muscimol and piperidines

muscimol has been researched along with piperidines in 34 studies

Research

Studies (34)

TimeframeStudies, this research(%)All Research%
pre-19907 (20.59)18.7374
1990's6 (17.65)18.2507
2000's12 (35.29)29.6817
2010's7 (20.59)24.3611
2020's2 (5.88)2.80

Authors

AuthorsStudies
Braestrup, C; Falch, E; Krogsgaard-Larsen, P; Nielsen, M2
Dziki, M; Ikonomidou, C; Parada-Turska, J; Turski, WA; Urbanska, E1
Kumasaka, Y; Ueki, S; Yamamoto, T1
Iversen, LL; Wong, EH1
Curtis, DR; Falch, E; Krogsgaard-Larsen, P; Nielsen, L1
Creveling, CR; Daly, JW; Hollingsworth, EB; Lewandowski, G; Waters, JA1
Mitchell, R; Wilson, LE1
Ammendola, D; De Sarro, A; De Sarro, G; Nava, F1
Ebert, B; Kemp, JA; Krogsgaard-Larsen, P; Wafford, KA; Whiting, PJ1
Ebert, B; Krogsgaard-Larsen, P; McKernan, R; Saounatsou, K; Thompson, SA; Wafford, KA1
Dement, WC; Mignot, E; Nishino, S; Reid, MS; Siegel, JM; Tafti, M1
Fields, HL; Manning, BH; Martin, WJ; Meng, ID1
Que, M; Witte, OW; Zilles, K1
Maksay, G; McKernan, R1
Engblom, C; Frølund, B; Kristiansen, U; Krogsgaard-Larsen, P; Liljefors, T; Stensbøl, TB; Tagmose, L1
Siemes, S; Szabo, B; Wallmichrath, I1
Ebert, B; Frølund, B; Kristiansen, U; Krogsgaard-Larsen, P; Liljefors, T1
Fukumori, R; Goshima, Y; Hagiwara, Y; Kanaya, T; Kubo, T; Okatani, H2
Dixon, HB; Dragoni, S; Frosini, M; Machetti, F; Palmi, M; Sesti, C; Sgaragli, G; Valoti, M1
Argiolas, A; Mascia, MS; Melis, MR; Melis, T; Sanna, F; Succu, S1
Fujii, Y; Kamei, C; Mikami, A; Yamamoto, Y1
Akabas, MH; Dannhardt, G; Debus, F; Dieler, S; Jansen, M; Lüddens, H; Rabe, H; Strehle, A1
Kovacs, FE; Szabo, B; Urbanski, MJ1
Abdel-Rahman, AA; Ibrahim, BM1
Cornélio, AM; Morgan, MM; Nunes-de-Souza, RL1
Arreto, CD; Bourgeais, L; Condes-Lara, M; Jay, T; Noseda, R; Robert, C; Villanueva, L1
Holmes, NM; Killcross, AS; Parkes, SL; Westbrook, RF1
Cui, CL; Ge, FF; Li, YJ; Ping, XJ; Qi, C; Shen, F; Sun, LL; Sun, XW; Xing, GG1
Chergui, K; Yao, N; Zhang, X1
Baillie, LD; Catton, JK; Davies, DA; Greba, Q; Howland, JG; Mulligan, SJ; Selk, JC1
Bertoglio, LJ; Troyner, F1
Axelsson, SFA; Horiguchi, N; Horst, NK; Robbins, TW; Roberts, AC1

Reviews

1 review(s) available for muscimol and piperidines

ArticleYear
GABA(A) receptor ligands and their therapeutic potentials.
    Current topics in medicinal chemistry, 2002, Volume: 2, Issue:8

    Topics: Animals; Central Nervous System Diseases; GABA Agents; GABA Agonists; GABA Antagonists; Humans; Isonicotinic Acids; Isoxazoles; Ligands; Muscimol; Piperidines; Protein Subunits; Receptors, GABA-A

