muscimol and pentobarbital

muscimol has been researched along with pentobarbital in 122 studies

Research

Studies (122)

TimeframeStudies, this research(%)All Research%
pre-199054 (44.26)18.7374
1990's49 (40.16)18.2507
2000's11 (9.02)29.6817
2010's8 (6.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ho, IK; Yu, S1
Bertrand, PP; Galligan, JJ1
Berger, T; Kettenmann, H; Schnitzer, J; Walz, W1
Shibata, S; Tominaga, K; Ueki, S; Watanabe, S1
Aibara, K; Akaike, N; Itabashi, S; Sasaki, H1
Allan, AM; Draski, LJ; Mayes, GG1
Gautam, SK; Kulkarni, SK1
Dohi, T; Kitayama, S; Morita, K; Tsujimoto, A1
Akaike, N; Shirasaki, T; Yakushiji, T1
Cano, J; Machado, A; Ruano, D; Vitorica, J1
Kang, T; Xiao-Hong, D; Xin-Quan, J1
Akaike, N; Nakagawa, T; Nakaye, T; Shirasaki, T; Wakamori, M1
Hori, S; Ito, T; Kadokawa, T; Miura, Y; Miyahara, T; Shimada, J1
Fincher, AS; Frye, GD; Griffith, WH; Lorenzetti, M; Trzeciakowski, J1
Balfour, DJ; Stevenson, IH; Yau, JL1
Kim, KH; Takeuchi, H1
Paul, SM; Schwartz, RD; Skolnick, P; Suzdak, PD1
Paul, SM; Schwartz, RD; Suzdak, PD1
Majewska, MD; Paul, SM; Schwartz, RD1
Moody, EJ; Paul, SM; Skolnick, P; Suzdak, PD1
Akaike, N; Ikemoto, Y; Kijima, H1
Allan, AM; Harris, RA2
Dudek, BC; Phillips, TJ1
Paul, SM; Schwartz, RD; Seale, TW; Skolnick, P1
Bédard, L; Roberge, AG; Seoane, JR; Thibault, L; Wandji, SA1
Akaike, N; Hattori, K; Inomata, N; Oomura, Y1
Nistri, A; Sivilotti, L1
Mehta, AK; Ticku, MK2
Hanada, S; Hashimoto, S; Tanaka, C; Taniyama, K1
Karanian, JW; Morrow, AL; Paul, SM; Suzdak, PD1
Hara, S; Morioka, S; Satoh, K; Yanagihara, S1
Callachan, H; Kirkness, EF; Lambert, JJ; Peters, JA; Turner, AJ1
Georgiev, V; Getova, D1
Handley, SL; Heaton, JC; Rea, PJ; Singh, L1
Iwai, S; Shirakawa, J; Tanaka, C; Taniyama, K1
Spealman, RD1
Olsen, RW; Snowman, AM2
Lee, RJ; Lomax, P; McCabe, RT; Olsen, RW; Wamsley, JK1
Simmonds, MA1
Sweetnam, PM; Tallman, JF1
Audi, EA; Brandão, ML; Graeff, FG; Schütz, MT1
Little, HJ; Nutt, DJ; Taylor, SC1
Maksay, G; Nielsen, M; Simonyi, M1
Lindgren, S; Simmonds, MA1
Olsen, RW; Yang, JS1
Bédard, L; Caron, N; Seoane, JR1
Biggio, G; Concas, A; Mele, S1
Girard, CL; Matte, JJ; Seoane, JR1
Jackson, MB1
Harrison, NL; Simmonds, MA1
Kamp, CW; Morgan, WW1
Borea, PA; Karobath, M; Supavilai, P1
Nicoll, RA; Wojtowicz, JM1
Davis, WC; Ticku, MK1
Burch, TP; Ticku, MK1
Ho, IK; Nabeshima, T; Sivam, SP1
Barker, JL; Jackson, MB; Lecar, H; Mathers, DA1
Olsen, RW; Stephenson, FA1
Itoga, E; Kishida, T; Kito, S; Togo, M1
Burch, TP; Thyagarajan, R; Ticku, MK1
Brenner, O; Quast, U1
Burch, TP; Ramanjaneyulu, R; Thyagarajan, R; Ticku, MK1
Barnard, EA; Sigel, E1
Brody, LE; Jacobs, R; Jones, EA; Pappas, SC; Schafer, DF1
Herling, S; Valentino, RJ; Winger, GD1
Harris, RA; Rohde, BH1
Collins, GG1
Amin, J; Weiss, DS1
Kelder, D; Ross, SB1
Hiemke, C; Jussofie, A; Schmiz, A1
Fukuda, H; Ito, Y; Segawa, K1
Araki, T; Kanai, Y; Kato, H; Kogure, K1
Peoples, RW; Weight, FF1
Auerbach, SB; Tao, R1
Garcia de Yebenes, E; Pelletier, G1
Belelli, D; Chen, R; Lambert, JJ; Lan, NC; Peters, JA; Reyes, A1
Lukasiewicz, PD; Maple, BR; Werblin, FS1
Ho, IK; Ito, Y1
Li, S; Pelletier, G1
Jussofie, A1
Ho, IK; Miyaoka, T; Tseng, YT1
Chikai, T; Oishi, R; Saeki, K1
Misawa, M; Motegi, H; Suzuki, T1
Dowling, JE; Qian, H1
Biggio, G; Ghiani, CA; Maciocco, E; Sanna, E; Serra, M; Tuligi, G1
Brozowski, SJ; Hadingham, KL; Harris, RA; Whatley, VJ; Whiting, PJ1
Reis, DJ; Sun, MK1
Davies, PA; Hales, TG; Hanna, MC; Kirkness, EF1
Brozowski, S; Hadingham, K; Harris, RA; Mihic, SJ; Whiting, PJ1
Barros, HM; Manitiu, A; Miczek, KA; Vivian, JA1
Brozowski, S; Chuang, L; Hadingham, K; Harris, RA; Valenzuela, CF; Whiting, PJ1
Dzoljic, M; Van Duijn, B1
Chang, X; Javors, MA; King, TS; Levinson, C; Ticku, MK1
Davies, M; Dunn, SM; Thuynsma, RP1
Lee, YP; Yin, HS1
Akhondzadeh, S; Stone, TW1
Isshiki, A; Ito, H; Uchino, H; Watanabe, Y1
Chau, C; Hales, TG; Kaufman, DL; Tian, J1
Chistina Grobin, A; Devaud, LL; Inglefield, JR; Morrow, AL; Schwartz-Bloom, RD1
Ho, IK; Oh, S1
Galligan, JJ; Zhou, X1
Azarov, A; Grant, KA; Green-Jordan, K; Szeliga, KT; Waters, CA1
Baufreton, J; Bioulac, B; Dovero, S; Dufy, B; Garret, M; Taupignon, A1
Adkins, CE; Bonnert, TP; Gonzalez, JE; Haldon, C; Kerby, J; McKernan, RM; Oades, K; Pillai, GV; Simpson, PB; Whiting, PJ1
Fregosi, RF; Iizuka, M; Luo, Z1
Eun, JS; Han, H; Hong, JT; Kim, HC; Ma, Y; Oh, KW1
Han, H; Hong, JT; Kim, YB; Ma, Y; Nam, SY; Oh, KW; Yun, YP1
Czajkowski, C; Sharkey, LM1
Eun, JS; Hong, JT; Kim, YB; Lee, MK; Ma, H; Ma, Y; Nam, SY; Oh, KW1
Leung, LS; Long, JJ; Luo, T; McMurran, TJ; Shen, B; Stewart, L1
Behan, M; Carey, HV; Hengen, KB; Johnson, SM; Jones, MV1
Baptiste, SL; Devinsky, O; French, JA; Kuzniecky, RI; Ludvig, N; Tang, HM1
Han, JY; Hong, JT; Moon, DC; Oh, KW; Park, KS1
Chong, MS; Han, JY; Hong, JT; Hu, Z; Kim, CS; Kim, JW; Kim, SK; Lee, K; Oh, KW; Yeo, YM; Yoo, SK1
Bordey, A; Ikeda-Matsuo, Y; Kubera, C; Taylor, MM; Wu, S; Young, SZ1
Constantin, S; Herbison, AE; Iremonger, KJ1
Han, JY; Hong, JT; Lee, CI; Oh, KW1
Grauer, M; Jabs, R; Passlick, S; Schäfer, C; Seifert, G; Steinhäuser, C1
Kilb, W; Luhmann, HJ; Winkler, P1

