muscimol has been researched along with oxazoles in 237 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 235 (99.16) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (0.84) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Kamioka, T; Matsui, Y | 3 |
Chase, TN; Crayton, JW; Tamminga, CA | 1 |
Arnt, J; Krogsgaard-Larsen, P; Magelund, G; Scheel-Krüger, J | 1 |
Kuhar, MJ; Niehoff, DL; Palacios, JM | 1 |
Crossman, AR; Lee, LA; Longman, DA; Slater, P | 1 |
Jobert, A; Soubrié, P; Thiébot, MH | 2 |
Horton, RW; Meldrum, BS; Pedley, TA | 1 |
Baker, HF; Ridley, RM; Scraggs, PR | 1 |
Charlton, M; Goldblatt, D; Joynt, RJ; Shoulson, I | 1 |
Bloch, R; Bousquet, P; Feldman, J; Schwartz, J | 3 |
Chase, TN; Frohman, LA; Neophytides, A; Tamminga, CA | 1 |
Fang, VS; Meltzer, HY; Simonovic, M | 1 |
Arnt, J; Krogsgaard-Larsen, P | 2 |
Longman, DA; Slater, P | 1 |
DeFeudis, FV; Mandel, P; Ossola, L; Schmitt, G | 2 |
Matthews, WD; McCafferty, GP | 1 |
Baraldi, M; Grandison, L; Guidotti, A | 1 |
Mantegazza, P; Restelli, A; Vicentini, L; Zambotti, F; Zonta, N | 1 |
Risley, EA; Williams, M | 2 |
Andén, NE; Grabowska-Andén, M; Wachtel, H | 1 |
Roberts, E; Salvaterra, P; Wang, YJ | 1 |
Curtis, DR; Hjeds, H; Johnston, GA; Krogsgaard-Larsen, P; Lodge, D | 1 |
Enna, SJ; Maggi, A | 1 |
Baldessarini, RJ; Herschel, M | 1 |
Maurer, R | 2 |
Jenner, P; Leigh, N; Marsden, CD; Reavill, C | 1 |
Betti, R; Cocchi, D; Frigerio, C; Krogsgaard-Larsen, P; Locatelli, V; Müller, EE; Racagni, G | 1 |
Bartholini, G; Scatton, B | 1 |
Cross, AJ; Waddington, JL | 1 |
McDonald, A | 1 |
Gross, DM; Sweet, CS; Wenger, HC | 1 |
Mantegazza, P; Tammiso, R; Vicentini, L; Zambotti, F; Zonta, N | 1 |
Karobath, M; Lippitsch, M | 1 |
Defrance, J; Enna, SJ; Marchand, J; Stanley, J | 1 |
DeFeudis, FV; Mandel, P; Ossola, L | 3 |
Andrews, PR; Johnston, GA | 1 |
Grossman, SP; Kelly, J; Rothstein, J | 1 |
Johnston, GA; Kennedy, SM; Lodge, D | 1 |
Curtis, DR; Johnston, GA; Lodge, D | 1 |
Chan-Palay, V | 1 |
Bacino, CB; Martin, GE; Papp, NL | 1 |
Haubrich, DR; Martin, GE | 1 |
Delini-Stula, A; Vassout, A | 1 |
Depoortere, H; Lloyd, KG; Worms, P | 1 |
Arnt, J; Scheel-Krüger, J | 1 |
Gower, M; MacNeil, D; Szymanska, I | 1 |
Carlà, V; Giotti, A; Magnani, M; Sgaragli, GP | 1 |
Antonaccio, MJ; Kerwin, L; Taylor, DG | 1 |
Cavalla, D; Neff, NH | 1 |
Chuang, DM; Majewska, MD | 1 |
Hansen, SH; Krogsgaard-Larsen, P; Nielsen, EO; Schousboe, A | 1 |
Hikosaka, O; Wurtz, RH | 2 |
Gähwiler, BH; Graff, P; Maurer, R; Nordmann, R | 1 |
Botez, MI; Lalonde, R | 1 |
Apud, JA; Masotto, C; Racagni, G | 1 |
Borsini, F; Evangelista, S; Meli, A | 1 |
Arbit, E; Fogel, R; Kaplan, RB | 1 |
Hikosaka, O; Iwamura, Y; Sakamoto, M; Tanaka, M | 1 |
Klockgether, T; Schwarz, M; Sontag, KH; Turski, L; Wolfarth, S | 1 |
Cynader, M; Needler, MC; Shaw, C | 2 |
Gale, K; Garant, DS; Lim, CR | 1 |
Belonogoff, OB; Lideman, RR | 1 |
Coloma, FM; Niles, LP | 1 |
Kamp, CW; Morgan, WW | 1 |
Hösli, E; Hösli, L; Möhler, H; Richards, JG | 1 |
Brecha, N; Yazulla, S | 2 |
Chweh, A; Ebadi, M | 1 |
Elde, RP; Grouse, LH; Robbins, MS; Sorenson, RL | 1 |
Atterwill, CK; Batts, C; Bloomfield, MR | 1 |
Ishida, M; Shinozaki, H | 1 |
Menon, MK; Vivonia, CA | 2 |
Collins, JF; Karobath, M; Mannonen, A; Supavilai, P | 1 |
Forchetti, MC; Guidotti, A; Krogsgaard-Larsen, P; Moroni, F | 1 |
Saano, V | 1 |
Borea, PA; Karobath, M; Supavilai, P | 1 |
Chweh, AY; Lin, YB; Swinyard, EA | 1 |
Ostrovskaia, RU | 1 |
Placheta, P; Singer, E | 1 |
Romandini, S; Samanin, R | 1 |
Chase, TN; Denaro, A; Durso, R; Ruggeri, S; Tamminga, CA | 1 |
Degener, P; Krause, DN; Roberts, E; Wong, E | 1 |
Edvinsson, L; Larsson, B; Skärby, T | 1 |
Hösli, E; Hösli, L | 1 |
Kuriyama, K; Yoneda, Y | 2 |
DeFeudis, FV | 2 |
Cananzi, AR; Costa, E; Guidotti, A | 1 |
DeFeudis, FV; Devilliers, G; Mandel, P; Sarliéve, LL; Varga, V | 1 |
Ito, Y; Kurihara, E; Kuriyama, K; Yoneda, Y | 1 |
Kilpatrick, IC; Starr, MS | 2 |
DeFeudis, FV; Mandel, P; Ossola, L; Sarliève, LL; Varga, V | 1 |
Besser, GM; Delitala, G; Grossman, A; Yeo, T | 1 |
Kelly, PA; McCulloch, J | 4 |
Gardell, MA; Neale, JH; Shibla, DB | 1 |
Barker, JL; Mathers, DA | 1 |
Yazulla, S | 1 |
DeFeudis, FV; Geffard, M; Mandel, P; Ossola, L; Varga, V | 2 |
Kolasiewicz, W; Sontag, KH; Wolfarth, S | 1 |
Mitchell, CK; Redburn, DA | 1 |
Dauth, GW; Frey, KA; Pan, HS; Penney, JB; Young, AB | 1 |
Grace, M; Kneip, J; Levine, AS; Morley, JE; Silvis, SE | 1 |
Brehm, L; Krogsgaard-Larsen, P; Schaumburg, K | 1 |
Goetz, IE; Hamel, E; Roberts, E | 1 |
Crawley, JN; Marangos, PJ | 1 |
Ho, IK; Nabeshima, T; Sivam, SP | 1 |
Fukuda, H; Matsumoto, K | 2 |
Jordan, CC; Matus, AI; Piotrowski, W; Wilkinson, D | 1 |
Barker, JL; Jackson, MB; Lecar, H; Mathers, DA | 1 |
Linnoila, M; Marangos, PJ; Stowell, L; Thurman, RG | 1 |
Agardh, E; Ehinger, B | 1 |
Curtis, DR; Hjeds, H; Krogsgaard-Larsen, P; Leah, JD; Peet, MJ | 1 |
Cagan, RH; Quinn, MR | 1 |
Armstrong, DR; Breckenridge, RJ; Suckling, CJ | 1 |
Engel, J; Liljequist, S | 1 |
Lorens, SA; Sainati, SM | 1 |
Patel, SC; Peck, EJ | 1 |
Frey, KA; Pan, HS; Penney, JB; Young, AB | 1 |
Rägo, LK; Zarkovsky, AM | 1 |
Canonico, PL; Di Chiara, G; Imperato, A; Nicoletti, F; Piacente, B; Raffaele, R; Scapagnini, U | 1 |
Brenner, O; Quast, U | 1 |
Lucacchini, A; Martini, C; Rigacci, T | 1 |
Johnston, GA; Skerritt, JH | 1 |
Quinn, MR; Somerville, RA | 1 |
Breese, GR; Frye, GD; McCown, TJ | 1 |
Becker, H; Dietz, R; Ganten, D; Lang, RE; Rettig, R; Schömig, A; Schwab, NA; Unger, T | 1 |
Dewhurst, IC; Ekuwem, CE; Griffiths, R; O'Neill, C; Sinclair, CD; Williams, DC | 1 |
Gonzalez, LP; Hettinger, MK | 1 |
Besson, MJ; Gauchy, C; Glowinski, J; Kemel, ML | 1 |
Fukuda, H; Goto, M; Hasebe, Y; Kaneko, T; Kato, K | 1 |
Beani, L; Bianchi, C; Tanganelli, S | 1 |
Simmonds, MA | 1 |
Apud, J; Cagiano, R; Cuomo, V; Masotto, C; Racagni, G | 1 |
Bereksi, B; Boggio, V; Guilland, JC; Klepping, J; Mack, G; Noirot, P | 1 |
Goebel, DJ; McReynolds, JS; Pourch, RG | 1 |
Hanada, S; Hosomi, T; Isoda, K; Kasai, T; Kuno, T; Kuyama, T; Mita, T; Nakai, H; Nishino, N; Uchida, S | 1 |
Sarhan, S; Seiler, N | 1 |
Dean, P; Redgrave, P; Taha, EB | 2 |
Allen, CN; Crawford, IL | 1 |
Brennan, TJ; Haywood, JR; Morris, M | 1 |
Gillis, RA; Quest, JA; Souza, JD | 1 |
Mitchell, R; Wilson, L | 1 |
Drower, EJ; Hammond, DL | 1 |
Essatara, MB; Levine, AS; McClain, CJ; Morley, JE | 1 |
Besson, MJ; Gauchy, C; Glowinski, J; Kemel, ML; Romo, R | 1 |
Goebel, DJ; Pourcho, RG | 1 |
Di Scala, G; Karli, P; Schmitt, P | 1 |
De Caro, G; Iovino, M; Massi, M; Poenaru, S; Steardo, L | 1 |
Fowler, LJ; John, RA; Lovell, DH | 1 |
Besson, MJ; Chéramy, A; Gauchy, C; Glowinski, J; Kemel, ML; Romo, R | 1 |
Bendotti, C; Borsini, F; Przewlocka, B; Samanin, R | 1 |
Gluckman, PD; Johnston, BM | 1 |
Chen, SQ; Geng, RL; Wang, SC | 1 |
Childs, JA; Gale, K | 1 |
Glusman, M; Potegal, M; Yoburn, B | 1 |
Chmielewska, B; Czuczwar, SJ; Kleinrok, Z; Turski, WA | 1 |
Albala, BJ; Moshé, SL | 1 |
Helén, P; London, ED | 1 |
Kaakkola, S; Kääriäinen, I | 1 |
Gent, JP; Phillips, NI | 1 |
Mandel, P; Puglisi-Allegra, S | 1 |
Moises, HC; Waterhouse, BD; Woodward, DJ; Yeh, HH | 1 |
Beart, PM; Gundlach, AL | 2 |
Amladi, SR; Kelkar, MR; Naik, SR; Sheth, UK | 1 |
Haddox, VG; Menon, MK; Vivonia, CA | 1 |
Claperon, N; Durussel, JJ; Rossignol, P | 1 |
Scholfield, CN | 2 |
Aloisi, F; Gallo, V; Levi, G | 1 |
Blaker, WD; Cheney, DL; Costa, E; Gandolfi, O | 1 |
Harris, RA; Rohde, BH | 1 |
Ho, IK; Sivam, SP | 1 |
Fung, YK; Kuruvilla, A; Uretsky, NJ | 1 |
Curtis, DR; Hansen, JJ; Honoré, T; Krogsgaard-Larsen, P; Lodge, D | 1 |
Cappelletti, G; Cavagnini, F; Dubini, A; Invitti, C; Pinto, M; Polli, EE | 1 |
Conci, F; Mantegazza, P; Parenti, M; Tommasi, R; Vicentini, L; Zambotti, F; Zonta, N | 1 |
