muscimol and oxazoles

muscimol has been researched along with oxazoles in 237 studies

Research

Studies (237)

TimeframeStudies, this research(%)All Research%
pre-1990235 (99.16)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (0.84)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kamioka, T; Matsui, Y3
Chase, TN; Crayton, JW; Tamminga, CA1
Arnt, J; Krogsgaard-Larsen, P; Magelund, G; Scheel-Krüger, J1
Kuhar, MJ; Niehoff, DL; Palacios, JM1
Crossman, AR; Lee, LA; Longman, DA; Slater, P1
Jobert, A; Soubrié, P; Thiébot, MH2
Horton, RW; Meldrum, BS; Pedley, TA1
Baker, HF; Ridley, RM; Scraggs, PR1
Charlton, M; Goldblatt, D; Joynt, RJ; Shoulson, I1
Bloch, R; Bousquet, P; Feldman, J; Schwartz, J3
Chase, TN; Frohman, LA; Neophytides, A; Tamminga, CA1
Fang, VS; Meltzer, HY; Simonovic, M1
Arnt, J; Krogsgaard-Larsen, P2
Longman, DA; Slater, P1
DeFeudis, FV; Mandel, P; Ossola, L; Schmitt, G2
Matthews, WD; McCafferty, GP1
Baraldi, M; Grandison, L; Guidotti, A1
Mantegazza, P; Restelli, A; Vicentini, L; Zambotti, F; Zonta, N1
Risley, EA; Williams, M2
Andén, NE; Grabowska-Andén, M; Wachtel, H1
Roberts, E; Salvaterra, P; Wang, YJ1
Curtis, DR; Hjeds, H; Johnston, GA; Krogsgaard-Larsen, P; Lodge, D1
Enna, SJ; Maggi, A1
Baldessarini, RJ; Herschel, M1
Maurer, R2
Jenner, P; Leigh, N; Marsden, CD; Reavill, C1
Betti, R; Cocchi, D; Frigerio, C; Krogsgaard-Larsen, P; Locatelli, V; Müller, EE; Racagni, G1
Bartholini, G; Scatton, B1
Cross, AJ; Waddington, JL1
McDonald, A1
Gross, DM; Sweet, CS; Wenger, HC1
Mantegazza, P; Tammiso, R; Vicentini, L; Zambotti, F; Zonta, N1
Karobath, M; Lippitsch, M1
Defrance, J; Enna, SJ; Marchand, J; Stanley, J1
DeFeudis, FV; Mandel, P; Ossola, L3
Andrews, PR; Johnston, GA1
Grossman, SP; Kelly, J; Rothstein, J1
Johnston, GA; Kennedy, SM; Lodge, D1
Curtis, DR; Johnston, GA; Lodge, D1
Chan-Palay, V1
Bacino, CB; Martin, GE; Papp, NL1
Haubrich, DR; Martin, GE1
Delini-Stula, A; Vassout, A1
Depoortere, H; Lloyd, KG; Worms, P1
Arnt, J; Scheel-Krüger, J1
Gower, M; MacNeil, D; Szymanska, I1
Carlà, V; Giotti, A; Magnani, M; Sgaragli, GP1
Antonaccio, MJ; Kerwin, L; Taylor, DG1
Cavalla, D; Neff, NH1
Chuang, DM; Majewska, MD1
Hansen, SH; Krogsgaard-Larsen, P; Nielsen, EO; Schousboe, A1
Hikosaka, O; Wurtz, RH2
Gähwiler, BH; Graff, P; Maurer, R; Nordmann, R1
Botez, MI; Lalonde, R1
Apud, JA; Masotto, C; Racagni, G1
Borsini, F; Evangelista, S; Meli, A1
Arbit, E; Fogel, R; Kaplan, RB1
Hikosaka, O; Iwamura, Y; Sakamoto, M; Tanaka, M1
Klockgether, T; Schwarz, M; Sontag, KH; Turski, L; Wolfarth, S1
Cynader, M; Needler, MC; Shaw, C2
Gale, K; Garant, DS; Lim, CR1
Belonogoff, OB; Lideman, RR1
Coloma, FM; Niles, LP1
Kamp, CW; Morgan, WW1
Hösli, E; Hösli, L; Möhler, H; Richards, JG1
Brecha, N; Yazulla, S2
Chweh, A; Ebadi, M1
Elde, RP; Grouse, LH; Robbins, MS; Sorenson, RL1
Atterwill, CK; Batts, C; Bloomfield, MR1
Ishida, M; Shinozaki, H1
Menon, MK; Vivonia, CA2
Collins, JF; Karobath, M; Mannonen, A; Supavilai, P1
Forchetti, MC; Guidotti, A; Krogsgaard-Larsen, P; Moroni, F1
Saano, V1
Borea, PA; Karobath, M; Supavilai, P1
Chweh, AY; Lin, YB; Swinyard, EA1
Ostrovskaia, RU1
Placheta, P; Singer, E1
Romandini, S; Samanin, R1
Chase, TN; Denaro, A; Durso, R; Ruggeri, S; Tamminga, CA1
Degener, P; Krause, DN; Roberts, E; Wong, E1
Edvinsson, L; Larsson, B; Skärby, T1
Hösli, E; Hösli, L1
Kuriyama, K; Yoneda, Y2
DeFeudis, FV2
Cananzi, AR; Costa, E; Guidotti, A1
DeFeudis, FV; Devilliers, G; Mandel, P; Sarliéve, LL; Varga, V1
Ito, Y; Kurihara, E; Kuriyama, K; Yoneda, Y1
Kilpatrick, IC; Starr, MS2
DeFeudis, FV; Mandel, P; Ossola, L; Sarliève, LL; Varga, V1
Besser, GM; Delitala, G; Grossman, A; Yeo, T1
Kelly, PA; McCulloch, J4
Gardell, MA; Neale, JH; Shibla, DB1
Barker, JL; Mathers, DA1
Yazulla, S1
DeFeudis, FV; Geffard, M; Mandel, P; Ossola, L; Varga, V2
Kolasiewicz, W; Sontag, KH; Wolfarth, S1
Mitchell, CK; Redburn, DA1
Dauth, GW; Frey, KA; Pan, HS; Penney, JB; Young, AB1
Grace, M; Kneip, J; Levine, AS; Morley, JE; Silvis, SE1
Brehm, L; Krogsgaard-Larsen, P; Schaumburg, K1
Goetz, IE; Hamel, E; Roberts, E1
Crawley, JN; Marangos, PJ1
Ho, IK; Nabeshima, T; Sivam, SP1
Fukuda, H; Matsumoto, K2
Jordan, CC; Matus, AI; Piotrowski, W; Wilkinson, D1
Barker, JL; Jackson, MB; Lecar, H; Mathers, DA1
Linnoila, M; Marangos, PJ; Stowell, L; Thurman, RG1
Agardh, E; Ehinger, B1
Curtis, DR; Hjeds, H; Krogsgaard-Larsen, P; Leah, JD; Peet, MJ1
Cagan, RH; Quinn, MR1
Armstrong, DR; Breckenridge, RJ; Suckling, CJ1
Engel, J; Liljequist, S1
Lorens, SA; Sainati, SM1
Patel, SC; Peck, EJ1
Frey, KA; Pan, HS; Penney, JB; Young, AB1
Rägo, LK; Zarkovsky, AM1
Canonico, PL; Di Chiara, G; Imperato, A; Nicoletti, F; Piacente, B; Raffaele, R; Scapagnini, U1
Brenner, O; Quast, U1
Lucacchini, A; Martini, C; Rigacci, T1
Johnston, GA; Skerritt, JH1
Quinn, MR; Somerville, RA1
Breese, GR; Frye, GD; McCown, TJ1
Becker, H; Dietz, R; Ganten, D; Lang, RE; Rettig, R; Schömig, A; Schwab, NA; Unger, T1
Dewhurst, IC; Ekuwem, CE; Griffiths, R; O'Neill, C; Sinclair, CD; Williams, DC1
Gonzalez, LP; Hettinger, MK1
Besson, MJ; Gauchy, C; Glowinski, J; Kemel, ML1
Fukuda, H; Goto, M; Hasebe, Y; Kaneko, T; Kato, K1
Beani, L; Bianchi, C; Tanganelli, S1
Simmonds, MA1
Apud, J; Cagiano, R; Cuomo, V; Masotto, C; Racagni, G1
Bereksi, B; Boggio, V; Guilland, JC; Klepping, J; Mack, G; Noirot, P1
Goebel, DJ; McReynolds, JS; Pourch, RG1
Hanada, S; Hosomi, T; Isoda, K; Kasai, T; Kuno, T; Kuyama, T; Mita, T; Nakai, H; Nishino, N; Uchida, S1
Sarhan, S; Seiler, N1
Dean, P; Redgrave, P; Taha, EB2
Allen, CN; Crawford, IL1
Brennan, TJ; Haywood, JR; Morris, M1
Gillis, RA; Quest, JA; Souza, JD1
Mitchell, R; Wilson, L1
Drower, EJ; Hammond, DL1
Essatara, MB; Levine, AS; McClain, CJ; Morley, JE1
Besson, MJ; Gauchy, C; Glowinski, J; Kemel, ML; Romo, R1
Goebel, DJ; Pourcho, RG1
Di Scala, G; Karli, P; Schmitt, P1
De Caro, G; Iovino, M; Massi, M; Poenaru, S; Steardo, L1
Fowler, LJ; John, RA; Lovell, DH1
Besson, MJ; Chéramy, A; Gauchy, C; Glowinski, J; Kemel, ML; Romo, R1
Bendotti, C; Borsini, F; Przewlocka, B; Samanin, R1
Gluckman, PD; Johnston, BM1
Chen, SQ; Geng, RL; Wang, SC1
Childs, JA; Gale, K1
Glusman, M; Potegal, M; Yoburn, B1
Chmielewska, B; Czuczwar, SJ; Kleinrok, Z; Turski, WA1
Albala, BJ; Moshé, SL1
Helén, P; London, ED1
Kaakkola, S; Kääriäinen, I1
Gent, JP; Phillips, NI1
Mandel, P; Puglisi-Allegra, S1
Moises, HC; Waterhouse, BD; Woodward, DJ; Yeh, HH1
Beart, PM; Gundlach, AL2
Amladi, SR; Kelkar, MR; Naik, SR; Sheth, UK1
Haddox, VG; Menon, MK; Vivonia, CA1
Claperon, N; Durussel, JJ; Rossignol, P1
Scholfield, CN2
Aloisi, F; Gallo, V; Levi, G1
Blaker, WD; Cheney, DL; Costa, E; Gandolfi, O1
Harris, RA; Rohde, BH1
Ho, IK; Sivam, SP1
Fung, YK; Kuruvilla, A; Uretsky, NJ1
Curtis, DR; Hansen, JJ; Honoré, T; Krogsgaard-Larsen, P; Lodge, D1
Cappelletti, G; Cavagnini, F; Dubini, A; Invitti, C; Pinto, M; Polli, EE1
Conci, F; Mantegazza, P; Parenti, M; Tommasi, R; Vicentini, L; Zambotti, F; Zonta, N1
Back, KC; George, ME; Pinkerton, MK1
Kuhar, MJ; London, ED; Palacios, JM; Rapoport, SI2
Blanks, JC; Roffler-Tarlov, S1
File, SE1
Bosh, TK; Fung, YK; Grassman, DR; Novin-Baheran, A1
Collins, RC1
Kozlowski, MR; Marshall, JF1
Cortese, I; Cuomo, V; Siro-Brigiani, G1
Dean, P; Eastwood, L; Redgrave, P1
Buescher, HH; Hill, RC; Maurer, R; Roemer, D1
Intoccia, AP; Matthews, WD; McCafferty, GP; Osborne, VL1
Huston, JP; Welzl, H1
DeFeudis, FV; Mandel, P; Ossola, L; Rebel, G; Sarliève, LL; Schmitt, G; Varga, V1
Pourcho, RG1
Setler, PE; Zarevics, P1
Constanti, A; Nistri, A1
Pizzi, WJ; Unnerstall, JR1
Kneip, J; Levine, AS; Morley, JE1
Menon, MK1
Javid, MJ; Stone, WE1
Bergstrom, DA; Walters, JR; Waszczak, BL1
Fukuda, H; Kaneko, T; Ono, H1
Liebman, JM; Pastor, G1
Eng, N; Walters, JR; Waszczak, BL1
Chieli, T; Cocchi, D; Fregnan, GB; Müller, EE1
DeFeudis, FV; Mandel, P; Ossola, L; Sarliève, LL1
Korf, J; van der Heyden, JA; Venema, K1
Hruska, RE; Walters, JR; Waszczak, BL1
Cooper, BR; Howard, JL; Ingold, K; Maxwell, RA; Soroko, F; White, HL1
DeFeudis, FV; Geffard, M; Mandel, P; Varga, V1
Schaeffer, JM1
Persson, B1
DeFeudis, FV; Mandel, P; Ossola, L; Schmitt, G; Wolff, P1
Osborne, NN1
Baraczka, K; Sperk, G1
Furuta, K; Liu, G; Ozoe, F; Ozoe, Y1
Antoni, FA; Barkóczy, J; Belelli, D; Brown, AR; Etherington, LA; Gacsályi, I; Gunn, BG; Kertész, S; Lambert, JJ; Ling, I; Livesey, MR; Mihalik, B; Monteiro, O; Pallagi, K; Pálvölgyi, A; Spedding, M; Varga, P1

