Page last updated: 2024-08-23

n-n-propylnorapomorphine and quinpirole

n-n-propylnorapomorphine has been researched along with quinpirole in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19904 (20.00)18.7374
1990's11 (55.00)18.2507
2000's4 (20.00)29.6817
2010's1 (5.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Griffon, N; Lévesque, D; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P1
Brusniak, MY; DuRand, C; Ginsburg, B; Neve, KA; Pearlman, RS; Starr, S; Teeter, M; Tseng, T; Wilcox, RE1
Brusniak, MY; DuRand, CJ; Huang, WH; Neve, KA; Pearlman, RS; Teeter, MM; Wiens, BL; Wilcox, DM; Wilcox, RE1
Barnes, JM; Barnes, NM; Costall, B; Naylor, RJ1
Axton, MS; Moore, NA1
Hizami, R; Kreuter, L; Meller, E1
D'Agostini, F; Da Prada, M; Haefely, WE; Pizzi, M; Spano, PF1
Bohmaker, K; Bordi, F; Meller, E1
Agnati, LF; Fuxe, K; Goldstein, M; Köhler, C; Lew, JY; Okada, K1
Senogles, SE1
Kozell, LB; Neve, KA; Starr, S1
Garrett, BE; Holtzman, SG1
DeSouza, EB; Grigoriadis, DE; Levant, B1
Allard, S; Falardeau, P; Lapointe, S1
Artaud, F; Borrelli, E; Chéramy, A; Glowinski, J; Godeheu, G; L'hirondel, M; Saiardi, A1
Cumps, J; Geurts, M; Hermans, E; Maloteaux, JM1
Cauli, O; Morelli, M; Pinna, A1
Platt, DM; Rowlett, JK; Spealman, RD; Yao, WD1
Cho, EY; Kim, JH; Kim, KM; Min, C; Park, JH1
Amodeo, LR; Crawford, CA; Der-Ghazarian, T; Gonzalez, AE; Gutierrez, A; Humphrey, DE; McDougall, SA; Valentine, JM; Widarma, CB1

Other Studies

20 other study(ies) available for n-n-propylnorapomorphine and quinpirole

ArticleYear
A functional test identifies dopamine agonists selective for D3 versus D2 receptors.
    Neuroreport, 1995, Jan-26, Volume: 6, Issue:2

    Topics: Animals; CHO Cells; Cricetinae; Dopamine Agents; Humans; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3

1995
CoMFA-based prediction of agonist affinities at recombinant D1 vs D2 dopamine receptors.
    Journal of medicinal chemistry, 1998, Oct-22, Volume: 41, Issue:22

    Topics: Animals; Binding Sites; Databases, Factual; Dopamine Agonists; Humans; Ligands; Macaca mulatta; Models, Molecular; Molecular Conformation; Protein Structure, Secondary; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Recombinant Proteins; Structure-Activity Relationship; Tumor Cells, Cultured

1998
CoMFA-based prediction of agonist affinities at recombinant wild type versus serine to alanine point mutated D2 dopamine receptors.
    Journal of medicinal chemistry, 2000, Aug-10, Volume: 43, Issue:16

    Topics: Alanine; Amino Acid Substitution; Animals; Bromocriptine; Combinatorial Chemistry Techniques; Dopamine Agonists; Models, Molecular; Pergolide; Point Mutation; Radioligand Assay; Rats; Receptors, Dopamine D2; Recombinant Proteins; Serine; Structure-Activity Relationship; Tumor Cells, Cultured

2000
The actions of (-)N-n-propylnorapomorphine and selective dopamine D1 and D2 receptor agonists to modify the release of [3H]dopamine from the rat nucleus accumbens.
    Neuropharmacology, 1990, Volume: 29, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Apomorphine; Benzazepines; Dopamine; Dopamine Agents; Ergolines; Female; Fluphenazine; Motor Activity; Nucleus Accumbens; Potassium; Quinpirole; Rats; Receptors, Dopamine; Septal Nuclei; Sulpiride

1990
The role of multiple dopamine receptors in apomorphine and N-n-propylnorapomorphine-induced climbing and hypothermia.
    European journal of pharmacology, 1990, Mar-20, Volume: 178, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Benzazepines; Body Temperature; Dose-Response Relationship, Drug; Ergolines; Female; Mice; Quinpirole; Receptors, Dopamine; Stereotyped Behavior

1990
Hypothermia in mice: D2 dopamine receptor mediation and absence of spare receptors.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Antagonists; Animals; Apomorphine; Benzazepines; Body Temperature; Dopamine Agents; Dopamine Antagonists; Ergolines; Hypothermia; Male; Mice; Mice, Inbred Strains; Quinolines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride

1989
Dopamine D2 receptor stimulation decreases the inositol trisphosphate level of rat striatal slices.
    European journal of pharmacology, 1987, Apr-14, Volume: 136, Issue:2

    Topics: Animals; Apomorphine; Corpus Striatum; Ergolines; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Sugar Phosphates

1987
Enhancement by the D1 dopamine agonist SKF 38393 of specific components of stereotypy elicited by the D2 agonists LY 171555 and RU 24213.
    Life sciences, 1988, Volume: 42, Issue:25