2002

Other Studies

33 other study(ies) available for muscimol and piperidines

ArticleYear
Partial agonists for brain GABA/benzodiazepine receptor complex.
    Nature, 1979, Jul-26, Volume: 280, Issue:5720

    Topics: Animals; Benzodiazepines; Bicuculline; Brain; Crotonates; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, Drug; Sulfonic Acids

1979
Excitatory amino acid antagonists protect mice against seizures induced by bicuculline.
    Brain research, 1990, Apr-23, Volume: 514, Issue:1

    Topics: Animals; Bicuculline; Dibenzocycloheptenes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Mice; Muscimol; Pipecolic Acids; Piperazines; Piperidines; Receptors, Amino Acid; Receptors, Cell Surface; Seizures

1990
Behavioral analysis of zopiclone on the basis of their discriminative stimulus properties in the rat.
    Japanese journal of pharmacology, 1989, Volume: 51, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Behavior, Animal; Benzodiazepines; Bicuculline; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Hypnotics and Sedatives; Male; Muscimol; Naphthyridines; Pentylenetetrazole; Piperazines; Piperidines; Rats; Rats, Inbred WKY; Ritanserin; Serotonin Antagonists; Sulfur Compounds

1989
Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Androstanes; Animals; Azasteroids; Bicuculline; Cell Membrane; Cerebral Cortex; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isonicotinic Acids; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, GABA-A; Taurine

1985
GABA agonists. Resolution, absolute stereochemistry, and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:11

    Topics: Animals; Bicuculline; Brain; Cats; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Molecular Conformation; Muscimol; Neurons; Oxazolidinones; Piperidines; Rats; Receptors, GABA-A; Spinal Cord; Stereoisomerism; Structure-Activity Relationship; Synaptic Membranes

1985
Anticonvulsant activity of piperidinol and (dialkylamino)alkanol esters.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:8

    Topics: Amino Alcohols; Animals; Anticonvulsants; Ataxia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Diazepam; Electroshock; Esters; Muscimol; Pentylenetetrazole; Phenytoin; Piperidines; Rats; Receptors, GABA-A; Structure-Activity Relationship

1986
Two or more conformations of benzodiazepine receptors depending on GABA receptors and other variables.
    Advances in biochemical psychopharmacology, 1980, Volume: 21

    Topics: Animals; Benzodiazepines; Bicuculline; Brain; Diazepam; gamma-Aminobutyric Acid; Macromolecular Substances; Male; Muscimol; Piperidines; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Structure-Activity Relationship; Synaptic Membranes

1980
Effects of GABA receptor agonists on [3H] flunitrazepam binding to rat cerebellar and hippocampal membranes.
    Neuropharmacology, 1983, Volume: 22, Issue:7

    Topics: Animals; Cerebellum; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Imidazoles; Male; Membranes; Muscimol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Effects of some excitatory amino acid antagonists on imipenem-induced seizures in DBA/2 mice.
    Brain research, 1995, Feb-06, Volume: 671, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Animals; Anticonvulsants; Dizocilpine Maleate; Excitatory Amino Acids; Glutamine; Imipenem; Kynurenic Acid; Mice; Mice, Inbred DBA; Muscimol; Piperazines; Piperidines; Quinoxalines; Seizures

1995
Molecular pharmacology of gamma-aminobutyric acid type A receptor agonists and partial agonists in oocytes injected with different alpha, beta, and gamma receptor subunit combinations.
    Molecular pharmacology, 1994, Volume: 46, Issue:5

    Topics: Animals; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Muscimol; Oocytes; Oxazolidinones; Piperidines; Receptors, GABA-A; Recombinant Proteins; Structure-Activity Relationship; Xenopus

1994
Differences in agonist/antagonist binding affinity and receptor transduction using recombinant human gamma-aminobutyric acid type A receptors.
    Molecular pharmacology, 1997, Volume: 52, Issue:6