Back, KC; George, ME; Pinkerton, MK | 1 |
Kuhar, MJ; London, ED; Palacios, JM; Rapoport, SI | 2 |
Blanks, JC; Roffler-Tarlov, S | 1 |
File, SE | 1 |
Bosh, TK; Fung, YK; Grassman, DR; Novin-Baheran, A | 1 |
Collins, RC | 1 |
Kozlowski, MR; Marshall, JF | 1 |
Cortese, I; Cuomo, V; Siro-Brigiani, G | 1 |
Dean, P; Eastwood, L; Redgrave, P | 1 |
Buescher, HH; Hill, RC; Maurer, R; Roemer, D | 1 |
Intoccia, AP; Matthews, WD; McCafferty, GP; Osborne, VL | 1 |
Huston, JP; Welzl, H | 1 |
DeFeudis, FV; Mandel, P; Ossola, L; Rebel, G; Sarliève, LL; Schmitt, G; Varga, V | 1 |
Pourcho, RG | 1 |
Setler, PE; Zarevics, P | 1 |
Constanti, A; Nistri, A | 1 |
Pizzi, WJ; Unnerstall, JR | 1 |
Kneip, J; Levine, AS; Morley, JE | 1 |
Menon, MK | 1 |
Javid, MJ; Stone, WE | 1 |
Bergstrom, DA; Walters, JR; Waszczak, BL | 1 |
Fukuda, H; Kaneko, T; Ono, H | 1 |
Liebman, JM; Pastor, G | 1 |
Eng, N; Walters, JR; Waszczak, BL | 1 |
Chieli, T; Cocchi, D; Fregnan, GB; Müller, EE | 1 |
DeFeudis, FV; Mandel, P; Ossola, L; Sarliève, LL | 1 |
Korf, J; van der Heyden, JA; Venema, K | 1 |
Hruska, RE; Walters, JR; Waszczak, BL | 1 |
Cooper, BR; Howard, JL; Ingold, K; Maxwell, RA; Soroko, F; White, HL | 1 |
DeFeudis, FV; Geffard, M; Mandel, P; Varga, V | 1 |
Schaeffer, JM | 1 |
Persson, B | 1 |
DeFeudis, FV; Mandel, P; Ossola, L; Schmitt, G; Wolff, P | 1 |
Osborne, NN | 1 |
Baraczka, K; Sperk, G | 1 |
Furuta, K; Liu, G; Ozoe, F; Ozoe, Y | 1 |
Antoni, FA; Barkóczy, J; Belelli, D; Brown, AR; Etherington, LA; Gacsályi, I; Gunn, BG; Kertész, S; Lambert, JJ; Ling, I; Livesey, MR; Mihalik, B; Monteiro, O; Pallagi, K; Pálvölgyi, A; Spedding, M; Varga, P | 1 |
5 review(s) available for muscimol and oxazoles
Article | Year |
---|---|
GABA receptor agonists: relationship between structure and biological activity in vivo and in vitro.
Topics: Animals; gamma-Aminobutyric Acid; Kinetics; Muscimol; Oxazoles; Receptors, Drug; Structure-Activity Relationship; Substantia Nigra | 1979 |
Binsing studies with muscimol; relation ty synaptic gamma-aminobutyrate receptors.
Topics: Animals; Astacoidea; Autoradiography; Blood Vessels; Brain; Cattle; Cerebellum; Culture Techniques; Freezing; gamma-Aminobutyric Acid; Kinetics; Muscimol; Muscles; Oxazoles; Pia Mater; Polyethylene Glycols; Rats; Receptors, Neurotransmitter; Sodium; Subcellular Fractions; Substrate Specificity | 1980 |
Physiological and behavioral studies with muscimol.
Topics: Animals; Behavior; Behavior, Animal; Blood-Brain Barrier; Dopamine; Feeding Behavior; gamma-Aminobutyric Acid; Humans; Learning; Memory; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Seizures | 1980 |
Muscimol, a psychoactive constituent of Amanita muscaria, as a medicinal chemical model structure.
Topics: Agaricales; Amanita; Animals; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Magnetic Resonance Spectroscopy; Models, Chemical; Models, Structural; Molecular Conformation; Muscimol; Nipecotic Acids; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Stereoisomerism | 1981 |
Structure-activity studies on ibotenic acid and related muscimol analogues.
Topics: Amino Acids; Animals; Cats; Ibotenic Acid; In Vitro Techniques; Muscimol; Neurons; Oxazoles; Structure-Activity Relationship | 1981 |
2 trial(s) available for muscimol and oxazoles
Article | Year |
---|---|
Huntington's disease: treatment with muscimol, a GABA-mimetic drug.
Topics: Activities of Daily Living; Adolescent; Adult; Clinical Trials as Topic; Cognition; Double-Blind Method; Female; gamma-Aminobutyric Acid; Humans; Huntington Disease; Male; Middle Aged; Muscimol; Oxazoles; Placebos | 1978 |
Effects of gamma aminobutyric acid (GABA) and muscimol on endocrine pancreatic function in man.
Topics: Adolescent; Adult; Blood Glucose; C-Peptide; Female; gamma-Aminobutyric Acid; Glucagon; Humans; Insulin; Islets of Langerhans; Male; Middle Aged; Muscimol; Oxazoles | 1982 |
230 other study(ies) available for muscimol and oxazoles
Article | Year |
---|---|
Cataleptic and anticataleptic effects of muscimol and gabaculine injected into globus pallidus and substantia nigra, and interactions with haloperidol or benzodiazepines.
Topics: 4-Aminobutyrate Transaminase; Animals; Anti-Anxiety Agents; Benzodiazepines; Catalepsy; Corpus Striatum; Cyclohexanecarboxylic Acids; Cyclohexylamines; Drug Interactions; gamma-Aminobutyric Acid; Globus Pallidus; Haloperidol; Homovanillic Acid; Humans; Injections; Male; Muscimol; Oxazoles; Rats; Substantia Nigra; Transaminases | 1978 |
Improvement in tardive dyskinesia after muscimol therapy.
Topics: Adult; Aged; Antipsychotic Agents; Dopamine; Drug Evaluation; Dyskinesia, Drug-Induced; Extrapyramidal Tracts; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Muscimol; Oxazoles; Receptors, Dopamine; Schizophrenia; Stimulation, Chemical; Synaptic Transmission | 1979 |
Muscimol and related GABA receptor agonists: the potency of GABAergic drugs in vivo determined after intranigral injection.
Topics: Animals; gamma-Aminobutyric Acid; Humans; Injections; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Stereotyped Behavior; Substantia Nigra; Time Factors | 1979 |
Potentiation of muscimol-induced hyperactivity by benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Drug Synergism; Injections; Male; Motor Activity; Muscimol; Oxazoles; Rats; Substantia Nigra; Time Factors | 1979 |
Ontogeny of GABA and benzodiazepine receptors: effects of Triton X-100, bromide and muscimol.
Topics: Age Factors; Animals; Anti-Anxiety Agents; Bromides; Cerebellum; Female; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Polyethylene Glycols; Pregnancy; Rats; Receptors, Drug | 1979 |
Effects of benzodiazepines and barbiturates in a GABA-dependent animal model: interactions with muscimol in the globus pallidus [proceedings].
Topics: Animals; Anti-Anxiety Agents; Barbiturates; Behavior, Animal; Benzodiazepines; Drug Interactions; Female; gamma-Aminobutyric Acid; Globus Pallidus; Muscimol; Oxazoles; Rats | 1979 |
[Effects of muscimol and diazepam: a comparative study on behavioral inhibiton induced by novelty, punishment, and nonreward (author's transl)].
Topics: Animals; Behavior, Animal; Conditioning, Operant; Diazepam; Environment; Feeding Behavior; Male; Muscimol; Oxazoles; Punishment; Rats; Reward | 1979 |
Electroencephalographic and behavioral effects of a GABA agonist (muscimol) on photosensitive epilepsy in the baboon, papio papio.
Topics: Animals; Anticonvulsants; Drug Evaluation, Preclinical; Electroencephalography; Haplorhini; Muscimol; Oxazoles; Papio; Photic Stimulation; Seizures | 1979 |
Modification of the behavioural effects of amphetamine by a GABA agonist in a primate species.
Topics: Animals; Behavior, Animal; Callitrichinae; Dextroamphetamine; Dopamine; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Haplorhini; Humans; Male; Motor Activity; Muscimol; Oxazoles; Stereotyped Behavior | 1979 |
[Ventrobulbular hypotensive action of muscimol].
Topics: Animals; Bradycardia; Brain Stem; Cats; Female; Hypotension; Male; Muscimol; Oxazoles | 1978 |
Stimulation of prolactin and growth hormone secretion by muscimol, a gamma-aminobutyric acid agonist.
Topics: Adult; Aged; Chronic Disease; Female; gamma-Aminobutyric Acid; Growth Hormone; Humans; Huntington Disease; Kinetics; Male; Middle Aged; Muscimol; Oxazoles; Prolactin; Schizophrenia | 1978 |
The effect of muscimol on prolactin secretion in male rats.
Topics: Animals; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Haloperidol; Male; Methyltyrosines; Muscimol; Oxazoles; Premedication; Prolactin; Rats; Receptors, Neurotransmitter | 1978 |
GABA agonists and potential antagonists related to muscimol.
