muscimol and alphaxalone

muscimol has been researched along with alphaxalone in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-199010 (41.67)18.7374
1990's12 (50.00)18.2507
2000's2 (8.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bertrand, PP; Galligan, JJ1
Kokka, N; Olsen, RW; Sapp, DW; Witte, U1
Bolger, MB; Chen, JS; Gee, KW; Lan, NC1
Simmonds, MA; Turner, JP2
Olsen, RW; Ransom, RW; Turner, DM; Yang, JS1
Harrison, NL; Simmonds, MA1
Akhondzadeh, S; Stone, TW3
Jussofie, A2
Biggio, G; Ghiani, CA; Maciocco, E; Sanna, E; Serra, M; Tuligi, G1
Andrés-Trelles, F; Baamonde, A; Hidalgo, A; Meana, A; Menendez, L; SanMartin, S1
Gavish, M; Paz, L; Peter, Y; Pick, CG; Schreiber, S; Weizman, R1
Bence, M; Everest, H; Forrest-Owen, W; Lightman, SL; McArdle, CA; Williams, B1
Adkins, CE; Bonnert, TP; Gonzalez, JE; Haldon, C; Kerby, J; McKernan, RM; Oades, K; Pillai, GV; Simpson, PB; Whiting, PJ1
Maksay, G1
Iversen, LL; Wong, EH1
Olsen, RW; Yang, JS1
Casida, JE; Cole, LM; Lawrence, LJ1
Olsen, RW1
Maksay, G; Ticku, MK1
Ai, J; Kahnberg, P; Nielsen, M; Saederup, E; Squires, RF; Sterner, O; Witt, MR1

Other Studies

24 other study(ies) available for muscimol and alphaxalone

ArticleYear
Alfaxalone, pentobarbital and diazepam potentiate gamma-aminobutyric acid-induced depolarizations in single myenteric neurons of guinea pig intestine.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Anesthetics; Animals; Diazepam; Drug Synergism; gamma-Aminobutyric Acid; Guinea Pigs; Hydrocortisone; Intestines; Male; Membrane Potentials; Muscimol; Pentobarbital; Pregnanediones; Receptors, GABA-A

1992
Sex differences in sensitivity to pentylenetetrazol but not in GABAA receptor binding.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: Anesthetics; Animals; Anticonvulsants; Autoradiography; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; Electroshock; Ethanol; Female; Flunitrazepam; Male; Muscimol; Orchiectomy; Ovariectomy; Pentylenetetrazole; Pregnanediones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sex Characteristics

1992
Differential responses of expressed recombinant human gamma-aminobutyric acidA receptors to neurosteroids.
    Journal of neurochemistry, 1991, Volume: 57, Issue:5

    Topics: Allosteric Regulation; Animals; Binding, Competitive; Brain; Cell Line; Flunitrazepam; Humans; Kinetics; Macromolecular Substances; Muscimol; Pregnanediones; Pregnanes; Progesterone; Rats; Receptors, GABA-A; Recombinant Proteins; Spinal Cord; Transfection

1991
Modulation of the GABAA receptor complex by steroids in slices of rat cuneate nucleus.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: Androsterone; Anesthetics; Animals; Electric Stimulation; In Vitro Techniques; Isomerism; Medulla Oblongata; Muscimol; Picrotoxin; Pregnanediones; Rats; Receptors, GABA-A; Steroids; Structure-Activity Relationship

1989
Steroid anesthetics and naturally occurring analogs modulate the gamma-aminobutyric acid receptor complex at a site distinct from barbiturates.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Anesthetics; Animals; Barbiturates; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; In Vitro Techniques; Male; Muscimol; Pregnanediones; Rats; Rats, Inbred Strains; Receptors, GABA-A; Steroids; Structure-Activity Relationship

1989
Modulation of the GABA receptor complex by a steroid anaesthetic.
    Brain research, 1984, Dec-10, Volume: 323, Issue:2

