muscimol has been researched along with tert-butylbicyclophosphorothionate in 96 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 46 (47.92) | 18.7374 |
1990's | 41 (42.71) | 18.2507 |
2000's | 8 (8.33) | 29.6817 |
2010's | 1 (1.04) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM | 1 |
Ehrmann, ML; Mileson, BE; Schwartz, RD | 1 |
Kukulka, KM; Mans, AM; McAvoy, KJ; Rokosz, NC | 1 |
Koenig, JA; Martin, IL | 1 |
Kokka, N; Olsen, RW; Sapp, DW; Witte, U | 1 |
Banerjee, PK; Depaulis, A; Hechler, V; Snead, OC; Vergnes, M | 1 |
Galpern, WR; Greenblatt, DJ; Lumpkin, M; Miller, LG; Shader, RI | 1 |
Chesley, S; Greenblatt, DJ; Lopez, F; Miller, LG; Schatzki, A; Shader, RI | 1 |
Chesley, S; Greenblatt, DJ; Lopez, F; Miller, LG; Schatzki, A; Shader, RI; Thompson, ML | 1 |
Niles, L | 1 |
Basile, AS | 1 |
Biggio, G; Concas, A; Sanna, E; Santoro, G; Serra, M | 1 |
Farb, DH; Farrant, M; Roca, DJ; Rozenberg, I | 1 |
Barnard, EA; Devine, J; Macdonald, RL; Moss, SJ; Nayeem, N; Porter, NM; Smart, TG; Stephenson, FA | 1 |
Braestrup, C; Honore, T; Nielsen, M | 1 |
Barnard, EA; Casalotti, SO; Mamalaki, C; Stephenson, FA | 1 |
Cole, RJ; Eldefrawi, AT; Eldefrawi, ME; Gant, DB; Valdes, JJ | 1 |
Majewska, MD | 1 |
Greenblatt, DJ; Miller, LG; Roy, RB; Shader, RI; Summer, WR | 1 |
Moody, EJ; Paul, SM; Skolnick, P; Suzdak, PD | 1 |
Bleck, V; Harris, RA; Lewin, E; Peris, J; Zahniser, NR | 2 |
Maggi, A; Perez, J; Zucchi, I | 1 |
Greenblatt, DJ; Kaplan, GB; Lopez, F; Miller, LG; Shader, RI | 1 |
Biggio, G; Cau, A; Corda, MG; Laudani, U; Longoni, B; Paci, S; Salvadori, S | 1 |
Ho, IK; Ito, Y; Lim, DK; Nabeshima, T | 1 |
Olsen, RW; Ransom, RW; Turner, DM; Yang, JS | 1 |
Paul, SM; Schwartz, RD; Seale, TW; Skolnick, P | 1 |
Biggio, G; Concas, A; Corda, MG; Serra, M | 1 |
Erdö, SL; Wolff, JR | 1 |
Bowen, DM; Cross, AJ; Francis, PT; Green, AR; Robinson, TN; Stirling, JM | 1 |
Lopez, F; Miller, LG; Roy, RB; Weill, CL | 1 |
Moguilewsky, M; Philibert, D; Shu, C; Vincens, M | 1 |
Allan, AM; Buck, KJ; Harris, RA | 1 |
Ho, IK; Hoskins, B; Ito, Y; Lim, DK | 1 |
Abalis, IM; Eldefrawi, AT; Eldefrawi, ME | 1 |
Hamon, M | 1 |
Chiu, TH; Ito, M; Yu, O | 1 |
Atsoggiu, T; Biggio, G; Concas, A; Serra, M | 1 |
Braestrup, C; Nielsen, M | 1 |
Barnes, EM; Tehrani, MH | 1 |
Haefely, W; Möhler, H; Richards, JG; Schoch, P | 1 |
Stephenson, FA | 2 |
Chiu, TH; Ito, M; Rosenberg, HC | 1 |
Creveling, CR; Daly, JW; Hollingsworth, EB; Lewandowski, G; Waters, JA | 1 |
Häring, P; Mohler, H; Richards, JG; Schoch, P; Takacs, B | 1 |
Chow, SC; Holan, G; Johnston, GA; Lummis, SC | 1 |
Crofton, KM; Mailman, RB; Reiter, LW | 1 |
Majewska, MD; Schwartz, RD | 1 |
Barker, JL; Harrington, JW; Harrison, NL; Majewska, MD | 1 |
Allan, AM; Harris, RA | 1 |
Gallo, V; Guidotti, A; Vaccarino, F; Wise, BC | 1 |
Casida, JE; Cole, LM; Lawrence, LJ | 1 |
Braestrup, C; Tacke, U | 1 |
Braunwalder, A; Cheney, DL; Loo, P; Wood, PL | 1 |
Borea, PA; Karobath, M; Supavilai, P | 1 |
Bymaster, FP; Squires, RF; Threlkeld, PG; Wong, DT | 1 |
Barnard, EA; Sigel, E | 1 |
Karobath, M; Supavilai, P | 1 |
Camón, L; Martínez, E; Pazos, A; Rodríguez-Farré, E; Solà, C | 1 |
Imaizumi, M; Machida, H; Miyazaki, S | 1 |
Burnham, WM; Lôscher, W; Nobrega, JN; Richter, A | 1 |
Biggio, G; Concas, A; Cuccheddu, T; Maciocco, E; Santoro, G; Serra, M | 1 |
Clark, M; Massenburg, GS; Post, RM; Weiss, SR | 1 |
Chen, DZ; Chen, SH; Katsura, M; Kuriyama, K; Ohkuma, S | 1 |