    Topics: Animals; Binding, Competitive; DNA, Complementary; Electrophysiology; GABA Agonists; GABA Antagonists; Humans; Isoxazoles; Kinetics; Macromolecular Substances; Muscimol; Oocytes; Piperidines; Receptors, GABA-A; Transduction, Genetic; Transfection; Tritium; Xenopus laevis

1997
Neuropharmacological characterization of basal forebrain cholinergic stimulated cataplexy in narcoleptic canines.
    Experimental neurology, 1998, Volume: 151, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Behavior, Animal; Carbachol; Cataplexy; Cholinergic Fibers; Dogs; Feeding Behavior; Female; GABA Agonists; Gallamine Triethiodide; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Muscimol; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Piperidines; Pirenzepine; Prosencephalon

1998
An analgesia circuit activated by cannabinoids.
    Nature, 1998, Sep-24, Volume: 395, Issue:6700

    Topics: Analgesia; Analgesics, Non-Narcotic; Animals; Benzoxazines; Cannabinoids; GABA Agonists; Male; Medulla Oblongata; Morphine; Morpholines; Motor Activity; Muscimol; Naphthalenes; Neural Pathways; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

1998
Transient up-regulation of gamma-aminobutyric acid(A) receptor binding by lubeluzole after neocortical specify lesion in rats.
    Neuroscience letters, 2000, Dec-22, Volume: 296, Issue:2-3

    Topics: Animals; Brain Ischemia; Male; Muscimol; Neocortex; Neuroprotective Agents; Photochemistry; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, AMPA; Receptors, GABA-A; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Rose Bengal; Thiazoles; Tritium; Up-Regulation

2000
Entropy as the predominant driving force of binding to human recombinant alpha(x)beta(3)gamma(2) GABA(A) receptors.
    European journal of pharmacology, 2001, Jan-05, Volume: 411, Issue:1-2

    Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Entropy; GABA Agonists; GABA Antagonists; Humans; Isoxazoles; L Cells; Membranes; Mice; Muscimol; Piperidines; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Temperature; Tritium

2001
A novel class of potent 3-isoxazolol GABA(A) antagonists: design, synthesis, and pharmacology.
    Journal of medicinal chemistry, 2000, Dec-28, Volume: 43, Issue:26

    Topics: Animals; Brain; Cells, Cultured; GABA Antagonists; Isoxazoles; Models, Molecular; Muscimol; Neurons; Patch-Clamp Techniques; Piperidines; Radioligand Assay; Rats; Receptors, GABA-A; Structure-Activity Relationship; Synaptic Membranes

2000
Inhibition of GABAergic neurotransmission in the ventral tegmental area by cannabinoids.
    The European journal of neuroscience, 2002, Volume: 15, Issue:12

    Topics: Analgesics; Animals; Animals, Newborn; Benzoxazines; Cannabinoids; Drug Interactions; GABA Agonists; gamma-Aminobutyric Acid; Membrane Potentials; Morpholines; Muscimol; Naphthalenes; Neural Inhibition; Neural Pathways; Neurons; Nucleus Accumbens; Organ Culture Techniques; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Receptors, GABA-A; Rimonabant; Synaptic Transmission; Ventral Tegmental Area

2002
Cholinergic mechanism in the lateral septal area is involved in the stress-induced blood pressure increase in rats.
    Brain research bulletin, 2003, Jan-30, Volume: 59, Issue:5

    Topics: Animals; Blood Pressure; Carbachol; Cholinergic Agonists; Cholinesterase Inhibitors; Epinephrine; GABA Agonists; Injections, Intraventricular; Male; Muscarinic Antagonists; Muscimol; Norepinephrine; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Restraint, Physical; Septal Nuclei; Stress, Physiological

2003
Interactions of taurine and structurally related analogues with the GABAergic system and taurine binding sites of rabbit brain.
    British journal of pharmacology, 2003, Volume: 138, Issue:6

    Topics: 4-Aminobutyrate Transaminase; Animals; Binding Sites; Brain; Drug Interactions; gamma-Aminobutyric Acid; Isomerism; Molecular Structure; Muscimol; Piperidines; Rabbits; Receptors, GABA-A; Receptors, GABA-B; Receptors, Neurotransmitter; Structure-Activity Relationship; Synaptic Membranes; Synaptosomes; Taurine; Tritium

