muscarine has been researched along with pirenzepine in 76 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 29 (38.16) | 18.7374 |
1990's | 42 (55.26) | 18.2507 |
2000's | 4 (5.26) | 29.6817 |
2010's | 1 (1.32) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Kimura, T; Satoh, S; Shimamura, T | 1 |
Dohi, T; Minami, N; Morita, K; Ohtsuki, H; Suemitsu, T; Tsujimoto, A | 1 |
Aguilar, JS; Ballesta, JJ; Criado, M; Palmero, M; Reig, JA; Viniegra, S | 1 |
Bungardt, E; Feifel, R; Lambrecht, G; Moser, U; Mutschler, E; Surprenant, A; Tacke, R; Vockert, E | 1 |
Akerman, KE; Heikkilä, J; Jansson, C | 1 |
Jiang, ZG; North, RA; Sugita, S; Uchimura, N | 1 |
North, RA; Uchimura, N | 1 |
Ringdahl, B; Vargas, HM | 1 |
Inoue, M; Kuriyama, H | 1 |
Nishimura, S; Sorimachi, M; Yamagami, K | 1 |
Barker, JL; Fiszman, ML; Jones, SV | 1 |
Black, JW; Durant, PA; Shankley, NP; Welsh, NJ | 1 |
Doods, HN | 1 |
Beume, R; Eltze, M; Häfner, D; Hanauer, G; Kilian, U; Schudt, C | 1 |
Fujimoto, K; Hayakawa, T; Kashima, Y; Kawashima, K; Oohata, H; Suzuki, T | 1 |
Aceves, J; Brassart, JL; Góngora-Alfaro, JL; Hernández-López, S; Martínez-Fong, D | 1 |
Felix, W; Schneider, E | 1 |
Angeli, P; Brasili, L; Cantalamessa, F; Marucci, G; Wess, J | 1 |
Angelici, O; Cereda, E; Donetti, A; Duranti, P; Giudici, L; Micheletti, R; Schiavone, A | 1 |
Burgard, EC; Sarvey, JM | 1 |
de Pont, JJ; Rodrigues de Miranda, JF; van Ginneken, CA; van Zwam, AJ; Willems, PH | 1 |
Allen, TG; Burnstock, G | 1 |
Black, JW; Shankley, NP | 2 |
Kahn, R; Malhotra, RK; Wakade, AR; Wakade, CG; Wakade, TD | 1 |
Kobayashi, H; Mochida, S | 1 |
Galvan, M | 1 |
Horwitz, J | 1 |
Rojas, E; Santos, RM | 1 |
Mihara, S; Nishi, S | 1 |
Kaneko, E; Ooi, S | 1 |
Connolly, GP; Newberry, NR | 1 |
Gilbert, MJ; Newberry, NR | 1 |
Ellerbrock, BR; Hoss, W; Messer, WS; Smith, DA | 1 |
Boer, R; Galvan, M; Schudt, C | 1 |
Boselli, C; Kenakin, T | 1 |
Giachetti, A; Micheletti, R; Montagna, E | 1 |
Angeli, P; Lambrecht, G; Melchiorre, C; Moser, U; Mutschler, E; Wess, J | 1 |
Broekkamp, CL; Hagan, JJ; van der Heijden, B | 1 |
Gallagher, JP; Hasuo, H; Shinnick-Gallagher, P | 1 |
Chung, FZ; Lai, J; Mei, L; Roeske, WR; Venter, JC; Yamamura, HI | 1 |
Falch, E; Krogsgaard-Larsen, P; Lembøl, HL; Meier, E; Sauerberg, P | 1 |
Ferkany, JW; Kinnier, WJ; Kirkien-Rzeszotarski, A; McPherson, DW; Noronha-Blob, L; Rzeszotarski, WJ | 1 |
Akiba, I; Bujo, H; Kubo, T; Maeda, A; Mishina, M; Nakai, J; Numa, S | 1 |
Newberry, NR; Priestley, T | 1 |
Brown, DA; Gähwiler, BH | 1 |
Kilbinger, H; Nafziger, M | 1 |
Beld, AJ; Klaassen, AB; Kuijpers, W; Rodrigues de Miranda, JF; Salden, HJ; Scheres, HM | 1 |
Newberry, NR; Priestley, T; Woodruff, GN | 1 |
Beld, AJ; Hermanussen, MW; Lammers, JW; Rodrigues de Miranda, JF; van Ginneken, CA; van Koppen, CJ | 1 |
Christophe, J; Dehaye, JP; Hermans, L; Poloczek, P; Winand, J | 1 |
Hackmiller, RC; Jumblatt, JE | 1 |