Other Studies

122 other study(ies) available for muscimol and pentobarbital

ArticleYear
Effects of acute pentobarbital administration on GABAA receptor-regulated chloride uptake in rat brain synaptoneurosomes.
    Brain research bulletin, 1992, Volume: 28, Issue:5

    Topics: Animals; Brain; Cerebellum; Cerebral Cortex; Chlorides; Flunitrazepam; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1992
Alfaxalone, pentobarbital and diazepam potentiate gamma-aminobutyric acid-induced depolarizations in single myenteric neurons of guinea pig intestine.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Anesthetics; Animals; Diazepam; Drug Synergism; gamma-Aminobutyric Acid; Guinea Pigs; Hydrocortisone; Intestines; Male; Membrane Potentials; Muscimol; Pentobarbital; Pregnanediones; Receptors, GABA-A

1992
GABA- and glutamate-activated currents in glial cells of the mouse corpus callosum slice.
    Journal of neuroscience research, 1992, Volume: 31, Issue:1

    Topics: Action Potentials; Animals; Bicuculline; Chloride Channels; Corpus Callosum; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Ion Channel Gating; Kainic Acid; Membrane Proteins; Mice; Muscimol; Oligodendroglia; Pentobarbital; Potassium Channels; Receptors, GABA-A; Receptors, Glutamate; Receptors, Neurotransmitter; Stem Cells

1992
Effects of inhibitory and excitatory drugs on the metabolic rhythm of the hamster suprachiasmatic nucleus in vitro.
    European journal of pharmacology, 1992, Jun-24, Volume: 217, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Circadian Rhythm; Cricetinae; Deoxyglucose; Dose-Response Relationship, Drug; Flurazepam; Glutamates; Glutamic Acid; Male; Mesocricetus; Muscimol; Neurons; Pentobarbital; Potassium Chloride; Suprachiasmatic Nucleus; Tetrodotoxin

1992
gamma-Aminobutyric acid-induced response in rat dissociated paratracheal ganglion cells.
    Journal of neurophysiology, 1992, Volume: 67, Issue:5

    Topics: Animals; Chlorides; Diazepam; Drug Synergism; Electric Conductivity; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Trachea

1992
gamma-Aminobutyric acid-activated chloride channels in rats selectively bred for differential acute sensitivity to alcohol.
    Alcoholism, clinical and experimental research, 1991, Volume: 15, Issue:2

    Topics: Alcohol Drinking; Animals; Chloride Channels; Diazepam; Female; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Proteins; Muscimol; Pentobarbital; Phenobarbital; Phenotype; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Selection, Genetic

1991
GABA/BZ-and NMDA-receptor interaction in digoxin-induced convulsions in rats.
    Indian journal of experimental biology, 1991, Volume: 29, Issue:7

    Topics: Animals; Baclofen; Diazepam; Digoxin; Dizocilpine Maleate; Female; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Salts; Seizures

1991
GABAergic modulation of catecholamine release from cultured bovine adrenal chromaffin cells. Evidence for the involvement of Cl(-)-dependent Ca2+ entry.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 341, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Glands; Animals; Calcium; Calcium Radioisotopes; Catecholamines; Cattle; Cells, Cultured; Chlorides; Chromaffin System; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Ion Channels; Muscimol; Pentobarbital; Time Factors; Veratridine

1990
Quinolones and fenbufen interact with GABAA receptor in dissociated hippocampal cells of rat.
    Journal of neurophysiology, 1991, Volume: 66, Issue:2

    Topics: 4-Quinolones; Animals; Anti-Infective Agents; Anti-Inflammatory Agents, Non-Steroidal; Chloride Channels; Drug Interactions; Electrophysiology; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Ion Channels; Membrane Proteins; Muscimol; Neurons; Pentobarbital; Phenylbutyrates; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship

1991
Pharmacologic characterization of GABAA/benzodiazepine receptor in rat hippocampus during aging.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:3

    Topics: Aging; Animals; Binding Sites; Cerebellum; Cerebral Cortex; Culture Techniques; Drug Interactions; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A

1991
Pentobarbital selectively blocks supraspinal morphine analgesia. Evidence for GABAA receptor involvement.
    Pain, 1990, Volume: 43, Issue:3

    Topics: Analgesia; Animals; Diazepam; Drug Synergism; Injections, Intraventricular; Injections, Spinal; Male; Morphine; Muscimol; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord

1990
gamma-Aminobutyric acid-induced response in acutely isolated nucleus solitarii neurons of the rat.
    The American journal of physiology, 1991, Volume: 260, Issue:4 Pt 1

    Topics: Animals; Bicuculline; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Medulla Oblongata; Membrane Potentials; Muscimol; Neurons; Penicillin G; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Strychnine

1991
Effects of enoxacin and its combination with 4-biphenylacetate, an active metabolite of fenbufen, on population spikes in rat hippocampal slices.
    Pharmacology & toxicology, 1991, Volume: 68, Issue:3

    Topics: Action Potentials; Animals; Anti-Inflammatory Agents, Non-Steroidal; Baclofen; Bicuculline; Clorazepate Dipotassium; Drug Interactions; Electric Stimulation; Enoxacin; Hippocampus; In Vitro Techniques; Male; Muscimol; Pentobarbital; Phenylacetates; Phenylbutyrates; Rats; Rats, Inbred Strains

1991
Comparison of contractile responses of the guinea pig ileum longitudinal muscle to ethanol and GABAA agonists.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:2

    Topics: Animals; Atropine; Bicuculline; Chlorides; Ethanol; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscimol; Muscle Contraction; Pentobarbital; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Taurine; Tetrodotoxin

1990
Postmortem stability of the GABAA receptor complex: a study using rat brain cerebrocortical membranes.
    Biochemical pharmacology, 1990, Aug-15, Volume: 40, Issue:4

    Topics: Animals; Cerebral Cortex; Male; Muscimol; Pentobarbital; Postmortem Changes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Time Factors

1990
Pharmacological characteristics of two different types of inhibitory GABA receptors on Achatina fulica neurones.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Crotonates; Diazepam; Dibenzazepines; Electrophysiology; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Muscimol; Neurons; Pentobarbital; Picrotoxin; Receptors, GABA-A; Snails

1990
Ethanol stimulates gamma-aminobutyric acid receptor-mediated chloride transport in rat brain synaptoneurosomes.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:11

    Topics: Animals; Bicuculline; Biological Transport; Brain; Cell-Free System; Chlorides; Ethanol; In Vitro Techniques; Ion Channels; Muscimol; Pentobarbital; Picrotoxin; Rats; Receptors, GABA-A; Synaptosomes

1986
gamma-Aminobutyric acid (GABA)- and barbiturate-mediated 36Cl- uptake in rat brain synaptoneurosomes: evidence for rapid desensitization of the GABA receptor-coupled chloride ion channel.
    Molecular pharmacology, 1986, Volume: 30, Issue:5