2003
Projections from the caudal part to the rostral part of the lateral septal area mediate blood pressure increase.
    Brain research bulletin, 2003, Sep-30, Volume: 61, Issue:5

    Topics: Animals; Blood Pressure; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Fluorescent Dyes; GABA Agonists; Hypertension; Male; Microinjections; Muscarinic Antagonists; Muscimol; Neural Pathways; Neurons; Piperidines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Reaction Time; Septum of Brain; Stress, Physiological

2003
The cannabinoid CB1 receptor antagonist SR 141716A induces penile erection by increasing extra-cellular glutamic acid in the paraventricular nucleus of male rats.
    Behavioural brain research, 2006, May-15, Volume: 169, Issue:2

    Topics: Anesthetics, Local; Animals; Baclofen; Behavior, Animal; Cannabinoid Receptor Antagonists; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Extracellular Space; GABA Agonists; Glutamic Acid; Male; Microdialysis; Microinjections; Models, Biological; Muscimol; Paraventricular Hypothalamic Nucleus; Penile Erection; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Tetrodotoxin

2006
Effect of histamine on muscimol-induced working memory deficits in radial maze performance.
    Journal of pharmacological sciences, 2007, Volume: 104, Issue:3

    Topics: Animals; Brain Chemistry; Cholinesterase Inhibitors; Donepezil; Dose-Response Relationship, Drug; GABA Agonists; GABA-A Receptor Agonists; Histamine; Histidine; Indans; Male; Maze Learning; Memory Disorders; Memory, Short-Term; Microinjections; Muscimol; Piperidines; Rats; Tacrine

2007
Synthesis of GABAA receptor agonists and evaluation of their alpha-subunit selectivity and orientation in the GABA binding site.
    Journal of medicinal chemistry, 2008, Aug-14, Volume: 51, Issue:15

    Topics: Animals; Binding Sites; Brain; Cell Line; Electrophysiology; Female; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Models, Molecular; Molecular Structure; Muscimol; Mutation; Oocytes; Patch-Clamp Techniques; Piperidines; Protein Subunits; Rats; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis

2008
Depolarizing GABAergic synaptic input triggers endocannabinoid-mediated retrograde synaptic signaling.
    Synapse (New York, N.Y.), 2009, Volume: 63, Issue:8

    Topics: Aniline Compounds; Animals; Animals, Newborn; Arachidonic Acids; Benzamides; Bicuculline; Biophysics; Calcium; Calcium Signaling; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Carbamates; Cerebellum; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Fluoresceins; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Lactones; Mice; Muscimol; Orlistat; Patch-Clamp Techniques; Piperidines; Purkinje Cells; Pyrazoles; Quinoxalines; Rimonabant; Signal Transduction; Synapses; Valine

2009
Role of brainstem GABAergic signaling in central cannabinoid receptor evoked sympathoexcitation and pressor responses in conscious rats.
    Brain research, 2011, Sep-26, Volume: 1414

    Topics: Analysis of Variance; Animals; Benzoxazines; Blood Pressure; Brain Stem; Dose-Response Relationship, Drug; Drug Interactions; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Heart Rate; Injections, Intraventricular; Male; Morpholines; Muscimol; Naphthalenes; Neurons; Norepinephrine; Piperidines; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Tyrosine 3-Monooxygenase; Wakefulness

2011
Contribution of the rostral ventromedial medulla to post-anxiety induced hyperalgesia.
    Brain research, 2012, Apr-23, Volume: 1450

    Topics: Animals; Anxiety; GABA-A Receptor Agonists; Hyperalgesia; Male; Medulla Oblongata; Muscimol; Pain Measurement; Pain Threshold; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1

2012
Paraventricular hypothalamic regulation of trigeminovascular mechanisms involved in headaches.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, May-15, Volume: 33, Issue:20