    Topics: Anesthetics; Animals; In Vitro Techniques; Male; Medulla Oblongata; Muscimol; Pentobarbital; Pregnanediones; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, GABA-A; Receptors, Muscarinic

1984
Potentiation by neurosteroids of muscimol/adenosine interactions in rat hippocampus.
    Brain research, 1995, Apr-24, Volume: 677, Issue:2

    Topics: Adenosine; Anesthetics; Animals; Anti-Anxiety Agents; Barium; Bicuculline; Chloride Channel Agonists; Drug Synergism; GABA-A Receptor Agonists; Hippocampus; Male; Muscimol; Neural Inhibition; Pregnanediones; Pregnanolone; Rats; Rats, Wistar

1995
Induction of a novel form of hippocampal long-term depression by muscimol: involvement of GABAA but not glutamate receptors.
    British journal of pharmacology, 1995, Volume: 115, Issue:3

    Topics: Action Potentials; Adenosine; Alanine; Anesthetics; Animals; Anti-Anxiety Agents; Bicuculline; Corpus Striatum; Culture Techniques; Dose-Response Relationship, Drug; Electric Stimulation; GABA Agonists; GABA Antagonists; Hippocampus; Male; Muscimol; Neuronal Plasticity; Pregnanediones; Pregnanolone; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA; Receptors, Metabotropic Glutamate; Valine

1995
Brain region-specific effects of neuroactive steroids on the affinity and density of the GABA-binding site.
    Biological chemistry Hoppe-Seyler, 1993, Volume: 374, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Brain; Cerebellum; Desoxycorticosterone; Female; Hippocampus; Hypothalamus; Medulla Oblongata; Muscimol; Pregnanediones; Pregnanolone; Progesterone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1993
A new highly sensitive procedure--a prerequisite to evaluate the density of GABAA receptors and to study their allosteric properties in distinct areas of rat brain.
    Biological chemistry Hoppe-Seyler, 1993, Volume: 374, Issue:1

    Topics: Allosteric Regulation; Animals; Binding Sites; Brain; Cerebellum; Desoxycorticosterone; Female; Frontal Lobe; Humans; Hydrogen-Ion Concentration; Muscimol; Pentobarbital; Pregnanediones; Pregnanolone; Progesterone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1993
Biochemical evaluations of the effects of loreclezole and propofol on the GABAA receptor in rat brain.
    Biochemical pharmacology, 1996, Jun-14, Volume: 51, Issue:11

    Topics: Anesthetics; Animals; Anticonvulsants; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Triazoles; Tritium

1996
Interaction among alfaxalone, pregnenolone sulfate, and two GABAA agonists on hippocampal slices.
    Cellular and molecular neurobiology, 1996, Volume: 16, Issue:3

    Topics: Allosteric Regulation; Animals; Evoked Potentials; GABA Agonists; GABA-A Receptor Agonists; Hippocampus; Male; Mice; Muscimol; Pregnanediones; Pregnenolone; Taurine

1996
Maintenance of muscimol-induced long-term depression by neurosteroids.
    Progress in neuro-psychopharmacology & biological psychiatry, 1996, Volume: 20, Issue:2

    Topics: Anesthetics; Animals; Evoked Potentials; Hippocampus; Male; Muscimol; Pregnanediones; Rats; Rats, Wistar; Time Factors

1996
Effect of the pregnane-related GABA-active steroid alphaxalone on mice performance in the staircase test.
    Brain research, 1997, Aug-08, Volume: 765, Issue:1

    Topics: Alprazolam; Anesthetics; Animals; Anti-Inflammatory Agents; Corticosterone; Dose-Response Relationship, Drug; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Muscimol; Pregnanediones; Pregnanes; Pregnenolone; Psychomotor Performance

1997
GABAA receptor mediated elevation of Ca2+ and modulation of gonadotrophin-releasing hormone action in alphaT3-1 gonadotropes.
    Journal of neuroendocrinology, 2000, Volume: 12, Issue:2