    Topics: Animals; Cerebral Cortex; Chlorides; Dose-Response Relationship, Drug; Ethanol; gamma-Aminobutyric Acid; Ion Channels; Male; Muscimol; Pentobarbital; Ranidae; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1986
Factors modulating the sensitivity of the GABA receptor-gated chloride ion channel.
    Clinical neuropharmacology, 1986, Volume: 9 Suppl 4

    Topics: Animals; Chlorides; Ion Channels; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1986
Modulation of the benzodiazepine/gamma-aminobutyric acid receptor chloride channel complex by inhalation anesthetics.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: Anesthesia, Inhalation; Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Enflurane; Ether; Halothane; Ion Channels; Male; Methoxyflurane; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1988
Kinetic and pharmacological properties of the GABA-induced chloride current in Aplysia neurones: a 'concentration clamp' study.
    British journal of pharmacology, 1988, Volume: 95, Issue:3

    Topics: Animals; Aplysia; beta-Alanine; Chlorides; Diazepam; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Muscimol; Neurons; Pentobarbital

1988
Sensitivity to ethanol hypnosis and modulation of chloride channels does not cosegregate with pentobarbital sensitivity in HS mice.
    Alcoholism, clinical and experimental research, 1989, Volume: 13, Issue:3

    Topics: Animals; Arousal; Brain; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Drug Tolerance; Ethanol; Flunitrazepam; Ion Channels; Male; Membrane Proteins; Mice; Muscimol; Pentobarbital; Receptors, GABA-A; Sleep Stages

1989
Genotype-dependent effects of GABAergic agents on sedative properties of ethanol.
    Psychopharmacology, 1989, Volume: 98, Issue:4

    Topics: Animals; Bicuculline; Ethanol; gamma-Aminobutyric Acid; Genetics, Behavioral; Genotype; Hypnotics and Sedatives; Male; Mice; Mice, Inbred A; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Inbred Strains; Muscimol; Pentobarbital; Picrotoxin; Species Specificity

1989
Differential seizure sensitivities to picrotoxinin in two inbred strains of mice (DBA/2J and BALB/c ByJ): parallel changes in GABA receptor-mediated chloride flux and receptor binding.
    Brain research, 1989, Feb-27, Volume: 481, Issue:1

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; Frontal Lobe; Male; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Muscimol; Pentobarbital; Picrotoxin; Receptors, GABA-A; Seizures; Species Specificity; Synaptosomes

1989
Effects of intrahypothalamic injections of GABA, muscimol, pentobarbital, and L-glutamic acid on feed intake of satiated sheep.
    Canadian journal of physiology and pharmacology, 1989, Volume: 67, Issue:1

    Topics: Animals; Feeding Behavior; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hypothalamus; Male; Muscimol; Pentobarbital; Satiation; Sheep; Time Factors

1989
gamma-Aminobutyric-acid- and pentobarbitone-gated chloride currents in internally perfused frog sensory neurones.
    The Journal of physiology, 1985, Volume: 360

    Topics: Action Potentials; Amino Acids; Animals; Chlorides; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Ganglia, Spinal; In Vitro Techniques; Ion Channels; Muscimol; Neurons, Afferent; Pentobarbital

1985
Pharmacology of a novel effect of gamma-aminobutyric acid on the frog optic tectum in vitro.
    European journal of pharmacology, 1989, May-19, Volume: 164, Issue:2

    Topics: Animals; Bicuculline; Chlorides; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Midazolam; Muscimol; Pentobarbital; Rana temporaria; Superior Colliculi

1989
Characteristics of flunitrazepam binding to intact primary cultured spinal cord neurons and its modulation by GABAergic drugs.
    Journal of neurochemistry, 1987, Volume: 49, Issue:5

    Topics: Animals; Benzodiazepines; Binding, Competitive; Carbolines; Cells, Cultured; Embryo, Mammalian; Etazolate; Etomidate; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Muscimol; Neurons; Pentobarbital; Receptors, GABA-A; Spinal Cord

1987
Benzodiazepines and barbiturate potentiate the pre- and postsynaptic gamma-aminobutyric acid (GABA)A receptor-mediated response in the enteric nervous system of guinea pig small intestine.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Acetylcholine; Animals; Barbiturates; Benzodiazepines; Clonazepam; Diazepam; Female; Flumazenil; Guinea Pigs; Intestine, Small; Male; Muscimol; Pentobarbital; Potassium; Receptors, GABA-A

1988
Chronic ethanol administration alters gamma-aminobutyric acid, pentobarbital and ethanol-mediated 36Cl- uptake in cerebral cortical synaptoneurosomes.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1

    Topics: Administration, Inhalation; Animals; Cerebral Cortex; Chlorides; Dose-Response Relationship, Drug; Ethanol; gamma-Aminobutyric Acid; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synapses

1988
Exacerbation of indomethacin-induced gastric ulceration by systemically administered GABA in rats: possible involvement of peripheral GABA receptors.
    Japanese journal of pharmacology, 1988, Volume: 47, Issue:4

    Topics: Animals; Anticonvulsants; Atropine; beta-Alanine; Bicuculline; Drug Synergism; gamma-Aminobutyric Acid; Glycine; Indomethacin; Male; Muscimol; Pentobarbital; Pentylenetetrazole; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stomach Ulcer; Taurine

1988
Modulation of the GABAA receptor by depressant barbiturates and pregnane steroids.
    British journal of pharmacology, 1988, Volume: 94, Issue:4

    Topics: Animals; Barbiturates; Cattle; Chromaffin System; In Vitro Techniques; Muscimol; Pentobarbital; Pregnanes; Receptors, GABA-A; Secobarbital; Swine

1988
GABA-ergic mechanisms in the anticonvulsive activity of newly synthesized barbiturates. II. Correlation of HB-7 with GABA-ergic agents.
    Acta physiologica et pharmacologica Bulgarica, 1988, Volume: 14, Issue:2

    Topics: Animals; Anticonvulsants; Baclofen; Barbiturates; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Mice; Muscimol; Pentobarbital; Receptors, GABA-A

1988
Involvement of noradrenaline in potentiation of the head-twitch response by GABA-related drugs.
    Psychopharmacology, 1986, Volume: 88, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Brain Chemistry; Catecholamines; Diazepam; Dopamine; Drug Synergism; gamma-Aminobutyric Acid; Male; Methoxydimethyltryptamines; Metoprolol; Mice; Muscimol; Norepinephrine; Pentobarbital; Picrotoxin; Stereotyped Behavior; Taurine

1986
Regulation of [3H]GABA release from strips of guinea pig urinary bladder.
    The American journal of physiology, 1988, Volume: 255, Issue:6 Pt 2

    Topics: Acetylcholine; Animals; Atropine; Baclofen; Bicuculline; Clonazepam; Clonidine; Female; gamma-Aminobutyric Acid; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Male; Muscimol; Pentobarbital; Phenylephrine; Pirenzepine; Potassium; Prazosin; Tritium; Urinary Bladder; Yohimbine

1988
Discriminative-stimulus effects of midazolam in squirrel monkeys: comparison with other drugs and antagonism by Ro 15-1788.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Azabicyclo Compounds; Barbital; Benzodiazepines; Benzodiazepinones; Buspirone; Caffeine; Chlordiazepoxide; Cinanserin; Clozapine; Conditioning, Operant; Cyproheptadine; Diazepam; Diphenhydramine; Discrimination Learning; Electroshock; Flumazenil; Male; Midazolam; Muscimol; Nordazepam; Pentobarbital; Piperazines; Pyridazines; Pyrimidines; Saimiri; Tripelennamine