Topics: Animals; Dose-Response Relationship, Drug; Functional Laterality; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Male; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter; Stereotyped Behavior; Substantia Nigra | 1979 |
Effects of diazepam and muscimol on GABA-mediated neurotransmission: interactions with inosine and nicotinamide.
Topics: Animals; Corpus Striatum; Diazepam; Drug Interactions; Female; gamma-Aminobutyric Acid; Globus Pallidus; Inosine; Muscimol; Niacinamide; Oxazoles; Rats; Synaptic Transmission; Time Factors | 1979 |
High-affinity binding of [3H]muscimol to subcellular particles of a neurone-enriched culture of embryonic rat brain.
Topics: Animals; Brain; Brain Chemistry; Culture Techniques; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter; Subcellular Fractions | 1979 |
Anticonvulsant activity of muscimol against seizures induced by impairment of GABA-mediated neurotransmission.
Topics: Animals; Anticonvulsants; Bicuculline; gamma-Aminobutyric Acid; Isoniazid; Male; Muscimol; Oxazoles; Pentylenetetrazole; Picrotoxin; Rats; Seizures; Strychnine; Synaptic Transmission | 1979 |
Distribution and metabolism of muscimol in the brain and other tissues of the rat.
Topics: Aminooxyacetic Acid; Animals; Brain; Injections, Intravenous; Injections, Intraventricular; Male; Muscimol; Oxazoles; Pargyline; Proadifen; Rats; Time Factors; Tissue Distribution | 1979 |
Modifications of DOPAC levels in the striatum and olfactory tubercles of the rat after muscimol.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Corpus Striatum; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscimol; Olfactory Bulb; Oxazoles; Phenylacetates; Rats; Time Factors | 1979 |
Characterization of the binding of [3H]muscimol, a potent gamma-aminobutyric acid agonist, to rat brain synaptosomal membranes using a filtration assay.
Topics: Animals; Binding, Competitive; Brain; Cerebellum; gamma-Aminobutyric Acid; Kinetics; Muscimol; Oxazoles; Rats; Receptors, Drug; Synaptic Membranes; Tissue Distribution | 1979 |
Effects of the GABA receptor agonist muscimol on the turnover of brain dopamine and on the motor activity of rats.
Topics: Animals; Brain; Cell Nucleus; Dihydroxyphenylalanine; Dopamine; gamma-Aminobutyric Acid; Male; Motor Activity; Muscimol; Norepinephrine; Oxazoles; Rats | 1979 |
Characterization of [3H]muscimol binding to mouse brain membranes.
Topics: Animals; Binding, Competitive; Brain; Detergents; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Mice; Muscimol; Osmolar Concentration; Oxazoles; Receptors, Drug | 1979 |
Dihydromuscimol, thiomuscimol and related heterocyclic compounds as GABA analogues.
Topics: Animals; Brain; Cats; Cell Membrane; gamma-Aminobutyric Acid; Muscimol; Neurons; Oxazoles; Oxazolidinones; Rats; Receptors, Drug; Spinal Cord; Structure-Activity Relationship | 1979 |
Enhancement of the binding of 3H-diazepam to rat brain membranes in vitro by SQ 20009, A novel anxiolytic, gamma-aminobutyric acid (GABA) and muscimol.
Topics: Animals; Bicuculline; Brain; Diazepam; Etazolate; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Nicotinic Acids; Oxazoles; Picrotoxin; Rats; Stimulation, Chemical | 1979 |
Characteristics of muscimol accumulation in mouse brain after systemic administration.
Topics: Animals; Bicuculline; Brain; gamma-Aminobutyric Acid; History, 18th Century; Injections, Intravenous; Mice; Muscimol; Oxazoles; Phenobarbital; Time Factors | 1979 |
Evidence for two types of binding of 3H-gaba and 3H-muscimol in rat cerebral cortex and cerebellum.
Topics: Animals; Brain Stem; Cerebellum; Cerebral Cortex; Corpus Striatum; gamma-Aminobutyric Acid; Male; Muscimol; Organ Specificity; Oxazoles; Radioligand Assay; Rats; Receptors, Drug; Substrate Specificity; Synaptosomes | 1979 |
The GABA agonist THIP a muscimol analogue, does not interfere with the benzodiazepine binding site on rats cortical membranes.
Topics: Animals; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Imidazoles; In Vitro Techniques; Isonicotinic Acids; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Taurine | 1979 |
Turning behaviour induced by injection of muscimol or picrotoxin into the substantia nigra demonstrates dual GABA components.
Topics: Animals; gamma-Aminobutyric Acid; Male; Movement; Muscimol; Organ Specificity; Oxazoles; Picrotoxin; Rats; Substantia Nigra | 1979 |
Dual gamma-aminobutyric acid control of prolactin secretion in the rat.
Topics: Animals; Bicuculline; Female; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Methyltyrosines; Muscimol; Oxazoles; Picrotoxin; Pituitary Gland, Anterior; Prolactin; Rats | 1979 |
Increase in striatal acetylcholine levels by GABA mimetic drugs: lack of involvement of the nigro-striatal dopaminergic neurons.
Topics: Acetylcholine; Animals; Corpus Striatum; gamma-Aminobutyric Acid; Hydroxydopamines; Male; Muscimol; Oxazoles; Rats | 1979 |
Baclofen and muscimol: behavioural and neurochemical sequelae of unilateral intranigral administration and effects on 3H-GABA receptor binding.
Topics: Aminobutyrates; Animals; Baclofen; Behavior, Animal; Brain Chemistry; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Hydroxydopamines; Injections; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Substantia Nigra; Time Factors | 1979 |
Unpleasant side effects of muscimol.
Topics: Humans; Muscimol; Oxazoles; Schizophrenia | 1979 |
Central antihypertensive properties of muscimol and related gamma-aminobutyric acid agonists and the interaction of muscimol with baroreceptor reflexes.
Topics: Animals; Blood Pressure; Cats; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Heart Rate; Male; Muscimol; Oxazoles; Pressoreceptors; Reflex; Vasomotor System | 1979 |
Muscimol antagonism of morphine analgesia in rats.
Topics: Animals; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Muscimol; Oxazoles; Rats; Reaction Time; Time Factors | 1979 |
THIP and isoguvacine are partial agonists of GABA-stimulated benzodiazepine receptor binding.
Topics: Animals; Benzodiazepines; Cerebral Cortex; Drug Synergism; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Muscimol; Oxazoles; Rats; Receptors, Drug | 1979 |
The effect of muscimol on hippocampal pyramidal cells.
Topics: Action Potentials; Animals; Bicuculline; Electric Stimulation; Hippocampus; Humans; In Vitro Techniques; Male; Muscimol; Oxazoles; Pyramidal Tracts; Rabbits; Strychnine; Synapses; Time Factors | 1979 |
[3H]Muscimol binding to rat cerebellar membranes.
Topics: Animals; Cell Membrane; Cerebellum; Female; gamma-Aminobutyric Acid; Kinetics; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Tritium | 1979 |
More muscimol binding sites than GABA binding sites in a particulate fraction of rat brain.
Topics: Animals; Binding Sites; Brain; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Muscimol; Oxazoles; Rats | 1979 |
Comparison of the "specific" binding of [3H]GABA and [3H]muscimol to a particulate fraction of rat brain.
Topics: Animals; Brain; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Muscimol; Nerve Tissue Proteins; Oxazoles; Protein Binding; Rats; Subcellular Fractions | 1979 |
Conformational analysis of muscimol, a GABA agonist.
Topics: Bicuculline; Binding Sites; gamma-Aminobutyric Acid; Isoxazoles; Models, Molecular; Molecular Conformation; Muscimol; Oxazoles; Quantum Theory | 1979 |
GABA and hypothalamic feeding systems. I. Topographic analysis of the effects of microinjections of muscimol.
Topics: Animals; Bicuculline; Brain Mapping; Digestive System; Eating; Female; gamma-Aminobutyric Acid; Gastric Juice; Hypothalamus; Hypothalamus, Middle; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats | 1979 |
Muscimol uptake, release and binding in rat brain slices.
Topics: Alanine; Animals; Binding, Competitive; Biological Transport; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Muscimol; Oxazoles; Rats; Receptors, Drug | 1978 |
Does uptake limit the actions of GABA agonists in vivo? Experiments with muscimol, isoguvacine and THIP in cat spinal cord.
Topics: Aminobutyrates; Animals; Biological Transport; Cats; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Muscimol; Neurons; Nipecotic Acids; Oxazoles; Spinal Cord | 1978 |
Recent advances in the morphological localization of gamma-aminobutyric acid receptors in the cerebellum by means of [3H]muscimol.
Topics: Animals; Brain; Cerebellar Nuclei; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Oxazoles; Purkinje Cells; Rats | 1979 |
Contralateral turning evoked by the intranigral microinjection of muscimol and other GABA agonists.
Topics: Animals; Behavior; Caudate Nucleus; Dopamine Antagonists; Dose-Response Relationship, Drug; Ethanolamines; Female; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Imidazoles; Muscimol; Oxazoles; Picrotoxin; Putamen; Rats; Stereotyped Behavior; Substantia Nigra | 1978 |
Striatal dopamine release and contraversive rotation elicited by intranigrally applied muscimol.
Topics: Animals; Behavior, Animal; Dopamine; Functional Laterality; Homovanillic Acid; Movement; Muscimol; Oxazoles; Substantia Nigra | 1978 |
A comparative study of the effects of muscimol and diazepam on the recall of noxious events.
Topics: Animals; Avoidance Learning; Diazepam; Dissociative Disorders; gamma-Aminobutyric Acid; Humans; Male; Memory; Mental Recall; Muscimol; Oxazoles; Rats | 1979 |
Modulatory effects of baclofen muscimol and GABA on interspecific aggressive behaviour in the rat.
Topics: Aggression; Aminobutyrates; Animals; Baclofen; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Olfactory Bulb; Oxazoles; Rats | 1978 |
Neuropharmacological spectrum of muscimol.
Topics: Animals; Anticonvulsants; Catalepsy; Drug Interactions; gamma-Aminobutyric Acid; Humans; Male; Mice; Motor Activity; Muscimol; Muscle Relaxants, Central; Nervous System; Oxazoles; Receptors, Drug | 1979 |
Behavioral differences induced by muscimol selectively injected into pars compacta and pars reticulata of Substantia nigra.
Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; Drug Interactions; Humans; Injections; Male; Muscimol; Oxazoles; Rats; Stereotyped Behavior; Substantia Nigra; Time Factors | 1979 |
Effects of intracerebral injection with muscimol on locomotor activity and catalepsy in rats.
Topics: Animals; Catalepsy; Humans; Injections, Intraventricular; Locomotion; Male; Muscimol; Oxazoles; Rats | 1979 |
Response of dopamine neurons in substantia nigra to muscimol.
Topics: Animals; Bicuculline; Dopamine; Dose-Response Relationship, Drug; Evoked Potentials; gamma-Aminobutyric Acid; Male; Muscimol; Neurons; Oxazoles; Picrotoxin; Rats; Substantia Nigra | 1978 |
Homotaurine and muscimol mimic taurine and GABA effects on muscle tone and temperature regulation.
