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n-methylscopolamine and colforsin

n-methylscopolamine has been researched along with colforsin in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's16 (94.12)18.2507
2000's1 (5.88)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aly, MH; el-Fakahany, EE; Forray, C; Mohamed, AS1
Chidiac, P; Nagy, A; Sole, MJ; Wells, JW1
Nathanson, NM; Scherer, NM1
Akerman, KE; Heikkilä, JE1
Barnes, PJ; Haddad, EB; Rousell, J1
Chowdhury, P; Doi, R; Inoue, K; Kaji, H; Rayford, PL1
el-Fakahany, EE; Wang, SZ1
Barnes, PJ; Haddad, EB; Mak, JC; Rousell, J1
Jones, SB; Liston, DR; Ward, KM; Zorn, SH1
Abello, J; Bernard, C; Bosshard, A; Chayvialle, JA; Cuber, JC; Ye, F1
Davis, RE; Jaen, JC; Schwarz, RD; Spencer, CJ; Tecle, H; Thomas, AJ1
Goldman, PS; Nathanson, NM; Schlador, ML; Shapiro, RA1
Alessandro, R; Brilley, E; Felder, CC; Jacobs, W; Kohn, EC; Probst, J1
Olianas, MC; Onali, P1
Maullu, C; Olianas, MC; Onali, P1
Lisá, V; Myslivecek, J; Trojan, S; Tucek, S1
Barak, D; Pittel, Z; Segall, Y1

Reviews

1 review(s) available for n-methylscopolamine and colforsin

ArticleYear
Characterization of muscarinic agonists in recombinant cell lines.
    Life sciences, 1993, Volume: 52, Issue:5-6

    Topics: Animals; Cell Line, Transformed; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; N-Methylscopolamine; Parasympatholytics; Parasympathomimetics; Phosphatidylinositols; Receptors, Muscarinic; Recombination, Genetic; Scopolamine Derivatives

1993

Other Studies

16 other study(ies) available for n-methylscopolamine and colforsin

ArticleYear
Lack of intrinsic activity and significant subtype selectivity of SR 95639A at muscarinic receptors.
    European journal of pharmacology, 1992, Oct-01, Volume: 227, Issue:2

    Topics: Acetylcholine; Animals; Binding Sites; Carbachol; Cerebral Cortex; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Female; Hydrolysis; Inositol Phosphates; Male; Morpholines; N-Methylscopolamine; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Scopolamine Derivatives; Transfection

1992
Inefficient muscarinic transduction in cardiomyopathic Syrian hamsters.
    Journal of molecular and cellular cardiology, 1991, Volume: 23, Issue:11

    Topics: Adenylyl Cyclases; Animals; Carbachol; Cardiomyopathies; Colforsin; Cricetinae; Cyclic AMP; GTP-Binding Proteins; Isoproterenol; Mesocricetus; N-Methylscopolamine; Parasympatholytics; Receptors, Muscarinic; Scopolamine Derivatives; Signal Transduction

1991
Differential regulation by agonist and phorbol ester of cloned m1 and m2 muscarinic acetylcholine receptors in mouse Y1 adrenal cells and in Y1 cells deficient in cAMP-dependent protein kinase.
    Biochemistry, 1990, Sep-11, Volume: 29, Issue:36

    Topics: Adenocarcinoma; Adrenal Gland Neoplasms; Animals; Colforsin; Concanavalin A; Cyclic AMP; Endocytosis; Mice; N-Methylscopolamine; Phorbol Esters; Pilocarpine; Protein Kinases; Quinuclidinyl Benzilate; Receptors, Muscarinic; Recombinant Fusion Proteins; Scopolamine Derivatives; Second Messenger Systems; Thionucleotides; Tumor Cells, Cultured

1990
12-O-tetradecanoylphorbol 13-acetate and forskolin modify muscarinic receptor-linked Ca2+ mobilization in SH-SY5Y neuroblastoma cells through different mechanisms.
    Journal of neurochemistry, 1990, Volume: 54, Issue:2

    Topics: Benzofurans; Binding, Competitive; Biomechanical Phenomena; Calcium; Carbachol; Colforsin; Cytosol; Fluorescent Dyes; Fura-2; Ionomycin; Membrane Potentials; N-Methylscopolamine; Neuroblastoma; Osmolar Concentration; Receptors, Muscarinic; Scopolamine Derivatives; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured

1990
Muscarinic M2 receptor synthesis: study of receptor turnover with propylbenzilylcholine mustard.
    European journal of pharmacology, 1995, Aug-15, Volume: 290, Issue:3

    Topics: Alkylation; Cell Line; Colforsin; Cyclic AMP; Cycloheximide; Fibroblasts; Humans; Kinetics; Muscarinic Antagonists; N-Methylscopolamine; Propylbenzilylcholine Mustard; Protein Synthesis Inhibitors; Radioligand Assay; Receptors, Muscarinic; Scopolamine Derivatives

1995
Structural and functional changes of exocrine pancreas induced by FK506 in rats.
    Gastroenterology, 1993, Volume: 104, Issue:4

    Topics: Amylases; Analysis of Variance; Animals; Atropine; Body Weight; Calcimycin; Calcium; Carbachol; Cholecystokinin; Colforsin; Cytosol; Dose-Response Relationship, Drug; Feeding Behavior; Kinetics; Male; N-Methylscopolamine; Pancreas; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Reference Values; Scopolamine; Scopolamine Derivatives; Secretin; Sincalide; Tacrolimus; Tetradecanoylphorbol Acetate; Time Factors; Trypsinogen; Vasoactive Intestinal Peptide