Reviews

5 review(s) available for muscimol and oxazoles

ArticleYear
GABA receptor agonists: relationship between structure and biological activity in vivo and in vitro.
    Advances in experimental medicine and biology, 1979, Volume: 123

    Topics: Animals; gamma-Aminobutyric Acid; Kinetics; Muscimol; Oxazoles; Receptors, Drug; Structure-Activity Relationship; Substantia Nigra

1979
Binsing studies with muscimol; relation ty synaptic gamma-aminobutyrate receptors.
    Neuroscience, 1980, Volume: 5, Issue:4

    Topics: Animals; Astacoidea; Autoradiography; Blood Vessels; Brain; Cattle; Cerebellum; Culture Techniques; Freezing; gamma-Aminobutyric Acid; Kinetics; Muscimol; Muscles; Oxazoles; Pia Mater; Polyethylene Glycols; Rats; Receptors, Neurotransmitter; Sodium; Subcellular Fractions; Substrate Specificity

1980
Physiological and behavioral studies with muscimol.
    Neurochemical research, 1980, Volume: 5, Issue:10

    Topics: Animals; Behavior; Behavior, Animal; Blood-Brain Barrier; Dopamine; Feeding Behavior; gamma-Aminobutyric Acid; Humans; Learning; Memory; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1980
Muscimol, a psychoactive constituent of Amanita muscaria, as a medicinal chemical model structure.
    Acta chemica Scandinavica. Series B: Organic chemistry and biochemistry, 1981, Volume: 35, Issue:5

    Topics: Agaricales; Amanita; Animals; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Magnetic Resonance Spectroscopy; Models, Chemical; Models, Structural; Molecular Conformation; Muscimol; Nipecotic Acids; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Stereoisomerism

1981
Structure-activity studies on ibotenic acid and related muscimol analogues.
    Advances in biochemical psychopharmacology, 1981, Volume: 27

    Topics: Amino Acids; Animals; Cats; Ibotenic Acid; In Vitro Techniques; Muscimol; Neurons; Oxazoles; Structure-Activity Relationship

1981

Trials

2 trial(s) available for muscimol and oxazoles

ArticleYear
Huntington's disease: treatment with muscimol, a GABA-mimetic drug.
    Annals of neurology, 1978, Volume: 4, Issue:3

    Topics: Activities of Daily Living; Adolescent; Adult; Clinical Trials as Topic; Cognition; Double-Blind Method; Female; gamma-Aminobutyric Acid; Humans; Huntington Disease; Male; Middle Aged; Muscimol; Oxazoles; Placebos

1978
Effects of gamma aminobutyric acid (GABA) and muscimol on endocrine pancreatic function in man.
    Metabolism: clinical and experimental, 1982, Volume: 31, Issue:1

    Topics: Adolescent; Adult; Blood Glucose; C-Peptide; Female; gamma-Aminobutyric Acid; Glucagon; Humans; Insulin; Islets of Langerhans; Male; Middle Aged; Muscimol; Oxazoles

1982

Other Studies

230 other study(ies) available for muscimol and oxazoles

ArticleYear
Cataleptic and anticataleptic effects of muscimol and gabaculine injected into globus pallidus and substantia nigra, and interactions with haloperidol or benzodiazepines.
    Naunyn-Schmiedeberg's archives of pharmacology, 1978, Volume: 305, Issue:3

    Topics: 4-Aminobutyrate Transaminase; Animals; Anti-Anxiety Agents; Benzodiazepines; Catalepsy; Corpus Striatum; Cyclohexanecarboxylic Acids; Cyclohexylamines; Drug Interactions; gamma-Aminobutyric Acid; Globus Pallidus; Haloperidol; Homovanillic Acid; Humans; Injections; Male; Muscimol; Oxazoles; Rats; Substantia Nigra; Transaminases

1978
Improvement in tardive dyskinesia after muscimol therapy.
    Archives of general psychiatry, 1979, Volume: 36, Issue:5

    Topics: Adult; Aged; Antipsychotic Agents; Dopamine; Drug Evaluation; Dyskinesia, Drug-Induced; Extrapyramidal Tracts; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Muscimol; Oxazoles; Receptors, Dopamine; Schizophrenia; Stimulation, Chemical; Synaptic Transmission

1979
Muscimol and related GABA receptor agonists: the potency of GABAergic drugs in vivo determined after intranigral injection.
    The Journal of pharmacy and pharmacology, 1979, Volume: 31, Issue:5

    Topics: Animals; gamma-Aminobutyric Acid; Humans; Injections; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Stereotyped Behavior; Substantia Nigra; Time Factors

1979
Potentiation of muscimol-induced hyperactivity by benzodiazepines.
    The Journal of pharmacy and pharmacology, 1979, Volume: 31, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Drug Synergism; Injections; Male; Motor Activity; Muscimol; Oxazoles; Rats; Substantia Nigra; Time Factors

1979
Ontogeny of GABA and benzodiazepine receptors: effects of Triton X-100, bromide and muscimol.
    Brain research, 1979, Dec-28, Volume: 179, Issue:2

    Topics: Age Factors; Animals; Anti-Anxiety Agents; Bromides; Cerebellum; Female; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Polyethylene Glycols; Pregnancy; Rats; Receptors, Drug

1979
Effects of benzodiazepines and barbiturates in a GABA-dependent animal model: interactions with muscimol in the globus pallidus [proceedings].
    British journal of pharmacology, 1979, Volume: 66, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Barbiturates; Behavior, Animal; Benzodiazepines; Drug Interactions; Female; gamma-Aminobutyric Acid; Globus Pallidus; Muscimol; Oxazoles; Rats

1979
[Effects of muscimol and diazepam: a comparative study on behavioral inhibiton induced by novelty, punishment, and nonreward (author's transl)].
    Psychopharmacology, 1979, Mar-14, Volume: 61, Issue:1

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Diazepam; Environment; Feeding Behavior; Male; Muscimol; Oxazoles; Punishment; Rats; Reward

1979
Electroencephalographic and behavioral effects of a GABA agonist (muscimol) on photosensitive epilepsy in the baboon, papio papio.
    Epilepsia, 1979, Volume: 20, Issue:4

    Topics: Animals; Anticonvulsants; Drug Evaluation, Preclinical; Electroencephalography; Haplorhini; Muscimol; Oxazoles; Papio; Photic Stimulation; Seizures

1979
Modification of the behavioural effects of amphetamine by a GABA agonist in a primate species.
    Psychopharmacology, 1979, Aug-08, Volume: 64, Issue:2

    Topics: Animals; Behavior, Animal; Callitrichinae; Dextroamphetamine; Dopamine; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Haplorhini; Humans; Male; Motor Activity; Muscimol; Oxazoles; Stereotyped Behavior

1979
[Ventrobulbular hypotensive action of muscimol].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1978, Volume: 172, Issue:4

    Topics: Animals; Bradycardia; Brain Stem; Cats; Female; Hypotension; Male; Muscimol; Oxazoles

1978
Stimulation of prolactin and growth hormone secretion by muscimol, a gamma-aminobutyric acid agonist.
    The Journal of clinical endocrinology and metabolism, 1978, Volume: 47, Issue:6

    Topics: Adult; Aged; Chronic Disease; Female; gamma-Aminobutyric Acid; Growth Hormone; Humans; Huntington Disease; Kinetics; Male; Middle Aged; Muscimol; Oxazoles; Prolactin; Schizophrenia

1978
The effect of muscimol on prolactin secretion in male rats.
    Communications in psychopharmacology, 1978, Volume: 2, Issue:3

    Topics: Animals; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Haloperidol; Male; Methyltyrosines; Muscimol; Oxazoles; Premedication; Prolactin; Rats; Receptors, Neurotransmitter

1978
GABA agonists and potential antagonists related to muscimol.
    Brain research, 1979, Nov-16, Volume: 177, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Functional Laterality; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Male; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter; Stereotyped Behavior; Substantia Nigra

1979
Effects of diazepam and muscimol on GABA-mediated neurotransmission: interactions with inosine and nicotinamide.
    Life sciences, 1979, Dec-03, Volume: 25, Issue:23

    Topics: Animals; Corpus Striatum; Diazepam; Drug Interactions; Female; gamma-Aminobutyric Acid; Globus Pallidus; Inosine; Muscimol; Niacinamide; Oxazoles; Rats; Synaptic Transmission; Time Factors

1979
High-affinity binding of [3H]muscimol to subcellular particles of a neurone-enriched culture of embryonic rat brain.
    Neuroscience letters, 1979, Volume: 14, Issue:2-3

    Topics: Animals; Brain; Brain Chemistry; Culture Techniques; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter; Subcellular Fractions

1979
Anticonvulsant activity of muscimol against seizures induced by impairment of GABA-mediated neurotransmission.
    Neuropharmacology, 1979, Volume: 18, Issue:11

    Topics: Animals; Anticonvulsants; Bicuculline; gamma-Aminobutyric Acid; Isoniazid; Male; Muscimol; Oxazoles; Pentylenetetrazole; Picrotoxin; Rats; Seizures; Strychnine; Synaptic Transmission

1979
Distribution and metabolism of muscimol in the brain and other tissues of the rat.
    Neuropharmacology, 1979, Volume: 18, Issue:1

    Topics: Aminooxyacetic Acid; Animals; Brain; Injections, Intravenous; Injections, Intraventricular; Male; Muscimol; Oxazoles; Pargyline; Proadifen; Rats; Time Factors; Tissue Distribution

1979
Modifications of DOPAC levels in the striatum and olfactory tubercles of the rat after muscimol.
    Pharmacological research communications, 1979, Volume: 11, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Corpus Striatum; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscimol; Olfactory Bulb; Oxazoles; Phenylacetates; Rats; Time Factors

1979
Characterization of the binding of [3H]muscimol, a potent gamma-aminobutyric acid agonist, to rat brain synaptosomal membranes using a filtration assay.
    Journal of neurochemistry, 1979, Volume: 32, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Cerebellum; gamma-Aminobutyric Acid; Kinetics; Muscimol; Oxazoles; Rats; Receptors, Drug; Synaptic Membranes; Tissue Distribution

1979
Effects of the GABA receptor agonist muscimol on the turnover of brain dopamine and on the motor activity of rats.
    Acta pharmacologica et toxicologica, 1979, Volume: 44, Issue:3

    Topics: Animals; Brain; Cell Nucleus; Dihydroxyphenylalanine; Dopamine; gamma-Aminobutyric Acid; Male; Motor Activity; Muscimol; Norepinephrine; Oxazoles; Rats

1979
Characterization of [3H]muscimol binding to mouse brain membranes.
    Biochemical pharmacology, 1979, Apr-01, Volume: 28, Issue:7

    Topics: Animals; Binding, Competitive; Brain; Detergents; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Mice; Muscimol; Osmolar Concentration; Oxazoles; Receptors, Drug

1979
Dihydromuscimol, thiomuscimol and related heterocyclic compounds as GABA analogues.
    Journal of neurochemistry, 1979, Volume: 32, Issue:6

    Topics: Animals; Brain; Cats; Cell Membrane; gamma-Aminobutyric Acid; Muscimol; Neurons; Oxazoles; Oxazolidinones; Rats; Receptors, Drug; Spinal Cord; Structure-Activity Relationship

1979
Enhancement of the binding of 3H-diazepam to rat brain membranes in vitro by SQ 20009, A novel anxiolytic, gamma-aminobutyric acid (GABA) and muscimol.
    Life sciences, 1979, Feb-26, Volume: 24, Issue:9

    Topics: Animals; Bicuculline; Brain; Diazepam; Etazolate; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Nicotinic Acids; Oxazoles; Picrotoxin; Rats; Stimulation, Chemical

