Page last updated: 2024-09-03

n(alpha)-tosyl-(3-amidinophenyl)alanine piperidide and n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide

n(alpha)-tosyl-(3-amidinophenyl)alanine piperidide has been researched along with n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide in 3 studies

Compound Research Comparison

Studies
(n(alpha)-tosyl-(3-amidinophenyl)alanine piperidide)
Trials
(n(alpha)-tosyl-(3-amidinophenyl)alanine piperidide)
Recent Studies (post-2010)
(n(alpha)-tosyl-(3-amidinophenyl)alanine piperidide)
Studies
(n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide)
Trials
(n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide)
Recent Studies (post-2010) (n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide)
11005202

Protein Interaction Comparison

ProteinTaxonomyn(alpha)-tosyl-(3-amidinophenyl)alanine piperidide (IC50)n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide (IC50)
ProthrombinHomo sapiens (human)0.69
Trypsin-1Homo sapiens (human)0.169
Trypsin-2Homo sapiens (human)0.169
Trypsin-3Homo sapiens (human)0.169

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19901 (33.33)18.7374
1990's2 (66.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hoffmann, J; Markwardt, F; Nowak, G1
Bauer, M; Bergner, A; Bode, W; Brandstetter, H; Stürzebecher, J1
Prasa, D; Stürzebecher, J; Vieweg, H; Wikström, P1

Other Studies

3 other study(ies) available for n(alpha)-tosyl-(3-amidinophenyl)alanine piperidide and n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide

ArticleYear
Comparative studies on thrombin inhibitors in experimental microthrombosis.
    Thrombosis and haemostasis, 1983, Jun-28, Volume: 49, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Arginine; Dipeptides; Female; Fibrinogen; Hirudins; Kinetics; Lung; Male; Microcirculation; para-Aminobenzoates; Piperidines; Rats; Rats, Inbred Strains; Thrombin; Thrombosis

1983
The X-ray crystal structure of thrombin in complex with N alpha-2-naphthylsulfonyl-L-3-amidino-phenylalanyl-4-methylpiperidide: the beneficial effect of filling out an empty cavity.
    Journal of enzyme inhibition, 1995, Volume: 9, Issue:1

    Topics: Alanine; Antithrombins; Binding Sites; Computer Graphics; Crystallography, X-Ray; Dipeptides; Models, Molecular; Piperidines; Protein Binding; Serine Proteinase Inhibitors; Thrombin

1995
Structure-activity relationships of inhibitors derived from 3-amidinophenylalanine.
    Journal of enzyme inhibition, 1995, Volume: 9, Issue:1

    Topics: Amidines; Animals; Antithrombins; Cattle; Crystallography, X-Ray; Dipeptides; Factor Xa Inhibitors; Molecular Structure; Piperidines; Serine Proteinase Inhibitors; Stereoisomerism; Structure-Activity Relationship; Thrombin

1995