Duranti, P; Giudici, L; Sagrada, A; Schiavone, A | 1 |
Akasu, T; Gallagher, JP; Hasuo, H | 2 |
Burgard, EC; Cote, TE; Sarvey, JM | 1 |
Changeux, JP; Vidal, C | 1 |
Akaike, N; Furukawa, K; Nabekura, J | 1 |
Iwamoto, ET; Marion, L | 1 |
Chen, FF; Hsu, HF; Sung, TC; Wu, D; Yang, CM | 1 |
Wills-Karp, M | 1 |
Desrues, L; Garnier, M; Lamacz, M; Louiset, E; Tonon, MC; Vaudry, H | 1 |
Eglen, RM; Sharif, NA; To, ZP | 1 |
Asano, T; Ito, S; Nakazato, Y; Ohta, T; Otsuguro, K | 1 |
Alvarez, R; Diez, N; Gil, MJ; Lizcano, F; Llorente, I; Salvador, J; Sopena, M | 1 |
Travagli, RA | 1 |
Bargas, J; Galarraga, E; Hernández-Echeagaray, E | 1 |
Hu, HZ; Li, ZW; Shao, M | 1 |
Bargas, J; Bermudez-Rattoni, F; Galarraga, E; Hernández-López, S; Miranda, I; Reyes, A; Vilchis, C | 1 |
Bernardi, G; Bonci, A; Grillner, P; Mercuri, NB; Svensson, TH | 1 |
Acs, Z; Makara, GB; Némethy, Z | 1 |
Kato, T; Ogasawara, M; Sato, K; Shimoda, N; Sugaya, K | 1 |
Arredondo, J; Chernyavsky, AI; Grando, SA; Ndoye, A; Nguyen, VT; Wess, J; Zia, S | 1 |
Chen, SR; Pan, HL | 1 |
Dudel, J | 1 |
Aceves, JJ; Bargas, J; Galarraga, E; Hernández-Flores, T; Hernández-González, O; Hernández-Martínez, R; Rueda-Orozco, PE; Tapia, D | 1 |
2 review(s) available for muscarine and pirenzepine
Article | Year |
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Selective muscarinic antagonists as bronchodilators.
Topics: Animals; Bronchodilator Agents; Humans; Muscarine; Pirenzepine; Receptors, Muscarinic; Respiratory System; Salivation | 1991 |
Telenzepine and its enantiomers, M1-selective antimuscarinics, in guinea pig lung function tests.
Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Muscarine; Parasympatholytics; Pirenzepine; Respiratory Function Tests; Stereoisomerism; Trachea | 1991 |
74 other study(ies) available for muscarine and pirenzepine
Article | Year |
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Effects of pirenzepine and hexamethonium on adrenal catecholamine release in responses to endogenous and exogenous acetylcholine in anesthetized dogs.
Topics: Acetylcholine; Adrenal Glands; Anesthesia; Animals; Catecholamines; Dogs; Epinephrine; Female; Hexamethonium Compounds; Male; Muscarine; Norepinephrine; Pirenzepine; Splanchnic Nerves | 1992 |
Involvement of Ca2+ entry and inositol trisphosphate-induced internal Ca2+ mobilization in muscarinic receptor-mediated catecholamine release in dog adrenal chromaffin cells.
Topics: Acetylcholine; Adrenal Medulla; Animals; Atropine; Bethanechol; Bethanechol Compounds; Biological Transport; Calcium; Calcium Channel Blockers; Catecholamines; Cells, Cultured; Dogs; Female; Gallic Acid; Inositol 1,4,5-Trisphosphate; Kinetics; Male; Muscarine; Neomycin; Nicotine; Oxotremorine; Pirenzepine; Polymyxin B; Potassium Chloride; Receptors, Muscarinic; Retinaldehyde; Tetradecanoylphorbol Acetate | 1992 |
Muscarinic receptor subtypes in bovine adrenal medulla.