1979
Characteristics of muscimol accumulation in mouse brain after systemic administration.
    Neuropharmacology, 1979, Volume: 18, Issue:4

    Topics: Animals; Bicuculline; Brain; gamma-Aminobutyric Acid; History, 18th Century; Injections, Intravenous; Mice; Muscimol; Oxazoles; Phenobarbital; Time Factors

1979
Evidence for two types of binding of 3H-gaba and 3H-muscimol in rat cerebral cortex and cerebellum.
    Life sciences, 1979, May-14, Volume: 24, Issue:20

    Topics: Animals; Brain Stem; Cerebellum; Cerebral Cortex; Corpus Striatum; gamma-Aminobutyric Acid; Male; Muscimol; Organ Specificity; Oxazoles; Radioligand Assay; Rats; Receptors, Drug; Substrate Specificity; Synaptosomes

1979
The GABA agonist THIP a muscimol analogue, does not interfere with the benzodiazepine binding site on rats cortical membranes.
    Neuroscience letters, 1979, Volume: 12, Issue:1

    Topics: Animals; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Imidazoles; In Vitro Techniques; Isonicotinic Acids; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Taurine

1979
Turning behaviour induced by injection of muscimol or picrotoxin into the substantia nigra demonstrates dual GABA components.
    Neuroscience letters, 1979, Volume: 12, Issue:2-3

    Topics: Animals; gamma-Aminobutyric Acid; Male; Movement; Muscimol; Organ Specificity; Oxazoles; Picrotoxin; Rats; Substantia Nigra

1979
Dual gamma-aminobutyric acid control of prolactin secretion in the rat.
    Endocrinology, 1979, Volume: 105, Issue:3

    Topics: Animals; Bicuculline; Female; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Methyltyrosines; Muscimol; Oxazoles; Picrotoxin; Pituitary Gland, Anterior; Prolactin; Rats

1979
Increase in striatal acetylcholine levels by GABA mimetic drugs: lack of involvement of the nigro-striatal dopaminergic neurons.
    European journal of pharmacology, 1979, Volume: 56, Issue:1-2

    Topics: Acetylcholine; Animals; Corpus Striatum; gamma-Aminobutyric Acid; Hydroxydopamines; Male; Muscimol; Oxazoles; Rats

1979
Baclofen and muscimol: behavioural and neurochemical sequelae of unilateral intranigral administration and effects on 3H-GABA receptor binding.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 306, Issue:3

    Topics: Aminobutyrates; Animals; Baclofen; Behavior, Animal; Brain Chemistry; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Hydroxydopamines; Injections; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Substantia Nigra; Time Factors

1979
Unpleasant side effects of muscimol.
    The American journal of psychiatry, 1979, Volume: 136, Issue:10

    Topics: Humans; Muscimol; Oxazoles; Schizophrenia

1979
Central antihypertensive properties of muscimol and related gamma-aminobutyric acid agonists and the interaction of muscimol with baroreceptor reflexes.
    Canadian journal of physiology and pharmacology, 1979, Volume: 57, Issue:6

    Topics: Animals; Blood Pressure; Cats; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Heart Rate; Male; Muscimol; Oxazoles; Pressoreceptors; Reflex; Vasomotor System

1979
Muscimol antagonism of morphine analgesia in rats.
    British journal of pharmacology, 1979, Volume: 67, Issue:1

    Topics: Animals; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Muscimol; Oxazoles; Rats; Reaction Time; Time Factors

1979
THIP and isoguvacine are partial agonists of GABA-stimulated benzodiazepine receptor binding.
    European journal of pharmacology, 1979, Oct-15, Volume: 58, Issue:4

    Topics: Animals; Benzodiazepines; Cerebral Cortex; Drug Synergism; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Muscimol; Oxazoles; Rats; Receptors, Drug

1979
The effect of muscimol on hippocampal pyramidal cells.
    European journal of pharmacology, 1979, Oct-26, Volume: 59, Issue:1-2

    Topics: Action Potentials; Animals; Bicuculline; Electric Stimulation; Hippocampus; Humans; In Vitro Techniques; Male; Muscimol; Oxazoles; Pyramidal Tracts; Rabbits; Strychnine; Synapses; Time Factors

1979
[3H]Muscimol binding to rat cerebellar membranes.
    Advances in experimental medicine and biology, 1979, Volume: 123

    Topics: Animals; Cell Membrane; Cerebellum; Female; gamma-Aminobutyric Acid; Kinetics; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Tritium

1979
More muscimol binding sites than GABA binding sites in a particulate fraction of rat brain.
    Biochemical pharmacology, 1979, Sep-01, Volume: 28, Issue:17

    Topics: Animals; Binding Sites; Brain; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Muscimol; Oxazoles; Rats

1979
Comparison of the "specific" binding of [3H]GABA and [3H]muscimol to a particulate fraction of rat brain.
    General pharmacology, 1979, Volume: 10, Issue:6

    Topics: Animals; Brain; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Muscimol; Nerve Tissue Proteins; Oxazoles; Protein Binding; Rats; Subcellular Fractions

1979
Conformational analysis of muscimol, a GABA agonist.
    Journal of theoretical biology, 1979, Aug-07, Volume: 79, Issue:3

    Topics: Bicuculline; Binding Sites; gamma-Aminobutyric Acid; Isoxazoles; Models, Molecular; Molecular Conformation; Muscimol; Oxazoles; Quantum Theory

1979
GABA and hypothalamic feeding systems. I. Topographic analysis of the effects of microinjections of muscimol.
    Physiology & behavior, 1979, Volume: 23, Issue:6

    Topics: Animals; Bicuculline; Brain Mapping; Digestive System; Eating; Female; gamma-Aminobutyric Acid; Gastric Juice; Hypothalamus; Hypothalamus, Middle; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats

1979
Muscimol uptake, release and binding in rat brain slices.
    Journal of neurochemistry, 1978, Volume: 31, Issue:6

    Topics: Alanine; Animals; Binding, Competitive; Biological Transport; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Muscimol; Oxazoles; Rats; Receptors, Drug

1978
Does uptake limit the actions of GABA agonists in vivo? Experiments with muscimol, isoguvacine and THIP in cat spinal cord.
    Journal of neurochemistry, 1978, Volume: 31, Issue:6

    Topics: Aminobutyrates; Animals; Biological Transport; Cats; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Muscimol; Neurons; Nipecotic Acids; Oxazoles; Spinal Cord

1978
Recent advances in the morphological localization of gamma-aminobutyric acid receptors in the cerebellum by means of [3H]muscimol.
    Progress in brain research, 1979, Volume: 51

    Topics: Animals; Brain; Cerebellar Nuclei; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Oxazoles; Purkinje Cells; Rats

1979
Contralateral turning evoked by the intranigral microinjection of muscimol and other GABA agonists.
    Brain research, 1978, Oct-27, Volume: 155, Issue:2

    Topics: Animals; Behavior; Caudate Nucleus; Dopamine Antagonists; Dose-Response Relationship, Drug; Ethanolamines; Female; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Imidazoles; Muscimol; Oxazoles; Picrotoxin; Putamen; Rats; Stereotyped Behavior; Substantia Nigra

1978
Striatal dopamine release and contraversive rotation elicited by intranigrally applied muscimol.
    Nature, 1978, Sep-21, Volume: 275, Issue:5677

    Topics: Animals; Behavior, Animal; Dopamine; Functional Laterality; Homovanillic Acid; Movement; Muscimol; Oxazoles; Substantia Nigra

1978
A comparative study of the effects of muscimol and diazepam on the recall of noxious events.
    Experientia, 1979, Feb-15, Volume: 35, Issue:2

    Topics: Animals; Avoidance Learning; Diazepam; Dissociative Disorders; gamma-Aminobutyric Acid; Humans; Male; Memory; Mental Recall; Muscimol; Oxazoles; Rats

1979
Modulatory effects of baclofen muscimol and GABA on interspecific aggressive behaviour in the rat.
    Neuropharmacology, 1978, Volume: 17, Issue:12

    Topics: Aggression; Aminobutyrates; Animals; Baclofen; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Olfactory Bulb; Oxazoles; Rats

1978
Neuropharmacological spectrum of muscimol.
    Life sciences, 1979, Aug-13, Volume: 25, Issue:7

    Topics: Animals; Anticonvulsants; Catalepsy; Drug Interactions; gamma-Aminobutyric Acid; Humans; Male; Mice; Motor Activity; Muscimol; Muscle Relaxants, Central; Nervous System; Oxazoles; Receptors, Drug

1979
Behavioral differences induced by muscimol selectively injected into pars compacta and pars reticulata of Substantia nigra.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 310, Issue:1

    Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; Drug Interactions; Humans; Injections; Male; Muscimol; Oxazoles; Rats; Stereotyped Behavior; Substantia Nigra; Time Factors

1979
Effects of intracerebral injection with muscimol on locomotor activity and catalepsy in rats.
    Japanese journal of pharmacology, 1979, Volume: 29, Issue:3

    Topics: Animals; Catalepsy; Humans; Injections, Intraventricular; Locomotion; Male; Muscimol; Oxazoles; Rats

1979
Response of dopamine neurons in substantia nigra to muscimol.
    Brain research, 1978, Oct-13, Volume: 154, Issue:2

    Topics: Animals; Bicuculline; Dopamine; Dose-Response Relationship, Drug; Evoked Potentials; gamma-Aminobutyric Acid; Male; Muscimol; Neurons; Oxazoles; Picrotoxin; Rats; Substantia Nigra

1978
Homotaurine and muscimol mimic taurine and GABA effects on muscle tone and temperature regulation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1978, Volume: 305, Issue:2

    Topics: Amino Acids; Animals; Body Temperature Regulation; Electroencephalography; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Injections, Intraventricular; Male; Muscimol; Muscle Tonus; Oxazoles; Rabbits; Taurine

1978
Reductions in blood pressure, heart rate and renal sympathetic nerve discharge in cats after the central administration of muscimol, a GABA agonist.
    Neuropharmacology, 1978, Volume: 17, Issue:10

    Topics: Animals; Bicuculline; Blood Pressure; Cats; Drug Interactions; Heart Rate; Kidney; Muscimol; Norepinephrine; Oxazoles; Pressoreceptors; Sympathetic Nervous System

1978
Photoaffinity labeling of the GABAA receptor with [3H]muscimol.
    Journal of neurochemistry, 1985, Volume: 44, Issue:3

    Topics: Affinity Labels; Animals; Baclofen; Diazepam; Glutamates; Glutamic Acid; Kinetics; Male; Molecular Weight; Muscimol; Oxazoles; Photochemistry; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spectrophotometry, Ultraviolet

1985
Benzodiazepines enhance the muscimol-dependent activation of phospholipase A2 in glioma C6 cells.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Arachidonic Acid; Arachidonic Acids; Cell Line; Chromatography, High Pressure Liquid; Diazepam; Drug Interactions; Enzyme Activation; Glioma; Muscimol; Neuroglia; Oxazoles; Phospholipases; Phospholipases A; Phospholipases A2; Prostaglandin D2; Prostaglandins D; Rats; Receptors, GABA-A

1985
Excitatory amino acids: studies on the biochemical and chemical stability of ibotenic acid and related compounds.
    Journal of neurochemistry, 1985, Volume: 45, Issue:3

    Topics: Animals; Brain; Chemical Phenomena; Chemistry; Chromatography, High Pressure Liquid; Decarboxylation; Glutamates; Glutamic Acid; Hot Temperature; Hydrogen-Ion Concentration; Ibotenic Acid; Isoxazoles; Liver; Mice; Muscimol; Oxazoles; Pregnancy Proteins

1985
Modification of saccadic eye movements by GABA-related substances. I. Effect of muscimol and bicuculline in monkey superior colliculus.
    Journal of neurophysiology, 1985, Volume: 53, Issue:1

    Topics: Animals; Bicuculline; Eye Movements; gamma-Aminobutyric Acid; Macaca mulatta; Muscimol; Oxazoles; Saccades; Superior Colliculi; Synaptic Transmission; Visual Fields

1985
Modification of saccadic eye movements by GABA-related substances. II. Effects of muscimol in monkey substantia nigra pars reticulata.
    Journal of neurophysiology, 1985, Volume: 53, Issue:1

    Topics: Animals; Brain Mapping; Eye Movements; gamma-Aminobutyric Acid; Macaca mulatta; Muscimol; Neural Pathways; Oxazoles; Saccades; Substantia Nigra; Superior Colliculi; Synaptic Transmission

