Page last updated: 2024-09-02

n-(1-methyl-2-phenylethyl)adenosine and colforsin

n-(1-methyl-2-phenylethyl)adenosine has been researched along with colforsin in 4 studies

Compound Research Comparison

Studies
(n-(1-methyl-2-phenylethyl)adenosine)
Trials
(n-(1-methyl-2-phenylethyl)adenosine)
Recent Studies (post-2010)
(n-(1-methyl-2-phenylethyl)adenosine)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
1340413,460461,298

Protein Interaction Comparison

ProteinTaxonomyn-(1-methyl-2-phenylethyl)adenosine (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19901 (25.00)18.7374
1990's2 (50.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
López-Novoa, JM; Olivera, A; Tomás, M1
Parsons, WJ; Pierson, G; Stiles, GL; Sunay, S1
Andrés, A; Cubero, A; Fernández, M; Gonzalez-Calero, G; Ros, M; Ruiz, A; Sanz, JM1
Erdmann, A; Gao, ZG; IJzerman, AP; Jacobson, KA; Kim, SG; Melman, N; Müller, CE1

Other Studies

4 other study(ies) available for n-(1-methyl-2-phenylethyl)adenosine and colforsin

ArticleYear
Effect of adenosine A1 and A2 agonists and antagonists on cAMP and Ca2+ in cultured rat mesangial cells.
    The American journal of physiology, 1992, Volume: 262, Issue:4 Pt 1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Glomerular Mesangium; Purines; Rats; Sulfonamides; Xanthines

1992
The rat testicular A1 adenosine receptor-adenylate cyclase system.
    Endocrinology, 1986, Volume: 119, Issue:4

    Topics: Adenosine; Adenylyl Cyclases; Affinity Labels; Animals; Colforsin; Guanylyl Imidodiphosphate; Iodine Radioisotopes; Isoproterenol; Male; Phenylisopropyladenosine; Photochemistry; Rats; Rats, Inbred Strains; Receptors, Purinergic; Solubility; Testis

1986
Desensitization and internalization of adenosine A1 receptors in rat brain by in vivo treatment with R-PIA: involvement of coated vesicles.
    Biochimica et biophysica acta, 1996, Jan-10, Volume: 1310, Issue:1

    Topics: Adenosine; Adenylyl Cyclase Inhibitors; Animals; Brain; Coated Vesicles; Colforsin; Enzyme Activation; Guanosine Triphosphate; Immunoblotting; Intracellular Membranes; Male; Microsomes; Purinergic P1 Receptor Agonists; Radioligand Assay; Rats; Rats, Wistar; Receptors, Purinergic P1; Vasodilator Agents; Xanthines

1996
Differential allosteric modulation by amiloride analogues of agonist and antagonist binding at A(1) and A(3) adenosine receptors.
    Biochemical pharmacology, 2003, Feb-15, Volume: 65, Issue:4

    Topics: Adenosine; Allosteric Regulation; Amiloride; Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Diuretics; Dose-Response Relationship, Drug; Drug Interactions; Humans; Imidazoles; Kinetics; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Radioligand Assay; Receptor, Adenosine A2A; Receptor, Adenosine A3; Receptors, Purinergic P1; Transfection; Tritium; Xanthines

2003