Allan, AM; Harris, RA; McQuilkin, SJ; Mihic, SJ; Whatley, VJ | 1 |
Samochocki, M; Strosznajder, J | 2 |
Belelli, D; Chen, R; Lambert, JJ; Lan, NC; Peters, JA; Reyes, A | 1 |
Ho, IK; Kim, HS; Kimura, T; Oh, KW; Rheu, HM; Saunders, PA | 1 |
Ho, IK; Ito, Y | 1 |
Crawley, JN; Drugan, RC; Paul, SM | 1 |
Airaksinen, MM; Nieminen, SA; Railoma, O; Titievsky, AV | 1 |
Korpi, ER; Seeburg, PH | 1 |
Liu, CC; Snead, OC | 1 |
Carter, DB; Im, WB; Pregenzer, JF; Thomsen, DR | 1 |
Ho, IK; Miyaoka, T; Tseng, YT | 1 |
Korpi, ER; Lüddens, H; Wong, G | 1 |
Biggio, G; Ghiani, CA; Maciocco, E; Sanna, E; Serra, M; Tuligi, G | 1 |
Sieghart, W; Slany, A; Zezula, J | 1 |
Karle, J; Nielsen, M; Witt, MR | 1 |
Hedblom, E; Kirkness, EF | 1 |
Mehta, AK; Ticku, MK | 2 |
Acosta-Burruel, M; Carter, RB; Chen, JS; Drewe, JA; Hawkinson, JE; Hogenkamp, DJ; Lan, NC; Upasani, RB; Whittemore, ER; Woodward, RM; Yang, KC | 1 |
Ho, IK; Jang, CG; Ma, T; Oh, S | 1 |
Cooper, RL; Meacham, CA; Shafer, TJ; Ward, TR | 1 |
Burton, G; Dodd, RH; Furtmüller, R; Ghini, AA; Nicoletti, D; Sieghart, W | 1 |
Korpi, ER; Lüddens, H; Panula, P; Särkioja, T; Sinkkonen, ST; Tiihonen, J; Tupala, E; Uusi-Oukari, M | 1 |
Atack, JR; Bromidge, F; Collinson, N; Dawson, GR; Hadingham, KL; Howell, O; Macaulay, A; McKernan, RM; Myers, J; Newman, R; O'Meara, G; Reynolds, DS; Rosahl, TW; Sur, C; Wafford, KA; Whiting, PJ | 1 |
Chigr, F; M'hamed, SB; Najimi, M | 1 |
Akk, G; Bracamontes, JR; Covey, DF; Darbandi-Tonkabon, R; Evers, AS; Hastings, WR; Manion, BD; Mennerick, SJ; Steinbach, JH; Zeng, CM | 1 |
Abuhamdah, S; Chazot, PL; Fürstner, A; Lees, G | 1 |
Fan, LW; Ho, IK; Loh, HH; Ma, T; Tien, LT | 1 |
Burton, G; Coirini, H; Ghini, AA; Kruse, MS; Rey, M; Veleiro, AS | 1 |
4 review(s) available for muscimol and tert-butylbicyclophosphorothionate
Article | Year |
---|---|
The role of receptor binding in drug discovery.
Topics: Animals; Drug Design; Humans; Receptors, Drug | 1993 |
[GABA receptors in the central nervous system. Biochemical and pharmacological aspects].
Topics: Allosteric Site; Animals; Anti-Anxiety Agents; Barbiturates; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; gamma-Aminobutyric Acid; Humans; Muscimol; Picrotoxin; Receptors, GABA-A | 1987 |
Benzodiazepine receptors resolved.
Topics: Animals; Antibodies, Monoclonal; Autoradiography; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Histocytochemistry; Humans; Immunologic Techniques; Ionophores; Muscimol; Neurons; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Spinal Cord; Synapses; Tissue Distribution | 1986 |
Distinction of benzodiazepine receptor agonists and inverse agonists by binding studies in vitro.
Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Etazolate; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Muscimol; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
92 other study(ies) available for muscimol and tert-butylbicyclophosphorothionate
Article | Year |
---|---|
Alterations in the gamma-aminobutyric acid-gated chloride channel following transient forebrain ischemia in the gerbil.
Topics: Animals; Autoradiography; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; gamma-Aminobutyric Acid; Gerbillinae; Ion Channel Gating; Ischemic Attack, Transient; Male; Membrane Proteins; Motor Activity; Muscimol | 1992 |
Regional distribution and kinetics of three sites on the GABAA receptor: lack of effect of portacaval shunting.