1985
Avermectin B1a modulation of gamma-aminobutyric acid/benzodiazepine receptor binding in mammalian brain.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Animals; Bicuculline; Brain; Cattle; Cell Membrane; Cerebral Cortex; Etazolate; gamma-Aminobutyric Acid; Isonicotinic Acids; Ivermectin; Lactones; Muscimol; Pentobarbital; Rats; Receptors, GABA-A

1985
Benzodiazepine/gamma-aminobutyric acid receptor deficit in the midbrain of the seizure-susceptible gerbil.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:19

    Topics: Animals; Bicuculline; Diazepam; Disease Models, Animal; Flunitrazepam; Gerbillinae; Mesencephalon; Muscimol; Pentobarbital; Receptors, GABA-A; Seizures

1985
Antagonism of flurazepam and other effects of Ro15-1788, PK8165 and Ro5-4864 on the GABA-A receptor complex in rat cuneate nucleus.
    European journal of pharmacology, 1985, Oct-29, Volume: 117, Issue:1

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Drug Synergism; Flumazenil; Flurazepam; In Vitro Techniques; Male; Medulla Oblongata; Muscimol; Pentobarbital; Picrotoxin; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Regional difference in brain benzodiazepine receptor carbohydrates.
    Molecular pharmacology, 1986, Volume: 29, Issue:3

    Topics: Acetylglucosaminidase; Animals; Asparagine; Benzodiazepinones; Brain Chemistry; Carbohydrates; Electrophoresis, Polyacrylamide Gel; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Male; Mannosyl-Glycoprotein Endo-beta-N-Acetylglucosaminidase; Molecular Weight; Muscimol; Neuraminidase; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sialic Acids; Tritium

1986
Modulation of the brain aversive system by GABAergic and serotonergic mechanisms.
    Behavioural brain research, 1986, Volume: 21, Issue:1

    Topics: Animals; Avoidance Learning; Benzodiazepines; Cerebral Ventricles; Chlordiazepoxide; Drug Interactions; gamma-Aminobutyric Acid; Isonicotinic Acids; Midazolam; Muscimol; Pentobarbital; Periaqueductal Gray; Rats; Receptors, GABA-A; Serotonin

1986
The effects of drugs acting at the GABAA-receptor/ionophore after chemical kindling with the benzodiazepine receptor ligand FG 7142.
    British journal of pharmacology, 1986, Volume: 88, Issue:3

    Topics: Animals; Bicuculline; Body Temperature; Carbolines; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Mice; Muscimol; Pentobarbital; Pentylenetetrazole; Picrotoxin; Receptors, GABA-A; Seizures; Time Factors

1986
The enhancement of diazepam and muscimol binding by pentobarbital and (+)-etomidate: size of the molecular arrangement estimated by electron irradiation inactivation of rat cortex.
    Neuroscience letters, 1986, Sep-25, Volume: 70, Issue:1

    Topics: Animals; Cerebral Cortex; Diazepam; Etomidate; gamma-Aminobutyric Acid; In Vitro Techniques; Molecular Weight; Muscimol; Pentobarbital; Rats; Receptors, GABA-A

1986
Comparison of anticonvulsant effect of pentobarbital and phenobarbital against seizures induced by maximal electroshock and picrotoxin in rats.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:5

    Topics: Amino Acids; Amino Acids, Neutral; Animals; Anticonvulsants; Bicuculline; Electroshock; Male; Muscimol; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1986
Adaptation of the GABAA-receptor complex in rat brain during chronic elevation of GABA by ethanolamine O-sulphate.
    British journal of pharmacology, 1987, Volume: 91, Issue:3

    Topics: 4-Aminobutyrate Transaminase; Animals; Brain Chemistry; Ethanolamines; Flurazepam; gamma-Aminobutyric Acid; Muscimol; Nipecotic Acids; Pentobarbital; Picrotoxin; Potassium; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
gamma-Aminobutyric acid receptor binding in fresh mouse brain membranes at 22 degrees C: ligand-induced changes in affinity.
    Molecular pharmacology, 1987, Volume: 32, Issue:1

    Topics: Allosteric Regulation; Animals; Brain; Cell Membrane; gamma-Aminobutyric Acid; Kinetics; Ligands; Mice; Microsomes; Mitochondria; Muscimol; Pentobarbital; Receptors, GABA-A; Temperature

1987
Comparison between pentobarbital- and muscimol-induced feeding in satiated sheep.
    Canadian journal of physiology and pharmacology, 1988, Volume: 66, Issue:6

    Topics: Aminocaproates; Animals; Calcium; Eating; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Pentobarbital; Picrotoxin; Sheep; Sodium; Vigabatrin

1988
Foot shock stress decreases chloride efflux from rat brain synaptoneurosomes.
    European journal of pharmacology, 1987, Mar-31, Volume: 135, Issue:3

    Topics: Animals; Brain; Chlorides; Electroshock; gamma-Aminobutyric Acid; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Stress, Psychological; Synaptosomes

1987
Gamma-aminobutyric acid and alcohol actions: neurochemical studies of long sleep and short sleep mice.
    Life sciences, 1986, Nov-24, Volume: 39, Issue:21

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebellum; Chlorides; Diencephalon; Drug Synergism; Ethanol; Female; gamma-Aminobutyric Acid; Hippocampus; Mice; Muscimol; Pentobarbital; Sleep; Telencephalon

1986
Studies of the role of gamma-aminobutyric acid in the hypothalamic control of feed intake in sheep.
    Canadian journal of physiology and pharmacology, 1985, Volume: 63, Issue:10

    Topics: Animals; Bicuculline; Brain; Eating; gamma-Aminobutyric Acid; Hypothalamus; Male; Muscimol; Pentobarbital; Picrotoxin; Sheep

1985
Chemically activated channels in muscle and spinal cord.
    Annals of neurology, 1984, Volume: 16 Suppl

    Topics: Acetylcholine; Animals; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Membrane Potentials; Muscimol; Neuromuscular Junction; Pentobarbital; Receptors, Cholinergic; Receptors, GABA-A; Spinal Cord; Stimulation, Chemical; Synaptic Transmission

1984
Modulation of the GABA receptor complex by a steroid anaesthetic.
    Brain research, 1984, Dec-10, Volume: 323, Issue:2

    Topics: Anesthetics; Animals; In Vitro Techniques; Male; Medulla Oblongata; Muscimol; Pentobarbital; Pregnanediones; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, GABA-A; Receptors, Muscarinic

1984
Some barbiturates enhance the effect of muscimol on dopamine turnover in the rat retina.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 213, Issue:2

    Topics: Animals; Barbital; Barbiturates; Convulsants; Dopamine; Drug Synergism; GABA Antagonists; gamma-Aminobutyric Acid; Light; Male; Methyltyrosines; Muscimol; Oxazoles; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Retina; Sesterterpenes

1980
Differential modulation of etazolate or pentobarbital enhanced [3H] muscimol binding by benzodiazepine agonists and inverse agonists.
    Brain research, 1983, Dec-05, Volume: 280, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Etazolate; Flumazenil; Flunitrazepam; Kinetics; Muscimol; Nicotinic Acids; Oxazoles; Pentobarbital; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
The effects of pentobarbital and related compounds on frog motoneurons.
    Brain research, 1980, Jun-02, Volume: 191, Issue:1

    Topics: Amino Acids; Animals; Anura; Bicuculline; Chloralose; Chlordiazepoxide; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Glutamates; Motor Neurons; Muscimol; Pentobarbital; Phenobarbital; Phenytoin; Picrotoxin; Spinal Cord; Strychnine; Synaptic Transmission

1980
Evidence that ethanol and pentobarbital enhance [3H]diazepam binding at the benzodiazepine-GABA receptor-ionophore complex indirectly.
    European journal of pharmacology, 1981, May-22, Volume: 71, Issue:4

    Topics: Animals; Diazepam; Ethanol; Muscimol; Pentobarbital; Picrotoxin; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium

1981
Histidine modification with diethyl pyrocarbonate shows heterogeneity of benzodiazepine receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1981, Volume: 78, Issue:6

    Topics: Animals; Benzodiazepines; Brain; Chemical Phenomena; Chemistry; Diazepam; Diethyl Pyrocarbonate; Formates; Histidine; Male; Muscimol; Pentobarbital; Rats; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter

1981
Acute and chronic effects of pentobarbital in relation to postsynaptic GABA receptors: a study with muscimol.
    Journal of neuroscience research, 1982, Volume: 7, Issue:1

    Topics: Animals; Brain; Drug Tolerance; gamma-Aminobutyric Acid; Humans; Male; Mice; Mice, Inbred ICR; Muscimol; Oxazoles; Pentobarbital; Receptors, Cell Surface; Receptors, GABA-A; Sleep; Substance Withdrawal Syndrome; Synaptic Membranes

1982
Single channel currents activated by gamma-aminobutyric acid, muscimol, and (-)-pentobarbital in cultured mouse spinal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1982, Volume: 2, Issue:7

    Topics: Animals; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Mice; Muscimol; Neurons; Oxazoles; Pentobarbital; Spinal Cord

1982
Solubilization by CHAPS detergent of barbiturate-enhanced benzodiazepine-GABA receptor complex.
    Journal of neurochemistry, 1982, Volume: 39, Issue:6

    Topics: Animals; Barbiturates; Cattle; Chlorides; Cholic Acids; Chromatography, Gel; Dose-Response Relationship, Drug; Muscimol; Pentobarbital; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Solubility; Time Factors

1982
Chloride-dependent enhancement by barbiturates of gamma-aminobutyric acid receptor binding.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1982, Volume: 2, Issue:12

    Topics: Animals; Barbiturates; Benzodiazepines; Brain; Cattle; Chlorides; Muscimol; Pentobarbital; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Membranes

1982
Morphological study of neurotransmitter receptors in the rat brain.
    Advances in biochemical psychopharmacology, 1983, Volume: 36

    Topics: Animals; Autoradiography; Brain; Cerebellum; Enkephalin, Methionine; In Vitro Techniques; Kinetics; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter

1983
Group-selective reagent modification of the benzodiazepine-gamma-aminobutyric acid receptor-ionophore complex reveals that low-affinity gamma-aminobutyric acid receptors stimulate benzodiazepine binding.
    Molecular pharmacology, 1983, Volume: 23, Issue:1

    Topics: Animals; Benzodiazepines; Cell Membrane; Cerebellum; Cerebral Cortex; Diazepam; Diazonium Compounds; Diethyl Pyrocarbonate; Flunitrazepam; Hippocampus; Male; Muscimol; Pentobarbital; Rats; Receptors, Cell Surface; Receptors, GABA-A; Sulfanilic Acids

1983
Modulation of [3H]muscimol binding in rat cerebellar and cerebral cortical membranes by picrotoxin, pentobarbitone, and etomidate.
    Journal of neurochemistry, 1983, Volume: 41, Issue:2

    Topics: Animals; Cell Membrane; Cerebellar Cortex; Cerebral Cortex; Etomidate; Imidazoles; Kinetics; Male; Muscimol; Organ Specificity; Oxazoles; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Barbiturate interactions with benzodiazepine-GABA receptor-ionophore complex.
    Advances in biochemical psychopharmacology, 1983, Volume: 37

    Topics: Animals; Barbiturates; Etomidate; In Vitro Techniques; Ionophores; Muscimol; Pentobarbital; Picrotoxin; Rats; Receptors, Cell Surface; Receptors, GABA-A; Sesterterpenes

1983
A gamma-aminobutyric acid/benzodiazepine receptor complex from bovine cerebral cortex. Improved purification with preservation of regulatory sites and their interactions.
    The Journal of biological chemistry, 1984, Jun-10, Volume: 259, Issue:11

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Cholic Acids; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Methods; Muscimol; Pentobarbital; Receptors, Cell Surface; Receptors, GABA-A; Solubility

1984
Visual evoked potentials in a rabbit model of hepatic encephalopathy. I. Sequential changes and comparisons with drug-induced comas.
    Gastroenterology, 1984, Volume: 86, Issue:3

    Topics: Animals; Diazepam; Disease Models, Animal; Electrodes; Electroencephalography; Evoked Potentials, Visual; Galactosamine; Hepatic Encephalopathy; Muscimol; Pentobarbital; Rabbits

1984
Discriminative stimulus effects of pentobarbital in pigeons.
    Psychopharmacology, 1980, Volume: 71, Issue:1

    Topics: Animals; Baclofen; Bemegride; Columbidae; Ethanol; gamma-Aminobutyric Acid; Muscimol; Pentobarbital; Prejudice

1980
Effects of barbiturates and ethanol on muscimol-induced release of [3H]-D-aspartate from rodent cerebellum.
    Neuropharmacology, 1983, Volume: 22, Issue:6

    Topics: Animals; Aspartic Acid; Cerebellum; Ethanol; gamma-Aminobutyric Acid; Kinetics; Male; Muscimol; Oxazoles; Pentobarbital; Potassium; Rats; Rats, Inbred Strains; Synaptosomes; Tritium

1983
Release of endogenous amino acid neurotransmitter candidates from rat olfactory cortex slices: possible regulatory mechanisms and the effects of pentobarbitone.
    Brain research, 1980, May-26, Volume: 190, Issue:2

    Topics: Animals; Aspartic Acid; Dose-Response Relationship, Drug; Electric Stimulation; gamma-Aminobutyric Acid; Male; Muscimol; Olfactory Bulb; Pentobarbital; Picrotoxin; Rats; Taurine

1980
GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital.
    Nature, 1993, Dec-09, Volume: 366, Issue:6455

    Topics: Amino Acid Sequence; Animals; Binding Sites; Cell Membrane; DNA Mutational Analysis; Female; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Macromolecular Substances; Molecular Sequence Data; Muscimol; Mutagenesis, Site-Directed; Oocytes; Pentobarbital; Point Mutation; Rats; Receptors, GABA-A; Xenopus laevis

1993
Counteraction of the rapid tolerance to 8-OH-DPAT-induced corticosterone secretion in rats by activation of the GABAA receptor-chloride channel complex.
    British journal of pharmacology, 1993, Volume: 109, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzodiazepines; Bicuculline; Chloride Channels; Chlormethiazole; Corticosterone; Drug Tolerance; Ion Channels; Male; Membrane Proteins; Muscimol; Pentobarbital; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1993
Kavapyrone enriched extract from Piper methysticum as modulator of the GABA binding site in different regions of rat brain.
    Psychopharmacology, 1994, Volume: 116, Issue:4

    Topics: Animals; Binding, Competitive; Brain Chemistry; Diazepam; Female; In Vitro Techniques; Muscimol; Ovariectomy; Pentobarbital; Plant Extracts; Plants, Medicinal; Pyrones; Rats; Rats, Sprague-Dawley; Receptors, GABA; Steroids

1994
Functional diversity of GABAA receptor ligand-gated chloride channels in rat synaptoneurosomes.
    Synapse (New York, N.Y.), 1995, Volume: 19, Issue:3

    Topics: Animals; Bicuculline; Brain; Chloride Channels; Chlorides; Desoxycorticosterone; Ion Channel Gating; Ligands; Male; Muscimol; Pentobarbital; Rats; Rats, Wistar; Receptors, GABA-A; Synaptosomes; Tissue Distribution

1995
Effect of pentobarbital on postischemic MK-801, muscimol, and naloxone bindings in the gerbil brain.
    Brain research, 1994, Sep-19, Volume: 657, Issue:1-2