1993
Application of transfected cell lines in studies of functional receptor subtype selectivity of muscarinic agonists.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Carbachol; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Hydrolysis; N-Methylscopolamine; Phosphatidylinositols; Pilocarpine; Receptors, Muscarinic; Scopolamine Derivatives; Stimulation, Chemical; Substrate Specificity; Transfection

1993
Transcriptional down-regulation of m2 muscarinic receptor gene expression in human embryonic lung (HEL 299) cells by protein kinase C.
    The Journal of biological chemistry, 1995, Mar-31, Volume: 270, Issue:13

    Topics: Blotting, Northern; Cell Line; Cell Nucleus; Colforsin; Cycloheximide; Dactinomycin; Embryo, Mammalian; Gene Expression Regulation; Half-Life; Humans; Indoles; Kinetics; Lung; Maleimides; N-Methylscopolamine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Muscarinic; RNA, Messenger; Scopolamine Derivatives; Time Factors; Transcription, Genetic

1995
Clozapine is a potent and selective muscarinic M4 receptor agonist.
    European journal of pharmacology, 1994, Nov-15, Volume: 269, Issue:3

    Topics: Animals; Carbachol; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Humans; Hydrolysis; Muscarinic Agonists; N-Methylscopolamine; Parasympatholytics; Phosphatidylinositols; Salivation; Scopolamine Derivatives

1994
Stimulation of glucagon-like peptide-1 secretion by muscarinic agonist in a murine intestinal endocrine cell line.
    Endocrinology, 1994, Volume: 134, Issue:5

    Topics: Calcium; Carbachol; Cell Line; Colforsin; Cyclic AMP; Endocrine Glands; Glucagon; Glucagon-Like Peptide 1; Intestinal Mucosa; Intestines; Kinetics; Muscarinic Antagonists; N-Methylscopolamine; Parasympathomimetics; Peptide Fragments; Protein Precursors; Receptors, Muscarinic; Scopolamine Derivatives; Tetradecanoylphorbol Acetate

1994
Identification of a region required for subtype-specific agonist-induced sequestration of the m2 muscarinic acetylcholine receptor.
    The Journal of biological chemistry, 1996, Feb-23, Volume: 271, Issue:8

    Topics: Amino Acid Sequence; Carbachol; Cell Line; Colforsin; Humans; Kinetics; Luciferases; Models, Structural; Molecular Sequence Data; Muscarinic Agonists; N-Methylscopolamine; Polymerase Chain Reaction; Protein Structure, Secondary; Quinuclidinyl Benzilate; Receptor, Muscarinic M2; Receptors, Muscarinic; Recombinant Fusion Proteins; Restriction Mapping; Scopolamine Derivatives; Sequence Homology, Amino Acid; Transfection; Tumor Cells, Cultured

1996
Identification and molecular characterization of a m5 muscarinic receptor in A2058 human melanoma cells. Coupling to inhibition of adenylyl cyclase and stimulation of phospholipase A2.
    The Journal of biological chemistry, 1996, Jul-19, Volume: 271, Issue:29

    Topics: Adenylyl Cyclase Inhibitors; Arachidonic Acid; Base Sequence; Blotting, Southern; Calcium; Carbachol; Cell Adhesion; Cell Division; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; DNA Primers; Egtazic Acid; Humans; Inositol 1,4,5-Trisphosphate; Kinetics; Melanoma; Molecular Sequence Data; N-Methylscopolamine; Phospholipases A; Phospholipases A2; Polymerase Chain Reaction; Receptor, Muscarinic M5; Receptors, Muscarinic; Scopolamine Derivatives; Signal Transduction; Time Factors; Tumor Cells, Cultured

1996
Impairment of muscarinic stimulation of adenylyl cyclase by heparin in rat olfactory bulb.
    Life sciences, 1997, Volume: 61, Issue:5

    Topics: Adenylyl Cyclases; Animals; Carbachol; Colforsin; Corpus Striatum; Enzyme Activation; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Heparin; In Vitro Techniques; Kinetics; Male; Muscarinic Agonists; N-Methylscopolamine; Olfactory Bulb; Parasympatholytics; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Scopolamine Derivatives

1997
Effects of clozapine on rat striatal muscarinic receptors coupled to inhibition of adenylyl cyclase activity and on the human cloned m4 receptor.
    British journal of pharmacology, 1997, Volume: 122, Issue:3

    Topics: Adenylyl Cyclases; Alkylation; Animals; Cell Membrane; CHO Cells; Clozapine; Colforsin; Corpus Striatum; Cricetinae; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Humans; In Vitro Techniques; Male; Muscarinic Antagonists; N-Methylscopolamine; Protein Binding; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Synaptosomes

1997
Heterologous regulation of muscarinic and beta-adrenergic receptors in rat cardiomyocytes in culture.
    Life sciences, 1998, Volume: 63, Issue:13

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; Bucladesine; Carbachol; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Inhibitors; Female; Indoles; Isoproterenol; Isoquinolines; Kinetics; Male; Maleimides; Muscarinic Agonists; Myocardium; N-Methylscopolamine; Propanolamines; Protein Kinase C; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Sulfonamides; Thionucleotides; Tritium

1998
Function-specific blockage of M(1) and M(3) muscarinic acetylcholine receptors by VX and echothiophate.
    Brain research, 2006, Apr-26, Volume: 1085, Issue:1

    Topics: Animals; Atropine; CHO Cells; Cholinesterase Inhibitors; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Echothiophate Iodide; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Organothiophosphorus Compounds; Oxotremorine; Phosphatidylinositols; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Transfection; Tritium

2006