Topics: Animals; Autoradiography; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Flumazenil; Flunitrazepam; Image Processing, Computer-Assisted; Kinetics; Male; Muscimol; Portacaval Shunt, Surgical; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tissue Distribution | 1992 |
Effect of free fatty acids on GABAA receptor ligand binding.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Fatty Acids, Nonesterified; Flunitrazepam; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1992 |
Sex differences in sensitivity to pentylenetetrazol but not in GABAA receptor binding.
Topics: Anesthetics; Animals; Anticonvulsants; Autoradiography; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; Electroshock; Ethanol; Female; Flunitrazepam; Male; Muscimol; Orchiectomy; Ovariectomy; Pentylenetetrazole; Pregnanediones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sex Characteristics | 1992 |
The GABAA receptor complex in experimental absence seizures in rat: an autoradiographic study.
Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Convulsants; Epilepsy, Absence; Flunitrazepam; GABA-A Receptor Antagonists; Ion Channels; Ionophores; Male; Membrane Proteins; Muscimol; Organ Specificity; Pyramidal Tracts; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Tritium | 1992 |
Chronic benzodiazepine administration. VII. Behavioral tolerance and withdrawal and receptor alterations associated with clonazepam administration.
Topics: Animals; Behavior, Animal; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Clonazepam; Convulsants; Drug Tolerance; Flumazenil; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome | 1991 |
Chronic administration of benzodiazepines--V. Rapid onset of behavioral and neurochemical alterations after discontinuation of alprazolam.
Topics: Alprazolam; Animals; Behavior, Animal; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Down-Regulation; Drug Tolerance; Ion Channels; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome; Sulfur Radioisotopes | 1990 |
Chronic morphine administration augments benzodiazepine binding and GABAA receptor function.
Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; Flunitrazepam; In Vitro Techniques; Ion Channels; Male; Mice; Morphine; Muscimol; Naltrexone; Radioisotopes; Receptors, GABA-A; Sulfur Radioisotopes | 1990 |
Melatonin interaction with the benzodiazepine-GABA receptor complex in the CNS.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Chlorides; Diazepam; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Ion Channels; Melatonin; Muscimol; Prosencephalon; Rats; Receptors, GABA-A; Serotonin; Synaptosomes | 1991 |
The contribution of endogenous benzodiazepine receptor ligands to the pathogenesis of hepatic encephalopathy.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Diazepam; Flumazenil; Hepatic Encephalopathy; Kinetics; Ligands; Male; Mass Spectrometry; Muscimol; Peripheral Nerves; Rabbits; Radioligand Assay; Receptors, GABA-A; Sulfur Radioisotopes | 1991 |
Neurochemical action of the general anaesthetic propofol on the chloride ion channel coupled with GABAA receptors.
Topics: Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Flunitrazepam; Male; Membrane Proteins; Muscimol; Propofol; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1991 |
Chronic agonist exposure induces down-regulation and allosteric uncoupling of the gamma-aminobutyric acid/benzodiazepine receptor complex.
Topics: Allosteric Regulation; Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Chick Embryo; Down-Regulation; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Muscimol; Pyridazines; Receptors, GABA-A | 1990 |
Cloned GABA receptors are maintained in a stable cell line: allosteric and channel properties.
Topics: Animals; Antibodies, Monoclonal; Barbiturates; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cell Line; Chlorides; Clone Cells; Convulsants; DNA; gamma-Aminobutyric Acid; Membrane Potentials; Muscimol; Neurons; Plasmids; Receptors, GABA-A; Spinal Cord; Transfection | 1990 |
Radiation inactivation of brain [35S]t-butylbicyclophosphorothionate binding sites reveals complicated molecular arrangements of the GABA/benzodiazepine receptor chloride channel complex.
Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebellum; Cerebral Cortex; Chlorides; Etazolate; Etomidate; In Vitro Techniques; Ion Channels; Molecular Weight; Muscimol; Organophosphorus Compounds; Radioligand Assay; Rats; Receptors, GABA-A; Sulfur Radioisotopes | 1985 |
Antibodies recognising the GABAA/benzodiazepine receptor including its regulatory sites.
Topics: Allosteric Regulation; Animals; Antibodies; Antibody Specificity; Antigens; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cattle; Cerebral Cortex; Electrophoresis, Polyacrylamide Gel; Epitopes; Flunitrazepam; Immunologic Techniques; Immunosorbent Techniques; Muscimol; Receptors, GABA-A | 1986 |
Action of tremorgenic mycotoxins on GABAA receptor.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Electric Organ; Flunitrazepam; In Vitro Techniques; Ion Channels; Male; Muscimol; Mycotoxins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Torpedo; Tremor | 1987 |
Antagonist-type interaction of glucocorticoids with the GABA receptor-coupled chloride channel.
Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Frontal Lobe; Glucocorticoids; Ion Channels; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes | 1987 |
Chronic benzodiazepine administration. II. Discontinuation syndrome is associated with upregulation of gamma-aminobutyric acidA receptor complex binding and function.
Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Drug Tolerance; Flumazenil; Flunitrazepam; Ion Channels; Lorazepam; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Time Factors | 1988 |
Modulation of the benzodiazepine/gamma-aminobutyric acid receptor chloride channel complex by inhalation anesthetics.
Topics: Anesthesia, Inhalation; Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Enflurane; Ether; Halothane; Ion Channels; Male; Methoxyflurane; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes | 1988 |
Chemical kindling decreases GABA-activated chloride channels of mouse brain.
Topics: Animals; Autoradiography; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; gamma-Aminobutyric Acid; Ion Channels; Kindling, Neurologic; Male; Mice; Mice, Inbred ICR; Muscimol; Sulfur Radioisotopes | 1989 |
Estrogen modulation of the gamma-aminobutyric acid receptor complex in the central nervous system of rat.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Dose-Response Relationship, Drug; Estrogens; Female; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; RNA; Seizures | 1988 |
Diazepam sensitizes mice to FG 7142 and reduces muscimol-stimulated 36Cl- flux.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Chlorides; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Ion Channels; Kindling, Neurologic; Mice; Mice, Inbred ICR; Muscimol | 1989 |
Interaction of caffeine with the GABAA receptor complex: alterations in receptor function but not ligand binding.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Caffeine; Cerebral Cortex; Chlorides; In Vitro Techniques; Ion Channels; Kinetics; Ligands; Male; Mice; Muscimol; Receptors, GABA-A; Sulfur Radioisotopes; Synaptosomes | 1989 |
Distribution and pharmacological properties of the GABAA/benzodiazepine/chloride ionophore receptor complex in the brain of the fish Anguilla anguilla.
Topics: Anguilla; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Flunitrazepam; gamma-Aminobutyric Acid; Ionophores; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Tissue Distribution | 1989 |
Effects of picrotoxin treatment on GABAA receptor supramolecular complexes in rat brain.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Flunitrazepam; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Tissue Distribution | 1989 |
Steroid anesthetics and naturally occurring analogs modulate the gamma-aminobutyric acid receptor complex at a site distinct from barbiturates.
Topics: Anesthetics; Animals; Barbiturates; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; In Vitro Techniques; Male; Muscimol; Pregnanediones; Rats; Rats, Inbred Strains; Receptors, GABA-A; Steroids; Structure-Activity Relationship | 1989 |
Differential seizure sensitivities to picrotoxinin in two inbred strains of mice (DBA/2J and BALB/c ByJ): parallel changes in GABA receptor-mediated chloride flux and receptor binding.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; Frontal Lobe; Male; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Muscimol; Pentobarbital; Picrotoxin; Receptors, GABA-A; Seizures; Species Specificity; Synaptosomes | 1989 |
Enhancement of GABAergic transmission by zolpidem, an imidazopyridine with preferential affinity for type I benzodiazepine receptors.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Muscimol; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission; Zolpidem | 1989 |
Age-related loss of t-[35S]butylbicyclophosphorothionate binding to the gamma-aminobutyric acidA receptor-coupled chloride ionophore in rat cerebral cortex.
Topics: Aging; Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Female; Ionophores; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes | 1989 |
The modulation by chlormethiazole of the GABAA-receptor complex in rat brain.
Topics: Animals; Baclofen; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlormethiazole; CLC-2 Chloride Channels; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Picrotoxin; Rats; Receptors, GABA-A | 1989 |
Persistent alterations in GABAA receptor binding and function after prenatal lorazepam administration in the chick.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chick Embryo; Chickens; Chlorides; Female; Flunitrazepam; Lorazepam; Muscimol; Pregnancy; Prenatal Exposure Delayed Effects; Radioligand Assay; Receptors, GABA-A | 1989 |
A progesterone metabolite enhances the activity of the GABAA receptor complex at the pituitary level.
Topics: 5-alpha-Dihydroprogesterone; Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; In Vitro Techniques; Male; Membranes; Muscimol; Picrotoxin; Pituitary Gland, Anterior; Pregnanediones; Progesterone; Prolactin; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Fluidization of brain membranes by A2C does not produce anesthesia and does not augment muscimol-stimulated 36Cl- influx.
Topics: Anesthesia; Animals; Benzyl Alcohols; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; gamma-Aminobutyric Acid; Male; Membrane Fluidity; Membranes; Mice; Mice, Inbred ICR; Muscimol; Radioisotopes; Stearates; Stearic Acids; Synaptosomes; Temperature | 1989 |
Bicuculline up-regulation of GABAA receptors in rat brain.
Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Corpus Striatum; Flunitrazepam; Frontal Lobe; gamma-Aminobutyric Acid; Male; Muscimol; Octoxynol; Polyethylene Glycols; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra; Synaptic Membranes | 1988 |
Actions of avermectin B1a on the gamma-aminobutyric acidA receptor and chloride channels in rat brain.
