n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine has been researched along with quisinostat in 1 studies
Studies (n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine) | Trials (n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine) | Recent Studies (post-2010) (n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine) | Studies (quisinostat) | Trials (quisinostat) | Recent Studies (post-2010) (quisinostat) |
---|---|---|---|---|---|
79 | 1 | 16 | 71 | 3 | 63 |
Protein | Taxonomy | n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine (IC50) | quisinostat (IC50) |
---|---|---|---|
Histone deacetylase 8 | Schistosoma mansoni | 0.3034 | |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | 0.039 | |
Histone deacetylase 3 | Homo sapiens (human) | 0.0039 | |
Cytochrome P450 3A4 | Homo sapiens (human) | 0.0001 | |
Cytochrome P450 2D6 | Homo sapiens (human) | 0.0001 | |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | 0.019 | |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | 0.054 | |
Histone deacetylase 4 | Homo sapiens (human) | 0.0026 | |
Histone deacetylase 1 | Homo sapiens (human) | 0.0009 | |
Histone deacetylase 7 | Homo sapiens (human) | 0.0424 | |
Histone deacetylase 2 | Homo sapiens (human) | 0.0018 | |
Polyamine deacetylase HDAC10 | Homo sapiens (human) | 0.0082 | |
Histone deacetylase 11 | Homo sapiens (human) | 0.0004 | |
Histone deacetylase 8 | Homo sapiens (human) | 0.078 | |
Histone deacetylase 6 | Homo sapiens (human) | 0.0664 | |
Histone deacetylase 9 | Homo sapiens (human) | 0.0151 | |
Histone deacetylase 5 | Homo sapiens (human) | 0.0049 | |
Nuclear receptor corepressor 2 | Homo sapiens (human) | 0.0049 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 1 (100.00) | 2.80 |
Authors | Studies |
---|---|
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M | 1 |
1 other study(ies) available for n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine and quisinostat
Article | Year |
---|---|
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries | 2023 |