n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide and benzamidine

n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide has been researched along with benzamidine in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bode, W; Brandstetter, H; Edwards, BF; Grosse, D; Hoeffken, HW; Martin, PD; Stürzebecher, J; Turk, D1
Banner, DW; Hadváry, P1
Jenneboer, AJ; Lucas, H; Noach, AB; Rewinkel, JB; Rood, AM; van Boeckel, CA; van Dinther, TG; van Galen, PJ1

Other Studies

3 other study(ies) available for n(alpha)-(2-naphthylsulfonylglycyl)-4-amidinophenylalanine piperidide and benzamidine

ArticleYear
Refined 2.3 A X-ray crystal structure of bovine thrombin complexes formed with the benzamidine and arginine-based thrombin inhibitors NAPAP, 4-TAPAP and MQPA. A starting point for improving antithrombotics.
    Journal of molecular biology, 1992, Aug-20, Volume: 226, Issue:4

    Topics: Amidines; Amino Acid Sequence; Animals; Antithrombins; Arginine; Benzamidines; Binding Sites; Cattle; Crystallography; Dipeptides; Fibrinolytic Agents; Hydrogen Bonding; Ligands; Models, Molecular; Molecular Sequence Data; Pipecolic Acids; Piperidines; Protein Conformation; Structure-Activity Relationship; Sulfonamides; Thrombin

1992
Crystallographic analysis at 3.0-A resolution of the binding to human thrombin of four active site-directed inhibitors.
    The Journal of biological chemistry, 1991, Oct-25, Volume: 266, Issue:30

    Topics: Amino Acid Chloromethyl Ketones; Antithrombins; Arginine; Benzamidines; Binding Sites; Dipeptides; Humans; Models, Molecular; Pipecolic Acids; Piperidines; Stereoisomerism; Sulfonamides; Thrombin; Trypsin

1991
1-Aminoisoquinoline as benzamidine isoster in the design and synthesis of orally active thrombin inhibitors.
    Bioorganic & medicinal chemistry letters, 1999, Mar-08, Volume: 9, Issue:5

    Topics: Administration, Oral; Anticoagulants; Benzamidines; Caco-2 Cells; Dipeptides; Drug Design; Humans; Isoquinolines; Piperidines; Thrombin; Trypsin Inhibitors

1999