Topics: Adrenal Medulla; Animals; Atropine; Binding Sites; Binding, Competitive; Cattle; Cell Membrane; Dicyclomine; Muscarine; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1992 |
Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Arterioles; Benzodiazepinones; Carbachol; Guinea Pigs; Ileum; Methacholine Chloride; Muscarine; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandin Endoperoxides, Synthetic; Receptors, Muscarinic; Vasodilation | 1992 |
Differential coupling of muscarinic receptors to Ca2+ mobilization and cyclic AMP in SH-SY5Y and IMR 32 neuroblastoma cells.
Topics: Acetylcholine; Alprostadil; Atropine; Calcium; Carbachol; Cyclic AMP; Humans; Methacholine Chloride; Muscarine; Neuroblastoma; Pertussis Toxin; Pirenzepine; Receptors, Muscarinic; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1991 |
Distinct muscarinic receptors inhibit release of gamma-aminobutyric acid and excitatory amino acids in mammalian brain.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Brain; Corpus Striatum; Diamines; gamma-Aminobutyric Acid; Glutamates; In Vitro Techniques; Kinetics; Muscarine; Neurons; Nucleus Accumbens; Organ Specificity; Parasympatholytics; Pirenzepine; Quinoxalines; Rats; Receptors, Muscarinic; Synapses | 1991 |
Muscarine reduces inwardly rectifying potassium conductance in rat nucleus accumbens neurones.
Topics: Action Potentials; Animals; Calcium; Cobalt; In Vitro Techniques; Ion Channels; Magnesium; Male; Muscarine; Neurons; Nucleus Accumbens; Phorbol Esters; Pirenzepine; Potassium; Rats; Receptors, Muscarinic; Septal Nuclei; Serotonin | 1990 |
Antimuscarinic potency and functional selectivity of oxotremorine analogs at muscarinic receptor subtypes in the rat.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Blood Pressure; Heart Rate; Male; Muscarine; Oxotremorine; Parasympathomimetics; Physostigmine; Pirenzepine; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1990 |
Muscarinic receptor is coupled with a cation channel through a GTP-binding protein in guinea-pig chromaffin cells.
Topics: Adrenal Medulla; Animals; Barium; Calcium; Dose-Response Relationship, Drug; Female; GTP-Binding Proteins; Guinea Pigs; Ion Channels; Male; Membrane Potentials; Muscarine; Oxotremorine; Pirenzepine; Receptors, Muscarinic; Tetraethylammonium; Tetraethylammonium Compounds | 1991 |
Internal Ca2+ mobilization by muscarinic stimulation increases secretion from adrenal chromaffin cells only in the presence of Ca2+ influx.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Atropine; Calcium; Catecholamines; Cats; Cattle; Cytosol; Gallopamil; Kinetics; Methacholine Chloride; Muscarine; Nicotine; Parasympatholytics; Pilocarpine; Pirenzepine; Receptors, Muscarinic | 1991 |
Electrophysiological responses to muscarinic receptor stimulation in cultured hippocampal neurons.
Topics: Action Potentials; Animals; Atropine; Carbachol; Cells, Cultured; Electrophysiology; Female; Hippocampus; Kinetics; Membrane Potentials; Muscarine; Muscarinic Antagonists; Neurons; Parasympathomimetics; Pirenzepine; Pregnancy; Rats; Receptors, Muscarinic; Stimulation, Chemical | 1991 |
Pharmacological analysis of agonist-antagonist interactions at acetylcholine muscarinic receptors in a new urinary bladder assay.
Topics: Animals; Atropine; Atropine Derivatives; Guinea Pigs; Hemicholinium 3; In Vitro Techniques; Male; Mice; Muscarine; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Pirenzepine; Receptors, Muscarinic; Trachea; Urinary Bladder | 1991 |
Determination of acetylcholine release in the striatum of anesthetized rats using in vivo microdialysis and a radioimmunoassay.
Topics: Acetylcholine; Administration, Topical; Animals; Atropine; Corpus Striatum; Dialysis; Male; Muscarine; Parasympatholytics; Physostigmine; Pirenzepine; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1991 |
Activation of nigral M1 and M2 muscarinic receptors produces opposing effects on striatal 3,4-dihydroxyphenylacetic acid measured by in vivo voltammetry.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Corpus Striatum; Electrochemistry; Functional Laterality; Male; Muscarine; Parasympatholytics; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereotaxic Techniques; Substantia Nigra | 1991 |
Effects of acetylcholine on different muscarinic receptors in the perfused porcine ear vein.