1985
Synthesis and pharmacological evaluation of cis-2,3,3a,4,5,6,7,7a-octahydro-3-oxoisoxazolo[5,4-c]pyridine: a structural analogue of the GABA agonist THIP.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:8

    Topics: Animals; Anticonvulsants; Cerebellum; Electrophysiology; Female; Isoxazoles; Male; Mice; Muscimol; Oxazoles; Rats; Receptors, GABA-A

1985
Subsensitivity to muscimol-induced catalepsy after long-term administration of phenytoin in rats.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: Animals; Bicuculline; Catalepsy; Drug Interactions; Humans; Male; Muscimol; Oxazoles; Phenytoin; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Effect of THIP and SL 76002, two clinically experimented GABA-mimetic compounds, on anterior pituitary GABA receptors and prolactin secretion in the rat.
    Life sciences, 1987, Mar-02, Volume: 40, Issue:9

    Topics: Animals; Anticonvulsants; Bicuculline; Binding, Competitive; Female; gamma-Aminobutyric Acid; Haloperidol; Isoxazoles; Kinetics; Male; Muscimol; Ovariectomy; Oxazoles; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Effect of GABAergic drugs in the behavioral 'despair' test in rats.
    European journal of pharmacology, 1986, Feb-18, Volume: 121, Issue:2

    Topics: Acetates; Aminooxyacetic Acid; Animals; Baclofen; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Muscimol; Oxazoles; Picrotoxin; Rats

1986
Central action of gamma-aminobutyric acid ligands to alter basal water and electrolyte absorption in the rat ileum.
    Gastroenterology, 1985, Volume: 88, Issue:2

    Topics: Animals; Bicuculline; Biological Transport; Body Fluids; Cholinergic Fibers; Electrolytes; GABA Antagonists; gamma-Aminobutyric Acid; Ileum; Intestinal Absorption; Ligands; Male; Muscimol; Oxazoles; Parasympathetic Nervous System; Rats; Rats, Inbred Strains; Receptors, Cholinergic

1985
Deficits in manipulative behaviors induced by local injections of muscimol in the first somatosensory cortex of the conscious monkey.
    Brain research, 1985, Jan-28, Volume: 325, Issue:1-2

    Topics: Animals; Brain Diseases; Brain Mapping; Female; gamma-Aminobutyric Acid; Hand; Macaca; Motor Skills; Muscimol; Oxazoles; Somatosensory Cortex

1985
Rigidity and catalepsy after injections of muscimol into the ventromedial thalamic nucleus: an electromyographic study in the rat.
    Experimental brain research, 1985, Volume: 58, Issue:3

    Topics: Animals; Bicuculline; Catalepsy; Electromyography; Humans; Male; Muscimol; Muscle Rigidity; Oxazoles; Rats; Rats, Inbred Strains; Restraint, Physical; Thalamic Nuclei

1985
Characteristics and distribution of muscimol binding sites in cat visual cortex.
    Brain research, 1984, Aug-13, Volume: 308, Issue:2

    Topics: Animals; Autoradiography; Cats; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Muscimol; Oxazoles; Receptors, GABA-A; Tissue Distribution; Tritium; Visual Cortex

1984
Ontogenesis of muscimol binding sites in cat visual cortex.
    Brain research bulletin, 1984, Volume: 13, Issue:2

    Topics: Animals; Binding Sites; Cats; gamma-Aminobutyric Acid; Kinetics; Muscimol; Neural Inhibition; Oxazoles; Receptors, GABA-A; Visual Cortex

1984
GABA agonist induced analgesia elicited from the lateral preoptic area in the rat.
    European journal of pharmacology, 1984, Dec-15, Volume: 107, Issue:1

    Topics: Analgesia; Animals; Baclofen; Male; Muscimol; Oxazoles; Preoptic Area; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A

1984
Single class of muscimol binding sites in the solubilized gamma-aminobutyrate-benzodiazepine receptor complex.
    Neuroscience, 1984, Volume: 13, Issue:4

    Topics: Animals; Brain; Brain Chemistry; Cattle; Cerebral Cortex; Chromatography, Gel; Flunitrazepam; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
In vitro effects of melatonin on [3H]muscimol binding in rat brain.
    Progress in neuro-psychopharmacology & biological psychiatry, 1984, Volume: 8, Issue:4-6

    Topics: Animals; Brain; Buffers; Corpus Striatum; Frontal Lobe; Male; Melatonin; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes

1984
Some barbiturates enhance the effect of muscimol on dopamine turnover in the rat retina.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 213, Issue:2

    Topics: Animals; Barbital; Barbiturates; Convulsants; Dopamine; Drug Synergism; GABA Antagonists; gamma-Aminobutyric Acid; Light; Male; Methyltyrosines; Muscimol; Oxazoles; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Retina; Sesterterpenes

1980
Autoradiographic localization of binding sites for [3H]gamma-aminobutyrate, [3H]muscimol,(+)[3H]bicuculline methiodide and [3H] flunitrazepam in cultures of rat cerebellum and spinal cord.
    Neuroscience, 1980, Volume: 5, Issue:9

    Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Autoradiography; Bicuculline; Binding Sites; Cells, Cultured; Cerebellum; Female; Fetus; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Pregnancy; Rats; Receptors, Drug; Spinal Cord; Tritium

1980
Binding and uptake of the GABA analogue, 3H-muscimol, in the retinas of goldfish and chicken.
    Investigative ophthalmology & visual science, 1980, Volume: 19, Issue:12

    Topics: Animals; Autoradiography; Chickens; gamma-Aminobutyric Acid; Goldfish; Muscimol; Neurons; Neurotransmitter Agents; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Retina

1980
Inhibition by arylsulphatase A of Na-independent [3H]-GABA and [3H]-muscimol binding to bovine cerebellar synaptic membranes.
    Neuropharmacology, 1980, Volume: 19, Issue:11

    Topics: Animals; Brain; Cattle; Cerebellum; Cerebroside-Sulfatase; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Oxazoles; Sodium; Sulfatases; Synaptic Membranes

1980
Effect of muscimol on glucose-stimulated somatostatin and insulin release from the isolated, perfused rat pancreas.
    Diabetes, 1981, Volume: 30, Issue:2

    Topics: Animals; Glucose; In Vitro Techniques; Insulin; Male; Muscimol; Oxazoles; Pancreas; Perfusion; Rats; Somatostatin

1981
Effect of single and repeated convulsions on glutamate decarboxylase (GAD) activity and [3H]muscimol binding in the rat brain.
    The Journal of pharmacy and pharmacology, 1981, Volume: 33, Issue:5

    Topics: Animals; Brain; Carboxy-Lyases; Electroshock; Glutamate Decarboxylase; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium

1981
Effects of muscimol on the crayfish neuromuscular junction.
    Comparative biochemistry and physiology. C: Comparative pharmacology, 1981, Volume: 70, Issue:1

    Topics: Animals; Astacoidea; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Kinetics; Membrane Potentials; Muscimol; Neuromuscular Junction; Oxazoles; Synapses

1981
Serotonergic drugs, benzodiazepines and baclofen block muscimol-induced myoclonic jerks in a strain of mice.
    European journal of pharmacology, 1981, Jul-17, Volume: 73, Issue:2-3

    Topics: 5-Hydroxytryptophan; Animals; Anti-Anxiety Agents; Baclofen; Benzodiazepines; Male; Mice; Muscimol; Myoclonus; Oxazoles; Piperazines; Pyrazines; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Serotonin; Serotonin

1981
Anion-dependent modulation of [3H]muscimol binding and of GABA-stimulated [3H]flunitrazepam binding by picrotoxin and related CNS convulsants.
    European journal of pharmacology, 1982, Jul-30, Volume: 81, Issue:4

    Topics: Animals; Anions; Anti-Anxiety Agents; Cerebral Cortex; Convulsants; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Receptors, Drug; Receptors, GABA-A; Strychnine; Tubocurarine

1982
Relative disposition of the GABA agonists THIP and muscimol in the brain of the rat.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:10

    Topics: Animals; Brain; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Time Factors

1982
Tofizopam affects binding of [3H]muscimol to gamma-amino-butyric acid receptors in rat and mouse brains.
    Pharmacological research communications, 1982, Volume: 14, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Brain; Diazepam; Kinetics; Male; Mice; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter

1982
Differential modulation of etazolate or pentobarbital enhanced [3H] muscimol binding by benzodiazepine agonists and inverse agonists.
    Brain research, 1983, Dec-05, Volume: 280, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Etazolate; Flumazenil; Flunitrazepam; Kinetics; Muscimol; Nicotinic Acids; Oxazoles; Pentobarbital; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Hypnotic action of benzodiazepines: a possible mechanism.
    Life sciences, 1984, Apr-30, Volume: 34, Issue:18

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Hypnotics and Sedatives; Male; Mice; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Reflex; Sleep

1984
[Differences in the mechanism of the antihypoxic action of benzodiazepine receptor agonists and muscimol].
    Biulleten' eksperimental'noi biologii i meditsiny, 1984, Volume: 98, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Drug Evaluation, Preclinical; gamma-Aminobutyric Acid; Hypoxia; Ligands; Mice; Muscimol; Oxazoles; Receptors, GABA-A

1984
Reduction of [3H]muscimol binding sites in rat dorsal spinal cord after neonatal capsaicin treatment.
    Brain research, 1980, Dec-08, Volume: 202, Issue:2

    Topics: Animals; Animals, Newborn; Capsaicin; Fatty Acids, Unsaturated; Ganglia, Spinal; Muscimol; Neurons; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Sodium; Strychnine; Substance P

1980
Muscimol injections in the nucleus raphé dorsalis block the antinociceptive effect of morphine in rats: apparent lack of 5-hydroxytryptamine involvement in muscimol's effect.
    British journal of pharmacology, 1984, Volume: 81, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Analgesics; Animals; Brain Chemistry; Hydroxyindoleacetic Acid; Injections; Male; Morphine; Muscimol; Oxazoles; Raphe Nuclei; Rats; Reaction Time; Serotonin; Time Factors

1984
Plasma growth hormone and prolactin response to dopaminergic GABAmimetic and cholinergic stimulation in Huntington's disease.
    Neurology, 1983, Volume: 33, Issue:9

    Topics: Adult; Apomorphine; Arecoline; Dopamine; Female; gamma-Aminobutyric Acid; Growth Hormone; Humans; Huntington Disease; Male; Muscimol; Oxazoles; Prolactin

1983
GABA receptors in bovine cerebral blood vessels: binding studies with [3H]muscimol.
    Brain research, 1980, Mar-03, Volume: 185, Issue:1

    Topics: Animals; Binding, Competitive; Cattle; Cerebral Arteries; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Pia Mater; Receptors, Neurotransmitter; Vasodilation

1980
Effect of the GABA receptor agonist muscimol on regional cerebral blood flow in the rat.
    Brain research, 1980, Mar-10, Volume: 185, Issue:2

    Topics: Animals; Caudate Nucleus; Cerebellum; Cerebral Cortex; Cerebrovascular Circulation; Female; gamma-Aminobutyric Acid; Mesencephalon; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter; Thalamus

1980
Autoradiographic localization of 3H-GABA and 3H-muscimol binding in rat cerebellar cultures.
    Experimental brain research, 1980, Volume: 38, Issue:2

    Topics: Animals; Autoradiography; Binding Sites; Cerebellum; Culture Techniques; Dendrites; gamma-Aminobutyric Acid; Muscimol; Neurons; Oxazoles; Purkinje Cells; Rats; Receptors, Neurotransmitter

1980
Substrate specificity of [3H]muscimol binding to a particulate fraction of a neuron-enriched culture of embryonic rat brain.
    Journal of neurochemistry, 1980, Volume: 34, Issue:4

    Topics: Animals; Binding, Competitive; Brain; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Kinetics; Muscimol; Neurons; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A

1980
Presence of a low molecular weight endogenous inhibitor on 3H-muscimol binding in synaptic membranes.
    Nature, 1980, Jun-26, Volume: 285, Issue:5767

    Topics: Animals; Brain Chemistry; GABA Antagonists; Molecular Weight; Muscimol; Neurons; Oxazoles; Polyethylene Glycols; Rats; Receptors, Neurotransmitter; Synaptic Membranes

1980
Potentiation by intraventricular muscimol of the anticonflict effect of benzodiazepines.
    Brain research, 1980, Sep-08, Volume: 196, Issue:2

    Topics: Animals; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drinking; Eating; Fear; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter

1980
Na+-independent binding of [3H]GABA and [3H]muscimol to a "microsomal" fraction, but not to a myelin fraction of rat brain; further evidence that glial elements do not possess GABA-receptors.
    General pharmacology, 1980, Volume: 11, Issue:4

    Topics: Animals; Brain; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Microscopy, Electron; Microsomes; Muscimol; Neuroglia; Oxazoles; Rats; Receptors, Neurotransmitter; Sodium; Tritium

1980
Increase in striatal [3H]muscimol binding following intrastriatal injection of kainic acid: a denervation supersensitivity phenomenon.
    Journal of neurochemistry, 1980, Volume: 35, Issue:2

    Topics: Animals; Corpus Striatum; gamma-Aminobutyric Acid; Kainic Acid; Male; Microinjections; Muscimol; Muscle Denervation; Octoxynol; Oxazoles; Polyethylene Glycols; Pyrrolidines; Rats; Receptors, Cell Surface; Receptors, GABA-A

1980
Nigral-derived muscimol circling--ipsiversive, contraversive or controversial?
    Nature, 1981, Apr-16, Volume: 290, Issue:5807

    Topics: Animals; Behavior, Animal; Dopamine; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra

1981
Development of [3H]muscimol binding to subcellular particles of a culture of mouse brain.
    Neurochemical research, 1980, Volume: 5, Issue:12

    Topics: Animals; Axons; Brain; Cells, Cultured; Female; Mice; Microscopy, Phase-Contrast; Muscimol; Neurons; Oxazoles; Pregnancy; Receptors, Cell Surface; Receptors, GABA-A; Subcellular Fractions

1980
GABA and muscimol inhibit the release of prolactin from dispersed rat anterior pituitary cells.
    Neuroendocrinology, 1981, Volume: 32, Issue:3

    Topics: Animals; Bicuculline; Dopamine; Female; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Oxazoles; Picrotoxin; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Cell Surface; Receptors, GABA-A

1981
Heterogeneous depression of glucose utilization in the caudate nucleus by GABA agonists.
    Brain research, 1981, Mar-30, Volume: 209, Issue:2

    Topics: Animals; Autoradiography; Blood Glucose; Caudate Nucleus; Isoxazoles; Male; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A

1981
The insensitivity of developing benzodiazepine receptors to chronic treatment with diazepam, GABA and muscimol in brain cell cultures.
    Brain research, 1981, Apr-06, Volume: 210, Issue:1-2

    Topics: Animals; Brain; Cell Membrane; Cells, Cultured; Diazepam; Female; Fetus; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Muscimol; Oxazoles; Pregnancy; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter

1981
Localized binding of [3H]muscimol to synapses in chicken retina.
    Proceedings of the National Academy of Sciences of the United States of America, 1981, Volume: 78, Issue:1

    Topics: Animals; Autoradiography; Binding, Competitive; Chickens; gamma-Aminobutyric Acid; Microscopy, Electron; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Retina; Synapses

1981
GABA and muscimol open ion channels of different lifetimes on cultured mouse spinal cord cells.
    Brain research, 1981, Jan-05, Volume: 204, Issue:1

    Topics: Animals; Cells, Cultured; Electric Conductivity; Embryo, Mammalian; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Membrane Potentials; Mice; Muscimol; Neurons; Oxazoles; Spinal Cord

1981
Involvement of dopamine in circling responses to muscimol depends on intranigral site of injection.
    European journal of pharmacology, 1981, Feb-19, Volume: 69, Issue:4

    Topics: Animals; Humans; Hydroxydopamines; Male; Motor Activity; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Stereotyped Behavior; Substantia Nigra

1981
GABAergic synapses in the goldfish retina: an autoradiographic study of 3H-muscimol and 3H-GABA binding.
    The Journal of comparative neurology, 1981, Jul-20, Volume: 200, Issue:1

    Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; Goldfish; Muscimol; Neurons; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Muscarinic; Retina; Synapses; Visual Pathways

1981
Na+ independent binding of [3H] muscimol to a membrane fraction of the brains of normal and dwarf mice.
    Experientia, 1981, Volume: 37, Issue:6

    Topics: Animals; Brain; Cell Membrane; Dwarfism, Pituitary; Kinetics; Mice; Muscimol; Organ Size; Oxazoles; Receptors, Drug; Receptors, GABA-A; Sodium

1981
The effects of muscimol and picrotoxin injections into the cat substantia nigra.
    Naunyn-Schmiedeberg's archives of pharmacology, 1981, Volume: 317, Issue:1

    Topics: Animals; Behavior, Animal; Cats; Female; Hindlimb; Humans; Injections; Male; Muscimol; Oxazoles; Picrotoxin; Receptors, Cell Surface; Receptors, GABA-A; Stereotyped Behavior; Substantia Nigra

1981
3H-muscimol binding in synaptosomal fractions from bovine and developing rabbit retinas.
    Journal of neuroscience research, 1981, Volume: 6, Issue:4

    Topics: Animals; Binding, Competitive; Cattle; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rabbits; Receptors, Cell Surface; Receptors, GABA-A; Retina; Synaptic Transmission; Synaptosomes

1981
Quantitative autoradiography of [3H]muscimol binding in rat brain.
    Science (New York, N.Y.), 1981, Nov-27, Volume: 214, Issue:4524

    Topics: Animals; Autoradiography; Brain; Kainic Acid; Kinetics; Muscimol; Oxazoles; Rats; Receptors, Drug; Receptors, GABA-A; Tritium

1981
Muscimol induces gastric acid secretion after central administration.
    Brain research, 1981, Dec-14, Volume: 229, Issue:1

    Topics: Animals; Gastric Acid; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Secretory Rate

1981
Glutamic acid decarboxylase and gamma-aminobutyric acid in Huntington's disease fibroblasts and other cultured cells, determined by a [3H]muscimol radioreceptor assay.
    Journal of neurochemistry, 1981, Volume: 37, Issue:4

    Topics: Carboxy-Lyases; Cells, Cultured; Fibroblasts; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Humans; Huntington Disease; Kinetics; Muscimol; Oxazoles; Radioligand Assay; Receptors, Cell Surface; Receptors, GABA-A; Skin

1981
Chronic benzodiazepine treatment increases [3H]muscimol binding in mouse brain.
    Neuropharmacology, 1982, Volume: 21, Issue:1

    Topics: Animals; Benzodiazepinones; Brain; Cerebellum; Chlordiazepoxide; Clonazepam; In Vitro Techniques; Mice; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A

1982
Acute and chronic effects of pentobarbital in relation to postsynaptic GABA receptors: a study with muscimol.
    Journal of neuroscience research, 1982, Volume: 7, Issue:1

    Topics: Animals; Brain; Drug Tolerance; gamma-Aminobutyric Acid; Humans; Male; Mice; Mice, Inbred ICR; Muscimol; Oxazoles; Pentobarbital; Receptors, Cell Surface; Receptors, GABA-A; Sleep; Substance Withdrawal Syndrome; Synaptic Membranes

1982
Stimulatory and protective effects of benzodiazepines on GABA receptors labeled with [3H]muscimol.
    Life sciences, 1982, Mar-15, Volume: 30, Issue:11

    Topics: Animals; Benzodiazepines; Hot Temperature; In Vitro Techniques; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium

1982
Binding of [3H]gamma-aminobutyric acid and [3H]muscimol in purified rat brain synaptic plasma membranes and the effects of bicuculline.
    Journal of neurochemistry, 1982, Volume: 39, Issue:1

    Topics: Animals; Bicuculline; Binding, Competitive; Brain; gamma-Aminobutyric Acid; Male; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Membranes; Tritium

1982
Single channel currents activated by gamma-aminobutyric acid, muscimol, and (-)-pentobarbital in cultured mouse spinal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1982, Volume: 2, Issue:7

    Topics: Animals; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Mice; Muscimol; Neurons; Oxazoles; Pentobarbital; Spinal Cord

1982
Effect of ethanol and ethanol withdrawal on 3H-muscimol binding and behaviour in the rat: a pilot study.
    Acta pharmacologica et toxicologica, 1981, Volume: 49, Issue:5

    Topics: Animals; Behavior, Animal; Brain; Ethanol; Humans; Male; Muscimol; Oxazoles; Pilot Projects; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substance Withdrawal Syndrome

1981
(3H)-muscimol, (3H)-nipecotic acid and (3H)-isoguvacine as autoradiographic markers for GABA neurotransmission.
    Journal of neural transmission, 1982, Volume: 54, Issue:1-2

    Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; Goldfish; Guinea Pigs; Isonicotinic Acids; Muscimol; Neuroglia; Neurons; Nipecotic Acids; Oxazoles; Rabbits; Receptors, Cell Surface; Receptors, GABA-A; Retina; Synaptic Transmission

1982
Glycine antagonists structurally related to muscimol, THIP, or isoguvacine.
    Journal of neurochemistry, 1982, Volume: 39, Issue:5

    Topics: Animals; Cats; gamma-Aminobutyric Acid; Glycine; Interneurons; Isonicotinic Acids; Isoxazoles; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Glycine; Spinal Cord; Structure-Activity Relationship

1982
High specific binding of [3H]GABA and [3H]muscimol to membranes from dendrodendritic synaptosomes of the rat olfactory bulb.
    Journal of neurochemistry, 1982, Volume: 39, Issue:5

    Topics: Animals; Dendrites; gamma-Aminobutyric Acid; Male; Muscimol; Olfactory Bulb; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Subcellular Fractions; Synaptic Membranes; Synaptosomes

1982
Muscimol and some aza analogues: molecular orbital calculations relating to their potency as GABA mimetics.
    Journal of theoretical biology, 1982, Jul-21, Volume: 97, Issue:2

    Topics: Binding Sites; Chemical Phenomena; Chemistry; Electrons; gamma-Aminobutyric Acid; Humans; Molecular Conformation; Muscimol; Oxazoles; Pyrazoles; Pyrazolones; Receptors, Neurotransmitter; Rotation; Structure-Activity Relationship; Triazoles

1982
Effects of GABAergic agonists and antagonists on various ethanol-induced behavioral changes.
    Psychopharmacology, 1982, Volume: 78, Issue:1

    Topics: Animals; Behavior, Animal; Bicuculline; Body Temperature Regulation; Dose-Response Relationship, Drug; Ethanol; Female; Motor Activity; Muridae; Muscimol; Oxazoles; Pentylenetetrazole; Picrotoxin; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Sleep Stages; Strychnine

1982
Intra-raphe muscimol induced hyperactivity depends on ascending serotonin projections.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:5

    Topics: Animals; Bicuculline; Brain Stem; Chlordiazepoxide; Dose-Response Relationship, Drug; Male; Mesencephalon; Motor Activity; Muscimol; Oxazoles; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Serotonin; Tegmentum Mesencephali

1982
Comparison of centrifugation and filtration assays of ligand binding: do multiple GABA receptive sites exist?
    Journal of neuroscience research, 1982, Volume: 8, Issue:4

    Topics: Animals; Brain; Cattle; Centrifugation; Cerebral Cortex; Filtration; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Membranes

1982
Changes in [3H]muscimol binding in substantia nigra, entopeduncular nucleus, globus pallidus, and thalamus after striatal lesions as demonstrated by quantitative receptor autoradiography.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1983, Volume: 3, Issue:6

    Topics: Animals; Autoradiography; Corpus Striatum; gamma-Aminobutyric Acid; Globus Pallidus; Kainic Acid; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Substantia Nigra; Thalamus

1983
Bicuculline insensitive effects of baclofen.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 322, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Bicuculline; Corpus Striatum; gamma-Aminobutyric Acid; Male; Motor Activity; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter

1983
Motor and postural effects of kainic acid or GABA agonist and antagonist injection into the cerebellar nucleus fastigii.
    Birth defects original article series, 1983, Volume: 19, Issue:4

    Topics: Animals; Cerebellar Nuclei; Kainic Acid; Motor Skills; Muscimol; Muscle Contraction; Oxazoles; Picrotoxin; Posture; Pyrrolidines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission

1983
Anisatin modulation of temperature-dependent inhibition [3H]muscimol binding by chloride ion.
    Brain research, 1983, Jun-27, Volume: 270, Issue:1

    Topics: Animals; Anions; Brain; Chlorides; Kinetics; Lactones; Male; Muscimol; Oxazoles; Plants, Toxic; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Sesquiterpenes; Spiro Compounds; Synaptic Membranes; Temperature

1983
Modulation of [3H]muscimol binding in rat cerebellar and cerebral cortical membranes by picrotoxin, pentobarbitone, and etomidate.
    Journal of neurochemistry, 1983, Volume: 41, Issue:2