Topics: Amino Acids; Animals; Body Temperature Regulation; Electroencephalography; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Injections, Intraventricular; Male; Muscimol; Muscle Tonus; Oxazoles; Rabbits; Taurine | 1978 |
Reductions in blood pressure, heart rate and renal sympathetic nerve discharge in cats after the central administration of muscimol, a GABA agonist.
Topics: Animals; Bicuculline; Blood Pressure; Cats; Drug Interactions; Heart Rate; Kidney; Muscimol; Norepinephrine; Oxazoles; Pressoreceptors; Sympathetic Nervous System | 1978 |
Photoaffinity labeling of the GABAA receptor with [3H]muscimol.
Topics: Affinity Labels; Animals; Baclofen; Diazepam; Glutamates; Glutamic Acid; Kinetics; Male; Molecular Weight; Muscimol; Oxazoles; Photochemistry; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spectrophotometry, Ultraviolet | 1985 |
Benzodiazepines enhance the muscimol-dependent activation of phospholipase A2 in glioma C6 cells.
Topics: Animals; Anti-Anxiety Agents; Arachidonic Acid; Arachidonic Acids; Cell Line; Chromatography, High Pressure Liquid; Diazepam; Drug Interactions; Enzyme Activation; Glioma; Muscimol; Neuroglia; Oxazoles; Phospholipases; Phospholipases A; Phospholipases A2; Prostaglandin D2; Prostaglandins D; Rats; Receptors, GABA-A | 1985 |
Excitatory amino acids: studies on the biochemical and chemical stability of ibotenic acid and related compounds.
Topics: Animals; Brain; Chemical Phenomena; Chemistry; Chromatography, High Pressure Liquid; Decarboxylation; Glutamates; Glutamic Acid; Hot Temperature; Hydrogen-Ion Concentration; Ibotenic Acid; Isoxazoles; Liver; Mice; Muscimol; Oxazoles; Pregnancy Proteins | 1985 |
Modification of saccadic eye movements by GABA-related substances. I. Effect of muscimol and bicuculline in monkey superior colliculus.
Topics: Animals; Bicuculline; Eye Movements; gamma-Aminobutyric Acid; Macaca mulatta; Muscimol; Oxazoles; Saccades; Superior Colliculi; Synaptic Transmission; Visual Fields | 1985 |
Modification of saccadic eye movements by GABA-related substances. II. Effects of muscimol in monkey substantia nigra pars reticulata.
Topics: Animals; Brain Mapping; Eye Movements; gamma-Aminobutyric Acid; Macaca mulatta; Muscimol; Neural Pathways; Oxazoles; Saccades; Substantia Nigra; Superior Colliculi; Synaptic Transmission | 1985 |
Synthesis and pharmacological evaluation of cis-2,3,3a,4,5,6,7,7a-octahydro-3-oxoisoxazolo[5,4-c]pyridine: a structural analogue of the GABA agonist THIP.
Topics: Animals; Anticonvulsants; Cerebellum; Electrophysiology; Female; Isoxazoles; Male; Mice; Muscimol; Oxazoles; Rats; Receptors, GABA-A | 1985 |
Subsensitivity to muscimol-induced catalepsy after long-term administration of phenytoin in rats.
Topics: Animals; Bicuculline; Catalepsy; Drug Interactions; Humans; Male; Muscimol; Oxazoles; Phenytoin; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Effect of THIP and SL 76002, two clinically experimented GABA-mimetic compounds, on anterior pituitary GABA receptors and prolactin secretion in the rat.
Topics: Animals; Anticonvulsants; Bicuculline; Binding, Competitive; Female; gamma-Aminobutyric Acid; Haloperidol; Isoxazoles; Kinetics; Male; Muscimol; Ovariectomy; Oxazoles; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Effect of GABAergic drugs in the behavioral 'despair' test in rats.
Topics: Acetates; Aminooxyacetic Acid; Animals; Baclofen; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Muscimol; Oxazoles; Picrotoxin; Rats | 1986 |
Central action of gamma-aminobutyric acid ligands to alter basal water and electrolyte absorption in the rat ileum.
Topics: Animals; Bicuculline; Biological Transport; Body Fluids; Cholinergic Fibers; Electrolytes; GABA Antagonists; gamma-Aminobutyric Acid; Ileum; Intestinal Absorption; Ligands; Male; Muscimol; Oxazoles; Parasympathetic Nervous System; Rats; Rats, Inbred Strains; Receptors, Cholinergic | 1985 |
Deficits in manipulative behaviors induced by local injections of muscimol in the first somatosensory cortex of the conscious monkey.
Topics: Animals; Brain Diseases; Brain Mapping; Female; gamma-Aminobutyric Acid; Hand; Macaca; Motor Skills; Muscimol; Oxazoles; Somatosensory Cortex | 1985 |
Rigidity and catalepsy after injections of muscimol into the ventromedial thalamic nucleus: an electromyographic study in the rat.
Topics: Animals; Bicuculline; Catalepsy; Electromyography; Humans; Male; Muscimol; Muscle Rigidity; Oxazoles; Rats; Rats, Inbred Strains; Restraint, Physical; Thalamic Nuclei | 1985 |
Characteristics and distribution of muscimol binding sites in cat visual cortex.
Topics: Animals; Autoradiography; Cats; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Muscimol; Oxazoles; Receptors, GABA-A; Tissue Distribution; Tritium; Visual Cortex | 1984 |
Ontogenesis of muscimol binding sites in cat visual cortex.
Topics: Animals; Binding Sites; Cats; gamma-Aminobutyric Acid; Kinetics; Muscimol; Neural Inhibition; Oxazoles; Receptors, GABA-A; Visual Cortex | 1984 |
GABA agonist induced analgesia elicited from the lateral preoptic area in the rat.
Topics: Analgesia; Animals; Baclofen; Male; Muscimol; Oxazoles; Preoptic Area; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A | 1984 |
Single class of muscimol binding sites in the solubilized gamma-aminobutyrate-benzodiazepine receptor complex.
Topics: Animals; Brain; Brain Chemistry; Cattle; Cerebral Cortex; Chromatography, Gel; Flunitrazepam; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1984 |
In vitro effects of melatonin on [3H]muscimol binding in rat brain.
Topics: Animals; Brain; Buffers; Corpus Striatum; Frontal Lobe; Male; Melatonin; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes | 1984 |
Some barbiturates enhance the effect of muscimol on dopamine turnover in the rat retina.
Topics: Animals; Barbital; Barbiturates; Convulsants; Dopamine; Drug Synergism; GABA Antagonists; gamma-Aminobutyric Acid; Light; Male; Methyltyrosines; Muscimol; Oxazoles; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Retina; Sesterterpenes | 1980 |
Autoradiographic localization of binding sites for [3H]gamma-aminobutyrate, [3H]muscimol,(+)[3H]bicuculline methiodide and [3H] flunitrazepam in cultures of rat cerebellum and spinal cord.
Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Autoradiography; Bicuculline; Binding Sites; Cells, Cultured; Cerebellum; Female; Fetus; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Pregnancy; Rats; Receptors, Drug; Spinal Cord; Tritium | 1980 |
Binding and uptake of the GABA analogue, 3H-muscimol, in the retinas of goldfish and chicken.
Topics: Animals; Autoradiography; Chickens; gamma-Aminobutyric Acid; Goldfish; Muscimol; Neurons; Neurotransmitter Agents; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Retina | 1980 |
Inhibition by arylsulphatase A of Na-independent [3H]-GABA and [3H]-muscimol binding to bovine cerebellar synaptic membranes.
Topics: Animals; Brain; Cattle; Cerebellum; Cerebroside-Sulfatase; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Oxazoles; Sodium; Sulfatases; Synaptic Membranes | 1980 |
Effect of muscimol on glucose-stimulated somatostatin and insulin release from the isolated, perfused rat pancreas.
Topics: Animals; Glucose; In Vitro Techniques; Insulin; Male; Muscimol; Oxazoles; Pancreas; Perfusion; Rats; Somatostatin | 1981 |
Effect of single and repeated convulsions on glutamate decarboxylase (GAD) activity and [3H]muscimol binding in the rat brain.
Topics: Animals; Brain; Carboxy-Lyases; Electroshock; Glutamate Decarboxylase; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium | 1981 |
Effects of muscimol on the crayfish neuromuscular junction.
Topics: Animals; Astacoidea; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Kinetics; Membrane Potentials; Muscimol; Neuromuscular Junction; Oxazoles; Synapses | 1981 |
Serotonergic drugs, benzodiazepines and baclofen block muscimol-induced myoclonic jerks in a strain of mice.
Topics: 5-Hydroxytryptophan; Animals; Anti-Anxiety Agents; Baclofen; Benzodiazepines; Male; Mice; Muscimol; Myoclonus; Oxazoles; Piperazines; Pyrazines; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Serotonin; Serotonin | 1981 |
Anion-dependent modulation of [3H]muscimol binding and of GABA-stimulated [3H]flunitrazepam binding by picrotoxin and related CNS convulsants.
Topics: Animals; Anions; Anti-Anxiety Agents; Cerebral Cortex; Convulsants; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Receptors, Drug; Receptors, GABA-A; Strychnine; Tubocurarine | 1982 |
Relative disposition of the GABA agonists THIP and muscimol in the brain of the rat.
Topics: Animals; Brain; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Time Factors | 1982 |
Tofizopam affects binding of [3H]muscimol to gamma-amino-butyric acid receptors in rat and mouse brains.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Brain; Diazepam; Kinetics; Male; Mice; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter | 1982 |
Differential modulation of etazolate or pentobarbital enhanced [3H] muscimol binding by benzodiazepine agonists and inverse agonists.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Etazolate; Flumazenil; Flunitrazepam; Kinetics; Muscimol; Nicotinic Acids; Oxazoles; Pentobarbital; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Hypnotic action of benzodiazepines: a possible mechanism.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Hypnotics and Sedatives; Male; Mice; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Reflex; Sleep | 1984 |
[Differences in the mechanism of the antihypoxic action of benzodiazepine receptor agonists and muscimol].
Topics: Animals; Anti-Anxiety Agents; Diazepam; Drug Evaluation, Preclinical; gamma-Aminobutyric Acid; Hypoxia; Ligands; Mice; Muscimol; Oxazoles; Receptors, GABA-A | 1984 |
Reduction of [3H]muscimol binding sites in rat dorsal spinal cord after neonatal capsaicin treatment.
Topics: Animals; Animals, Newborn; Capsaicin; Fatty Acids, Unsaturated; Ganglia, Spinal; Muscimol; Neurons; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Sodium; Strychnine; Substance P | 1980 |
Muscimol injections in the nucleus raphé dorsalis block the antinociceptive effect of morphine in rats: apparent lack of 5-hydroxytryptamine involvement in muscimol's effect.
Topics: 5,7-Dihydroxytryptamine; Analgesics; Animals; Brain Chemistry; Hydroxyindoleacetic Acid; Injections; Male; Morphine; Muscimol; Oxazoles; Raphe Nuclei; Rats; Reaction Time; Serotonin; Time Factors | 1984 |
Plasma growth hormone and prolactin response to dopaminergic GABAmimetic and cholinergic stimulation in Huntington's disease.