Topics: Acetylcholine; Animals; Atropine; Carbachol; Ear; Feedback; Gallamine Triethiodide; Indomethacin; Muscarine; Muscle, Smooth, Vascular; Organ Culture Techniques; Perfusion; Pirenzepine; Receptors, Muscarinic; Swine; Vasomotor System | 1991 |
Determination of muscarinic agonist potencies at M1 and M2 muscarinic receptors in a modified pithed rat preparation.
Topics: Animals; Bradycardia; Diamines; Dimethylamines; Dose-Response Relationship, Drug; Heart Rate; Heterocyclic Compounds; Male; Muscarine; Muscarinic Antagonists; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic; Stereoisomerism; Thiophenes | 1990 |
Affinity profile of the novel muscarinic antagonist, guanylpirenzepine.
Topics: Animals; Atrial Function; Duodenum; Guanine; Guinea Pigs; Ileum; Male; Muscarine; Muscarinic Antagonists; Muscle Relaxation; Pirenzepine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Vas Deferens | 1990 |
Muscarinic receptor activation facilitates the induction of long-term potentiation (LTP) in the rat dentate gyrus.
Topics: Animals; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Kinetics; Muscarine; Pirenzepine; Rats; Receptors, Muscarinic | 1990 |
Binding characteristics of the muscarinic receptor subtype in rabbit pancreas.
Topics: Animals; Binding, Competitive; Carbachol; Kinetics; Muscarine; Oxotremorine; Pancreas; Parasympathomimetics; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Time Factors; Tritium | 1990 |
M1 and M2 muscarinic receptors mediate excitation and inhibition of guinea-pig intracardiac neurones in culture.
Topics: Action Potentials; Animals; Cells, Cultured; Ganglia; Guinea Pigs; Heart; Membrane Potentials; Muscarine; Neural Inhibition; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic | 1990 |
Pharmacological analysis of the muscarinic receptors involved when McN-A 343 stimulates acid secretion in the mouse isolated stomach.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Benzodiazepinones; Cimetidine; Drug Interactions; Gastric Acid; Histamine H2 Antagonists; In Vitro Techniques; Mice; Muscarine; Parietal Cells, Gastric; Pirenzepine; Quaternary Ammonium Compounds; Receptors, Muscarinic; Tetrodotoxin | 1985 |
McN-A-343, a specific agonist of M1-muscarinic receptors, exerts antinicotinic and antimuscarinic effects in the rat adrenal medulla.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adrenal Medulla; Animals; Catecholamines; Male; Muscarine; Nicotine; Oxotremorine; Parasympatholytics; Pirenzepine; Quaternary Ammonium Compounds; Rats | 1986 |
Activation of M2 muscarinic receptors causes an alteration of action potentials by modulation of Ca entry in isolated sympathetic neurons of rabbits.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Action Potentials; Animals; Calcium; Cells, Cultured; Ganglia, Sympathetic; Male; Muscarine; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic | 1986 |
Modulation of synaptic transmission in autonomic ganglia mediated via the activation of postganglionic muscarinic M1 receptors.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Action Potentials; Animals; Ganglia, Autonomic; Ganglia, Sympathetic; In Vitro Techniques; Muscarine; Pirenzepine; Rabbits; Rats; Receptors, Muscarinic; Synapses; Synaptic Transmission | 1988 |
Muscarinic receptor stimulation increases inositol-phospholipid metabolism and inhibits cyclic AMP accumulation in PC12 cells.
Topics: Animals; Cyclic AMP; Muscarine; N-Methylscopolamine; Pheochromocytoma; Phorbol Esters; Phosphatidylinositols; Phosphodiesterase Inhibitors; Pirenzepine; Protein Kinase C; Receptors, Muscarinic; Scopolamine Derivatives; Stimulation, Chemical; Tumor Cells, Cultured | 1989 |
Muscarinic receptor modulation of glucose-induced electrical activity in mouse pancreatic B-cells.
Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Cells, Cultured; Glucose; In Vitro Techniques; Membrane Potentials; Mice; Muscarine; Pancreas; Pirenzepine; Receptors, Muscarinic | 1989 |
Muscarinic excitation and inhibition of neurons in the submucous plexus of the guinea-pig caecum.
Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Electric Stimulation; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscarine; Parasympathomimetics; Pirenzepine; Potassium; Receptors, Muscarinic; Submucous Plexus; Thionucleotides | 1989 |
Gastric acid secretion stimulated by modified sham-feeding, and the effects of histamine H2-antagonist and anti-muscarinic agent in patients with duodenal ulcer.