    Topics: Animals; Brain; Dizocilpine Maleate; Gerbillinae; Ischemic Attack, Transient; Male; Muscimol; Naloxone; Pentobarbital; Radioligand Assay

1994
Trichloroethanol potentiation of gamma-aminobutyric acid-activated chloride current in mouse hippocampal neurones.
    British journal of pharmacology, 1994, Volume: 113, Issue:2

    Topics: Animals; Cells, Cultured; Chloride Channels; Drug Synergism; Ethanol; Ethylene Chlorohydrin; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Mice; Muscimol; Neurons; Patch-Clamp Techniques; Pentobarbital; Receptors, GABA-A; Up-Regulation

1994
Anesthetics block morphine-induced increases in serotonin release in rat CNS.
    Synapse (New York, N.Y.), 1994, Volume: 18, Issue:4

    Topics: Anesthetics; Animals; Betaine; Brain Chemistry; Chloral Hydrate; Extracellular Space; Hippocampus; Injections; Male; Microdialysis; Morphine; Muscimol; Neurons; Nucleus Accumbens; Pentobarbital; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin

1994
Negative regulation of proopiomelanocortin gene expression by GABAA receptor activation in the rat arcuate nucleus.
    Peptides, 1994, Volume: 15, Issue:4

    Topics: Animals; Arcuate Nucleus of Hypothalamus; GABA-A Receptor Agonists; Gene Expression Regulation; In Situ Hybridization; Male; Muscimol; Pentobarbital; Pro-Opiomelanocortin; Rats; Rats, Sprague-Dawley

1994
Cloning and functional expression of a Drosophila gamma-aminobutyric acid receptor.
    Proceedings of the National Academy of Sciences of the United States of America, 1994, Jun-21, Volume: 91, Issue:13

    Topics: Amino Acid Sequence; Animals; Base Sequence; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cloning, Molecular; Convulsants; DNA Primers; DNA, Complementary; Drosophila melanogaster; Female; Flunitrazepam; gamma-Aminobutyric Acid; Gene Expression; Macromolecular Substances; Molecular Sequence Data; Muscimol; Oocytes; Pentobarbital; Picrotoxin; Polymerase Chain Reaction; Receptors, GABA; Receptors, GABA-A; Transcription, Genetic; Xenopus laevis

1994
A novel GABA receptor on bipolar cell terminals in the tiger salamander retina.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:3 Pt 1

    Topics: Animals; Bicuculline; Chlorides; Crotonates; Electrophysiology; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Muscimol; Pentobarbital; Picrotoxin; Pyridazines; Receptors, GABA; Receptors, GABA-A; Retina; Retinal Ganglion Cells; Urodela

1994
Studies on picrotoxin binding sites of GABAA receptors in rat cortical synaptoneurosomes.
    Brain research bulletin, 1994, Volume: 33, Issue:4

    Topics: Animals; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorine; Desoxycorticosterone; Diazepam; In Vitro Techniques; Male; Membranes; Muscimol; Pentobarbital; Picrotoxin; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Steroids; Synaptosomes

1994
Chronic administration of muscimol and pentobarbital decreases gonadotropin-releasing hormone mRNA levels in the male rat hypothalamus determined by quantitative in situ hybridization.
    Neuroendocrinology, 1993, Volume: 58, Issue:1

    Topics: Animals; Gonadotropin-Releasing Hormone; Hypothalamus; In Situ Hybridization; Male; Muscimol; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Time Factors

1993
A new highly sensitive procedure--a prerequisite to evaluate the density of GABAA receptors and to study their allosteric properties in distinct areas of rat brain.
    Biological chemistry Hoppe-Seyler, 1993, Volume: 374, Issue:1

    Topics: Allosteric Regulation; Animals; Binding Sites; Brain; Cerebellum; Desoxycorticosterone; Female; Frontal Lobe; Humans; Hydrogen-Ion Concentration; Muscimol; Pentobarbital; Pregnanediones; Pregnanolone; Progesterone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1993
Region-specific changes of GABAA receptors by tolerance to and dependence upon pentobarbital.
    European journal of pharmacology, 1993, May-12, Volume: 236, Issue:1

    Topics: Animals; Body Temperature; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Corpus Striatum; Drug Tolerance; Flunitrazepam; Frontal Lobe; In Vitro Techniques; Injections, Intraventricular; Male; Muscimol; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Substance-Related Disorders; Sulfur Radioisotopes; Synaptic Membranes

1993
Microdialysis study of the effects of sedative drugs on extracellular histamine in the striatum of freely moving rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: Animals; Corpus Striatum; Dialysis; Diazepam; Dronabinol; Extracellular Space; Histamine; Hypnotics and Sedatives; Male; Muscimol; Pentobarbital; Rats; Rats, Wistar; Reserpine

1993
Attenuation of anticonvulsant effects of diazepam after chronic treatment with bicuculline.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:4

    Topics: Animals; Anticonvulsants; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred F344; Rats, Inbred Lew; Receptors, GABA; Sleep

1993
Novel GABA responses from rod-driven retinal horizontal cells.
    Nature, 1993, Jan-14, Volume: 361, Issue:6408

    Topics: Animals; Bicuculline; Chlorides; Crotonates; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Muscimol; Pentobarbital; Perches; Photoreceptor Cells; Receptors, GABA; Retina

1993
Biochemical evaluations of the effects of loreclezole and propofol on the GABAA receptor in rat brain.
    Biochemical pharmacology, 1996, Jun-14, Volume: 51, Issue:11

    Topics: Anesthetics; Animals; Anticonvulsants; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Triazoles; Tritium

1996
Microtubule depolymerization inhibits ethanol-induced enhancement of GABAA responses in stably transfected cells.
    Journal of neurochemistry, 1996, Volume: 66, Issue:3

    Topics: Animals; Cattle; Cell Line; Chlorides; Colchicine; Ethanol; Flunitrazepam; Humans; Mice; Microtubules; Muscimol; Pentobarbital; Polymers; Receptor Aggregation; Receptors, GABA-A; Transfection

1996
Medullary vasomotor activity and hypoxic sympathoexcitation in pentobarbital-anesthetized rats.
    The American journal of physiology, 1996, Volume: 270, Issue:2 Pt 2

    Topics: Anesthesia; Animals; Blood Pressure; Hypoxia; Male; Medulla Oblongata; Microinjections; Muscimol; Neural Inhibition; Neurons; Pentobarbital; Rats; Rats, Sprague-Dawley; Spinal Cord; Sympathetic Nervous System; Vasomotor System

1996
Insensitivity to anaesthetic agents conferred by a class of GABA(A) receptor subunit.
    Nature, 1997, Feb-27, Volume: 385, Issue:6619

    Topics: Amino Acid Sequence; Anesthetics, Intravenous; Animals; Bicuculline; Brain; Cell Line; Consensus Sequence; DNA, Complementary; Flumazenil; Flunitrazepam; GABA Agents; gamma-Aminobutyric Acid; Humans; Molecular Sequence Data; Muscimol; Pentobarbital; Picrotoxin; Pregnanolone; Propofol; Rats; Receptors, GABA-A; Recombinant Proteins; RNA, Messenger; Transfection

1997
Ethanol, flunitrazepam, and pentobarbital modulation of GABAA receptors expressed in mammalian cells and Xenopus oocytes.
    Alcoholism, clinical and experimental research, 1997, Volume: 21, Issue:3

    Topics: Animals; Cattle; Cell Line, Transformed; Chloride Channels; Dose-Response Relationship, Drug; Ethanol; Flunitrazepam; Gene Expression; Humans; Mice; Muscimol; Oocytes; Pentobarbital; Protein Processing, Post-Translational; Receptors, GABA-A; Xenopus