    Topics: Animals; Cell Membrane; Cerebellar Cortex; Cerebral Cortex; Etomidate; Imidazoles; Kinetics; Male; Muscimol; Organ Specificity; Oxazoles; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
[3H]muscimol binding site on purified benzodiazepine receptor.
    Journal of neurochemistry, 1983, Volume: 41, Issue:4

    Topics: Animals; Binding Sites; Brain; Flunitrazepam; gamma-Aminobutyric Acid; Molecular Weight; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Diazepam stimulates the binding of GABA and muscimol but not THIP to rat brain membranes.
    Neuroscience letters, 1983, Aug-08, Volume: 38, Issue:3

    Topics: Analgesics; Animals; Brain; Diazepam; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Decreased high-affinity binding of [3H]muscimol to cerebral synaptic membranes of scrapie-infected mice.
    Journal of neurochemistry, 1984, Volume: 42, Issue:1

    Topics: Animals; Brain; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Mice, Inbred C57BL; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Scrapie; Sheep; Synaptic Membranes

1984
Characterization of susceptibility to audiogenic seizures in ethanol-dependent rats after microinjection of gamma-aminobutyric acid (GABA) agonists into the inferior colliculus, substantia nigra or medial septum.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:3

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Bicuculline; Ethanol; GABA Antagonists; Humans; Inferior Colliculi; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures; Septum Pellucidum; Substance Withdrawal Syndrome; Substantia Nigra

1983
Antihypertensive effect of the GABA receptor agonist muscimol in spontaneously hypertensive rats. Role of the sympathoadrenal axis.
    Circulation research, 1984, Volume: 54, Issue:1

    Topics: Adrenal Glands; Animals; Atropine; Blood Pressure; Catecholamines; Clonidine; Efferent Pathways; Heart Rate; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Splanchnic Nerves; Sympathectomy, Chemical; Sympathetic Nervous System; Vagotomy

1984
Synergistic inhibition of [3H]muscimol binding to calf-brain synaptic membranes in the presence of L-homocysteine and pyridoxal 5'-phosphate. A possible mechanism for homocysteine-induced seizures.
    European journal of biochemistry, 1983, Dec-15, Volume: 137, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Cattle; Drug Synergism; Homocysteine; In Vitro Techniques; Kinetics; Models, Chemical; Muscimol; Oxazoles; Pyridoxal Phosphate; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Synaptic Membranes

1983
Intranigral muscimol suppresses ethanol withdrawal seizures.
    Brain research, 1984, Apr-23, Volume: 298, Issue:1

    Topics: Acoustic Stimulation; Alcoholism; Animals; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Substance Withdrawal Syndrome; Substantia Nigra

1984
In vivo release of [3H]GABA in cat caudate nucleus and substantia nigra. II. Involvement of different thalamic nuclei in the bilateral changes induced by a nigral application of muscimol.
    Brain research, 1984, Jun-15, Volume: 303, Issue:2

    Topics: Animals; Cats; Caudate Nucleus; Dominance, Cerebral; Female; gamma-Aminobutyric Acid; Male; Muscimol; Neural Pathways; Neurons; Oxazoles; Substantia Nigra; Synaptic Transmission; Thalamic Nuclei

1984
Effects of valproic acid on spinal reflexes and [3H]muscimol and [3H]diazepam binding in brain membranes in rats.
    Journal of pharmacobio-dynamics, 1983, Volume: 6, Issue:3

    Topics: Animals; Brain; Diazepam; Male; Membranes; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Reflex; Spinal Cord; Valproic Acid

1983
Diazepam antagonizes GABA- and muscimol-induced changes of acetylcholine release in slices of guinea-pig cerebral cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:1

    Topics: Acetylcholine; Animals; Benzodiazepinones; Cerebral Cortex; Diazepam; Flumazenil; GABA Antagonists; Guinea Pigs; In Vitro Techniques; Muscimol; Oxazoles

1983
Depolarizing responses to glycine, beta-alanine and muscimol in isolated optic nerve and cuneate nucleus.
    British journal of pharmacology, 1983, Volume: 79, Issue:3

    Topics: Alanine; Animals; beta-Alanine; Bicuculline; Dose-Response Relationship, Drug; Glycine; Male; Medulla Oblongata; Muscimol; Optic Nerve; Oxazoles; Picrotoxin; Rats; Rats, Inbred Strains; Strychnine; Time Factors

1983
Behavioural responsiveness to muscimol and apomorphine 2 months after prolonged treatment with estradiol in rats.
    Psychopharmacology, 1984, Volume: 84, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Castration; Estradiol; Female; Humans; Motor Activity; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Stereotyped Behavior

1984
[Influence of the GABAergic system on eating behavior induced by the tail pinching technic in rats].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1981, Volume: 175, Issue:3

    Topics: Animals; Energy Intake; Feeding Behavior; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Rats, Inbred Strains; Stress, Psychological; Valproic Acid

1981
Autoradiographic studies of [3H]-glycine, [3H]-GABA, and [3H]-muscimol uptake in the mudpuppy retina.
    Experimental eye research, 1984, Volume: 39, Issue:1

    Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Microscopy, Electron; Muscimol; Necturus; Oxazoles; Retina; Tritium

1984
[Increased 3H-muscimol binding in post-mortem brains of chronic schizophrenics].
    Seishin shinkeigaku zasshi = Psychiatria et neurologia Japonica, 1984, Volume: 86, Issue:3

    Topics: Adult; Aged; Binding Sites; Chronic Disease; Female; Frontal Lobe; Glutamate Decarboxylase; Humans; Male; Middle Aged; Muscimol; Oxazoles; Putamen; Schizophrenia

1984
Synergistic anticonvulsant effects of a GABA agonist and glycine.
    General pharmacology, 1984, Volume: 15, Issue:4

    Topics: 3-Mercaptopropionic Acid; Animals; Anticonvulsants; Drug Synergism; gamma-Aminobutyric Acid; Glycine; Male; Mice; Muscimol; Oxazoles; Seizures

1984
Feeding induced by injections of muscimol into the substantia nigra of rats: unaffected by haloperidol but abolished by large lesions of the superior colliculus.
    Neuroscience, 1984, Volume: 13, Issue:1

    Topics: Animals; Brain Mapping; Corpus Striatum; Dopamine; Feeding Behavior; gamma-Aminobutyric Acid; Haloperidol; Male; Muscimol; Neural Pathways; Oxazoles; Rats; Substantia Nigra; Superior Colliculi

1984
GABAergic agents in the medial septal nucleus affect hippocampal theta rhythm and acetylcholine utilization.
    Brain research, 1984, Nov-26, Volume: 322, Issue:2

    Topics: Acetylcholine; Animals; Bicuculline; gamma-Aminobutyric Acid; Hippocampus; Male; Muscimol; Neural Pathways; Oxazoles; Rats; Rats, Inbred Strains; Septal Nuclei; Theta Rhythm

1984
GABA agonists inhibit the vasopressin-dependent pressor effects of central angiotensin II.
    Neuroendocrinology, 1984, Volume: 39, Issue:5

    Topics: Angiotensin II; Animals; Arginine Vasopressin; Blood Pressure; Brain; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Sympathetic Nervous System

1984
Blockade of bicuculline-induced pressor and tachycardic responses by forebrain administration of muscimol.
    Neuropharmacology, 1984, Volume: 23, Issue:11

    Topics: Animals; Bicuculline; Blood Pressure; Cats; Female; Heart Rate; Injections, Intraventricular; Male; Muscimol; Oxazoles

1984
Investigation of the effects of muscimol on different components of [3H]propyl beta-carboline-3-carboxylate binding to rat hippocampal and cerebellar membranes.
    European journal of pharmacology, 1984, Jan-27, Volume: 97, Issue:3-4

    Topics: Animals; Binding Sites; Carbolines; Cell Membrane; Cerebellum; Hippocampus; Indoles; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains

1984
Effects of intrathecally administered THIP, baclofen and muscimol on nociceptive threshold.
    European journal of pharmacology, 1984, Aug-03, Volume: 103, Issue:1-2

    Topics: Animals; Baclofen; Injections, Spinal; Isoxazoles; Male; Muscimol; Muscle Hypotonia; Nociceptors; Oxazoles; Rats; Rats, Inbred Strains; Reaction Time; Sensory Thresholds

1984
Zinc deficiency and anorexia in rats: the effect of central administration of norepinephrine, muscimol and bromerogocryptine.
    Physiology & behavior, 1984, Volume: 32, Issue:3

    Topics: Animals; Anorexia; Bromocriptine; Dose-Response Relationship, Drug; Drug Resistance; Eating; Feeding and Eating Disorders; Humans; Male; Muscimol; Norepinephrine; Oxazoles; Rats; Rats, Inbred Strains; Zinc

1984
In vivo release of [3H]GABA in cat caudate nucleus and substantia nigra. I. Bilateral changes induced by a unilateral nigral application of muscimol.
    Brain research, 1983, Aug-08, Volume: 272, Issue:2

    Topics: Animals; Brain Mapping; Cats; Caudate Nucleus; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Substantia Nigra

1983
Neuronal subpopulations in cat retina which accumulate the GABA agonist, (3H)muscimol: a combined Golgi and autoradiographic study.
    The Journal of comparative neurology, 1983, Sep-01, Volume: 219, Issue:1

    Topics: Animals; Autoradiography; Cats; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Muscimol; Oxazoles; Retina

1983
Unilateral injection of GABA agonists in the superior colliculus: asymmetry to tactile stimulation.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:2

    Topics: Analgesics; Animals; Baclofen; Functional Laterality; gamma-Aminobutyric Acid; Isoxazoles; Motor Activity; Muscimol; Oxazoles; Physical Stimulation; Rats; Rats, Inbred Strains; Superior Colliculi; Touch

1983
Muscimol inhibits ADH release induced by hypertonic sodium chloride in rats.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:2

    Topics: Animals; Bicuculline; Dose-Response Relationship, Drug; Male; Muscimol; Osmolar Concentration; Oxazoles; Radioimmunoassay; Rats; Rats, Inbred Strains; Sodium Chloride; Vasopressins

1983
Reaction of muscimol with 4-aminobutyrate aminotransferase.
    Journal of neurochemistry, 1983, Volume: 41, Issue:6

    Topics: 4-Aminobutyrate Transaminase; Animals; Brain; Kinetics; Liver; Muscimol; Ornithine-Oxo-Acid Transaminase; Oxazoles; Rabbits; Spectrophotometry

1983
Effects of nigral application of muscimol on release of [3H] gamma-aminobutyrate and on multiunit activity in various cat thalamic nuclei.
    Neuroscience, 1983, Volume: 10, Issue:3

    Topics: Animals; Cats; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Substantia Nigra; Thalamic Nuclei; Tritium

1983
Monoamine involvement in the overeating caused by muscimol injection in the rat nucleus raphe dorsalis and the effects of d-fenfluramine and d-amphetamine.
    European journal of pharmacology, 1983, Oct-14, Volume: 94, Issue:1-2

    Topics: 5,7-Dihydroxytryptamine; Animals; Biogenic Amines; Dextroamphetamine; Feeding Behavior; Fenfluramine; Food Deprivation; Injections; Male; Muscimol; Oxazoles; Penfluridol; Phenoxybenzamine; Raphe Nuclei; Rats

1983
GABA-mediated inhibition of breathing in the late gestation sheep fetus.
    Journal of developmental physiology, 1983, Volume: 5, Issue:6

    Topics: Animals; Apnea; Female; Fetal Hypoxia; Fetus; gamma-Aminobutyric Acid; Gestational Age; Muscimol; Oxazoles; Picrotoxin; Pregnancy; Respiration; Sheep

1983
[A new simplified method for the synthesis of muscimol (5-aminomethyl-3-hydroxyisoxazole)].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1983, Volume: 18, Issue:11

    Topics: Muscimol; Oxazoles

1983
Evidence that the nigrotegmental GABAergic projection mediates stereotypy induced by apomorphine and intranigral muscimol.
    Life sciences, 1983, Sep-05, Volume: 33, Issue:10

    Topics: Animals; Apomorphine; Corpus Striatum; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Neural Pathways; Oxazoles; Pons; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substantia Nigra; Tegmentum Mesencephali

1983
Disinhibition of muricide and irritability by intraseptal muscimol.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:4

    Topics: Aggression; Animals; Brain; Catheterization; Dose-Response Relationship, Drug; Feeding Behavior; Humans; Male; Metergoline; Muscimol; Oxazoles; Quipazine; Rats; Semicarbazides