Topics: Adult; Cimetidine; Duodenal Ulcer; Gastric Acid; Histamine H2 Antagonists; Humans; Middle Aged; Muscarine; Pirenzepine; Reference Values | 1989 |
Muscarinic pharmacology of the spinal cord of the neonatal rat in vitro.
Topics: Action Potentials; Animals; Animals, Newborn; Atropine; In Vitro Techniques; Muscarine; Pirenzepine; Rats; Rats, Inbred Strains; Spinal Cord | 1989 |
Biphasic dose-response curve to muscarine on the rat superior cervical ganglion.
Topics: Animals; Dose-Response Relationship, Drug; Gallamine Triethiodide; Ganglia, Spinal; In Vitro Techniques; Muscarine; Pertussis Toxin; Pirenzepine; Rats; Virulence Factors, Bordetella | 1989 |
Regional differences in the binding of selective muscarinic receptor antagonists in rat brain: comparison with minimum-energy conformations.
Topics: Animals; Autoradiography; Brain; Computer Simulation; Diencephalon; Mesencephalon; Molecular Conformation; Molecular Structure; Muscarine; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Rhombencephalon; Structure-Activity Relationship; Telencephalon; Thermodynamics; Tissue Distribution | 1989 |
Interaction of telenzepine with muscarinic receptors in mammalian sympathetic ganglia.
Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Ganglia, Sympathetic; Male; Membrane Potentials; Muscarine; Parasympatholytics; Pirenzepine; Rabbits; Rats; Receptors, Muscarinic; Time Factors | 1989 |
Pharmacologic discrimination between receptor heterogeneity and allosteric interaction: resultant analysis of gallamine and pirenzepine antagonism of muscarinic responses in rat trachea.
Topics: Allosteric Regulation; Animals; Atropine; Binding Sites; Carbachol; Dose-Response Relationship, Drug; Gallamine Triethiodide; In Vitro Techniques; Male; Muscarine; Oxotremorine; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine; Trachea | 1989 |
Pharmacological analysis of muscarinic receptors coupled to oxyntic cell secretion in the mouse stomach.
Topics: Animals; Atropine; Atropine Derivatives; Benzodiazepinones; Binding, Competitive; Cimetidine; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Mice; Muscarine; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Parietal Cells, Gastric; Pirenzepine; Receptors, Muscarinic; Trachea | 1985 |
AF-DX 116, a cardioselective muscarinic antagonist.
Topics: Animals; Atropine; Bethanechol; Bethanechol Compounds; Carbachol; Cats; Dimethylphenylpiperazinium Iodide; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gastric Acid; Gastric Emptying; Guinea Pigs; Heart; Heart Rate; Male; Muscarine; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Pirenzepine; Rats; Receptors, Muscarinic | 1987 |
Methoctramine selectively blocks cardiac muscarinic M2 receptors in vivo.
Topics: Animals; Atropine; Blood Pressure; Diamines; Heart Rate; Male; Methacholine Chloride; Methacholine Compounds; Muscarine; Myocardium; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1988 |
The relative potencies of cholinomimetics and muscarinic antagonists on the rat iris in vivo: effects of pH on potency of pirenzepine and telenzepine.
Topics: Animals; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Iris; Male; Muscarine; Ophthalmic Solutions; Parasympathomimetics; Pirenzepine; Pupil; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1988 |
Disinhibition in the rat septum mediated by M1 muscarinic receptors.
Topics: Action Potentials; Animals; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Muscarine; Neural Inhibition; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Septal Nuclei | 1988 |
The cloned murine M1 muscarinic receptor is associated with the hydrolysis of phosphatidylinositols in transfected murine B82 cells.
Topics: Animals; Atropine; Binding, Competitive; Carbachol; Cell Line; Cell Membrane; DNA, Recombinant; Fibroblasts; Guanylyl Imidodiphosphate; Hydrolysis; Mice; Muscarine; Nucleic Acid Hybridization; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Recombinant Proteins; Sequence Homology, Nucleic Acid; Transfection | 1988 |
Heterocyclic muscarinic agonists. Synthesis and biological activity of some bicyclic sulfonium arecoline bioisosteres.
Topics: Animals; Arecoline; Brain; Chemical Phenomena; Chemistry; Guinea Pigs; Ileum; Muscarine; Myocardium; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Structure-Activity Relationship | 1988 |
Affinity and selectivity of the optical isomers of 3-quinuclidinyl benzilate and related muscarinic antagonists.
