muscimol and nipecotic acid

muscimol has been researched along with nipecotic acid in 40 studies

Research

Studies (40)

TimeframeStudies, this research(%)All Research%
pre-199014 (35.00)18.7374
1990's15 (37.50)18.2507
2000's9 (22.50)29.6817
2010's2 (5.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ali, FE; Bondinell, WE; Dandridge, PA; Frazee, JS; Garvey, E; Girard, GR; Kaiser, C; Ku, TW; Lafferty, JJ; Moonsammy, GI1
Enna, SJ; Patch, RJ; Tomita, K; Witiak, DT1
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO1
Dutia, MB; Johnston, AR; McQueen, DS1
Balcar, VJ1
Andrioli, GC; Bonanno, G; Raiteri, M; Ruelle, A1
Blakeman, DP; Davis, JP; Im, WB1
Sved, AF; Sved, JC1
Georgiev, V; Kambourova, T; Yonkov, D1
Arakawa, T; Okada, Y1
Dalkara, T1
Ciesielski, L; Gobaille, S; Mandel, P; Molina, V1
Lindgren, S; Simmonds, MA1
Catelli, JM; Sved, AF1
Catelli, JM; Giakas, WJ; Sved, AF1
Brown, DA; Scholfield, CN1
Madtes, P; Redburn, DA1
Madtes, PC; Redburn, DA1
Deisz, RA; Dose, M1
Cherubini, E; North, RA1
Horvitz, HR; Jorgensen, E; McIntire, SL1
Kocsis, JD; Lim, JY; Sakatani, K; Utzschneider, DA1
el Manira, A; Grillner, S; Matsushima, T; Tegnér, J1
Draguhn, A; Heinemann, U; Meierkord, H; Pfeiffer, M1
Hashimoto, T; Kuriyama, K1
Kelley, AE; Stratford, TR1
Nicklas, WJ; Zeevalk, GD1
Abraini, JH; Bouquet, C; Cagniard, B; Kriem, B; Rostain, JC1
Falch, E; Frølund, BF; Krogsgaard-Larsen, P1
Durgam, VR; Mifflin, SW; Vitela, M1
Bernard, LP; Nicklas, WJ; Stokes, AH; Zeevalk, GD1
Auer, M; Gownley, C; Kim, MJ; Li, XD; Song, J; Villa, A; Wang, DN1
Hopp, FA; Krolo, M; McCrimmon, DR; Stucke, AG; Stuth, EA; Tonkovic-Capin, M; Tonkovic-Capin, V; Zuperku, EJ1
Ferreira, M; Gillis, RA; Hernandez, YM; Sahibzada, N; Wasserman, AM1
Bungo, T; Furuse, M; Izumi, T; Kawamura, K; Takagi, T; Ueda, H1
Frosini, M; Sgaragli, G; Valoti, M1
Isogai, O; Ito, S; Masubuchi, Y; Saito, S; Tsukamoto, K; Uchiyama, T; Yajima, Y1
Hablitz, JJ; Keros, S1
Gao, H; Smith, BN1
Arisawa, M; Hayakawa, W; Ide, S; Ito, Y; Katayama, T; Kawamura, S; Kobayashi, T; Masuda, E; Minami, M; Nakada, K; Shuto, S; Suemasa, A; Yamada, S; Yoshikawa, M1

Other Studies

40 other study(ies) available for muscimol and nipecotic acid

ArticleYear
Orally active and potent inhibitors of gamma-aminobutyric acid uptake.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:5

    Topics: 4-Aminobutyrate Transaminase; Administration, Oral; Alkylation; Amino Acids; Animals; Brain; Carboxylic Acids; gamma-Aminobutyric Acid; Glutamate Decarboxylase; In Vitro Techniques; Male; Neurotransmitter Uptake Inhibitors; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter; Stereoisomerism; Synaptosomes

1985
Epimeric cis-decahydroquinoline-5-carboxylic acids: effects on gamma-aminobutyric acid uptake and receptor binding in vitro.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:7

    Topics: Animals; Brain; Chemical Phenomena; Chemistry; gamma-Aminobutyric Acid; In Vitro Techniques; Molecular Conformation; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Stereoisomerism; Synaptosomes