1983
Extrastriatal circuits activated by intrastriatal muscimol: a [14C]2-deoxyglucose investigation.
    Brain research, 1984, Feb-06, Volume: 292, Issue:2

    Topics: Animals; Brain; Brain Mapping; Corpus Striatum; gamma-Aminobutyric Acid; Glucose; Male; Muscimol; Neural Pathways; Oxazoles; Rats; Rats, Inbred Strains

1984
Differential effects of baclofen, gamma-hydroxybutyric acid and muscimol on the protective action of phenobarbital and diphenylhydantoin against maximal electroshock-induced seizures in mice.
    Neuropharmacology, 1984, Volume: 23, Issue:2A

    Topics: Animals; Anticonvulsants; Baclofen; Drug Interactions; Electroshock; gamma-Aminobutyric Acid; Hydroxybutyrates; Injections, Intraventricular; Male; Mice; Muscimol; Oxazoles; Phenobarbital; Phenytoin; Sodium Oxybate

1984
Nigral muscimol infusions facilitate the development of seizures in immature rats.
    Brain research, 1984, Volume: 315, Issue:2

    Topics: Age Factors; Animals; Flurothyl; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rats; Seizures; Substantia Nigra

1984
Muscimol-scopolamine interactions in the rat brain: a study with 2-deoxy-D-[1-14C]glucose.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1984, Volume: 4, Issue:6

    Topics: Animals; Brain; Deoxyglucose; gamma-Aminobutyric Acid; Glucose; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Scopolamine

1984
Circling behavior induced by intranigral injections of GABA and muscimol in rats.
    Psychopharmacology, 1980, Volume: 68, Issue:1

    Topics: Animals; Atropine; Behavior; Bicuculline; Brain Chemistry; Female; gamma-Aminobutyric Acid; Haloperidol; Humans; Injections; Muscimol; Oxazoles; Rats; Stereotyped Behavior; Strychnine; Substantia Nigra; Time Factors

1980
Sodium di-n-propylacetate (valproate) potentiates responses to GABA and muscimol on single central neurones.
    Brain research, 1980, Sep-15, Volume: 197, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Evoked Potentials; gamma-Aminobutyric Acid; Medulla Oblongata; Muscimol; Neurons; Oxazoles; Rats; Reticular Formation; Valproic Acid

1980
Effects of sodium n-dipropylacetate, muscimol hydrobromide and (R,S) nipecotic acid amide on isolation-induced aggressive behavior in mice.
    Psychopharmacology, 1980, Volume: 70, Issue:3

    Topics: Aggression; Animals; gamma-Aminobutyric Acid; Humans; Male; Mice; Motor Activity; Muscimol; Nipecotic Acids; Oxazoles; Social Isolation; Time Factors; Valproic Acid

1980
Modulatory interactions between norepinephrine and taurine, beta-alanine, gamma-aminobutyric acid and muscimol, applied iontophoretically to cerebellar Purkinje cells.
    Neuropharmacology, 1981, Volume: 20, Issue:6

    Topics: Alanine; Animals; beta-Alanine; Cerebellum; Female; gamma-Aminobutyric Acid; Iontophoresis; Muscimol; Nerve Endings; Norepinephrine; Oxazoles; Purkinje Cells; Rats; Taurine

1981
Differential effects of IV and IP muscimol on central dopamine metabolism.
    Psychopharmacology, 1981, Volume: 74, Issue:1

    Topics: Animals; Brain; Dopamine; Injections, Intraperitoneal; Injections, Intravenous; Male; Muscimol; Oxazoles; Rats; Receptors, Dopamine

1981
Effect of muscimol, a central GABA receptor agonist, on the catalepsy, striatal homovanillic acid increase, and analgesia induced by pilocarpine in rats.
    Psychopharmacology, 1981, Volume: 74, Issue:4

    Topics: Analgesics; Animals; Catalepsy; Corpus Striatum; Drug Interactions; Homovanillic Acid; Humans; Male; Muscimol; Oxazoles; Phenylacetates; Pilocarpine; Rats; Rats, Inbred Strains

1981
A new method for the evaluation of benzodiazepines based on their ability to block muscimol-induced myoclonic jerks in mice.
    Psychopharmacology, 1981, Volume: 75, Issue:3

    Topics: Animals; Benzodiazepines; Diazepam; Drug Evaluation; Flunitrazepam; Male; Mice; Muscimol; Myoclonus; Oxazoles; Spinal Cord

1981
[Protective effects of muscimol on acute brain ischemia in the rat (author's transl)].
    Comptes rendus des seances de l'Academie des sciences. Serie III, Sciences de la vie, 1982, Mar-15, Volume: 294, Issue:11

    Topics: Animals; Baclofen; gamma-Aminobutyric Acid; Ischemic Attack, Transient; Kinetics; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1982
Oral behaviour induced by intranigral muscimol is unaffected by haloperidol but abolished by large lesions of superior colliculus.
    Psychopharmacology, 1982, Volume: 77, Issue:3

    Topics: Animals; Behavior, Animal; Brain; Haloperidol; Humans; Injections; Male; Muscimol; Oxazoles; Rats; Stereotyped Behavior; Substantia Nigra; Superior Colliculi

1982
Baclofen blocks postsynaptic inhibition but not the effect of muscimol in the olfactory cortex.
    British journal of pharmacology, 1983, Volume: 78, Issue:1

    Topics: Animals; Baclofen; Cerebral Cortex; Drug Interactions; Electric Stimulation; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscimol; Neural Conduction; Neural Inhibition; Olfactory Pathways; Oxazoles; Synapses

1983
The effects of the GABAergic agonist muscimol upon the relationship between local cerebral blood flow and glucose utilization.
    Brain research, 1983, Jan-10, Volume: 258, Issue:2

    Topics: Animals; Brain; Cerebrovascular Circulation; Deoxyglucose; Glucose; Kinetics; Muscimol; Organ Specificity; Oxazoles; Rats

1983
Muscimol potentiation of acidic amino acid release from cerebellar synaptosomes is chloride dependent.
    Journal of neurochemistry, 1983, Volume: 40, Issue:4

    Topics: Animals; Aspartic Acid; Cerebellum; Chlorides; Drug Synergism; Ions; Kinetics; Male; Muscimol; Osmolar Concentration; Oxazoles; Potassium; Rats; Rats, Inbred Strains; Synaptosomes

1983
Simultaneous modulation of hippocampal cholinergic activity and extinction by intraseptal muscimol.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:2

    Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Extinction, Psychological; Hippocampus; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Reaction Time; Reinforcement, Psychology

1983
Effects of barbiturates and ethanol on muscimol-induced release of [3H]-D-aspartate from rodent cerebellum.
    Neuropharmacology, 1983, Volume: 22, Issue:6

    Topics: Animals; Aspartic Acid; Cerebellum; Ethanol; gamma-Aminobutyric Acid; Kinetics; Male; Muscimol; Oxazoles; Pentobarbital; Potassium; Rats; Rats, Inbred Strains; Synaptosomes; Tritium

1983
GABAergic drugs, morphine and morphine tolerance: a study in relation to nociception and gastrointestinal transit in mice.
    Neuropharmacology, 1983, Volume: 22, Issue:6

    Topics: Aminooxyacetic Acid; Analgesia; Animals; Baclofen; Bicuculline; Cyclohexanecarboxylic Acids; Digestion; Digestive System; Digestive System Physiological Phenomena; Drug Tolerance; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Morphine; Muscimol; Naloxone; Nociceptors; Oxazoles; Picrotoxin

1983
BehavioraL and biochemical changes caused by muscimol in mice withdrawN from haloperidol administration.
    Neuropharmacology, 1982, Volume: 21, Issue:9

    Topics: Animals; Behavior, Animal; Corpus Striatum; Dopamine; Haloperidol; Homovanillic Acid; Humans; Male; Mice; Mice, Inbred ICR; Motor Activity; Muscimol; Oxazoles; Substance Withdrawal Syndrome

1982
The ventromedullary hypotensive effect of muscimol in the anaesthetized cat.
    Clinical and experimental hypertension, 1981, Volume: 3, Issue:2

    Topics: Anesthesia; Animals; Bicuculline; Blood Pressure; Brain Stem; Cats; Hypotension; Muscimol; Oxazoles; Stereotaxic Techniques

1981
Antagonism of gamma-aminobutyric acid and muscimol by picrotoxin, bicuculline, strychnine, bemegride, leptazol, D-tubocurarine and theophylline in the isolated olfactory cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1982, Volume: 318, Issue:4

    Topics: Animals; Bicuculline; GABA Antagonists; Guinea Pigs; In Vitro Techniques; Muscimol; Olfactory Bulb; Oxazoles; Pentylenetetrazole; Picrotoxin; Strychnine; Theophylline; Tubocurarine

1982
Periaqueductal gray matter involvement in the muscimol-induced decrease of morphine antinociception.
    Naunyn-Schmiedeberg's archives of pharmacology, 1982, Volume: 318, Issue:4

    Topics: Analgesia; Animals; Cerebral Aqueduct; Male; Morphine; Muscimol; Oxazoles; Rats; Rats, Inbred Strains

1982
Therapeutics of monomethylhydrazine intoxication.
    Toxicology and applied pharmacology, 1982, Volume: 63, Issue:2

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Therapy, Combination; Male; Methylhydrazines; Mice; Mice, Inbred ICR; Monomethylhydrazine; Muscimol; Oxazoles; Pyridoxine; Seizures

1982
Effects of the putative GABAergic agonists, muscimol and THIP, upon local cerebral glucose utilisation.
    Journal of neurochemistry, 1982, Volume: 39, Issue:3

    Topics: Analgesics; Animals; Brain; Deoxy Sugars; Deoxyglucose; gamma-Aminobutyric Acid; Glycolysis; Isoxazoles; Male; Muscimol; Organ Specificity; Oxazoles; Rats; Rats, Inbred Strains

1982
Effects of gamma-aminobutyric acid agonist and antagonist drugs on local cerebral glucose utilization.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1982, Volume: 2, Issue:7

    Topics: Animals; Autoradiography; Bicuculline; Brain; Carbon Radioisotopes; Deoxy Sugars; Deoxyglucose; gamma-Aminobutyric Acid; Glycolysis; Male; Muscimol; Organ Specificity; Oxazoles; Rats

1982
Differential localization of radioactive gamma-aminobutyric acid and muscimol in isolated and in vivo mouse retina.
    Experimental eye research, 1982, Volume: 35, Issue:6

    Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; In Vitro Techniques; Mice; Muscimol; Neuroglia; Oxazoles; Retina; Time Factors; Tissue Distribution

1982
Chlordiazepoxide-induced ataxia, muscle relaxation and sedation in the rat: effects of muscimol, picrotoxin and naloxone.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:6

    Topics: Animals; Arousal; Chlordiazepoxide; Exploratory Behavior; Male; Motor Activity; Motor Skills; Muridae; Muscimol; Muscle Contraction; Muscle Relaxation; Naloxone; Oxazoles; Picrotoxin; Rats; Reaction Time

1982
An in vivo method for testing GABAergic compounds.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:4

    Topics: Animals; Apomorphine; gamma-Aminobutyric Acid; Injections, Intraventricular; Injections, Subcutaneous; Male; Mice; Mice, Inbred ICR; Motor Activity; Muscimol; Oxazoles; Picrotoxin

1982
Anticonvulsant effects of muscimol.
    Neurology, 1980, Volume: 30, Issue:6

    Topics: Animals; Bicuculline; GABA Antagonists; Muscimol; Neurons; Oxazoles; Penicillins; Picrotoxin; Rats; Receptors, Drug; Seizures; Strychnine

1980
Rotation induced by intranigral injections of GABA agonists and antagonists: zone-specific effects.
    Pharmacology, biochemistry, and behavior, 1980, Volume: 13, Issue:4

    Topics: Animals; Bicuculline; GABA Antagonists; Humans; Hydroxydopamines; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Rotation; Stereotyped Behavior; Substantia Nigra

1980
Effects of muscimol alone and in combination with diazepam on shuttle-box performance in rats.
    Arzneimittel-Forschung, 1981, Volume: 31, Issue:10

    Topics: Animals; Avoidance Learning; Bicuculline; Diazepam; Drug Interactions; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains

1981
Suppression of apomorphine-induced oral stereotypy in rats by microinjection of muscimol into midbrain.
    Life sciences, 1982, Jun-21, Volume: 30, Issue:25

    Topics: Animals; Apomorphine; Humans; Male; Mesencephalon; Muscimol; Oxazoles; Rats; Stereotyped Behavior; Superior Colliculi