Topics: Adenylyl Cyclase Inhibitors; Animals; Cattle; Chemical Phenomena; Chemistry; Corpus Striatum; Inositol Phosphates; Male; Muscarine; Myocardium; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship | 1988 |
Primary structure of porcine muscarinic acetylcholine receptor III and antagonist binding studies.
Topics: Amino Acid Sequence; Animals; Base Sequence; DNA, Recombinant; Glycosylation; Molecular Sequence Data; Muscarine; Oocytes; Piperidines; Pirenzepine; Protein Conformation; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; RNA, Messenger; Sequence Homology, Nucleic Acid; Swine; Xenopus laevis | 1988 |
Pharmacological differences between two muscarinic responses of the rat superior cervical ganglion in vitro.
Topics: Acetylcholine; Animals; Atropine Derivatives; Calcium Chloride; Carbachol; Evoked Potentials; Ganglia, Spinal; In Vitro Techniques; Male; Muscarine; Neuromuscular Depolarizing Agents; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic | 1987 |
Muscarine affects calcium-currents in rat hippocampal pyramidal cells in vitro.
Topics: Animals; Atropine; Calcium; Electric Conductivity; Hippocampus; In Vitro Techniques; Membrane Potentials; Muscarine; Neurons; Pirenzepine; Rats; Tubocurarine | 1987 |
Two types of neuronal muscarine receptors modulating acetylcholine release from guinea-pig myenteric plexus.
Topics: Acetylcholine; Animals; Benzodiazepinones; Guinea Pigs; Ileum; In Vitro Techniques; Muscarine; Muscle Contraction; Myenteric Plexus; Oxotremorine; Pilocarpine; Pirenzepine; Receptors, Muscarinic; Scopolamine | 1985 |
Muscarinic receptors in rat nasal mucosa are predominantly of the low affinity agonist type.
Topics: Animals; Benzodiazepinones; Female; In Vitro Techniques; Kinetics; Male; Methacholine Compounds; Muscarine; Nasal Mucosa; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism | 1985 |
Pharmacological distinction between two muscarinic responses on the isolated superior cervical ganglion of the rat.
Topics: Animals; Atropine Derivatives; Benzodiazepinones; Calcium Chloride; Carbachol; Evoked Potentials; Gallamine Triethiodide; Ganglia, Spinal; In Vitro Techniques; Muscarine; Pirenzepine; Rats; Receptors, Muscarinic | 1985 |
Characterization of the muscarinic receptor in human tracheal smooth muscle.
Topics: Adolescent; Adult; Aged; Airway Resistance; Benzodiazepinones; Binding, Competitive; Child; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Kinetics; Methacholine Chloride; Methacholine Compounds; Middle Aged; Muscarine; Muscle, Smooth; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Trachea | 1985 |
Inhibitory effects of pirenzepine on muscarinic stimulation of rat pancreas.
Topics: alpha-Amylases; Animals; Atropine; Benzodiazepinones; Calcium; Carbachol; Male; Muscarine; Pancreas; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1983 |
M2-type muscarinic receptors mediate prejunctional inhibition of norepinephrine release in the human iris-ciliary body.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Carbachol; Child; Ciliary Body; Diamines; Dose-Response Relationship, Drug; Electric Stimulation; Humans; In Vitro Techniques; Iris; Middle Aged; Muscarine; Norepinephrine; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic | 1994 |
Himbacine discriminates between putative muscarinic M1 receptor-mediated responses.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Alkaloids; Animals; Binding, Competitive; Dogs; Female; Furans; Male; Muscarine; Naphthalenes; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Saphenous Vein; Superior Cervical Ganglion; Vas Deferens | 1994 |
Muscarine increases a voltage-independent potassium conductance through an M4 receptor in rat dorsolateral septal nucleus neurons.
Topics: Animals; Electrophysiology; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Male; Membrane Potentials; Muscarine; Neurons; Patch-Clamp Techniques; Pertussis Toxin; Pirenzepine; Potassium Channels; Rats; Rats, Inbred WKY; Receptors, Muscarinic; Septal Nuclei; Virulence Factors, Bordetella | 1995 |
Muscarinic depression of synaptic transmission and blockade of norepinephrine-induced long-lasting potentiation in the dentate gyrus.