Topics: Adult; Apomorphine; Arecoline; Dopamine; Female; gamma-Aminobutyric Acid; Growth Hormone; Humans; Huntington Disease; Male; Muscimol; Oxazoles; Prolactin | 1983 |
GABA receptors in bovine cerebral blood vessels: binding studies with [3H]muscimol.
Topics: Animals; Binding, Competitive; Cattle; Cerebral Arteries; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Pia Mater; Receptors, Neurotransmitter; Vasodilation | 1980 |
Effect of the GABA receptor agonist muscimol on regional cerebral blood flow in the rat.
Topics: Animals; Caudate Nucleus; Cerebellum; Cerebral Cortex; Cerebrovascular Circulation; Female; gamma-Aminobutyric Acid; Mesencephalon; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter; Thalamus | 1980 |
Autoradiographic localization of 3H-GABA and 3H-muscimol binding in rat cerebellar cultures.
Topics: Animals; Autoradiography; Binding Sites; Cerebellum; Culture Techniques; Dendrites; gamma-Aminobutyric Acid; Muscimol; Neurons; Oxazoles; Purkinje Cells; Rats; Receptors, Neurotransmitter | 1980 |
Substrate specificity of [3H]muscimol binding to a particulate fraction of a neuron-enriched culture of embryonic rat brain.
Topics: Animals; Binding, Competitive; Brain; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Kinetics; Muscimol; Neurons; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1980 |
Presence of a low molecular weight endogenous inhibitor on 3H-muscimol binding in synaptic membranes.
Topics: Animals; Brain Chemistry; GABA Antagonists; Molecular Weight; Muscimol; Neurons; Oxazoles; Polyethylene Glycols; Rats; Receptors, Neurotransmitter; Synaptic Membranes | 1980 |
Potentiation by intraventricular muscimol of the anticonflict effect of benzodiazepines.
Topics: Animals; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drinking; Eating; Fear; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter | 1980 |
Na+-independent binding of [3H]GABA and [3H]muscimol to a "microsomal" fraction, but not to a myelin fraction of rat brain; further evidence that glial elements do not possess GABA-receptors.
Topics: Animals; Brain; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Microscopy, Electron; Microsomes; Muscimol; Neuroglia; Oxazoles; Rats; Receptors, Neurotransmitter; Sodium; Tritium | 1980 |
Increase in striatal [3H]muscimol binding following intrastriatal injection of kainic acid: a denervation supersensitivity phenomenon.
Topics: Animals; Corpus Striatum; gamma-Aminobutyric Acid; Kainic Acid; Male; Microinjections; Muscimol; Muscle Denervation; Octoxynol; Oxazoles; Polyethylene Glycols; Pyrrolidines; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1980 |
Nigral-derived muscimol circling--ipsiversive, contraversive or controversial?
Topics: Animals; Behavior, Animal; Dopamine; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra | 1981 |
Development of [3H]muscimol binding to subcellular particles of a culture of mouse brain.
Topics: Animals; Axons; Brain; Cells, Cultured; Female; Mice; Microscopy, Phase-Contrast; Muscimol; Neurons; Oxazoles; Pregnancy; Receptors, Cell Surface; Receptors, GABA-A; Subcellular Fractions | 1980 |
GABA and muscimol inhibit the release of prolactin from dispersed rat anterior pituitary cells.
Topics: Animals; Bicuculline; Dopamine; Female; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Oxazoles; Picrotoxin; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1981 |
Heterogeneous depression of glucose utilization in the caudate nucleus by GABA agonists.
Topics: Animals; Autoradiography; Blood Glucose; Caudate Nucleus; Isoxazoles; Male; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1981 |
The insensitivity of developing benzodiazepine receptors to chronic treatment with diazepam, GABA and muscimol in brain cell cultures.
Topics: Animals; Brain; Cell Membrane; Cells, Cultured; Diazepam; Female; Fetus; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Muscimol; Oxazoles; Pregnancy; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter | 1981 |
Localized binding of [3H]muscimol to synapses in chicken retina.
Topics: Animals; Autoradiography; Binding, Competitive; Chickens; gamma-Aminobutyric Acid; Microscopy, Electron; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Retina; Synapses | 1981 |
GABA and muscimol open ion channels of different lifetimes on cultured mouse spinal cord cells.
Topics: Animals; Cells, Cultured; Electric Conductivity; Embryo, Mammalian; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Membrane Potentials; Mice; Muscimol; Neurons; Oxazoles; Spinal Cord | 1981 |
Involvement of dopamine in circling responses to muscimol depends on intranigral site of injection.
Topics: Animals; Humans; Hydroxydopamines; Male; Motor Activity; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Stereotyped Behavior; Substantia Nigra | 1981 |
GABAergic synapses in the goldfish retina: an autoradiographic study of 3H-muscimol and 3H-GABA binding.
Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; Goldfish; Muscimol; Neurons; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Muscarinic; Retina; Synapses; Visual Pathways | 1981 |
Na+ independent binding of [3H] muscimol to a membrane fraction of the brains of normal and dwarf mice.
Topics: Animals; Brain; Cell Membrane; Dwarfism, Pituitary; Kinetics; Mice; Muscimol; Organ Size; Oxazoles; Receptors, Drug; Receptors, GABA-A; Sodium | 1981 |
The effects of muscimol and picrotoxin injections into the cat substantia nigra.
Topics: Animals; Behavior, Animal; Cats; Female; Hindlimb; Humans; Injections; Male; Muscimol; Oxazoles; Picrotoxin; Receptors, Cell Surface; Receptors, GABA-A; Stereotyped Behavior; Substantia Nigra | 1981 |
3H-muscimol binding in synaptosomal fractions from bovine and developing rabbit retinas.
Topics: Animals; Binding, Competitive; Cattle; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rabbits; Receptors, Cell Surface; Receptors, GABA-A; Retina; Synaptic Transmission; Synaptosomes | 1981 |
Quantitative autoradiography of [3H]muscimol binding in rat brain.
Topics: Animals; Autoradiography; Brain; Kainic Acid; Kinetics; Muscimol; Oxazoles; Rats; Receptors, Drug; Receptors, GABA-A; Tritium | 1981 |
Muscimol induces gastric acid secretion after central administration.
Topics: Animals; Gastric Acid; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Secretory Rate | 1981 |
Glutamic acid decarboxylase and gamma-aminobutyric acid in Huntington's disease fibroblasts and other cultured cells, determined by a [3H]muscimol radioreceptor assay.
Topics: Carboxy-Lyases; Cells, Cultured; Fibroblasts; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Humans; Huntington Disease; Kinetics; Muscimol; Oxazoles; Radioligand Assay; Receptors, Cell Surface; Receptors, GABA-A; Skin | 1981 |
Chronic benzodiazepine treatment increases [3H]muscimol binding in mouse brain.
Topics: Animals; Benzodiazepinones; Brain; Cerebellum; Chlordiazepoxide; Clonazepam; In Vitro Techniques; Mice; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A | 1982 |
Acute and chronic effects of pentobarbital in relation to postsynaptic GABA receptors: a study with muscimol.
Topics: Animals; Brain; Drug Tolerance; gamma-Aminobutyric Acid; Humans; Male; Mice; Mice, Inbred ICR; Muscimol; Oxazoles; Pentobarbital; Receptors, Cell Surface; Receptors, GABA-A; Sleep; Substance Withdrawal Syndrome; Synaptic Membranes | 1982 |
Stimulatory and protective effects of benzodiazepines on GABA receptors labeled with [3H]muscimol.
Topics: Animals; Benzodiazepines; Hot Temperature; In Vitro Techniques; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium | 1982 |
Binding of [3H]gamma-aminobutyric acid and [3H]muscimol in purified rat brain synaptic plasma membranes and the effects of bicuculline.
Topics: Animals; Bicuculline; Binding, Competitive; Brain; gamma-Aminobutyric Acid; Male; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Membranes; Tritium | 1982 |
Single channel currents activated by gamma-aminobutyric acid, muscimol, and (-)-pentobarbital in cultured mouse spinal neurons.
Topics: Animals; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Mice; Muscimol; Neurons; Oxazoles; Pentobarbital; Spinal Cord | 1982 |
Effect of ethanol and ethanol withdrawal on 3H-muscimol binding and behaviour in the rat: a pilot study.
Topics: Animals; Behavior, Animal; Brain; Ethanol; Humans; Male; Muscimol; Oxazoles; Pilot Projects; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substance Withdrawal Syndrome | 1981 |
(3H)-muscimol, (3H)-nipecotic acid and (3H)-isoguvacine as autoradiographic markers for GABA neurotransmission.
Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; Goldfish; Guinea Pigs; Isonicotinic Acids; Muscimol; Neuroglia; Neurons; Nipecotic Acids; Oxazoles; Rabbits; Receptors, Cell Surface; Receptors, GABA-A; Retina; Synaptic Transmission | 1982 |
Glycine antagonists structurally related to muscimol, THIP, or isoguvacine.
Topics: Animals; Cats; gamma-Aminobutyric Acid; Glycine; Interneurons; Isonicotinic Acids; Isoxazoles; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Glycine; Spinal Cord; Structure-Activity Relationship | 1982 |
High specific binding of [3H]GABA and [3H]muscimol to membranes from dendrodendritic synaptosomes of the rat olfactory bulb.
Topics: Animals; Dendrites; gamma-Aminobutyric Acid; Male; Muscimol; Olfactory Bulb; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Subcellular Fractions; Synaptic Membranes; Synaptosomes | 1982 |
Muscimol and some aza analogues: molecular orbital calculations relating to their potency as GABA mimetics.
Topics: Binding Sites; Chemical Phenomena; Chemistry; Electrons; gamma-Aminobutyric Acid; Humans; Molecular Conformation; Muscimol; Oxazoles; Pyrazoles; Pyrazolones; Receptors, Neurotransmitter; Rotation; Structure-Activity Relationship; Triazoles | 1982 |
Effects of GABAergic agonists and antagonists on various ethanol-induced behavioral changes.
Topics: Animals; Behavior, Animal; Bicuculline; Body Temperature Regulation; Dose-Response Relationship, Drug; Ethanol; Female; Motor Activity; Muridae; Muscimol; Oxazoles; Pentylenetetrazole; Picrotoxin; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Sleep Stages; Strychnine | 1982 |
Intra-raphe muscimol induced hyperactivity depends on ascending serotonin projections.
Topics: Animals; Bicuculline; Brain Stem; Chlordiazepoxide; Dose-Response Relationship, Drug; Male; Mesencephalon; Motor Activity; Muscimol; Oxazoles; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Serotonin; Tegmentum Mesencephali | 1982 |
Comparison of centrifugation and filtration assays of ligand binding: do multiple GABA receptive sites exist?