1981
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
    Journal of medicinal chemistry, 2005, Nov-03, Volume: 48, Issue:22

    Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles

2005
Tonic activity of rat medial vestibular nucleus neurones in vitro and its inhibition by GABA.
    Experimental brain research, 1992, Volume: 88, Issue:3

    Topics: Action Potentials; Animals; Baclofen; Cobalt; Dose-Response Relationship, Drug; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Neurons; Nipecotic Acids; Picrotoxin; Proline; Rats; Rats, Inbred Strains; Vestibular Nuclei

1992
Presence of a highly efficient "binding" to bacterial contamination can distort data from binding studies.
    Neurochemical research, 1990, Volume: 15, Issue:12

    Topics: Animals; Cats; Cerebral Cortex; GABA Antagonists; gamma-Aminobutyric Acid; Gram-Positive Bacteria; Isonicotinic Acids; Muscimol; Nipecotic Acids; Proline; Pyridazines; Radioligand Assay; Receptors, GABA-A; Tritium

1990
Cholinergic nerve terminals of human cerebral cortex possess a GABA transporter whose activation induces release of acetylcholine.
    Brain research, 1991, Jan-25, Volume: 539, Issue:2

    Topics: Acetylcholine; Anticonvulsants; Baclofen; Bicuculline; Biotransformation; Carrier Proteins; Cerebral Cortex; Choline; Female; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Male; Membrane Proteins; Membrane Transport Proteins; Middle Aged; Muscimol; Nerve Endings; Nerve Tissue Proteins; Nipecotic Acids; Organic Anion Transporters; Parasympathetic Nervous System; Proline; Synaptosomes

1991
Na(+)-dependent GABA transport system scavenges endogenous external GABA and prevents desensitization of GABAA receptors in rat cerebrocortical synaptoneurosomes.
    Brain research, 1990, Jun-25, Volume: 521, Issue:1-2

    Topics: Animals; Cerebral Cortex; Chlorides; gamma-Aminobutyric Acid; Male; Muscimol; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sodium; Synaptosomes

1990
Endogenous GABA acts on GABAB receptors in nucleus tractus solitarius to increase blood pressure.
    Brain research, 1990, Sep-03, Volume: 526, Issue:2

    Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Baclofen; Blood Pressure; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Medulla Oblongata; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vigabatrin

1990
Further evidence for the GABAergic influence on memory. Interaction of GABAergic transmission with angiotensin II on memory processes.
    Methods and findings in experimental and clinical pharmacology, 1989, Volume: 11, Issue:10

    Topics: Angiotensin II; Animals; Avoidance Learning; Bicuculline; gamma-Aminobutyric Acid; Male; Memory; Muscimol; Nipecotic Acids; Picrotoxin; Proline; Rats; Rats, Inbred Strains; Synaptic Transmission

1989
Excitatory and inhibitory action of GABA on synaptic transmission in slices of guinea pig superior colliculus.
    European journal of pharmacology, 1988, Dec-13, Volume: 158, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Muscimol; Nipecotic Acids; Perfusion; Proline; Receptors, GABA-A; Superior Colliculi; Synaptic Membranes; Synaptic Transmission

1988
Nipecotic acid, an uptake blocker, prevents fading of the gamma-aminobutyric acid effect.
    Brain research, 1986, Feb-26, Volume: 366, Issue:1-2

    Topics: Animals; Drug Synergism; gamma-Aminobutyric Acid; Hippocampus; Male; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
Effects of the potentiation of the GABAergic neurotransmission in the olfactory bulbs on mouse-killing behavior.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:3

    Topics: Aggression; Aminocaproates; Animals; Brain Chemistry; Drug Synergism; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Male; Motor Activity; Muscimol; Nipecotic Acids; Olfactory Bulb; Proline; Rats; Rats, Inbred Strains; Synaptic Transmission; Valproic Acid; Vigabatrin

1986
Adaptation of the GABAA-receptor complex in rat brain during chronic elevation of GABA by ethanolamine O-sulphate.
    British journal of pharmacology, 1987, Volume: 91, Issue:3