Topics: Animals; Bicuculline; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Flunitrazepam; Ivermectin; Kinetics; Male; Membrane Proteins; Muscimol; Rats; Receptors, GABA-A | 1986 |
Interactions of ACTH4-10 and ACTH1-24 with L-[3H]glutamate binding sites and GABA/benzodiazepine/picrotoxin receptor complexes in vitro.
Topics: Adrenocorticotropic Hormone; Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Flunitrazepam; Glutamates; Glutamic Acid; Male; Muscimol; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Glutamate; Receptors, Neurotransmitter | 1988 |
Foot-shock stress and anxiogenic beta-carbolines increase t-[35S]butylbicyclophosphorothionate binding in the rat cerebral cortex, an effect opposite to anxiolytics and gamma-aminobutyric acid mimetics.
Topics: Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Diazepam; Electroshock; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological | 1988 |
Interaction of pitrazepin with the GABA/benzodiazepine receptor complex and with glycine receptors.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Dibenzazepines; In Vitro Techniques; Kinetics; Male; Membranes; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Glycine; Receptors, Neurotransmitter; Strychnine | 1985 |
Ontogeny of the GABA receptor complex in chick brain: studies in vivo and in vitro.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Chick Embryo; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Receptors, GABA-A | 1986 |
Isolation of the gamma-aminobutyric acid/benzodiazepine receptor.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Chromatography, Affinity; Flunitrazepam; Isoelectric Point; Molecular Weight; Muscimol; Radioimmunoassay; Rats; Receptors, GABA-A | 1985 |
Effects of pentylenetetrazol on GABA-A/benzodiazepine/picrotoxinin receptor complexes in rat brain regions.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Corpus Striatum; Flunitrazepam; gamma-Aminobutyric Acid; Male; Muscimol; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Tissue Distribution | 1986 |
Anticonvulsant activity of piperidinol and (dialkylamino)alkanol esters.
Topics: Amino Alcohols; Animals; Anticonvulsants; Ataxia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Diazepam; Electroshock; Esters; Muscimol; Pentylenetetrazole; Phenytoin; Piperidines; Rats; Receptors, GABA-A; Structure-Activity Relationship | 1986 |
Structural analysis and localization of GABA/benzodiazepine/TBPS-receptor complex using monoclonal antibodies.
Topics: Animals; Antibodies, Monoclonal; Autoradiography; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Convulsants; Flunitrazepam; Humans; Immunoenzyme Techniques; Mice; Muscimol; Rats; Receptors, GABA-A; Sulfur Radioisotopes; Tritium | 1986 |
gamma-Aminobutyric acid receptor ionophore complexes: differential effects of deltamethrin, dichlorodiphenyltrichloroethane, and some novel insecticides in a rat brain membrane preparation.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; DDT; Diazepam; Insecticides; Ionophores; Male; Muscimol; Nitriles; Pyrethrins; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Pyrethroid insecticides and radioligand displacement from the GABA receptor chloride ionophore complex.
Topics: Animals; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; Male; Muscimol; Nitriles; Permethrin; Pyrethrins; Rats; Receptors, GABA-A | 1987 |
Pregnenolone-sulfate: an endogenous antagonist of the gamma-aminobutyric acid receptor complex in brain?
Topics: Adrenal Glands; Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Male; Muscimol; Picrotoxin; Pregnenolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical | 1987 |
Structure-activity relationships for steroid interaction with the gamma-aminobutyric acidA receptor complex.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Desoxycorticosterone; Electric Conductivity; Ethanol; Evoked Potentials; Flunitrazepam; Muscimol; Pregnanes; Progesterone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Steroids; Structure-Activity Relationship | 1987 |
Progress towards the understanding of the GABAA receptor structure.
Topics: Allosteric Site; Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cholic Acids; Deoxycholic Acid; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Protein Binding; Receptors, GABA-A | 1987 |
Gamma-aminobutyric acid and alcohol actions: neurochemical studies of long sleep and short sleep mice.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebellum; Chlorides; Diencephalon; Drug Synergism; Ethanol; Female; gamma-Aminobutyric Acid; Hippocampus; Mice; Muscimol; Pentobarbital; Sleep; Telencephalon | 1986 |
gamma-Aminobutyric acid- and benzodiazepine-induced modulation of [35S]-t-butylbicyclophosphorothionate binding to cerebellar granule cells.
Topics: Animals; Benzodiazepines; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebellum; Diazepam; gamma-Aminobutyric Acid; Granulocytes; Muscimol; Picrotoxin; Rats; Sulfur Radioisotopes; Temperature | 1985 |
Similar properties of [35S]t-butylbicyclophosphorothionate receptor and coupled components of the GABA receptor-ionophore complex in brains of human, cow, rat, chicken and fish.
Topics: Androstanes; Animals; Azasteroids; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cattle; Chickens; Convulsants; Female; Fishes; Humans; Ivermectin; Lactones; Male; Middle Aged; Muscimol; Rats; Receptors, GABA-A; Taurine | 1984 |
A study on benzodiazepine receptor binding in audiogenic seizure-susceptible rats.
