muscimol has been researched along with piperidines in 34 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (20.59) | 18.7374 |
1990's | 6 (17.65) | 18.2507 |
2000's | 12 (35.29) | 29.6817 |
2010's | 7 (20.59) | 24.3611 |
2020's | 2 (5.88) | 2.80 |
Authors | Studies |
---|---|
Braestrup, C; Falch, E; Krogsgaard-Larsen, P; Nielsen, M | 2 |
Dziki, M; Ikonomidou, C; Parada-Turska, J; Turski, WA; Urbanska, E | 1 |
Kumasaka, Y; Ueki, S; Yamamoto, T | 1 |
Iversen, LL; Wong, EH | 1 |
Curtis, DR; Falch, E; Krogsgaard-Larsen, P; Nielsen, L | 1 |
Creveling, CR; Daly, JW; Hollingsworth, EB; Lewandowski, G; Waters, JA | 1 |
Mitchell, R; Wilson, LE | 1 |
Ammendola, D; De Sarro, A; De Sarro, G; Nava, F | 1 |
Ebert, B; Kemp, JA; Krogsgaard-Larsen, P; Wafford, KA; Whiting, PJ | 1 |
Ebert, B; Krogsgaard-Larsen, P; McKernan, R; Saounatsou, K; Thompson, SA; Wafford, KA | 1 |
Dement, WC; Mignot, E; Nishino, S; Reid, MS; Siegel, JM; Tafti, M | 1 |
Fields, HL; Manning, BH; Martin, WJ; Meng, ID | 1 |
Que, M; Witte, OW; Zilles, K | 1 |
Maksay, G; McKernan, R | 1 |
Engblom, C; Frølund, B; Kristiansen, U; Krogsgaard-Larsen, P; Liljefors, T; Stensbøl, TB; Tagmose, L | 1 |
Siemes, S; Szabo, B; Wallmichrath, I | 1 |
Ebert, B; Frølund, B; Kristiansen, U; Krogsgaard-Larsen, P; Liljefors, T | 1 |
Fukumori, R; Goshima, Y; Hagiwara, Y; Kanaya, T; Kubo, T; Okatani, H | 2 |
Dixon, HB; Dragoni, S; Frosini, M; Machetti, F; Palmi, M; Sesti, C; Sgaragli, G; Valoti, M | 1 |
Argiolas, A; Mascia, MS; Melis, MR; Melis, T; Sanna, F; Succu, S | 1 |
Fujii, Y; Kamei, C; Mikami, A; Yamamoto, Y | 1 |
Akabas, MH; Dannhardt, G; Debus, F; Dieler, S; Jansen, M; Lüddens, H; Rabe, H; Strehle, A | 1 |
Kovacs, FE; Szabo, B; Urbanski, MJ | 1 |
Abdel-Rahman, AA; Ibrahim, BM | 1 |
Cornélio, AM; Morgan, MM; Nunes-de-Souza, RL | 1 |
Arreto, CD; Bourgeais, L; Condes-Lara, M; Jay, T; Noseda, R; Robert, C; Villanueva, L | 1 |
Holmes, NM; Killcross, AS; Parkes, SL; Westbrook, RF | 1 |
Cui, CL; Ge, FF; Li, YJ; Ping, XJ; Qi, C; Shen, F; Sun, LL; Sun, XW; Xing, GG | 1 |
Chergui, K; Yao, N; Zhang, X | 1 |
Baillie, LD; Catton, JK; Davies, DA; Greba, Q; Howland, JG; Mulligan, SJ; Selk, JC | 1 |
Bertoglio, LJ; Troyner, F | 1 |
Axelsson, SFA; Horiguchi, N; Horst, NK; Robbins, TW; Roberts, AC | 1 |
1 review(s) available for muscimol and piperidines
Article | Year |
---|---|
GABA(A) receptor ligands and their therapeutic potentials.
Topics: Animals; Central Nervous System Diseases; GABA Agents; GABA Agonists; GABA Antagonists; Humans; Isonicotinic Acids; Isoxazoles; Ligands; Muscimol; Piperidines; Protein Subunits; Receptors, GABA-A | 2002 |
33 other study(ies) available for muscimol and piperidines
Article | Year |
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Partial agonists for brain GABA/benzodiazepine receptor complex.
Topics: Animals; Benzodiazepines; Bicuculline; Brain; Crotonates; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, Drug; Sulfonic Acids | 1979 |
Excitatory amino acid antagonists protect mice against seizures induced by bicuculline.