    Topics: 4-Aminobutyrate Transaminase; Animals; Brain Chemistry; Ethanolamines; Flurazepam; gamma-Aminobutyric Acid; Muscimol; Nipecotic Acids; Pentobarbital; Picrotoxin; Potassium; Proline; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Enhanced pressor response to GABA in the nucleus tractus solitarii of the spontaneously hypertensive rat.
    European journal of pharmacology, 1988, Jul-07, Volume: 151, Issue:2

    Topics: Animals; Baclofen; Blood Pressure; Brain Stem; gamma-Aminobutyric Acid; Heart Rate; Hypertension; Male; Muscimol; Nipecotic Acids; Proline; Rats; Rats, Inbred SHR; Rats, Inbred Strains

1988
GABAergic mechanisms in nucleus tractus solitarius alter blood pressure and vasopressin release.
    Brain research, 1987, Feb-17, Volume: 403, Issue:2

    Topics: Animals; Bicuculline; Blood Pressure; gamma-Aminobutyric Acid; Heart Rate; Male; Medulla Oblongata; Muscimol; Nipecotic Acids; Pressoreceptors; Proline; Rats; Rats, Inbred Strains; Vasopressins

1987
Inhibition of GABA uptake potentiates the conductance increase produced by GABA-mimetic compounds on single neurones in isolated olfactory cortex slices of the guinea-pig.
    British journal of pharmacology, 1984, Volume: 83, Issue:1

    Topics: Animals; Central Nervous System; Cerebral Cortex; Electric Stimulation; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Isonicotinic Acids; Muscimol; Neural Conduction; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Olfactory Pathways; Proline; Sodium; Taurine

1984
GABA as a trophic factor during development.
    Life sciences, 1983, Sep-05, Volume: 33, Issue:10

    Topics: Animals; Animals, Newborn; gamma-Aminobutyric Acid; Isoxazoles; Muscimol; Nipecotic Acids; Proline; Rabbits; Receptors, Cell Surface; Receptors, GABA-A; Retina

1983
Synaptic interactions in the GABA system during postnatal development in retina.
    Brain research bulletin, 1983, Volume: 10, Issue:6

    Topics: Animals; Cell Differentiation; gamma-Aminobutyric Acid; Muscimol; Nipecotic Acids; Proline; Rabbits; Receptors, Cell Surface; Receptors, GABA-A; Retina; Synaptic Transmission

1983
Comparison of GABA analogues at the crayfish stretch receptor neurone.
    Brain research bulletin, 1983, Volume: 11, Issue:3

    Topics: Animals; Astacoidea; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channels; Isoxazoles; Mechanoreceptors; Membrane Potentials; Muscimol; Nipecotic Acids; Proline; Sodium

1983
Actions of gamma-aminobutyric acid on neurones of guinea-pig myenteric plexus.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: Acetylcholine; Alanine; Animals; Baclofen; Bicuculline; gamma-Aminobutyric Acid; Glycine; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscimol; Myenteric Plexus; Neural Conduction; Neuromuscular Depolarizing Agents; Neurons; Nipecotic Acids; Picrotoxin; Proline; Tetrodotoxin

1984
Genes required for GABA function in Caenorhabditis elegans.
    Nature, 1993, Jul-22, Volume: 364, Issue:6435

    Topics: Animals; Behavior, Animal; Caenorhabditis elegans; Cell Differentiation; gamma-Aminobutyric Acid; Genes, Helminth; Muscimol; Mutation; Neurons; Nipecotic Acids; Proline

1993
The attenuation of GABA sensitivity in the maturing myelin-deficient rat optic nerve.
    Brain research. Developmental brain research, 1993, Mar-19, Volume: 72, Issue:1

    Topics: Action Potentials; Aging; Animals; Bicuculline; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Myelin Sheath; Nipecotic Acids; Optic Nerve; Proline; Rats; Rats, Mutant Strains; Receptors, GABA-A; Reference Values

1993
The spinal GABA system modulates burst frequency and intersegmental coordination in the lamprey: differential effects of GABAA and GABAB receptors.
    Journal of neurophysiology, 1993, Volume: 69, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Culture Techniques; Diazepam; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Lampreys; Locomotion; Motor Neurons; Muscimol; Muscles; N-Methylaspartate; Nerve Net; Neurons; Nipecotic Acids; Proline; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Spinal Nerve Roots; Synaptic Transmission