Topics: Animals; Brain; Cattle; Centrifugation; Cerebral Cortex; Filtration; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Membranes | 1982 |
Changes in [3H]muscimol binding in substantia nigra, entopeduncular nucleus, globus pallidus, and thalamus after striatal lesions as demonstrated by quantitative receptor autoradiography.
Topics: Animals; Autoradiography; Corpus Striatum; gamma-Aminobutyric Acid; Globus Pallidus; Kainic Acid; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Substantia Nigra; Thalamus | 1983 |
Bicuculline insensitive effects of baclofen.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Bicuculline; Corpus Striatum; gamma-Aminobutyric Acid; Male; Motor Activity; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter | 1983 |
Motor and postural effects of kainic acid or GABA agonist and antagonist injection into the cerebellar nucleus fastigii.
Topics: Animals; Cerebellar Nuclei; Kainic Acid; Motor Skills; Muscimol; Muscle Contraction; Oxazoles; Picrotoxin; Posture; Pyrrolidines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission | 1983 |
Anisatin modulation of temperature-dependent inhibition [3H]muscimol binding by chloride ion.
Topics: Animals; Anions; Brain; Chlorides; Kinetics; Lactones; Male; Muscimol; Oxazoles; Plants, Toxic; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Sesquiterpenes; Spiro Compounds; Synaptic Membranes; Temperature | 1983 |
Modulation of [3H]muscimol binding in rat cerebellar and cerebral cortical membranes by picrotoxin, pentobarbitone, and etomidate.
Topics: Animals; Cell Membrane; Cerebellar Cortex; Cerebral Cortex; Etomidate; Imidazoles; Kinetics; Male; Muscimol; Organ Specificity; Oxazoles; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
[3H]muscimol binding site on purified benzodiazepine receptor.
Topics: Animals; Binding Sites; Brain; Flunitrazepam; gamma-Aminobutyric Acid; Molecular Weight; Muscimol; Oxazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Diazepam stimulates the binding of GABA and muscimol but not THIP to rat brain membranes.
Topics: Analgesics; Animals; Brain; Diazepam; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Decreased high-affinity binding of [3H]muscimol to cerebral synaptic membranes of scrapie-infected mice.
Topics: Animals; Brain; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Mice, Inbred C57BL; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Scrapie; Sheep; Synaptic Membranes | 1984 |
Characterization of susceptibility to audiogenic seizures in ethanol-dependent rats after microinjection of gamma-aminobutyric acid (GABA) agonists into the inferior colliculus, substantia nigra or medial septum.
Topics: Acoustic Stimulation; Animals; Anticonvulsants; Bicuculline; Ethanol; GABA Antagonists; Humans; Inferior Colliculi; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures; Septum Pellucidum; Substance Withdrawal Syndrome; Substantia Nigra | 1983 |
Antihypertensive effect of the GABA receptor agonist muscimol in spontaneously hypertensive rats. Role of the sympathoadrenal axis.
Topics: Adrenal Glands; Animals; Atropine; Blood Pressure; Catecholamines; Clonidine; Efferent Pathways; Heart Rate; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Splanchnic Nerves; Sympathectomy, Chemical; Sympathetic Nervous System; Vagotomy | 1984 |
Synergistic inhibition of [3H]muscimol binding to calf-brain synaptic membranes in the presence of L-homocysteine and pyridoxal 5'-phosphate. A possible mechanism for homocysteine-induced seizures.
Topics: Animals; Binding, Competitive; Brain; Cattle; Drug Synergism; Homocysteine; In Vitro Techniques; Kinetics; Models, Chemical; Muscimol; Oxazoles; Pyridoxal Phosphate; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Synaptic Membranes | 1983 |
Intranigral muscimol suppresses ethanol withdrawal seizures.
Topics: Acoustic Stimulation; Alcoholism; Animals; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Substance Withdrawal Syndrome; Substantia Nigra | 1984 |
In vivo release of [3H]GABA in cat caudate nucleus and substantia nigra. II. Involvement of different thalamic nuclei in the bilateral changes induced by a nigral application of muscimol.
Topics: Animals; Cats; Caudate Nucleus; Dominance, Cerebral; Female; gamma-Aminobutyric Acid; Male; Muscimol; Neural Pathways; Neurons; Oxazoles; Substantia Nigra; Synaptic Transmission; Thalamic Nuclei | 1984 |
Effects of valproic acid on spinal reflexes and [3H]muscimol and [3H]diazepam binding in brain membranes in rats.
Topics: Animals; Brain; Diazepam; Male; Membranes; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Reflex; Spinal Cord; Valproic Acid | 1983 |
Diazepam antagonizes GABA- and muscimol-induced changes of acetylcholine release in slices of guinea-pig cerebral cortex.
Topics: Acetylcholine; Animals; Benzodiazepinones; Cerebral Cortex; Diazepam; Flumazenil; GABA Antagonists; Guinea Pigs; In Vitro Techniques; Muscimol; Oxazoles | 1983 |
Depolarizing responses to glycine, beta-alanine and muscimol in isolated optic nerve and cuneate nucleus.
Topics: Alanine; Animals; beta-Alanine; Bicuculline; Dose-Response Relationship, Drug; Glycine; Male; Medulla Oblongata; Muscimol; Optic Nerve; Oxazoles; Picrotoxin; Rats; Rats, Inbred Strains; Strychnine; Time Factors | 1983 |
Behavioural responsiveness to muscimol and apomorphine 2 months after prolonged treatment with estradiol in rats.
Topics: Animals; Apomorphine; Behavior, Animal; Castration; Estradiol; Female; Humans; Motor Activity; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Stereotyped Behavior | 1984 |
[Influence of the GABAergic system on eating behavior induced by the tail pinching technic in rats].
Topics: Animals; Energy Intake; Feeding Behavior; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Rats, Inbred Strains; Stress, Psychological; Valproic Acid | 1981 |
Autoradiographic studies of [3H]-glycine, [3H]-GABA, and [3H]-muscimol uptake in the mudpuppy retina.
Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Microscopy, Electron; Muscimol; Necturus; Oxazoles; Retina; Tritium | 1984 |
[Increased 3H-muscimol binding in post-mortem brains of chronic schizophrenics].
Topics: Adult; Aged; Binding Sites; Chronic Disease; Female; Frontal Lobe; Glutamate Decarboxylase; Humans; Male; Middle Aged; Muscimol; Oxazoles; Putamen; Schizophrenia | 1984 |
Synergistic anticonvulsant effects of a GABA agonist and glycine.
Topics: 3-Mercaptopropionic Acid; Animals; Anticonvulsants; Drug Synergism; gamma-Aminobutyric Acid; Glycine; Male; Mice; Muscimol; Oxazoles; Seizures | 1984 |
Feeding induced by injections of muscimol into the substantia nigra of rats: unaffected by haloperidol but abolished by large lesions of the superior colliculus.
Topics: Animals; Brain Mapping; Corpus Striatum; Dopamine; Feeding Behavior; gamma-Aminobutyric Acid; Haloperidol; Male; Muscimol; Neural Pathways; Oxazoles; Rats; Substantia Nigra; Superior Colliculi | 1984 |
GABAergic agents in the medial septal nucleus affect hippocampal theta rhythm and acetylcholine utilization.
Topics: Acetylcholine; Animals; Bicuculline; gamma-Aminobutyric Acid; Hippocampus; Male; Muscimol; Neural Pathways; Oxazoles; Rats; Rats, Inbred Strains; Septal Nuclei; Theta Rhythm | 1984 |
GABA agonists inhibit the vasopressin-dependent pressor effects of central angiotensin II.
Topics: Angiotensin II; Animals; Arginine Vasopressin; Blood Pressure; Brain; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Sympathetic Nervous System | 1984 |
Blockade of bicuculline-induced pressor and tachycardic responses by forebrain administration of muscimol.
Topics: Animals; Bicuculline; Blood Pressure; Cats; Female; Heart Rate; Injections, Intraventricular; Male; Muscimol; Oxazoles | 1984 |
Investigation of the effects of muscimol on different components of [3H]propyl beta-carboline-3-carboxylate binding to rat hippocampal and cerebellar membranes.
Topics: Animals; Binding Sites; Carbolines; Cell Membrane; Cerebellum; Hippocampus; Indoles; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains | 1984 |
Effects of intrathecally administered THIP, baclofen and muscimol on nociceptive threshold.
Topics: Animals; Baclofen; Injections, Spinal; Isoxazoles; Male; Muscimol; Muscle Hypotonia; Nociceptors; Oxazoles; Rats; Rats, Inbred Strains; Reaction Time; Sensory Thresholds | 1984 |
Zinc deficiency and anorexia in rats: the effect of central administration of norepinephrine, muscimol and bromerogocryptine.
Topics: Animals; Anorexia; Bromocriptine; Dose-Response Relationship, Drug; Drug Resistance; Eating; Feeding and Eating Disorders; Humans; Male; Muscimol; Norepinephrine; Oxazoles; Rats; Rats, Inbred Strains; Zinc | 1984 |
In vivo release of [3H]GABA in cat caudate nucleus and substantia nigra. I. Bilateral changes induced by a unilateral nigral application of muscimol.
Topics: Animals; Brain Mapping; Cats; Caudate Nucleus; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Substantia Nigra | 1983 |
Neuronal subpopulations in cat retina which accumulate the GABA agonist, (3H)muscimol: a combined Golgi and autoradiographic study.
Topics: Animals; Autoradiography; Cats; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Muscimol; Oxazoles; Retina | 1983 |
Unilateral injection of GABA agonists in the superior colliculus: asymmetry to tactile stimulation.
Topics: Analgesics; Animals; Baclofen; Functional Laterality; gamma-Aminobutyric Acid; Isoxazoles; Motor Activity; Muscimol; Oxazoles; Physical Stimulation; Rats; Rats, Inbred Strains; Superior Colliculi; Touch | 1983 |
Muscimol inhibits ADH release induced by hypertonic sodium chloride in rats.
Topics: Animals; Bicuculline; Dose-Response Relationship, Drug; Male; Muscimol; Osmolar Concentration; Oxazoles; Radioimmunoassay; Rats; Rats, Inbred Strains; Sodium Chloride; Vasopressins | 1983 |
Reaction of muscimol with 4-aminobutyrate aminotransferase.
Topics: 4-Aminobutyrate Transaminase; Animals; Brain; Kinetics; Liver; Muscimol; Ornithine-Oxo-Acid Transaminase; Oxazoles; Rabbits; Spectrophotometry | 1983 |
Effects of nigral application of muscimol on release of [3H] gamma-aminobutyrate and on multiunit activity in various cat thalamic nuclei.
Topics: Animals; Cats; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Substantia Nigra; Thalamic Nuclei; Tritium | 1983 |
Monoamine involvement in the overeating caused by muscimol injection in the rat nucleus raphe dorsalis and the effects of d-fenfluramine and d-amphetamine.
Topics: 5,7-Dihydroxytryptamine; Animals; Biogenic Amines; Dextroamphetamine; Feeding Behavior; Fenfluramine; Food Deprivation; Injections; Male; Muscimol; Oxazoles; Penfluridol; Phenoxybenzamine; Raphe Nuclei; Rats | 1983 |
GABA-mediated inhibition of breathing in the late gestation sheep fetus.