1997
Ultrasonic vocalizations in rat pups: modulation at the gamma-aminobutyric acidA receptor complex and the neurosteroid recognition site.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:1

    Topics: Alprazolam; Animals; Diazepam; Female; Male; Muscimol; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Vocalization, Animal

1997
Adaptation of gamma-aminobutyric acid type A receptors to alcohol exposure: studies with stably transfected cells.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:1

    Topics: Animals; Cells, Cultured; Drug Tolerance; Ethanol; Flunitrazepam; Humans; Mice; Muscimol; Pentobarbital; Pregnanolone; Protein Kinase C; Receptors, GABA-A; Transfection; Zinc

1998
Nitrous oxide-induced enhancement of gamma-aminobutyric acidA-mediated chloride currents in acutely dissociated hippocampal neurons.
    Anesthesiology, 1998, Volume: 88, Issue:2

    Topics: Anesthetics, Inhalation; Animals; Chloride Channels; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; GABA Agonists; Hippocampus; Male; Muscimol; Nitrous Oxide; Patch-Clamp Techniques; Pentobarbital; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA

1998
Characterization of chloride efflux from GT1-7 neurons: lack of effect of ethanol on GABAA response.
    Brain research, 1998, Jan-12, Volume: 780, Issue:2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Bicuculline; Bumetanide; Cells, Cultured; Central Nervous System Stimulants; Chlorides; Diuretics; Ethanol; GABA Agonists; GABA Antagonists; GABA Modulators; Mice; Muscimol; Neurons; Pentobarbital; Receptors, GABA-A; Temperature

1998
Effects of propofol and pentobarbital on ligand binding to GABAA receptors suggest a similar mechanism of action.
    Canadian journal of physiology and pharmacology, 1998, Volume: 76, Issue:1

    Topics: Allosteric Site; Anesthetics, Intravenous; Animals; Azides; Benzodiazepines; Brain; Cattle; Flunitrazepam; GABA Agonists; In Vitro Techniques; Ligands; Membranes; Muscimol; Pentobarbital; Propofol; Receptors, GABA-A

1998
Effects of pentobarbital on the expression of GABAA receptor beta 1 mRNA in the hippocampus: differential responses of CA1 and CA3.
    Synapse (New York, N.Y.), 1998, Volume: 29, Issue:4

    Topics: Animals; Behavior, Animal; Hippocampus; In Situ Hybridization; Male; Muscimol; Pentobarbital; Rats; Rats, Wistar; Receptors, GABA-A; RNA, Messenger; Tissue Distribution

1998
Potentiation of muscimol-induced long-term depression by benzodiazepines and prevention or reversal by pregnenolone sulfate.
    Pharmacological research, 1998, Volume: 38, Issue:6

    Topics: Amnesia; Animals; Barbiturates; Benzodiazepines; Cognition Disorders; Depression; Diazepam; Drug Synergism; Hippocampus; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanolone; Pregnenolone; Rats; Rats, Wistar; Time Factors

1998
Neuroprotective properties of propofol and midazolam, but not pentobarbital, on neuronal damage induced by forebrain ischemia, based on the GABAA receptors.
    Acta anaesthesiologica Scandinavica, 1999, Volume: 43, Issue:2

    Topics: Anesthetics, Intravenous; Animals; Baclofen; Brain Ischemia; Dose-Response Relationship, Drug; GABA Agonists; GABA Modulators; Gerbillinae; Histocytochemistry; Male; Midazolam; Muscimol; Neurons; Neuroprotective Agents; Pentobarbital; Propofol; Prosencephalon; Receptors, GABA-A; Reperfusion Injury

1999
GABA(A) receptors mediate inhibition of T cell responses.
    Journal of neuroimmunology, 1999, Apr-01, Volume: 96, Issue:1

    Topics: Amidines; Animals; Autocrine Communication; Bicuculline; CD3 Complex; Cell Division; Enzyme Inhibitors; Female; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hypersensitivity, Delayed; Immunosuppression Therapy; Interleukin-2; Lymphocyte Activation; Male; Mice; Mice, Inbred NOD; Muscimol; Pentobarbital; Picrotoxin; Receptors, GABA-A; Receptors, GABA-B; Signal Transduction; T-Lymphocytes; Vigabatrin

1999
Fluorescence imaging of GABAA receptor-mediated intracellular [Cl-] in P19-N cells reveals unique pharmacological properties.
    Brain research, 1999, May-08, Volume: 827, Issue:1-2

    Topics: Animals; Central Nervous System Depressants; Chlorides; Diazepam; DNA Primers; Ethanol; Flunitrazepam; Fluorescent Dyes; GABA Agonists; GABA Modulators; Gene Expression; Mice; Muscimol; Neoplastic Stem Cells; Neuroglia; Pentobarbital; Pregnanolone; Quinolinium Compounds; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tritium

1999
Changes of [3H]muscimol binding and GABA(A) receptor beta2-subunit mRNA level by tolerance to and withdrawal from pentobarbital in rats.
    Neurochemical research, 1999, Volume: 24, Issue:12

    Topics: Animals; Autoradiography; Brain; Cerebellum; Drug Tolerance; Frontal Lobe; Gene Expression Regulation; Hippocampus; Inferior Colliculi; Male; Muscimol; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Substance Withdrawal Syndrome; Tritium

1999
GABA(A) receptors on calbindin-immunoreactive myenteric neurons of guinea pig intestine.
    Journal of the autonomic nervous system, 2000, Jan-14, Volume: 78, Issue:2-3

    Topics: Animals; Calbindins; Cells, Cultured; Diazepam; Dose-Response Relationship, Drug; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Guinea Pigs; Immunohistochemistry; Intestine, Small; Membrane Potentials; Muscimol; Myenteric Plexus; Neurons; Pentobarbital; Receptors, GABA-A; S100 Calcium Binding Protein G

2000
Characterization of the discriminative stimulus effects of GABA(A) receptor ligands in Macaca fascicularis monkeys under different ethanol training conditions.
    Psychopharmacology, 2000, Volume: 152, Issue:2

    Topics: Animals; Discrimination Learning; Ethanol; Female; Macaca fascicularis; Male; Midazolam; Muscimol; Pentobarbital; Receptors, GABA-A; Sex Factors

2000
Activation of GABA(A) receptors in subthalamic neurons in vitro: properties of native receptors and inhibition mechanisms.
    Journal of neurophysiology, 2001, Volume: 86, Issue:1

    Topics: Animals; Bicarbonates; Bicuculline; Chlorides; Diazepam; Electrophysiology; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA Modulators; Membrane Potentials; Muscimol; Neural Inhibition; Neurons; Organ Culture Techniques; Pentobarbital; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Sesterterpenes; Subthalamic Nucleus

2001
alpha4beta3delta GABA(A) receptors characterized by fluorescence resonance energy transfer-derived measurements of membrane potential.
    The Journal of biological chemistry, 2001, Oct-19, Volume: 276, Issue:42

    Topics: Animals; Benzodiazepines; Cell Line; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Mice; Models, Biological; Muscimol; Pentobarbital; Pregnanediones; Pregnanolone; Protein Binding; Protein Conformation; Receptors, GABA-A; Spectrometry, Fluorescence; Time Factors; Transfection

2001
GABAA receptors mediate postnatal depression of respiratory frequency by barbiturates.
    Respiratory physiology & neurobiology, 2004, Jun-25, Volume: 140, Issue:3

    Topics: Animals; Animals, Newborn; Bicuculline; Drug Interactions; Female; GABA Agents; Hypnotics and Sedatives; In Vitro Techniques; Muscimol; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Respiratory Center; Respiratory Insufficiency; Respiratory Mechanics; Spinal Cord; Spinal Nerve Roots