Topics: Acoustic Stimulation; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Convulsants; Diazepam; Female; Flunitrazepam; In Vitro Techniques; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures | 1984 |
In vitro characterization of agonist, antagonist, inverse agonist and agonist/antagonist benzodiazepines.
Topics: Animals; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Etazolate; Ion Channels; Muscimol; Rats; Receptors, GABA-A | 1984 |
Saturable binding of 35S-t-butylbicyclophosphorothionate to the sites linked to the GABA receptor and the interaction with GABAergic agents.
Topics: Animals; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; gamma-Aminobutyric Acid; Male; Muscimol; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Sulfur Radioisotopes; Triazines | 1984 |
A gamma-aminobutyric acid/benzodiazepine receptor complex from bovine cerebral cortex. Improved purification with preservation of regulatory sites and their interactions.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Cholic Acids; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Methods; Muscimol; Pentobarbital; Receptors, Cell Surface; Receptors, GABA-A; Solubility | 1984 |
[35S]-t-butylbicyclophosphorothionate binding sites are constituents of the gamma-aminobutyric acid benzodiazepine receptor complex.
Topics: Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cerebral Cortex; gamma-Aminobutyric Acid; Kinetics; Macromolecular Substances; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Lindane administration to the rat induces modifications in the regional cerebral binding of [3H]Muscimol, [3H]-flunitrazepam, and t-[35S]butylbicyclophosphorothionate: an autoradiographic study.
Topics: Animals; Autoradiography; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Flunitrazepam; Hexachlorocyclohexane; Male; Muscimol; Rats; Rats, Wistar; Reference Values; Sulfur Radioisotopes; Tissue Distribution; Tritium | 1993 |
Effects of 1-amino-5-bromouracil on the benzodiazepine-GABAA receptor complex.
Topics: Anesthesia; Animals; Anti-Anxiety Agents; Anticonvulsants; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bromouracil; Convulsants; Dehydroepiandrosterone; Male; Mice; Mice, Inbred ICR; Muscimol; Picrotoxin; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Seizures; Synaptic Membranes | 1994 |
Alterations in the brain GABAA/benzodiazepine receptor-chloride ionophore complex in a genetic model of paroxysmal dystonia: a quantitative autoradiographic analysis.
Topics: Animals; Autoradiography; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Cricetinae; Dystonia; Flunitrazepam; Ionophores; Male; Models, Genetic; Muscimol; Radiography; Receptors, GABA-A | 1995 |
The effect of cyclopyrrolones on GABAA receptor function is different from that of benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Chlorine; Flumazenil; Hypnotics and Sedatives; Kinetics; Male; Mice; Mice, Inbred Strains; Muscimol; Naphthyridines; Piperazines; Radioisotopes; Receptors, GABA-A; Sulfur Compounds; Sulfur Radioisotopes; Tritium | 1994 |
Analysis of the hippocampal GABAA receptor system in kindled rats by autoradiographic and in situ hybridization techniques: contingent tolerance to carbamazepine.
Topics: Affinity Labels; Amygdala; Animals; Autoradiography; Azides; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbamazepine; Convulsants; Drug Tolerance; Electric Stimulation; Electroencephalography; Flunitrazepam; Functional Laterality; Gene Expression; Hippocampus; In Situ Hybridization; Kindling, Neurologic; Macromolecular Substances; Muscimol; Neurons; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Seizures; Tritium | 1994 |
GABAA receptor stimulation enhances NMDA-induced Ca2+ influx in mouse cerebral cortical neurons in primary culture.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Cerebral Cortex; Chloride Channels; Dizocilpine Maleate; Dose-Response Relationship, Drug; GABA Agonists; Isonicotinic Acids; Mice; Muscimol; N-Methylaspartate; Neurons; Picrotoxin; Potassium; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate | 1994 |
Gamma-aminobutyric acidA receptor function is inhibited by microtubule depolymerization.
Topics: Animals; Biological Transport; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Chlorides; Colchicine; Convulsants; Dose-Response Relationship, Drug; Flunitrazepam; Histones; Humans; Lumicolchicines; Membranes; Mice; Microtubules; Muscimol; Nocodazole; Paclitaxel; Phosphorylation; Receptors, GABA-A; Vinblastine; Xenopus | 1994 |
Age-related changes of GABA-activated chloride channel properties in brain cortex synaptic plasma membrane: evidence for phospholipase involvement.
Topics: Aging; Animals; Arachidonic Acid; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Convulsants; Diglycerides; gamma-Aminobutyric Acid; Kinetics; Muscimol; Phospholipases; Picrotoxin; Rats; Rats, Wistar; Sulfur Radioisotopes; Synaptic Membranes; Synaptosomes | 1994 |
Cloning and functional expression of a Drosophila gamma-aminobutyric acid receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cloning, Molecular; Convulsants; DNA Primers; DNA, Complementary; Drosophila melanogaster; Female; Flunitrazepam; gamma-Aminobutyric Acid; Gene Expression; Macromolecular Substances; Molecular Sequence Data; Muscimol; Oocytes; Pentobarbital; Picrotoxin; Polymerase Chain Reaction; Receptors, GABA; Receptors, GABA-A; Transcription, Genetic; Xenopus laevis | 1994 |
Interactions of ginsenosides with ligand-bindings of GABA(A) and GABA(B) receptors.