Topics: 1-Methyl-3-isobutylxanthine; Analysis of Variance; Animals; Cyclic AMP; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; Muscarine; Norepinephrine; Parasympatholytics; Pertussis Toxin; Piperidines; Pirenzepine; Pyramidal Tracts; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Synapses; Synaptic Transmission; Virulence Factors, Bordetella | 1993 |
Nicotinic and muscarinic modulations of excitatory synaptic transmission in the rat prefrontal cortex in vitro.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Atropine; Bungarotoxins; Cerebral Cortex; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Evoked Potentials; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Male; Mecamylamine; Membrane Potentials; Muscarine; Neurons; Nicotine; Pirenzepine; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Scopolamine; Synaptic Transmission; Tubocurarine | 1993 |
Nicotinic and muscarinic acetylcholine responses in differentiated PC12 cells.
Topics: Acetylcholine; Animals; Atropine; Carbachol; Cell Differentiation; Cell Membrane Permeability; Egtazic Acid; Hexamethonium; Hexamethonium Compounds; Membrane Potentials; Muscarine; Nerve Growth Factors; Nicotine; Nystatin; Parasympatholytics; PC12 Cells; Pirenzepine; Potassium; Receptors, Muscarinic; Receptors, Nicotinic; Tubocurarine | 1994 |
Characterization of the antinociception produced by intrathecally administered muscarinic agonists in rats.
Topics: Adrenergic alpha-Antagonists; Analgesia; Animals; Carbachol; Diamines; Dioxolanes; Dose-Response Relationship, Drug; Drug Interactions; Injections, Spinal; Male; Mecamylamine; Muscarine; Narcotic Antagonists; Nociceptors; Pain Measurement; Parasympathomimetics; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Receptors, Serotonin; Spinal Cord; Time Factors; Tissue Distribution | 1993 |
Pharmacological characterization of muscarinic receptors in neonatal rat cardiomyocytes.
Topics: Animals; Animals, Newborn; Cells, Cultured; Cyclic AMP; Inositol Phosphates; Kinetics; Muscarine; Muscarinic Antagonists; Myocardium; N-Methylscopolamine; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine Derivatives | 1993 |
Age-related changes in pulmonary muscarinic receptor binding properties.
Topics: Aging; Animals; Binding, Competitive; Guinea Pigs; Lung; Male; Muscarine; Parasympathomimetics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1993 |
Nicotine-induced stimulation of alpha-MSH release in frog pituitary melanotrophs is mediated through a novel type of receptor.
Topics: alpha-MSH; Animals; Atropine; Calcium; Gallamine Triethiodide; In Vitro Techniques; Muscarine; Nicotine; Nifedipine; Pirenzepine; Pituitary Gland, Posterior; Ranidae; Receptors, Muscarinic; Tetrodotoxin | 1993 |
Muscarinic M3 receptors mediate total inositol phosphates accumulation in murine HSDM1C1 fibrosarcoma cells.
Topics: Animals; Binding, Competitive; Carbachol; Dioxolanes; Fibrosarcoma; Inositol Phosphates; Mice; Muscarine; Muscarinic Antagonists; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pirenzepine; Radioligand Assay; Receptors, Muscarinic; Scopolamine Derivatives; Tumor Cells, Cultured | 1993 |
Muscarinic receptor subtypes mediating catecholamine secretion and increase in intracellular Ca2+ concentration in adrenal chromaffin cells of the guinea pig.
Topics: Adrenal Medulla; Animals; Calcium; Cells, Cultured; Cholinergic Agents; Chromatography, High Pressure Liquid; Diamines; Dose-Response Relationship, Drug; Epinephrine; Female; Guinea Pigs; Kinetics; Male; Methacholine Chloride; Muscarine; Norepinephrine; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic | 1995 |
Cholinergic modulation of spontaneous hypothalamic-pituitary-adrenal activity and its circadian variation in man.
Topics: Adrenocorticotropic Hormone; Adult; Cholinesterase Inhibitors; Circadian Rhythm; Drug Combinations; Growth Hormone; Humans; Hydrocortisone; Hypothalamo-Hypophyseal System; Male; Muscarine; Parasympathetic Nervous System; Pirenzepine; Pituitary-Adrenal System; Pyridostigmine Bromide | 1996 |
Muscarine activates a nonselective cation current through a M3 muscarinic receptor subtype in rat dorsolateral septal nucleus neurons.