Topics: Animals; Apnea; Female; Fetal Hypoxia; Fetus; gamma-Aminobutyric Acid; Gestational Age; Muscimol; Oxazoles; Picrotoxin; Pregnancy; Respiration; Sheep | 1983 |
[A new simplified method for the synthesis of muscimol (5-aminomethyl-3-hydroxyisoxazole)].
Topics: Muscimol; Oxazoles | 1983 |
Evidence that the nigrotegmental GABAergic projection mediates stereotypy induced by apomorphine and intranigral muscimol.
Topics: Animals; Apomorphine; Corpus Striatum; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Neural Pathways; Oxazoles; Pons; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substantia Nigra; Tegmentum Mesencephali | 1983 |
Disinhibition of muricide and irritability by intraseptal muscimol.
Topics: Aggression; Animals; Brain; Catheterization; Dose-Response Relationship, Drug; Feeding Behavior; Humans; Male; Metergoline; Muscimol; Oxazoles; Quipazine; Rats; Semicarbazides | 1983 |
Extrastriatal circuits activated by intrastriatal muscimol: a [14C]2-deoxyglucose investigation.
Topics: Animals; Brain; Brain Mapping; Corpus Striatum; gamma-Aminobutyric Acid; Glucose; Male; Muscimol; Neural Pathways; Oxazoles; Rats; Rats, Inbred Strains | 1984 |
Differential effects of baclofen, gamma-hydroxybutyric acid and muscimol on the protective action of phenobarbital and diphenylhydantoin against maximal electroshock-induced seizures in mice.
Topics: Animals; Anticonvulsants; Baclofen; Drug Interactions; Electroshock; gamma-Aminobutyric Acid; Hydroxybutyrates; Injections, Intraventricular; Male; Mice; Muscimol; Oxazoles; Phenobarbital; Phenytoin; Sodium Oxybate | 1984 |
Nigral muscimol infusions facilitate the development of seizures in immature rats.
Topics: Age Factors; Animals; Flurothyl; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rats; Seizures; Substantia Nigra | 1984 |
Muscimol-scopolamine interactions in the rat brain: a study with 2-deoxy-D-[1-14C]glucose.
Topics: Animals; Brain; Deoxyglucose; gamma-Aminobutyric Acid; Glucose; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Scopolamine | 1984 |
Circling behavior induced by intranigral injections of GABA and muscimol in rats.
Topics: Animals; Atropine; Behavior; Bicuculline; Brain Chemistry; Female; gamma-Aminobutyric Acid; Haloperidol; Humans; Injections; Muscimol; Oxazoles; Rats; Stereotyped Behavior; Strychnine; Substantia Nigra; Time Factors | 1980 |
Sodium di-n-propylacetate (valproate) potentiates responses to GABA and muscimol on single central neurones.
Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Evoked Potentials; gamma-Aminobutyric Acid; Medulla Oblongata; Muscimol; Neurons; Oxazoles; Rats; Reticular Formation; Valproic Acid | 1980 |
Effects of sodium n-dipropylacetate, muscimol hydrobromide and (R,S) nipecotic acid amide on isolation-induced aggressive behavior in mice.
Topics: Aggression; Animals; gamma-Aminobutyric Acid; Humans; Male; Mice; Motor Activity; Muscimol; Nipecotic Acids; Oxazoles; Social Isolation; Time Factors; Valproic Acid | 1980 |
Modulatory interactions between norepinephrine and taurine, beta-alanine, gamma-aminobutyric acid and muscimol, applied iontophoretically to cerebellar Purkinje cells.
Topics: Alanine; Animals; beta-Alanine; Cerebellum; Female; gamma-Aminobutyric Acid; Iontophoresis; Muscimol; Nerve Endings; Norepinephrine; Oxazoles; Purkinje Cells; Rats; Taurine | 1981 |
Differential effects of IV and IP muscimol on central dopamine metabolism.
Topics: Animals; Brain; Dopamine; Injections, Intraperitoneal; Injections, Intravenous; Male; Muscimol; Oxazoles; Rats; Receptors, Dopamine | 1981 |
Effect of muscimol, a central GABA receptor agonist, on the catalepsy, striatal homovanillic acid increase, and analgesia induced by pilocarpine in rats.
Topics: Analgesics; Animals; Catalepsy; Corpus Striatum; Drug Interactions; Homovanillic Acid; Humans; Male; Muscimol; Oxazoles; Phenylacetates; Pilocarpine; Rats; Rats, Inbred Strains | 1981 |
A new method for the evaluation of benzodiazepines based on their ability to block muscimol-induced myoclonic jerks in mice.
Topics: Animals; Benzodiazepines; Diazepam; Drug Evaluation; Flunitrazepam; Male; Mice; Muscimol; Myoclonus; Oxazoles; Spinal Cord | 1981 |
[Protective effects of muscimol on acute brain ischemia in the rat (author's transl)].
Topics: Animals; Baclofen; gamma-Aminobutyric Acid; Ischemic Attack, Transient; Kinetics; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Structure-Activity Relationship | 1982 |
Oral behaviour induced by intranigral muscimol is unaffected by haloperidol but abolished by large lesions of superior colliculus.
Topics: Animals; Behavior, Animal; Brain; Haloperidol; Humans; Injections; Male; Muscimol; Oxazoles; Rats; Stereotyped Behavior; Substantia Nigra; Superior Colliculi | 1982 |
Baclofen blocks postsynaptic inhibition but not the effect of muscimol in the olfactory cortex.
Topics: Animals; Baclofen; Cerebral Cortex; Drug Interactions; Electric Stimulation; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscimol; Neural Conduction; Neural Inhibition; Olfactory Pathways; Oxazoles; Synapses | 1983 |
The effects of the GABAergic agonist muscimol upon the relationship between local cerebral blood flow and glucose utilization.
Topics: Animals; Brain; Cerebrovascular Circulation; Deoxyglucose; Glucose; Kinetics; Muscimol; Organ Specificity; Oxazoles; Rats | 1983 |
Muscimol potentiation of acidic amino acid release from cerebellar synaptosomes is chloride dependent.
Topics: Animals; Aspartic Acid; Cerebellum; Chlorides; Drug Synergism; Ions; Kinetics; Male; Muscimol; Osmolar Concentration; Oxazoles; Potassium; Rats; Rats, Inbred Strains; Synaptosomes | 1983 |
Simultaneous modulation of hippocampal cholinergic activity and extinction by intraseptal muscimol.
Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Extinction, Psychological; Hippocampus; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Reaction Time; Reinforcement, Psychology | 1983 |
Effects of barbiturates and ethanol on muscimol-induced release of [3H]-D-aspartate from rodent cerebellum.
Topics: Animals; Aspartic Acid; Cerebellum; Ethanol; gamma-Aminobutyric Acid; Kinetics; Male; Muscimol; Oxazoles; Pentobarbital; Potassium; Rats; Rats, Inbred Strains; Synaptosomes; Tritium | 1983 |
GABAergic drugs, morphine and morphine tolerance: a study in relation to nociception and gastrointestinal transit in mice.
Topics: Aminooxyacetic Acid; Analgesia; Animals; Baclofen; Bicuculline; Cyclohexanecarboxylic Acids; Digestion; Digestive System; Digestive System Physiological Phenomena; Drug Tolerance; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Morphine; Muscimol; Naloxone; Nociceptors; Oxazoles; Picrotoxin | 1983 |
BehavioraL and biochemical changes caused by muscimol in mice withdrawN from haloperidol administration.
Topics: Animals; Behavior, Animal; Corpus Striatum; Dopamine; Haloperidol; Homovanillic Acid; Humans; Male; Mice; Mice, Inbred ICR; Motor Activity; Muscimol; Oxazoles; Substance Withdrawal Syndrome | 1982 |
The ventromedullary hypotensive effect of muscimol in the anaesthetized cat.
Topics: Anesthesia; Animals; Bicuculline; Blood Pressure; Brain Stem; Cats; Hypotension; Muscimol; Oxazoles; Stereotaxic Techniques | 1981 |
Antagonism of gamma-aminobutyric acid and muscimol by picrotoxin, bicuculline, strychnine, bemegride, leptazol, D-tubocurarine and theophylline in the isolated olfactory cortex.
Topics: Animals; Bicuculline; GABA Antagonists; Guinea Pigs; In Vitro Techniques; Muscimol; Olfactory Bulb; Oxazoles; Pentylenetetrazole; Picrotoxin; Strychnine; Theophylline; Tubocurarine | 1982 |
Periaqueductal gray matter involvement in the muscimol-induced decrease of morphine antinociception.
Topics: Analgesia; Animals; Cerebral Aqueduct; Male; Morphine; Muscimol; Oxazoles; Rats; Rats, Inbred Strains | 1982 |
Therapeutics of monomethylhydrazine intoxication.
Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Therapy, Combination; Male; Methylhydrazines; Mice; Mice, Inbred ICR; Monomethylhydrazine; Muscimol; Oxazoles; Pyridoxine; Seizures | 1982 |
Effects of the putative GABAergic agonists, muscimol and THIP, upon local cerebral glucose utilisation.
Topics: Analgesics; Animals; Brain; Deoxy Sugars; Deoxyglucose; gamma-Aminobutyric Acid; Glycolysis; Isoxazoles; Male; Muscimol; Organ Specificity; Oxazoles; Rats; Rats, Inbred Strains | 1982 |
Effects of gamma-aminobutyric acid agonist and antagonist drugs on local cerebral glucose utilization.
Topics: Animals; Autoradiography; Bicuculline; Brain; Carbon Radioisotopes; Deoxy Sugars; Deoxyglucose; gamma-Aminobutyric Acid; Glycolysis; Male; Muscimol; Organ Specificity; Oxazoles; Rats | 1982 |
Differential localization of radioactive gamma-aminobutyric acid and muscimol in isolated and in vivo mouse retina.
Topics: Animals; Autoradiography; gamma-Aminobutyric Acid; In Vitro Techniques; Mice; Muscimol; Neuroglia; Oxazoles; Retina; Time Factors; Tissue Distribution | 1982 |
Chlordiazepoxide-induced ataxia, muscle relaxation and sedation in the rat: effects of muscimol, picrotoxin and naloxone.
Topics: Animals; Arousal; Chlordiazepoxide; Exploratory Behavior; Male; Motor Activity; Motor Skills; Muridae; Muscimol; Muscle Contraction; Muscle Relaxation; Naloxone; Oxazoles; Picrotoxin; Rats; Reaction Time | 1982 |
An in vivo method for testing GABAergic compounds.
Topics: Animals; Apomorphine; gamma-Aminobutyric Acid; Injections, Intraventricular; Injections, Subcutaneous; Male; Mice; Mice, Inbred ICR; Motor Activity; Muscimol; Oxazoles; Picrotoxin | 1982 |
Anticonvulsant effects of muscimol.
