n-dansyl-3-aminobenzeneboronic acid and benzo(b)thiophene-2-boronic acid

n-dansyl-3-aminobenzeneboronic acid has been researched along with benzo(b)thiophene-2-boronic acid in 2 studies

Compound Research Comparison

Studies (n-dansyl-3-aminobenzeneboronic acid)	Trials (n-dansyl-3-aminobenzeneboronic acid)	Recent Studies (post-2010) (n-dansyl-3-aminobenzeneboronic acid)	Studies (benzo(b)thiophene-2-boronic acid)	Trials (benzo(b)thiophene-2-boronic acid)	Recent Studies (post-2010) (benzo(b)thiophene-2-boronic acid)
6	0	0	17	0	3

Protein Interaction Comparison

Protein	Taxonomy	benzo(b)thiophene-2-boronic acid (IC50)
B2 bradykinin receptor	Cavia porcellus (domestic guinea pig)	0.2
Acyl-protein thioesterase 1	Homo sapiens (human)	1.4145
Acyl-protein thioesterase 2	Homo sapiens (human)	1.4145
Chymotrypsinogen A	Bos taurus (cattle)	5
Beta-lactamase	Escherichia coli K-12	0.2083
5-hydroxytryptamine receptor 1A	Rattus norvegicus (Norway rat)	2.6
5-hydroxytryptamine receptor 1B	Rattus norvegicus (Norway rat)	5
5-hydroxytryptamine receptor 1D	Rattus norvegicus (Norway rat)	5
5-hydroxytryptamine receptor 1F	Rattus norvegicus (Norway rat)	5
Fatty-acid amide hydrolase 1	Rattus norvegicus (Norway rat)	0.15
Monoglyceride lipase	Homo sapiens (human)	0.15

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	1 (50.00)	18.2507
2000's	1 (50.00)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Baquero, F; Blázquez, J; Shoichet, BK; Weston, GS	1
Fischer, DS; Gerards, T; Inglis, SR; Luxen, A; Schofield, CJ; Teller, N; Woon, EC; Zervosen, A	1

Other Studies

2 other study(ies) available for n-dansyl-3-aminobenzeneboronic acid and benzo(b)thiophene-2-boronic acid

Article	Year
Structure-based enhancement of boronic acid-based inhibitors of AmpC beta-lactamase. Journal of medicinal chemistry, 1998, Nov-05, Volume: 41, Issue:23 Topics: Anti-Bacterial Agents; Bacterial Proteins; beta-Lactam Resistance; beta-Lactamase Inhibitors; beta-Lactamases; Binding Sites; Boronic Acids; Crystallography, X-Ray; Drug Synergism; Enterobacter cloacae; Enzyme Inhibitors; Escherichia coli; Microbial Sensitivity Tests; Models, Molecular; Structure-Activity Relationship; Thiophenes	1998
Synthesis and evaluation of 3-(dihydroxyboryl)benzoic acids as D,D-carboxypeptidase R39 inhibitors. Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19 Topics: Actinomycetales; Anti-Bacterial Agents; Bacterial Proteins; Benzoic Acid; Boronic Acids; Carboxypeptidases; Enzyme Inhibitors; Inhibitory Concentration 50; Structure-Activity Relationship	2009

Article

Year

Structure-based enhancement of boronic acid-based inhibitors of AmpC beta-lactamase.

Journal of medicinal chemistry, 1998, Nov-05, Volume: 41, Issue:23

Topics: Anti-Bacterial Agents; Bacterial Proteins; beta-Lactam Resistance; beta-Lactamase Inhibitors; beta-Lactamases; Binding Sites; Boronic Acids; Crystallography, X-Ray; Drug Synergism; Enterobacter cloacae; Enzyme Inhibitors; Escherichia coli; Microbial Sensitivity Tests; Models, Molecular; Structure-Activity Relationship; Thiophenes

1998

Synthesis and evaluation of 3-(dihydroxyboryl)benzoic acids as D,D-carboxypeptidase R39 inhibitors.

Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

Topics: Actinomycetales; Anti-Bacterial Agents; Bacterial Proteins; Benzoic Acid; Boronic Acids; Carboxypeptidases; Enzyme Inhibitors; Inhibitory Concentration 50; Structure-Activity Relationship

2009