    Topics: Action Potentials; Animals; Biotin; Corticosterone; Dextrans; Disease Models, Animal; GABA Antagonists; GABA-A Receptor Agonists; Male; Muscimol; Neural Pathways; Neurons; Paraventricular Hypothalamic Nucleus; Physical Stimulation; Piperidines; Pituitary Adenylate Cyclase-Activating Polypeptide; Pyridazines; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Stilbamidines; Stress, Psychological; Trigeminal Nuclei; Tryptamines

2013
The basolateral amygdala is critical for learning about neutral stimuli in the presence of danger, and the perirhinal cortex is critical in the absence of danger.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Aug-07, Volume: 33, Issue:32

    Topics: Acoustic Stimulation; Amygdala; Animals; Association Learning; Conditioning, Classical; Environment; Excitatory Amino Acid Antagonists; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; GABA-A Receptor Agonists; Male; Muscimol; Photic Stimulation; Piperidines; Prefrontal Cortex; Rats; Rats, Wistar

2013
Re-exposure to morphine-associated context facilitated long-term potentiation in the vSUB-NAc glutamatergic pathway via GluN2B-containing receptor activation.
    Addiction biology, 2017, Volume: 22, Issue:2

    Topics: Analgesics, Opioid; Animals; Baclofen; Behavior, Animal; Conditioning, Operant; GABA-A Receptor Agonists; GABA-B Receptor Agonists; Hippocampus; Long-Term Potentiation; Male; Memory; Morphine; Muscimol; Nucleus Accumbens; Phenols; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

2017
The GABAA receptor agonist muscimol induces an age- and region-dependent form of long-term depression in the mouse striatum.
    Learning & memory (Cold Spring Harbor, N.Y.), 2016, Volume: 23, Issue:9

    Topics: Animals; Corpus Striatum; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA-A Receptor Agonists; Long-Term Synaptic Depression; Male; Mice, Inbred C57BL; Muscimol; Piperidines; Pyrazoles; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, GABA-A; TRPV Cation Channels

2016
Interactions between medial prefrontal cortex and dorsomedial striatum are necessary for odor span capacity in rats: role of GluN2B-containing NMDA receptors.
    Learning & memory (Cold Spring Harbor, N.Y.), 2017, Volume: 24, Issue:10

    Topics: Animals; Catheters, Indwelling; Corpus Striatum; Excitatory Amino Acid Antagonists; GABA-A Receptor Agonists; Male; Memory, Short-Term; Muscimol; Neural Pathways; Neuropsychological Tests; Odorants; Olfactory Perception; Phenols; Piperidines; Prefrontal Cortex; Rats, Long-Evans; Receptors, N-Methyl-D-Aspartate

2017
Thalamic nucleus reuniens regulates fear memory destabilization upon retrieval.
    Neurobiology of learning and memory, 2020, Volume: 175

    Topics: Amygdala; Animals; Anisomycin; CA1 Region, Hippocampal; Clonidine; Cognition; Cysteine Proteinase Inhibitors; Early Growth Response Protein 1; Excitatory Amino Acid Antagonists; Fear; GABA-A Receptor Agonists; Lactones; Memory; Midline Thalamic Nuclei; Muscimol; Neurons; Piperidines; Prefrontal Cortex; Rats; Receptors, N-Methyl-D-Aspartate

2020
Flexible versus Fixed Spatial Self-Ordered Response Sequencing: Effects of Inactivation and Neurochemical Modulation of Ventrolateral Prefrontal Cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2021, 08-25, Volume: 41, Issue:34

    Topics: Animals; Antipsychotic Agents; Baclofen; Callithrix; Cognition Disorders; Dopamine; Dopamine D2 Receptor Antagonists; Fluorobenzenes; GABA Agonists; gamma-Aminobutyric Acid; Goals; Memory, Short-Term; Muscimol; Piperidines; Prefrontal Cortex; Psychomotor Performance; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Spatial Behavior; Sulpiride

2021