2004
Sanjoinine A isolated from Zizyphi Spinosi Semen augments pentobarbital-induced sleeping behaviors through the modification of GABA-ergic systems.
    Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:9

    Topics: Animals; Cerebellum; Chlorides; Drug Interactions; GABA Agonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hypnotics and Sedatives; Isoenzymes; Male; Mice; Mice, Inbred ICR; Muscimol; Pentobarbital; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sleep; Ziziphus

2007
Cyclopeptide alkaloid fraction from Zizyphi Spinosi Semen enhances pentobarbital-induced sleeping behaviors.
    Journal of ethnopharmacology, 2008, May-08, Volume: 117, Issue:2

    Topics: Alkaloids; Animals; Cells, Cultured; Cerebellum; Chlorides; Drug Synergism; GABA Agonists; gamma-Aminobutyric Acid; Glyceraldehyde-3-Phosphate Dehydrogenases; Hypnotics and Sedatives; Male; Mice; Mice, Inbred ICR; Muscimol; Neurons; Pentobarbital; Plant Extracts; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sleep; Synaptic Transmission; Ziziphus

2008
Individually monitoring ligand-induced changes in the structure of the GABAA receptor at benzodiazepine binding site and non-binding-site interfaces.
    Molecular pharmacology, 2008, Volume: 74, Issue:1

    Topics: Animals; Benzodiazepines; Binding Sites; Cysteine; Dose-Response Relationship, Drug; Electrophysiology; Female; Flumazenil; Flurazepam; GABA Agonists; GABA Antagonists; GABA Modulators; Inhibitory Concentration 50; Ligands; Microinjections; Muscimol; Mutagenesis, Site-Directed; Oocytes; Patch-Clamp Techniques; Pentobarbital; Pyridazines; Rats; Receptors, GABA-A; Xenopus

2008
Methanol extract of Longanae Arillus augments pentobarbital-induced sleep behaviors through the modification of GABAergic systems.
    Journal of ethnopharmacology, 2009, Mar-18, Volume: 122, Issue:2

    Topics: Animals; Chlorine; Drug Synergism; GABA Modulators; Glutamate Decarboxylase; Hypnotics and Sedatives; Male; Mice; Mice, Inbred ICR; Muscimol; Pentobarbital; Plant Extracts; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sapindaceae; Sleep

2009
Pilocarpine model of temporal lobe epilepsy shows enhanced response to general anesthetics.
    Experimental neurology, 2009, Volume: 219, Issue:1

    Topics: Anesthetics, General; Animals; Brain; Consciousness Disorders; Convulsants; Disease Models, Animal; Electroencephalography; Entorhinal Cortex; Epilepsy, Temporal Lobe; GABA Agonists; Halothane; Kindling, Neurologic; Male; Muscimol; Nerve Degeneration; Olfactory Pathways; Pentobarbital; Pilocarpine; Propofol; Rats; Rats, Sprague-Dawley; Status Epilepticus

2009
Hibernation induces pentobarbital insensitivity in medulla but not cortex.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2009, Volume: 297, Issue:4

    Topics: Action Potentials; Allosteric Regulation; Animals; Bicuculline; Body Temperature; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA Modulators; Hibernation; In Vitro Techniques; Ligands; Medulla Oblongata; Muscimol; Pentobarbital; Protein Conformation; Protein Subunits; Receptors, GABA-A; Respiratory Center; Sciuridae; Seasons; Solitary Nucleus; Time Factors

2009
Comparison of the antiepileptic properties of transmeningeally delivered muscimol, lidocaine, midazolam, pentobarbital and GABA, in rats.
    Neuroscience letters, 2010, Jan-29, Volume: 469, Issue:3

    Topics: Acetylcholine; Animals; Anticonvulsants; Electrodes, Implanted; Electroencephalography; gamma-Aminobutyric Acid; Lidocaine; Midazolam; Muscimol; Pentobarbital; Rats; Seizures; Somatosensory Cortex; Time Factors

2010
(-)-epigallocatechin-3-O-gallate augments pentobarbital-induced sleeping behaviors through Cl- channel activation.
    Journal of medicinal food, 2011, Volume: 14, Issue:11

    Topics: Animals; Catechin; Cells, Cultured; Cerebellum; Chloride Channels; Chlorides; Glutamate Decarboxylase; Hippocampus; Male; Mice; Mice, Inbred ICR; Muscimol; Neuroprotective Agents; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA; Sleep

2011
Enhancement of pentobarbital-induced sleep by apigenin through chloride ion channel activation.
    Archives of pharmacal research, 2012, Volume: 35, Issue:2

    Topics: Animals; Apigenin; Cerebellum; Chloride Channel Agonists; Dose-Response Relationship, Drug; Drug Synergism; Glutamate Decarboxylase; Hippocampus; Hypnotics and Sedatives; Male; Mice; Mice, Inbred ICR; Muscimol; Pentobarbital; Primary Cell Culture; Rats; Receptors, GABA-A; Sleep

2012
NKCC1 knockdown decreases neuron production through GABA(A)-regulated neural progenitor proliferation and delays dendrite development.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Sep-26, Volume: 32, Issue:39

    Topics: Age Factors; Analysis of Variance; Animals; Animals, Newborn; Calcium; Cell Count; Cell Differentiation; Cell Proliferation; Cells, Cultured; Cerebral Ventricles; Dendrites; Egtazic Acid; Electroporation; Female; GABA Modulators; GABA-A Receptor Agonists; Green Fluorescent Proteins; In Vitro Techniques; Ki-67 Antigen; Luminescent Proteins; Male; Mice; Muscimol; Neural Stem Cells; Neurons; Olfactory Bulb; Patch-Clamp Techniques; Pentobarbital; Receptors, GABA-A; Red Fluorescent Protein; RNA, Small Interfering; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2; SOXB1 Transcription Factors; Transfection

2012
In vivo recordings of GnRH neuron firing reveal heterogeneity and dependence upon GABAA receptor signaling.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, May-29, Volume: 33, Issue:22

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Electrodes, Implanted; Electrophysiological Phenomena; Excitatory Amino Acid Agonists; Female; GABA Agonists; GABA Antagonists; Gonadotropin-Releasing Hormone; Kisspeptins; Male; Mice; Muscimol; Neurons; Patch-Clamp Techniques; Pentobarbital; Pharynx; Picrotoxin; Receptors, GABA-A; Signal Transduction; Tetrodotoxin

2013
3,4,5-Trimethoxycinnamic acid (TMCA), one of the constituents of Polygalae Radix enhances pentobarbital-induced sleeping behaviors via GABAAergic systems in mice.
    Archives of pharmacal research, 2013, Volume: 36, Issue:10

    Topics: Animals; Cerebellum; Chlorides; Cinnamates; Drug Synergism; GABA Agonists; GABAergic Neurons; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hypnotics and Sedatives; Male; Mice; Motor Activity; Muscimol; Neurons; Pentobarbital; Polygala; Primary Cell Culture; Receptors, GABA-A; Sleep; Sleep Stages

2013
Expression of the γ2-subunit distinguishes synaptic and extrasynaptic GABA(A) receptors in NG2 cells of the hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Jul-17, Volume: 33, Issue:29

    Topics: Animals; Benzodiazepines; Bicuculline; Diazepam; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Muscimol; Neuroglia; Neurons; Patch-Clamp Techniques; Pentobarbital; Protein Subunits; Receptors, GABA-A; Synapses

2013
Taurine potentiates the anticonvulsive effect of the GABA
    Epilepsia, 2019, Volume: 60, Issue:3

    Topics: Animals; Animals, Newborn; Anticonvulsants; Drug Synergism; GABA-A Receptor Agonists; Hippocampus; Mice; Mice, Inbred C57BL; Muscimol; Pentobarbital; Seizures; Taurine

2019