Compounds > n(alpha)-(4-toluenesulfonyl)-4-amidinophenylalanylpiperidine
Page last updated: 2024-09-04

n(alpha)-(4-toluenesulfonyl)-4-amidinophenylalanylpiperidine and piperidines

n(alpha)-(4-toluenesulfonyl)-4-amidinophenylalanylpiperidine has been researched along with piperidines in 4 studies

Compound Research Comparison

Studies
(n(alpha)-(4-toluenesulfonyl)-4-amidinophenylalanylpiperidine)		Trials
(n(alpha)-(4-toluenesulfonyl)-4-amidinophenylalanylpiperidine)		Recent Studies (post-2010)
(n(alpha)-(4-toluenesulfonyl)-4-amidinophenylalanylpiperidine)		Studies
(piperidines)		Trials
(piperidines)		Recent Studies (post-2010) (piperidines)
50040,2355,22114,545

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (50.00)18.2507
2000's2 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bode, W; Brandstetter, H; Edwards, BF; Grosse, D; Hoeffken, HW; Martin, PD; Stürzebecher, J; Turk, D1
Bode, W; Stürzebecher, J; Turk, D1
O'Brien, LA; Sutherland, JJ; Weaver, DF1
Fonseca, N; Henriques, ES; Ramos, MJ1

Other Studies

4 other study(ies) available for n(alpha)-(4-toluenesulfonyl)-4-amidinophenylalanylpiperidine and piperidines

ArticleYear
Refined 2.3 A X-ray crystal structure of bovine thrombin complexes formed with the benzamidine and arginine-based thrombin inhibitors NAPAP, 4-TAPAP and MQPA. A starting point for improving antithrombotics.
    Journal of molecular biology, 1992, Aug-20, Volume: 226, Issue:4

    Topics: Amidines; Amino Acid Sequence; Animals; Antithrombins; Arginine; Benzamidines; Binding Sites; Cattle; Crystallography; Dipeptides; Fibrinolytic Agents; Hydrogen Bonding; Ligands; Models, Molecular; Molecular Sequence Data; Pipecolic Acids; Piperidines; Protein Conformation; Structure-Activity Relationship; Sulfonamides; Thrombin

1992
Geometry of binding of the N alpha-tosylated piperidides of m-amidino-, p-amidino- and p-guanidino phenylalanine to thrombin and trypsin. X-ray crystal structures of their trypsin complexes and modeling of their thrombin complexes.
    FEBS letters, 1991, Aug-05, Volume: 287, Issue:1-2

    Topics: Amidines; Animals; Binding Sites; Cattle; Guanidines; Models, Molecular; Molecular Structure; Piperidines; Stereoisomerism; Thrombin; Trypsin; X-Ray Diffraction

1991
Pruned receptor surface models and pharmacophores for three-dimensional database searching.
    Journal of medicinal chemistry, 2004, Jul-15, Volume: 47, Issue:15

    Topics: Amidines; Angiotensin-Converting Enzyme Inhibitors; Benzodiazepines; Celecoxib; Cholinesterase Inhibitors; Cyclooxygenase 2; Databases, Factual; Donepezil; Enalapril; Enzymes; Estradiol; Imidazoles; Indans; Isoenzymes; Ligands; Models, Molecular; Molecular Structure; Naphthalenes; Piperidines; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Quantitative Structure-Activity Relationship; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Estrogen; Receptors, GABA-A; Sulfonamides; Thrombin

2004
On the modeling of snake venom serine proteinase interactions with benzamidine-based thrombin inhibitors.
    Protein science : a publication of the Protein Society, 2004, Volume: 13, Issue:9

    Topics: Amidines; Amino Acid Sequence; Animals; Benzamidines; Binding Sites; Bothrops; Crotalid Venoms; Dipeptides; Glycoproteins; Kallikreins; Models, Molecular; Molecular Sequence Data; Piperidines; Protein Conformation; Sequence Homology, Amino Acid; Serine Endopeptidases; Serine Proteinase Inhibitors; Static Electricity; Structural Homology, Protein; Thrombin; Water

2004