Topics: Animals; Baclofen; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbohydrate Sequence; Flunitrazepam; Ginsenosides; Herb-Drug Interactions; Ligands; Male; Molecular Sequence Data; Muscimol; Panax; Plants, Medicinal; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Saponins; Sulfur Radioisotopes; Tritium | 1994 |
Studies on picrotoxin binding sites of GABAA receptors in rat cortical synaptoneurosomes.
Topics: Animals; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorine; Desoxycorticosterone; Diazepam; In Vitro Techniques; Male; Membranes; Muscimol; Pentobarbital; Picrotoxin; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Steroids; Synaptosomes | 1994 |
Decreased forebrain [35S]TBPS binding and increased [3H]muscimol binding in rats that do not develop stress-induced behavioral depression.
Topics: Adrenalectomy; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Depression; Desoxycorticosterone; Electroshock; Flunitrazepam; Helplessness, Learned; Male; Muscimol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stress, Psychological | 1993 |
Influence of flumazenil on the learning-enhancing effect of ambocarb in rats.
Topics: Animals; Behavior, Animal; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Discrimination Learning; Discrimination, Psychological; Flumazenil; Flunitrazepam; Harmine; Learning; Ligands; Male; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A | 1994 |
Modulatory action of arachidonic acid on GABAA/chloride channel receptor function in adult and aged brain cortex membranes.
Topics: Aging; Animals; Arachidonic Acid; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Chloride Channels; Chlorides; Convulsants; Docosahexaenoic Acids; Fatty Acids, Nonesterified; Kinetics; Male; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Stearic Acids; Synaptic Membranes; Synaptosomes | 1993 |
Natural mutation of GABAA receptor alpha 6 subunit alters benzodiazepine affinity but not allosteric GABA effects.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cerebellum; Cloning, Molecular; Convulsants; Diazepam; gamma-Aminobutyric Acid; Granulocytes; Humans; Kidney; Muscimol; Mutation; Picrotoxin; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection | 1993 |
GABAA receptor function in the gamma-hydroxybutyrate model of generalized absence seizures.
Topics: Aminocaproates; Animals; Anticonvulsants; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; Convulsants; Electroencephalography; Epilepsy, Absence; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Muscimol; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sodium Oxybate; Synaptosomes; Vigabatrin | 1993 |
Comparison of interactions of [3H]muscimol, t-butylbicyclophosphoro[35S]thionate, and [3H]flunitrazepam with cloned gamma-aminobutyric acidA receptors of the alpha 1 beta 2 and alpha 1 beta 2 gamma 2 subtypes.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cloning, Molecular; Flunitrazepam; Moths; Muscimol; Radioligand Assay; Receptors, GABA-A; Recombinant Proteins; Zinc | 1993 |
Region-specific changes of GABAA receptors by tolerance to and dependence upon pentobarbital.
Topics: Animals; Body Temperature; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Corpus Striatum; Drug Tolerance; Flunitrazepam; Frontal Lobe; In Vitro Techniques; Injections, Intraventricular; Male; Muscimol; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Substance-Related Disorders; Sulfur Radioisotopes; Synaptic Membranes | 1993 |
Subtype specificity of gamma-aminobutyric acid type A receptor antagonism by clozapine.
Topics: Animals; Antipsychotic Agents; Brain; Bridged Bicyclo Compounds, Heterocyclic; Clozapine; GABA Antagonists; GABA-A Receptor Antagonists; Male; Muscimol; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A | 1995 |
Biochemical evaluations of the effects of loreclezole and propofol on the GABAA receptor in rat brain.
Topics: Anesthetics; Animals; Anticonvulsants; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Triazoles; Tritium | 1996 |
Interaction of allosteric ligands with GABAA receptors containing one, two, or three different subunits.
Topics: Allosteric Site; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Convulsants; Flunitrazepam; GABA Agonists; GABA Modulators; GABA-A Receptor Antagonists; Humans; Kidney; Membranes; Muscimol; Radioligand Assay; Receptors, GABA-A | 1996 |
Antisense oligonucleotide to GABAA receptor gamma 2 subunit induces loss of neurones in rat hippocampus.
Topics: Animals; Base Sequence; Behavior, Animal; Benzodiazepines; Bridged Bicyclo Compounds, Heterocyclic; Cell Count; Convulsants; Flunitrazepam; GABA Agonists; GABA Modulators; Hippocampus; Male; Molecular Sequence Data; Muscimol; Neurons; Oligonucleotides, Antisense; Rats; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Tritium | 1995 |
A novel class of GABAA receptor subunit in tissues of the reproductive system.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cloning, Molecular; DNA, Complementary; Flumazenil; Humans; Molecular Sequence Data; Muscimol; Radioligand Assay; Rats; Receptors, GABA-A; RNA, Messenger | 1997 |
Chronic ethanol administration alters the modulatory effect of 5alpha-pregnan-3alpha-ol-20-one on the binding characteristics of various radioligands of GABAA receptors.
