Page last updated: 2024-09-03

n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine and metergoline

n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine has been researched along with metergoline in 1 studies

Compound Research Comparison

Studies
(n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine)
Trials
(n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine)
Recent Studies (post-2010)
(n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine)
Studies
(metergoline)
Trials
(metergoline)
Recent Studies (post-2010) (metergoline)
791166563744

Protein Interaction Comparison

ProteinTaxonomyn-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine (IC50)metergoline (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.0007
Bile salt export pumpHomo sapiens (human)10
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)0.366
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.0041
Alpha-2A adrenergic receptorHomo sapiens (human)0.058
Cytochrome P450 2D6Homo sapiens (human)0.2
D(2) dopamine receptorHomo sapiens (human)0.063
Alpha-2B adrenergic receptorHomo sapiens (human)0.016
Alpha-2C adrenergic receptorHomo sapiens (human)0.189
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0062
Substance-K receptorHomo sapiens (human)4.071
D(1A) dopamine receptorHomo sapiens (human)0.074
AcetylcholinesteraseHomo sapiens (human)1.344
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.366
Histamine H2 receptorHomo sapiens (human)0.975
Alpha-1D adrenergic receptorHomo sapiens (human)0.136
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0004
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0007
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.0062
Sodium-dependent serotonin transporterHomo sapiens (human)0.59
Histamine H1 receptorHomo sapiens (human)4.133
D(3) dopamine receptorHomo sapiens (human)0.0077
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0004
5-hydroxytryptamine receptor 6Homo sapiens (human)0.028
Sodium-dependent dopamine transporter Homo sapiens (human)0.063

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1

Other Studies

1 other study(ies) available for n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamine and metergoline

ArticleYear
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016