1993
Effects of gamma-aminobutyric acid (GABA) agonists and GABA uptake inhibitors on pharmacosensitive and pharmacoresistant epileptiform activity in vitro.
    British journal of pharmacology, 1996, Volume: 119, Issue:3

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Entorhinal Cortex; Epilepsy; Female; GABA Agonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Magnesium; Male; Membrane Potentials; Muscimol; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Proline; Rats; Rats, Wistar; Tiagabine

1996
GABAA receptor-mediated K(+)-evoked GABA release from globus pallidus--analysis using microdialysis.
    Neurochemistry international, 1997, Volume: 30, Issue:3

    Topics: Animals; Baclofen; Dinucleoside Phosphates; GABA Agonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Microdialysis; Muscimol; Nipecotic Acids; Potassium Chloride; Proline; Rats; Rats, Wistar; Receptors, GABA-A

1997
GABA in the nucleus accumbens shell participates in the central regulation of feeding behavior.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jun-01, Volume: 17, Issue:11

    Topics: Animals; Baclofen; Eating; Enzyme Inhibitors; Feeding Behavior; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microinjections; Muscimol; Nipecotic Acids; Nucleus Accumbens; Proline; Rats; Rats, Sprague-Dawley; Vigabatrin

1997
Activity at the GABA transporter contributes to acute cellular swelling produced by metabolic impairment in retina.
    Vision research, 1997, Volume: 37, Issue:24

    Topics: Animals; Biological Transport; Carbon Radioisotopes; Carrier Proteins; Chick Embryo; Culture Techniques; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Glycolysis; Iodoacetates; Ischemia; Isoxazoles; Membrane Proteins; Membrane Transport Proteins; Muscimol; Nipecotic Acids; Organic Anion Transporters; Oximes; Proline; Retina

1997
Modulation by GABA transmission in the substantia nigra compacta and reticulata of locomotor activity in rats exposed to high pressure.
    Neuroreport, 1998, May-11, Volume: 9, Issue:7

    Topics: Animals; Baclofen; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Helium; High Pressure Neurological Syndrome; Male; Motor Activity; Muscimol; Myoclonus; Nipecotic Acids; Proline; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra; Synaptic Transmission; Time Factors; Vigabatrin

1998
Inhibitors of gamma-aminobutyric acid transport as experimental tools and therapeutic agents.
    Methods in enzymology, 1998, Volume: 296

    Topics: Animals; Brain; Carrier Proteins; Cloning, Molecular; Drug Design; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Membrane Proteins; Membrane Transport Proteins; Molecular Structure; Muscimol; Neuroglia; Neurons; Nipecotic Acids; Organic Anion Transporters; Proline; Radioligand Assay; Recombinant Proteins; Tritium

1998
Enhanced gamma-aminobutyric acid-B receptor agonist responses and mRNA within the nucleus of the solitary tract in hypertension.
    Hypertension (Dallas, Tex. : 1979), 1999, Volume: 33, Issue:1 Pt 2

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; GABA Agonists; GABA Antagonists; Hypertension, Renovascular; Male; Muscimol; Nephrectomy; Nipecotic Acids; Phosphinic Acids; Proline; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Solitary Nucleus; Transcription, Genetic

1999
Attenuation of malonate toxicity in primary mesencephalic cultures using the GABA transport blocker, NO-711.
    Journal of neuroscience research, 2001, Apr-01, Volume: 64, Issue:1

    Topics: Animals; Cells, Cultured; Dopamine; Dose-Response Relationship, Drug; Drug Synergism; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Malonates; Mesencephalon; Muscimol; Neurons; Nipecotic Acids; Oximes; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species

2001
Monomeric state and ligand binding of recombinant GABA transporter from Escherichia coli.
    FEBS letters, 2001, Apr-13, Volume: 494, Issue:3

    Topics: Bacterial Proteins; Carrier Proteins; Detergents; Escherichia coli; Escherichia coli Proteins; Fluorescence; GABA Agonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Ligands; Membrane Proteins; Membrane Transport Proteins; Muscimol; Nipecotic Acids; Organic Anion Transporters; Protein Binding; Protein Structure, Quaternary; Recombinant Fusion Proteins; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Thrombin