Topics: Animals; Bicuculline; Dibenzocycloheptenes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Mice; Muscimol; Pipecolic Acids; Piperazines; Piperidines; Receptors, Amino Acid; Receptors, Cell Surface; Seizures | 1990 |
Behavioral analysis of zopiclone on the basis of their discriminative stimulus properties in the rat.
Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Behavior, Animal; Benzodiazepines; Bicuculline; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Hypnotics and Sedatives; Male; Muscimol; Naphthyridines; Pentylenetetrazole; Piperazines; Piperidines; Rats; Rats, Inbred WKY; Ritanserin; Serotonin Antagonists; Sulfur Compounds | 1989 |
Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.
Topics: Androstanes; Animals; Azasteroids; Bicuculline; Cell Membrane; Cerebral Cortex; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isonicotinic Acids; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, GABA-A; Taurine | 1985 |
GABA agonists. Resolution, absolute stereochemistry, and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol.
Topics: Animals; Bicuculline; Brain; Cats; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Molecular Conformation; Muscimol; Neurons; Oxazolidinones; Piperidines; Rats; Receptors, GABA-A; Spinal Cord; Stereoisomerism; Structure-Activity Relationship; Synaptic Membranes | 1985 |
Anticonvulsant activity of piperidinol and (dialkylamino)alkanol esters.
Topics: Amino Alcohols; Animals; Anticonvulsants; Ataxia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Diazepam; Electroshock; Esters; Muscimol; Pentylenetetrazole; Phenytoin; Piperidines; Rats; Receptors, GABA-A; Structure-Activity Relationship | 1986 |
Two or more conformations of benzodiazepine receptors depending on GABA receptors and other variables.
Topics: Animals; Benzodiazepines; Bicuculline; Brain; Diazepam; gamma-Aminobutyric Acid; Macromolecular Substances; Male; Muscimol; Piperidines; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Structure-Activity Relationship; Synaptic Membranes | 1980 |
Effects of GABA receptor agonists on [3H] flunitrazepam binding to rat cerebellar and hippocampal membranes.
Topics: Animals; Cerebellum; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Imidazoles; Male; Membranes; Muscimol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Effects of some excitatory amino acid antagonists on imipenem-induced seizures in DBA/2 mice.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Animals; Anticonvulsants; Dizocilpine Maleate; Excitatory Amino Acids; Glutamine; Imipenem; Kynurenic Acid; Mice; Mice, Inbred DBA; Muscimol; Piperazines; Piperidines; Quinoxalines; Seizures | 1995 |
Molecular pharmacology of gamma-aminobutyric acid type A receptor agonists and partial agonists in oocytes injected with different alpha, beta, and gamma receptor subunit combinations.
Topics: Animals; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Muscimol; Oocytes; Oxazolidinones; Piperidines; Receptors, GABA-A; Recombinant Proteins; Structure-Activity Relationship; Xenopus | 1994 |
Differences in agonist/antagonist binding affinity and receptor transduction using recombinant human gamma-aminobutyric acid type A receptors.
Topics: Animals; Binding, Competitive; DNA, Complementary; Electrophysiology; GABA Agonists; GABA Antagonists; Humans; Isoxazoles; Kinetics; Macromolecular Substances; Muscimol; Oocytes; Piperidines; Receptors, GABA-A; Transduction, Genetic; Transfection; Tritium; Xenopus laevis | 1997 |
Neuropharmacological characterization of basal forebrain cholinergic stimulated cataplexy in narcoleptic canines.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Behavior, Animal; Carbachol; Cataplexy; Cholinergic Fibers; Dogs; Feeding Behavior; Female; GABA Agonists; Gallamine Triethiodide; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Muscimol; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Piperidines; Pirenzepine; Prosencephalon | 1998 |
An analgesia circuit activated by cannabinoids.
Topics: Analgesia; Analgesics, Non-Narcotic; Animals; Benzoxazines; Cannabinoids; GABA Agonists; Male; Medulla Oblongata; Morphine; Morpholines; Motor Activity; Muscimol; Naphthalenes; Neural Pathways; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant | 1998 |
Transient up-regulation of gamma-aminobutyric acid(A) receptor binding by lubeluzole after neocortical specify lesion in rats.
Topics: Animals; Brain Ischemia; Male; Muscimol; Neocortex; Neuroprotective Agents; Photochemistry; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, AMPA; Receptors, GABA-A; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Rose Bengal; Thiazoles; Tritium; Up-Regulation | 2000 |
Entropy as the predominant driving force of binding to human recombinant alpha(x)beta(3)gamma(2) GABA(A) receptors.
Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Entropy; GABA Agonists; GABA Antagonists; Humans; Isoxazoles; L Cells; Membranes; Mice; Muscimol; Piperidines; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Temperature; Tritium | 2001 |
A novel class of potent 3-isoxazolol GABA(A) antagonists: design, synthesis, and pharmacology.
Topics: Animals; Brain; Cells, Cultured; GABA Antagonists; Isoxazoles; Models, Molecular; Muscimol; Neurons; Patch-Clamp Techniques; Piperidines; Radioligand Assay; Rats; Receptors, GABA-A; Structure-Activity Relationship; Synaptic Membranes | 2000 |
Inhibition of GABAergic neurotransmission in the ventral tegmental area by cannabinoids.
Topics: Analgesics; Animals; Animals, Newborn; Benzoxazines; Cannabinoids; Drug Interactions; GABA Agonists; gamma-Aminobutyric Acid; Membrane Potentials; Morpholines; Muscimol; Naphthalenes; Neural Inhibition; Neural Pathways; Neurons; Nucleus Accumbens; Organ Culture Techniques; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Receptors, GABA-A; Rimonabant; Synaptic Transmission; Ventral Tegmental Area | 2002 |
Cholinergic mechanism in the lateral septal area is involved in the stress-induced blood pressure increase in rats.
Topics: Animals; Blood Pressure; Carbachol; Cholinergic Agonists; Cholinesterase Inhibitors; Epinephrine; GABA Agonists; Injections, Intraventricular; Male; Muscarinic Antagonists; Muscimol; Norepinephrine; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Restraint, Physical; Septal Nuclei; Stress, Physiological | 2003 |
Interactions of taurine and structurally related analogues with the GABAergic system and taurine binding sites of rabbit brain.
Topics: 4-Aminobutyrate Transaminase; Animals; Binding Sites; Brain; Drug Interactions; gamma-Aminobutyric Acid; Isomerism; Molecular Structure; Muscimol; Piperidines; Rabbits; Receptors, GABA-A; Receptors, GABA-B; Receptors, Neurotransmitter; Structure-Activity Relationship; Synaptic Membranes; Synaptosomes; Taurine; Tritium | 2003 |
Projections from the caudal part to the rostral part of the lateral septal area mediate blood pressure increase.
Topics: Animals; Blood Pressure; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Fluorescent Dyes; GABA Agonists; Hypertension; Male; Microinjections; Muscarinic Antagonists; Muscimol; Neural Pathways; Neurons; Piperidines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Reaction Time; Septum of Brain; Stress, Physiological | 2003 |
The cannabinoid CB1 receptor antagonist SR 141716A induces penile erection by increasing extra-cellular glutamic acid in the paraventricular nucleus of male rats.
Topics: Anesthetics, Local; Animals; Baclofen; Behavior, Animal; Cannabinoid Receptor Antagonists; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Extracellular Space; GABA Agonists; Glutamic Acid; Male; Microdialysis; Microinjections; Models, Biological; Muscimol; Paraventricular Hypothalamic Nucleus; Penile Erection; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Tetrodotoxin | 2006 |
Effect of histamine on muscimol-induced working memory deficits in radial maze performance.
Topics: Animals; Brain Chemistry; Cholinesterase Inhibitors; Donepezil; Dose-Response Relationship, Drug; GABA Agonists; GABA-A Receptor Agonists; Histamine; Histidine; Indans; Male; Maze Learning; Memory Disorders; Memory, Short-Term; Microinjections; Muscimol; Piperidines; Rats; Tacrine | 2007 |
Synthesis of GABAA receptor agonists and evaluation of their alpha-subunit selectivity and orientation in the GABA binding site.
Topics: Animals; Binding Sites; Brain; Cell Line; Electrophysiology; Female; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Models, Molecular; Molecular Structure; Muscimol; Mutation; Oocytes; Patch-Clamp Techniques; Piperidines; Protein Subunits; Rats; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis | 2008 |
Depolarizing GABAergic synaptic input triggers endocannabinoid-mediated retrograde synaptic signaling.
Topics: Aniline Compounds; Animals; Animals, Newborn; Arachidonic Acids; Benzamides; Bicuculline; Biophysics; Calcium; Calcium Signaling; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Carbamates; Cerebellum; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Fluoresceins; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Lactones; Mice; Muscimol; Orlistat; Patch-Clamp Techniques; Piperidines; Purkinje Cells; Pyrazoles; Quinoxalines; Rimonabant; Signal Transduction; Synapses; Valine | 2009 |
Role of brainstem GABAergic signaling in central cannabinoid receptor evoked sympathoexcitation and pressor responses in conscious rats.
