsulosin; Urethra; Vas Deferens

2008
Differential effects of prazosin and naftopidil on pelvic blood flow and nitric oxide synthase levels in spontaneously hypertensive rats.
    Journal of receptor and signal transduction research, 2008, Volume: 28, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Hypertension; Male; Naphthalenes; Nitric Oxide Synthase; Pelvis; Penis; Piperazines; Prazosin; Prostate; Quinazolines; Quinoxalines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha; Regional Blood Flow; Urinary Bladder

2008
Role of alpha1-adrenergic receptors in detrusor overactivity induced by cold stress in conscious rats.
    Neurourology and urodynamics, 2009, Volume: 28, Issue:3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Body Temperature; Cold Temperature; Female; Indoles; Naphthalenes; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Urinary Bladder; Urinary Bladder, Overactive

2009
Excitatory effect of propiverine hydrochloride on urethral activity in rats.
    International journal of urology : official journal of the Japanese Urological Association, 2012, Volume: 19, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Benzilates; Female; Imidazoles; Indoles; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperazines; Prazosin; Pressure; Rats; Rats, Sprague-Dawley; Urethra; Urinary Bladder

2012
Antitumor action of α(1)-adrenoceptor blockers on human bladder, prostate and renal cancer cells.
    Pharmacology, 2012, Volume: 90, Issue:5-6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Antineoplastic Agents; Cell Line, Tumor; Cell Survival; Humans; Kidney Neoplasms; Male; Naphthalenes; Piperazines; Prazosin; Prostatic Neoplasms; Urinary Bladder Neoplasms

2012
Analyses of the Mode of Action of an Alpha-Adrenoceptor Blocker in Substantia Gelatinosa Neurons in Rats.
    International journal of molecular sciences, 2021, Sep-06, Volume: 22, Issue:17

    Topics: Adrenergic alpha-Antagonists; Animals; Excitatory Postsynaptic Potentials; Inhibitory Postsynaptic Potentials; Male; Membrane Potentials; Naphthalenes; Neurons; Norepinephrine; Patch-Clamp Techniques; Piperazines; Prazosin; Rats, Sprague-Dawley; Serotonin; Substantia Gelatinosa; Synaptic Transmission

2021