2001
Differential modulation of respiratory neuronal discharge patterns by GABA(A) receptor and apamin-sensitive K(+) channel antagonism.
    Journal of neurophysiology, 2001, Volume: 86, Issue:5

    Topics: Alkaloids; Animals; Apamin; Benzylisoquinolines; Bicuculline; Dogs; Electrophysiology; GABA Agonists; Muscimol; Neurons; Nipecotic Acids; Potassium Channel Blockers; Potassium Channels; Receptors, GABA-A; Respiratory Physiological Phenomena

2001
GABA-mediated neurotransmission in the ventrolateral NTS plays a role in respiratory regulation in the rat.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2002, Volume: 283, Issue:6

    Topics: Animals; Apnea; Baclofen; Bicuculline; Cardiovascular System; Fluorescent Antibody Technique; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Immunohistochemistry; Kynurenic Acid; Male; Microinjections; Muscimol; Nipecotic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA; Respiration; Synaptic Transmission; Ventral Thalamic Nuclei

2002
Intracerebroventricular injection of muscimol, baclofen or nipecotic acid stimulates food intake in layer-type, but not meat-type, chicks.
    Brain research, 2003, Dec-12, Volume: 993, Issue:1-2

    Topics: Animals; Animals, Newborn; Baclofen; Behavior, Animal; Chickens; Dose-Response Relationship, Drug; Eating; GABA Agonists; Injections, Intraventricular; Male; Muscimol; Nipecotic Acids; Species Specificity

2003
Changes in rectal temperature and ECoG spectral power of sensorimotor cortex elicited in conscious rabbits by i.c.v. injection of GABA, GABA(A) and GABA(B) agonists and antagonists.
    British journal of pharmacology, 2004, Volume: 141, Issue:1

    Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Body Temperature Regulation; Electroencephalography; GABA Agonists; GABA Antagonists; Injections, Intraventricular; Isoxazoles; Lateral Ventricles; Male; Muscimol; Nipecotic Acids; Preoptic Area; Rabbits; Receptors, GABA-A; Receptors, GABA-B; Rectum; Somatosensory Cortex

2004
Effect of a high-salt diet on gamma-aminobutyric acid-mediated responses in the nucleus tractus solitarius of Sprague-Dawley rats.
    Brain research bulletin, 2004, Sep-30, Volume: 64, Issue:3

    Topics: Animals; Baclofen; Baroreflex; Bicuculline; Blood Pressure; Cardiovascular Physiological Phenomena; Dose-Response Relationship, Drug; Food, Formulated; GABA Agonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Heart Rate; Male; Muscimol; Neural Inhibition; Nipecotic Acids; Nitroprusside; Organophosphorus Compounds; Phenylephrine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Sodium Chloride, Dietary; Solitary Nucleus

2004
Subtype-specific GABA transporter antagonists synergistically modulate phasic and tonic GABAA conductances in rat neocortex.
    Journal of neurophysiology, 2005, Volume: 94, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Animals, Newborn; Anisoles; Bicuculline; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Synergism; Electric Stimulation; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Membrane Transport Modulators; Membrane Transport Proteins; Models, Neurological; Muscimol; Neocortex; Neural Inhibition; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Time Factors

2005
Zolpidem modulation of phasic and tonic GABA currents in the rat dorsal motor nucleus of the vagus.
    Neuropharmacology, 2010, Volume: 58, Issue:8

    Topics: Action Potentials; Animals; Brain Stem; GABA Agonists; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Miniature Postsynaptic Potentials; Motor Neurons; Muscimol; Nipecotic Acids; Patch-Clamp Techniques; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Vagus Nerve; Zolpidem

2010
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: identification of an efficient lead for potent inhibitors of GABA transports.
    Bioorganic & medicinal chemistry, 2013, Sep-01, Volume: 21, Issue:17

    Topics: Animals; Anticonvulsants; Brain; Cyclopropanes; GABA Modulators; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Ligands; Mice; Protein Binding; Rats; Seizures; Stereoisomerism; Structure-Activity Relationship

2013