1982
Analgesic properties of the GABA-mimetic THIP.
    European journal of pharmacology, 1981, Jan-16, Volume: 69, Issue:2

    Topics: Analgesics; Animals; Arthritis, Experimental; Baclofen; Electric Stimulation; Isoxazoles; Macaca mulatta; Mice; Morphine; Muscimol; Oxazoles; Reaction Time

1981
Correlation of [14C]muscimol concentration in rat brain with anticonvulsant activity.
    European journal of pharmacology, 1981, Jan-29, Volume: 69, Issue:3

    Topics: Animals; Anticonvulsants; Bicuculline; Brain; Half-Life; Male; Muscimol; Oxazoles; Rats

1981
Sensitization of the perioral biting reflex by intranigral GABA agonist after detelencephalization.
    Neuroscience letters, 1981, Feb-06, Volume: 21, Issue:3

    Topics: Animals; Functional Laterality; Male; Muscimol; Oxazoles; Physical Stimulation; Rats; Reflex; Substantia Nigra; Telencephalon

1981
Muscimol-induced myoclonic jerks in mice.
    Neuropharmacology, 1981, Volume: 20, Issue:5

    Topics: Animals; Drug Interactions; Kinetics; Male; Mice; Muscimol; Oxazoles; Picrotoxin; Seizures

1981
Increases and decreases in local cerebral glucose utilization in response to GABA agonists.
    European journal of pharmacology, 1981, May-08, Volume: 71, Issue:2-3

    Topics: Animals; Brain; gamma-Aminobutyric Acid; Glucose; Isoxazoles; Male; Muscimol; Oxazoles; Rats

1981
GABA and muscimol binding processes in CNS tissue culture preparations.
    Advances in biochemical psychopharmacology, 1981, Volume: 29

    Topics: Animals; Astrocytes; Brain; Culture Media; Culture Techniques; gamma-Aminobutyric Acid; Mice; Muscimol; Neurons; Oxazoles; Rats

1981
Autoradiographic localization of [3H]muscimol in the cat retina.
    Brain research, 1981, Jun-29, Volume: 215, Issue:1-2

    Topics: Animals; Autoradiography; Cats; gamma-Aminobutyric Acid; Microscopy, Electron; Muscimol; Neurons; Oxazoles; Retina; Tritium

1981
Effects of GABAergic drugs on brain stimulation reward as assessed by a 'threshold' method.
    Brain research, 1981, Jun-29, Volume: 215, Issue:1-2

    Topics: Animals; Brain; Dose-Response Relationship, Drug; Electric Conductivity; Electric Stimulation; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Reward; Self Stimulation

1981
Differential effects of sodium-free media on gamma-aminobutyrate and muscimol-evoked conductance increases recorded from lobster muscle fibres.
    Neuroscience, 1981, Volume: 6, Issue:7

    Topics: Animals; Dose-Response Relationship, Drug; Electric Conductivity; Evoked Potentials; gamma-Aminobutyric Acid; Kinetics; Lithium; Muscimol; Muscles; Nephropidae; Nipecotic Acids; Oxazoles; Sodium

1981
Muscimol and gamma-hydroxybutyrate: similar interactions with convulsant agents.
    Life sciences, 1981, Jul-27, Volume: 29, Issue:4

    Topics: 3-Mercaptopropionic Acid; Animals; Anticonvulsants; Bicuculline; Dose-Response Relationship, Drug; Drug Synergism; Hydroxybutyrates; Male; Mice; Muscimol; Oxazoles; Pentylenetetrazole; Seizures; Sodium Oxybate; Strychnine; Sulfhydryl Compounds

1981
Central cardiovascular effects of taurine: comparison with homotaurine and muscimol.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 219, Issue:1

    Topics: Animals; Bicuculline; Cats; Central Nervous System; Hemodynamics; Injections, Intraventricular; Muscimol; Oxazoles; Strychnine; Taurine

1981
Muscimol induced feeding: a model to study the hypothalamic regulation of appetite.
    Life sciences, 1981, Sep-21, Volume: 29, Issue:12

    Topics: Animals; Appetite; Atropine; Calcitonin; Dose-Response Relationship, Drug; Eating; Haloperidol; Hypothalamus; Male; Models, Biological; Muscimol; Naloxone; Oxazoles; Rats; Rats, Inbred Strains

1981
Paradoxical blockade of a muscimol response by THIP, a GABA agonist and also by GABA-transaminase inhibitors.
    Neuropharmacology, 1981, Volume: 20, Issue:12A

    Topics: 4-Aminobutyrate Transaminase; Animals; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Muscimol; Myoclonus; Oxazoles; Time Factors; Transaminases

1981
Muscimol as an antagonist of chemical convulsants.
    Archives internationales de pharmacodynamie et de therapie, 1981, Volume: 253, Issue:2

    Topics: Animals; Anticonvulsants; Convulsants; Male; Mice; Mice, Inbred ICR; Muscimol; Oxazoles

1981
Single unit responses of substantia nigra and globus pallidus neurons to GABA agonist and antagonist drugs.
    Advances in biochemical psychopharmacology, 1981, Volume: 30

    Topics: Animals; gamma-Aminobutyric Acid; Globus Pallidus; Iontophoresis; Isoxazoles; Kainic Acid; Male; Muscimol; Neurons; Oxazoles; Rats; Rats, Inbred Strains; Substantia Nigra

1981
Decrease in effects of muscimol on the dorsal root after repeated administration of diazepam in rats.
    Journal of pharmacobio-dynamics, 1981, Volume: 4, Issue:12

    Topics: Animals; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Male; Membrane Potentials; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Spinal Nerve Roots; Time Factors

1981
Lack of Na"-independent binding of [3H]GABA or [3H]muscimol to particulate fractions of cultured astroblasts.
    Journal of neurochemistry, 1980, Volume: 34, Issue:4

    Topics: Animals; Astrocytes; Brain; Cells, Cultured; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Radioligand Assay; Rats; Sodium; Tritium

1980
Antinociceptive effects of baclofen and muscimol upon intraventricular administration.
    European journal of pharmacology, 1980, Feb-08, Volume: 61, Issue:3

    Topics: Analgesics; Animals; Baclofen; Injections, Intraperitoneal; Injections, Intraventricular; Male; Motor Activity; Muscimol; Oxazoles; Rats

1980
Effects of muscimol and picrotoxin on single unit activity of substantia nigra neurons.
    Brain research, 1980, Apr-21, Volume: 188, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Electric Conductivity; gamma-Aminobutyric Acid; Male; Muscimol; Neurons; Oxazoles; Picrotoxin; Rats; Substantia Nigra

1980
Neuroleptic-induced prolactin rise: influence of pharmacological alterations of different neurotransmitter system.
    Experientia, 1980, Apr-15, Volume: 36, Issue:4

    Topics: Animals; Apomorphine; Diazepam; Diphenhydramine; Haloperidol; Kinetics; Male; Metergoline; Muscimol; Oxazoles; Piperazines; Prolactin; Rats

1980
Binding of [3H]GABA and [3H]muscimol to subcellular particles of a neurone-enriched culture of mouse brain.
    Experientia, 1980, May-15, Volume: 36, Issue:5

    Topics: Animals; Binding, Competitive; Brain; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Kinetics; Ligands; Mice; Muscimol; Neurons; Oxazoles; Protein Binding; Receptors, Drug; Tritium

1980
In vivo release of endogenous gamma-aminobutyric acid from rat striatum: effects of muscimol, oxotremorine, and morphine.
    Journal of neurochemistry, 1980, Volume: 34, Issue:6

    Topics: Animals; Corpus Striatum; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Haloperidol; Male; Morphine; Muscimol; Nalorphine; Oxazoles; Oxotremorine; Potassium; Rats; Tetrodotoxin

1980
Binding of muscimol and GABA in sub-fractions of a crude membrane fraction of rat brain.
    Biochemical pharmacology, 1980, Apr-01, Volume: 29, Issue:7

    Topics: Animals; Brain; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Oxazoles; Rats; Synaptic Membranes

1980
GABAergic actions of THIP in vivo and vitro: a comparison with muscimol and GABA.
    European journal of pharmacology, 1980, Jul-11, Volume: 65, Issue:1

    Topics: Animals; Binding Sites; Brain; Cerebellum; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; In Vitro Techniques; Iontophoresis; Isoxazoles; Male; Muscimol; Neurons; Oxazoles; Rats; Substantia Nigra

1980
Anorexic effects of ethanolamine-O-sulfate and muscimol in the rat: evidence that GABA inhibits ingestive behavior.
    Life sciences, 1980, Jun-09, Volume: 26, Issue:23

    Topics: 4-Aminobutyrate Transaminase; Animals; Appetite Depressants; Body Weight; Brain Chemistry; Dextroamphetamine; Ethanolamines; Feeding Behavior; gamma-Aminobutyric Acid; Male; Motor Activity; Muscimol; Oxazoles; Rats

1980
Some characteristics of [3H]muscimol binding to synaptic membrane from rat brain.
    Brain research, 1980, Sep-22, Volume: 197, Issue:2

    Topics: Animals; Binding Sites; Brain; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Muscimol; Oxazoles; Polyethylene Glycols; Rats; Synaptic Membranes; Temperature

1980
Decreases in the binding of [3H]GABA and [3H]muscimol to a particulate fraction of rat brain produced by human sera; some speculations.
    General pharmacology, 1980, Volume: 11, Issue:5

    Topics: Animals; Blood Physiological Phenomena; Brain; gamma-Aminobutyric Acid; Male; Muscimol; Nerve Tissue Proteins; Oxazoles; Protein Binding; Rats; Synaptic Membranes

1980
[3H]Muscimol binding in the rat retina.
    Life sciences, 1980, Sep-29, Volume: 27, Issue:13

    Topics: Animals; Binding Sites; Female; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Membranes; Muscimol; Octoxynol; Oxazoles; Polyethylene Glycols; Rats; Retina

1980
Cardiovascular effects of intracerebroventricular GABA, glycine and muscimol in the rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1980, Volume: 313, Issue:3

    Topics: Anesthesia; Animals; Dopamine; gamma-Aminobutyric Acid; Glycine; Hemodynamics; Injections, Intraventricular; Male; Muscimol; Oxazoles; Parasympathetic Nervous System; Rats; Serotonin; Sympathetic Nervous System

1980
Effect of muscimol on dopamine metabolism of the rat hypothalamus.
    Experientia, 1980, Nov-15, Volume: 36, Issue:11

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Hypothalamus; Male; Muscimol; Norepinephrine; Oxazoles; Rats

1980
Na+-independent binding of [3H]GABA and [3H]muscimol to subcellular particles of neural primary cultures and whole brain.
    Journal of neurochemistry, 1980, Volume: 34, Issue:1

    Topics: Animals; Animals, Newborn; Astrocytes; Binding Sites; Brain; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rats; Sodium

1980
Binding of [3H]-muscimol, a potent gamma-aminobutyric acid receptor agonist, to membranes of the bovine retina.
    British journal of pharmacology, 1980, Volume: 71, Issue:1

    Topics: Animals; Cattle; In Vitro Techniques; Kinetics; Membranes; Muscimol; Oxazoles; Retina; Subcellular Fractions

1980
Measurement of gamma-aminobutyric acid in human cerebrospinal fluid: radioreceptor assay using [3H]muscimol.
    Clinica chimica acta; international journal of clinical chemistry, 1981, Jan-08, Volume: 109, Issue:1

    Topics: Animals; Cattle; gamma-Aminobutyric Acid; Humans; Muscimol; Oxazoles; Radioligand Assay; Tritium

1981
4,5-Substituted 3-Isoxazolols with Insecticidal Activity Act as Competitive Antagonists of Housefly GABA Receptors.
    Journal of agricultural and food chemistry, 2015, Jul-22, Volume: 63, Issue:28

    Topics: Animals; Binding, Competitive; GABA Antagonists; Gene Expression; Houseflies; Insecticides; Isoxazoles; Models, Molecular; Molecular Structure; Muscimol; Oocytes; Oxazoles; Receptors, GABA; Xenopus laevis

2015
Selective inhibition of extra-synaptic α5-GABA
    Neuropharmacology, 2017, Volume: 125

    Topics: Animals; Benzodiazepines; Binding, Competitive; Brain; Female; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Long-Term Potentiation; Male; Memory; Mice, Inbred C57BL; Muscimol; Neural Inhibition; Nootropic Agents; Oxazoles; Rats, Sprague-Dawley; Receptors, GABA-A; Tissue Culture Techniques

2017