Topics: Animals; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Ethanol; Flunitrazepam; GABA Agonists; GABA Modulators; Hippocampus; Male; Muscimol; Pregnanolone; Rats; Rats, Sprague-Dawley; Time Factors | 1998 |
Substituted 3beta-phenylethynyl derivatives of 3alpha-hydroxy-5alpha-pregnan-20-one: remarkably potent neuroactive steroid modulators of gamma-aminobutyric acidA receptors.
Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Flunitrazepam; GABA Modulators; Humans; Male; Mice; Muscimol; Pregnanolone; Rats; Receptors, GABA-A; Recombinant Proteins; Structure-Activity Relationship; Xenopus | 1998 |
Activation of protein kinase C by phorbol dibutyrate modulates GABAA receptor binding in rat brain slices.
Topics: Animals; Autoradiography; Brain Chemistry; Bridged Bicyclo Compounds, Heterocyclic; Enzyme Activation; Flunitrazepam; GABA Agonists; GABA Modulators; In Vitro Techniques; Ligands; Muscimol; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Receptors, GABA-A | 1999 |
Effects of the chlorotriazine herbicide, cyanazine, on GABA(A) receptors in cortical tissue from rat brain.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorine; GABA Agonists; Herbicides; Male; Muscimol; Radioisotopes; Rats; Rats, Long-Evans; Receptors, GABA-A; Synaptosomes; Triazines | 1999 |
Synthesis and GABA(A) receptor activity of 6-oxa-analogs of neurosteroids.
Topics: Animals; Antipsychotic Agents; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cholestanones; Flunitrazepam; GABA Modulators; Hydrogen Bonding; Inhibitory Concentration 50; Molecular Structure; Muscimol; Rats; Receptors, GABA-A; Steroids; Structure-Activity Relationship | 2000 |
Characterization of gamma-aminobutyrate type A receptors with atypical coupling between agonist and convulsant binding sites in discrete brain regions.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Chickens; Convulsants; GABA Agonists; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Picrotoxin; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Sesterterpenes; Sulfur Radioisotopes; Thalamus; Tritium | 2001 |
Unsulfated and sulfated neurosteroids differentially modulate the binding characteristics of various radioligands of GABA(A) receptors following chronic ethanol administration.
Topics: Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Central Nervous System Depressants; Cerebellum; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Ethanol; Flunitrazepam; GABA Agonists; Muscimol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Steroids | 2001 |
Loss of the major GABA(A) receptor subtype in the brain is not lethal in mice.
Topics: Animals; Autoradiography; Behavior, Animal; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Electrophysiology; Flumazenil; Gait Disorders, Neurologic; Gene Expression; Homozygote; Ligands; Mice; Mice, Inbred Strains; Mice, Knockout; Motor Activity; Muscimol; Protein Subunits; Purkinje Cells; Radioligand Assay; Receptors, GABA-A; Survival Rate; Tissue Distribution | 2001 |
Modulation Of [35S]-tert-butylbicyclophosphorothionate binding by somatostatin in rat hypothalamus.
Topics: Animals; Bicuculline; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Dose-Response Relationship, Drug; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Male; Muscimol; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A; Somatostatin; Sulfur Radioisotopes | 2002 |
Photoaffinity labeling with a neuroactive steroid analogue. 6-azi-pregnanolone labels voltage-dependent anion channel-1 in rat brain.
Topics: Affinity Labels; Animals; Aziridines; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cell Membrane; Female; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Kinetics; Membrane Potentials; Muscimol; Oocytes; Porins; Pregnanolone; Rats; Recombinant Proteins; Steroids; Telencephalon; Transfection; Voltage-Dependent Anion Channel 1; Voltage-Dependent Anion Channels; Xenopus laevis | 2003 |
Radioligand binding studies of caloporoside and novel congeners with contrasting effects upon [35S] TBPS binding to the mammalian GABA(A) receptor.
Topics: Animals; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Flunitrazepam; gamma-Aminobutyric Acid; Glucosides; Male; Mannose; Muscimol; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Salicylates; Structure-Activity Relationship; Sulfur Radioisotopes | 2005 |
Autoradiographic analysis of GABAA receptors in mu-opioid receptor knockout mice.
Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Down-Regulation; Flunitrazepam; Male; Mice; Mice, Knockout; Muscimol; Receptors, GABA-A; Receptors, Opioid, mu; Tritium; Up-Regulation | 2007 |
Effect of synthetic steroids on GABAA receptor binding in rat brain.
Topics: Animals; Autoradiography; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Flunitrazepam; GABA-A Receptor Agonists; Hippocampus; Male; Muscimol; Pregnanolone; Protein Binding; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Tritium | 2015 |