Topics: Animals; Bicuculline; GABA Antagonists; Muscimol; Neurons; Oxazoles; Penicillins; Picrotoxin; Rats; Receptors, Drug; Seizures; Strychnine | 1980 |
Rotation induced by intranigral injections of GABA agonists and antagonists: zone-specific effects.
Topics: Animals; Bicuculline; GABA Antagonists; Humans; Hydroxydopamines; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Rotation; Stereotyped Behavior; Substantia Nigra | 1980 |
Effects of muscimol alone and in combination with diazepam on shuttle-box performance in rats.
Topics: Animals; Avoidance Learning; Bicuculline; Diazepam; Drug Interactions; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains | 1981 |
Suppression of apomorphine-induced oral stereotypy in rats by microinjection of muscimol into midbrain.
Topics: Animals; Apomorphine; Humans; Male; Mesencephalon; Muscimol; Oxazoles; Rats; Stereotyped Behavior; Superior Colliculi | 1982 |
Analgesic properties of the GABA-mimetic THIP.
Topics: Analgesics; Animals; Arthritis, Experimental; Baclofen; Electric Stimulation; Isoxazoles; Macaca mulatta; Mice; Morphine; Muscimol; Oxazoles; Reaction Time | 1981 |
Correlation of [14C]muscimol concentration in rat brain with anticonvulsant activity.
Topics: Animals; Anticonvulsants; Bicuculline; Brain; Half-Life; Male; Muscimol; Oxazoles; Rats | 1981 |
Sensitization of the perioral biting reflex by intranigral GABA agonist after detelencephalization.
Topics: Animals; Functional Laterality; Male; Muscimol; Oxazoles; Physical Stimulation; Rats; Reflex; Substantia Nigra; Telencephalon | 1981 |
Muscimol-induced myoclonic jerks in mice.
Topics: Animals; Drug Interactions; Kinetics; Male; Mice; Muscimol; Oxazoles; Picrotoxin; Seizures | 1981 |
Increases and decreases in local cerebral glucose utilization in response to GABA agonists.
Topics: Animals; Brain; gamma-Aminobutyric Acid; Glucose; Isoxazoles; Male; Muscimol; Oxazoles; Rats | 1981 |
GABA and muscimol binding processes in CNS tissue culture preparations.
Topics: Animals; Astrocytes; Brain; Culture Media; Culture Techniques; gamma-Aminobutyric Acid; Mice; Muscimol; Neurons; Oxazoles; Rats | 1981 |
Autoradiographic localization of [3H]muscimol in the cat retina.
Topics: Animals; Autoradiography; Cats; gamma-Aminobutyric Acid; Microscopy, Electron; Muscimol; Neurons; Oxazoles; Retina; Tritium | 1981 |
Effects of GABAergic drugs on brain stimulation reward as assessed by a 'threshold' method.
Topics: Animals; Brain; Dose-Response Relationship, Drug; Electric Conductivity; Electric Stimulation; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Reward; Self Stimulation | 1981 |
Differential effects of sodium-free media on gamma-aminobutyrate and muscimol-evoked conductance increases recorded from lobster muscle fibres.
Topics: Animals; Dose-Response Relationship, Drug; Electric Conductivity; Evoked Potentials; gamma-Aminobutyric Acid; Kinetics; Lithium; Muscimol; Muscles; Nephropidae; Nipecotic Acids; Oxazoles; Sodium | 1981 |
Muscimol and gamma-hydroxybutyrate: similar interactions with convulsant agents.
Topics: 3-Mercaptopropionic Acid; Animals; Anticonvulsants; Bicuculline; Dose-Response Relationship, Drug; Drug Synergism; Hydroxybutyrates; Male; Mice; Muscimol; Oxazoles; Pentylenetetrazole; Seizures; Sodium Oxybate; Strychnine; Sulfhydryl Compounds | 1981 |
Central cardiovascular effects of taurine: comparison with homotaurine and muscimol.
Topics: Animals; Bicuculline; Cats; Central Nervous System; Hemodynamics; Injections, Intraventricular; Muscimol; Oxazoles; Strychnine; Taurine | 1981 |
Muscimol induced feeding: a model to study the hypothalamic regulation of appetite.
Topics: Animals; Appetite; Atropine; Calcitonin; Dose-Response Relationship, Drug; Eating; Haloperidol; Hypothalamus; Male; Models, Biological; Muscimol; Naloxone; Oxazoles; Rats; Rats, Inbred Strains | 1981 |
Paradoxical blockade of a muscimol response by THIP, a GABA agonist and also by GABA-transaminase inhibitors.
Topics: 4-Aminobutyrate Transaminase; Animals; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Muscimol; Myoclonus; Oxazoles; Time Factors; Transaminases | 1981 |
Muscimol as an antagonist of chemical convulsants.
Topics: Animals; Anticonvulsants; Convulsants; Male; Mice; Mice, Inbred ICR; Muscimol; Oxazoles | 1981 |
Single unit responses of substantia nigra and globus pallidus neurons to GABA agonist and antagonist drugs.
Topics: Animals; gamma-Aminobutyric Acid; Globus Pallidus; Iontophoresis; Isoxazoles; Kainic Acid; Male; Muscimol; Neurons; Oxazoles; Rats; Rats, Inbred Strains; Substantia Nigra | 1981 |
Decrease in effects of muscimol on the dorsal root after repeated administration of diazepam in rats.
Topics: Animals; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Male; Membrane Potentials; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Spinal Nerve Roots; Time Factors | 1981 |
Lack of Na"-independent binding of [3H]GABA or [3H]muscimol to particulate fractions of cultured astroblasts.
Topics: Animals; Astrocytes; Brain; Cells, Cultured; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Radioligand Assay; Rats; Sodium; Tritium | 1980 |
Antinociceptive effects of baclofen and muscimol upon intraventricular administration.
Topics: Analgesics; Animals; Baclofen; Injections, Intraperitoneal; Injections, Intraventricular; Male; Motor Activity; Muscimol; Oxazoles; Rats | 1980 |
Effects of muscimol and picrotoxin on single unit activity of substantia nigra neurons.
Topics: Animals; Dose-Response Relationship, Drug; Electric Conductivity; gamma-Aminobutyric Acid; Male; Muscimol; Neurons; Oxazoles; Picrotoxin; Rats; Substantia Nigra | 1980 |
Neuroleptic-induced prolactin rise: influence of pharmacological alterations of different neurotransmitter system.
Topics: Animals; Apomorphine; Diazepam; Diphenhydramine; Haloperidol; Kinetics; Male; Metergoline; Muscimol; Oxazoles; Piperazines; Prolactin; Rats | 1980 |
Binding of [3H]GABA and [3H]muscimol to subcellular particles of a neurone-enriched culture of mouse brain.
Topics: Animals; Binding, Competitive; Brain; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Kinetics; Ligands; Mice; Muscimol; Neurons; Oxazoles; Protein Binding; Receptors, Drug; Tritium | 1980 |
In vivo release of endogenous gamma-aminobutyric acid from rat striatum: effects of muscimol, oxotremorine, and morphine.
Topics: Animals; Corpus Striatum; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Haloperidol; Male; Morphine; Muscimol; Nalorphine; Oxazoles; Oxotremorine; Potassium; Rats; Tetrodotoxin | 1980 |
Binding of muscimol and GABA in sub-fractions of a crude membrane fraction of rat brain.
Topics: Animals; Brain; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Oxazoles; Rats; Synaptic Membranes | 1980 |
GABAergic actions of THIP in vivo and vitro: a comparison with muscimol and GABA.
Topics: Animals; Binding Sites; Brain; Cerebellum; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; In Vitro Techniques; Iontophoresis; Isoxazoles; Male; Muscimol; Neurons; Oxazoles; Rats; Substantia Nigra | 1980 |
Anorexic effects of ethanolamine-O-sulfate and muscimol in the rat: evidence that GABA inhibits ingestive behavior.
Topics: 4-Aminobutyrate Transaminase; Animals; Appetite Depressants; Body Weight; Brain Chemistry; Dextroamphetamine; Ethanolamines; Feeding Behavior; gamma-Aminobutyric Acid; Male; Motor Activity; Muscimol; Oxazoles; Rats | 1980 |
Some characteristics of [3H]muscimol binding to synaptic membrane from rat brain.
Topics: Animals; Binding Sites; Brain; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Muscimol; Oxazoles; Polyethylene Glycols; Rats; Synaptic Membranes; Temperature | 1980 |
Decreases in the binding of [3H]GABA and [3H]muscimol to a particulate fraction of rat brain produced by human sera; some speculations.
Topics: Animals; Blood Physiological Phenomena; Brain; gamma-Aminobutyric Acid; Male; Muscimol; Nerve Tissue Proteins; Oxazoles; Protein Binding; Rats; Synaptic Membranes | 1980 |
[3H]Muscimol binding in the rat retina.
Topics: Animals; Binding Sites; Female; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Membranes; Muscimol; Octoxynol; Oxazoles; Polyethylene Glycols; Rats; Retina | 1980 |
Cardiovascular effects of intracerebroventricular GABA, glycine and muscimol in the rat.
Topics: Anesthesia; Animals; Dopamine; gamma-Aminobutyric Acid; Glycine; Hemodynamics; Injections, Intraventricular; Male; Muscimol; Oxazoles; Parasympathetic Nervous System; Rats; Serotonin; Sympathetic Nervous System | 1980 |
Effect of muscimol on dopamine metabolism of the rat hypothalamus.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Hypothalamus; Male; Muscimol; Norepinephrine; Oxazoles; Rats | 1980 |
Na+-independent binding of [3H]GABA and [3H]muscimol to subcellular particles of neural primary cultures and whole brain.
Topics: Animals; Animals, Newborn; Astrocytes; Binding Sites; Brain; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rats; Sodium | 1980 |
Binding of [3H]-muscimol, a potent gamma-aminobutyric acid receptor agonist, to membranes of the bovine retina.
Topics: Animals; Cattle; In Vitro Techniques; Kinetics; Membranes; Muscimol; Oxazoles; Retina; Subcellular Fractions | 1980 |
Measurement of gamma-aminobutyric acid in human cerebrospinal fluid: radioreceptor assay using [3H]muscimol.
Topics: Animals; Cattle; gamma-Aminobutyric Acid; Humans; Muscimol; Oxazoles; Radioligand Assay; Tritium | 1981 |
4,5-Substituted 3-Isoxazolols with Insecticidal Activity Act as Competitive Antagonists of Housefly GABA Receptors.
Topics: Animals; Binding, Competitive; GABA Antagonists; Gene Expression; Houseflies; Insecticides; Isoxazoles; Models, Molecular; Molecular Structure; Muscimol; Oocytes; Oxazoles; Receptors, GABA; Xenopus laevis | 2015 |
Selective inhibition of extra-synaptic α5-GABA
Topics: Animals; Benzodiazepines; Binding, Competitive; Brain; Female; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Long-Term Potentiation; Male; Memory; Mice, Inbred C57BL; Muscimol; Neural Inhibition; Nootropic Agents; Oxazoles; Rats, Sprague-Dawley; Receptors, GABA-A; Tissue Culture Techniques | 2017 |