Topics: Analysis of Variance; Animals; Benzoxazines; Blood Pressure; Brain Stem; Dose-Response Relationship, Drug; Drug Interactions; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Heart Rate; Injections, Intraventricular; Male; Morpholines; Muscimol; Naphthalenes; Neurons; Norepinephrine; Piperidines; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Tyrosine 3-Monooxygenase; Wakefulness | 2011 |
Contribution of the rostral ventromedial medulla to post-anxiety induced hyperalgesia.
Topics: Animals; Anxiety; GABA-A Receptor Agonists; Hyperalgesia; Male; Medulla Oblongata; Muscimol; Pain Measurement; Pain Threshold; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1 | 2012 |
Paraventricular hypothalamic regulation of trigeminovascular mechanisms involved in headaches.
Topics: Action Potentials; Animals; Biotin; Corticosterone; Dextrans; Disease Models, Animal; GABA Antagonists; GABA-A Receptor Agonists; Male; Muscimol; Neural Pathways; Neurons; Paraventricular Hypothalamic Nucleus; Physical Stimulation; Piperidines; Pituitary Adenylate Cyclase-Activating Polypeptide; Pyridazines; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Stilbamidines; Stress, Psychological; Trigeminal Nuclei; Tryptamines | 2013 |
The basolateral amygdala is critical for learning about neutral stimuli in the presence of danger, and the perirhinal cortex is critical in the absence of danger.
Topics: Acoustic Stimulation; Amygdala; Animals; Association Learning; Conditioning, Classical; Environment; Excitatory Amino Acid Antagonists; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; GABA-A Receptor Agonists; Male; Muscimol; Photic Stimulation; Piperidines; Prefrontal Cortex; Rats; Rats, Wistar | 2013 |
Re-exposure to morphine-associated context facilitated long-term potentiation in the vSUB-NAc glutamatergic pathway via GluN2B-containing receptor activation.
Topics: Analgesics, Opioid; Animals; Baclofen; Behavior, Animal; Conditioning, Operant; GABA-A Receptor Agonists; GABA-B Receptor Agonists; Hippocampus; Long-Term Potentiation; Male; Memory; Morphine; Muscimol; Nucleus Accumbens; Phenols; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate | 2017 |
The GABAA receptor agonist muscimol induces an age- and region-dependent form of long-term depression in the mouse striatum.
Topics: Animals; Corpus Striatum; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA-A Receptor Agonists; Long-Term Synaptic Depression; Male; Mice, Inbred C57BL; Muscimol; Piperidines; Pyrazoles; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, GABA-A; TRPV Cation Channels | 2016 |
Interactions between medial prefrontal cortex and dorsomedial striatum are necessary for odor span capacity in rats: role of GluN2B-containing NMDA receptors.
Topics: Animals; Catheters, Indwelling; Corpus Striatum; Excitatory Amino Acid Antagonists; GABA-A Receptor Agonists; Male; Memory, Short-Term; Muscimol; Neural Pathways; Neuropsychological Tests; Odorants; Olfactory Perception; Phenols; Piperidines; Prefrontal Cortex; Rats, Long-Evans; Receptors, N-Methyl-D-Aspartate | 2017 |
Thalamic nucleus reuniens regulates fear memory destabilization upon retrieval.
Topics: Amygdala; Animals; Anisomycin; CA1 Region, Hippocampal; Clonidine; Cognition; Cysteine Proteinase Inhibitors; Early Growth Response Protein 1; Excitatory Amino Acid Antagonists; Fear; GABA-A Receptor Agonists; Lactones; Memory; Midline Thalamic Nuclei; Muscimol; Neurons; Piperidines; Prefrontal Cortex; Rats; Receptors, N-Methyl-D-Aspartate | 2020 |
Flexible versus Fixed Spatial Self-Ordered Response Sequencing: Effects of Inactivation and Neurochemical Modulation of Ventrolateral Prefrontal Cortex.
Topics: Animals; Antipsychotic Agents; Baclofen; Callithrix; Cognition Disorders; Dopamine; Dopamine D2 Receptor Antagonists; Fluorobenzenes; GABA Agonists; gamma-Aminobutyric Acid; Goals; Memory, Short-Term; Muscimol; Piperidines; Prefrontal Cortex; Psychomotor Performance; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Spatial Behavior; Sulpiride | 2021 |