    Topics: Anesthetics; Animals; Baclofen; Bicuculline; Biological Transport; Calcium; Calcium Channel Blockers; Cells, Cultured; Chlorides; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Mice; Muscimol; Nifedipine; Picrotoxin; Pituitary Gland; Pregnanediones; Receptors, GABA-A; Receptors, GABA-B

2000
alpha4beta3delta GABA(A) receptors characterized by fluorescence resonance energy transfer-derived measurements of membrane potential.
    The Journal of biological chemistry, 2001, Oct-19, Volume: 276, Issue:42

    Topics: Animals; Benzodiazepines; Cell Line; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Mice; Models, Biological; Muscimol; Pentobarbital; Pregnanediones; Pregnanolone; Protein Binding; Protein Conformation; Receptors, GABA-A; Spectrometry, Fluorescence; Time Factors; Transfection

2001
GABAA receptor populations bind agonists and antagonists differentially and with opposite affinities.
    Journal of neurochemistry, 1988, Volume: 50, Issue:6

    Topics: Affinity Labels; Androstanes; Animals; Azasteroids; Brain; Diazepam; Diazonium Compounds; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Photochemistry; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfanilic Acids; Synaptic Membranes

1988
Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Androstanes; Animals; Azasteroids; Bicuculline; Cell Membrane; Cerebral Cortex; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isonicotinic Acids; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, GABA-A; Taurine

1985
gamma-Aminobutyric acid receptor-regulated 36Cl- flux in mouse cortical slices.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: Androstanes; Animals; Azasteroids; Barbiturates; Cerebral Cortex; Chlorides; Dose-Response Relationship, Drug; Electrophysiology; Flunitrazepam; Male; Mathematics; Mice; Muscimol; Receptors, GABA-A

1987
Antagonism of inhibitory amino acids by the steroid derivative RU5135.
    British journal of pharmacology, 1985, Volume: 84, Issue:3

    Topics: Amino Acids; Androstanes; Animals; Azasteroids; Bicuculline; Electrophysiology; Glycine; In Vitro Techniques; Medulla Oblongata; Muscimol; Optic Nerve; Picrotoxin; Rats; Steroids, Heterocyclic; Strychnine

1985
Similar properties of [35S]t-butylbicyclophosphorothionate receptor and coupled components of the GABA receptor-ionophore complex in brains of human, cow, rat, chicken and fish.
    Life sciences, 1984, Oct-22, Volume: 35, Issue:17

    Topics: Androstanes; Animals; Azasteroids; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cattle; Chickens; Convulsants; Female; Fishes; Humans; Ivermectin; Lactones; Male; Middle Aged; Muscimol; Rats; Receptors, GABA-A; Taurine

1984
gamma-Aminobutyric acid receptor binding antagonism by the amidine steroid RU5135.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Androstanes; Animals; Azasteroids; Barbiturates; Benzodiazepines; Bicuculline; Binding, Competitive; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Rats; Receptors, GABA-A; Steroids, Heterocyclic

1984
Diazotization and thiocyanate differentiate agonists from antagonists for the high- and low-affinity receptors of gamma-aminobutyric acid.
    Journal of neurochemistry, 1984, Volume: 43, Issue:1

    Topics: Androstanes; Animals; Azasteroids; Benzenesulfonates; Bicuculline; Cerebral Cortex; Diazonium Compounds; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Sulfanilic Acids; Thiocyanates; Tubocurarine

1984
Honokiol and magnolol increase the number of [3H] muscimol binding sites three-fold in rat forebrain membranes in vitro using a filtration assay, by allosterically increasing the affinities of low-affinity sites.
    Neurochemical research, 1999, Volume: 24, Issue:12

    Topics: Allosteric Regulation; Androstanes; Animals; Azasteroids; Binding Sites; Biphenyl Compounds; Cell Membrane; Central Nervous System Depressants; Cerebellum; Diflunisal; Drugs, Chinese Herbal; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Lignans; Muscimol; Picrotoxin; Propofol; Prosencephalon; Rats; Receptors, GABA-A; Tritium

1999