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Dose-Response Relationship, Drug; Ergolines; Male; Phenethylamines; Quinpirole; Rats; Receptors, Dopamine; Stereotyped Behavior

1988
Interactions of a partial ergoline with dopamine receptors in vivo and in vitro.
    Acta physiologica Scandinavica, 1983, Volume: 117, Issue:2

    Topics: Animals; Apomorphine; Butyrophenones; Cell Membrane; Corpus Striatum; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1983
The D2 dopamine receptor mediates inhibition of growth in GH4ZR7 cells: involvement of protein kinase-C epsilon.
    Endocrinology, 1994, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alprenolol; Animals; Apomorphine; Benzazepines; Butaclamol; Carcinogens; Cell Division; Cell Line; DNA; Dopamine; Ergolines; Humans; Isoenzymes; Kinetics; Norepinephrine; Pertussis Toxin; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Quinpirole; Receptors, Dopamine D2; Salicylamides; Spiperone; Thymidine; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella

1994
Drug-induced up-regulation of dopamine D2 receptors on cultured cells.
    Journal of neurochemistry, 1995, Volume: 65, Issue:2

    Topics: Animals; Apomorphine; Dopamine Agonists; Dopamine Antagonists; Down-Regulation; Ergolines; Macaca mulatta; Quinpirole; Receptors, Dopamine D2; Tumor Cells, Cultured; Up-Regulation

1995
Caffeine cross-tolerance to selective dopamine D1 and D2 receptor agonists but not to their synergistic interaction.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Administration, Oral; Analysis of Variance; Animals; Apomorphine; Caffeine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Drug Tolerance; Ergolines; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2

1994
Monoamine oxidase inhibitors inhibit [3H]quinpirole binding in rat striatal membranes.
    European journal of pharmacology, 1993, Jul-15, Volume: 246, Issue:2

    Topics: Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine Agents; Ergolines; In Vitro Techniques; Kinetics; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenazocine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Spiperone

1993
Specific induction of a functional endogenous D2 short dopamine receptor in GH4C1 cells.
    Biochemical and biophysical research communications, 1993, Jun-15, Volume: 193, Issue:2

    Topics: Animals; Apomorphine; Base Sequence; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Kanamycin Kinase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Phosphotransferases; Pituitary Neoplasms; Polymerase Chain Reaction; Potassium Chloride; Prolactin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Sulpiride; Transfection; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1993
Lack of autoreceptor-mediated inhibitory control of dopamine release in striatal synaptosomes of D2 receptor-deficient mice.
    Brain research, 1998, May-11, Volume: 792, Issue:2

    Topics: 4-Aminopyridine; Amphetamine; Animals; Apomorphine; Autoreceptors; Benzopyrans; Cocaine; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluoresceins; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Mutation; Neural Inhibition; Oxazines; Potassium Chloride; Presynaptic Terminals; Quinpirole; Receptors, Dopamine D2; Synaptosomes; Tritium

1998
Dopamine receptor-modulated [35S]GTPgammaS binding in striatum of 6-hydroxydopamine-lesioned rats.
    Brain research, 1999, Sep-11, Volume: 841, Issue:1-2

    Topics: Animals; Apomorphine; Benzazepines; Bromocriptine; Cell Membrane; Corpus Striatum; Domperidone; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Ligands; Male; Oxidopamine; Piperazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulfur Radioisotopes; Tritium

1999
Subchronic intermittent caffeine administration to unilaterally 6-hydroxydopamine-lesioned rats sensitizes turning behaviour in response to dopamine D(1) but not D(2) receptor agonists.
    Behavioural pharmacology, 2005, Volume: 16, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Caffeine; Central Nervous System Stimulants; Dopamine Agents; Dopamine Agonists; Levodopa; Male; Oxidopamine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Sympathectomy, Chemical; Sympatholytics

2005
Modulation of heroin and cocaine self-administration by dopamine D1- and D2-like receptor agonists in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: Animals; Apomorphine; Behavior, Animal; Benzazepines; Cocaine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Female; Heroin; Injections, Intravenous; Macaca mulatta; Male; Narcotics; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement, Psychology; Self Administration; Vasoconstrictor Agents

2007
Characterization of functional roles of DRY motif in the 2nd intracellular loop of dopamine D2 and D3 receptors.
    Archives of pharmacal research, 2008, Volume: 31, Issue:4

    Topics: Amino Acid Motifs; Apomorphine; Arginine; Aspartic Acid; Cell Line; Cell Membrane; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Mutation; Protein Conformation; Protein Structure, Tertiary; Protein Transport; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Signal Transduction; Spiperone; Sulpiride; Transfection

2008
Behavioral effects of dopamine receptor inactivation in the caudate-putamen of preweanling rats: role of the D2 receptor.
    Psychopharmacology, 2014, Volume: 231, Issue:4

    Topics: Aging; Alkylating Agents; Animals; Apomorphine; Benzazepines; Caudate Nucleus; Dimethyl Sulfoxide; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Lisuride; Male; Motor Activity; Putamen; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Weaning

2014