Topics: Animals; Cations; Diamines; Electric Conductivity; GTP-Binding Proteins; In Vitro Techniques; Ion Channels; Membrane Potentials; Microelectrodes; Muscarine; Muscarinic Agonists; Neurons; Patch-Clamp Techniques; Pirenzepine; Rats; Receptors, Muscarinic; Septal Nuclei | 1996 |
Muscarine receptor activation in the substantia gelatinosa of the spinal trigeminal nucleus of the guinea pig.
Topics: Animals; Carbachol; Cricetinae; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Patch-Clamp Techniques; Pirenzepine; Receptors, Glutamate; Substantia Gelatinosa; Trigeminal Nucleus, Spinal | 1996 |
3-Alpha-chloro-imperialine, a potent blocker of cholinergic presynaptic modulation of glutamatergic afferents in the rat neostriatum.
Topics: 4-Aminopyridine; Afferent Pathways; Animals; Atropine; Bicuculline; Carbachol; Cevanes; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA-A Receptor Antagonists; Gallamine Triethiodide; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Neurons; Pirenzepine; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Muscarinic; Synapses | 1998 |
Enhancement of GABA-activated current by muscarine in rat dorsal root ganglion neurons.
Topics: Acetylcholine; Action Potentials; Animals; Atropine; Bicuculline; Carbachol; Carbolines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Female; GABA Agonists; GABA Modulators; Gallamine Triethiodide; gamma-Aminobutyric Acid; Ganglia, Spinal; Ion Channel Gating; Ion Channels; Male; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nerve Tissue Proteins; Nicotinic Antagonists; Patch-Clamp Techniques; Pentobarbital; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Muscarinic | 1999 |
Cholinergic modulation of neostriatal output: a functional antagonism between different types of muscarinic receptors.
Topics: Acetylcholine; Animals; Cadmium Chloride; Cesium; Chlorides; Electric Stimulation; In Vitro Techniques; Membrane Potentials; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Neurons; Physostigmine; Pirenzepine; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptor, Muscarinic M4; Receptors, Muscarinic; Tetrodotoxin | 1999 |
Presynaptic muscarinic (M3) receptors reduce excitatory transmission in dopamine neurons of the rat mesencephalon.
Topics: 4-Aminopyridine; Acetylcholine; Animals; Atropine; Carbachol; Diamines; Dicyclomine; Dopamine; Electric Stimulation; Excitatory Postsynaptic Potentials; Mesencephalon; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Reaction Time; Receptor, Muscarinic M3; Receptors, Muscarinic; Synaptic Transmission; Tetrodotoxin | 1999 |
Effect of cholinergic drugs on the concentration of intracellular free calcium of rat pituitary intermediate lobe cells.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Age Factors; Animals; Atropine; Calcium; Carbachol; Cells, Cultured; Cholinergic Agonists; Cytosol; Female; Male; Melanocytes; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nicotinic Agonists; Piperidines; Pirenzepine; Pituitary Gland; Rats; Rats, Wistar; Vasodilator Agents | 1999 |
[The effects of the antagonists of muscarinic acetylcholine receptor subtypes in rat brain on urinary bladder contraction].
Topics: Animals; Atropine; Brain; Female; Muscarine; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Urinary Bladder; Urination | 2002 |
The M4 muscarinic receptor-selective effects on keratinocyte crawling locomotion.
Topics: Animals; Atropine; Cell Movement; Humans; Infant, Newborn; Keratinocytes; Mice; Mice, Knockout; Muscarine; Muscarinic Agonists; Piperidines; Pirenzepine; Receptor, Muscarinic M4; Receptors, Muscarinic; Stimulation, Chemical | 2003 |
Up-regulation of spinal muscarinic receptors and increased antinociceptive effect of intrathecal muscarine in diabetic rats.
Topics: Analgesics; Animals; Binding Sites; Diabetic Neuropathies; Guanosine 5'-O-(3-Thiotriphosphate); Injections, Spinal; Male; Muscarine; Muscarinic Agonists; Pain; Pain Measurement; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Spinal Cord; Sulfur Radioisotopes; Tritium; Up-Regulation | 2003 |
The time course of transmitter release in mouse motor nerve terminals is differentially affected by activation of muscarinic M1 or M2 receptors.
Topics: Animals; Diamines; Diaphragm; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; In Vitro Techniques; Mice; Mice, Inbred BALB C; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neuromuscular Junction; Neurotransmitter Agents; Pirenzepine; Presynaptic Terminals; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Time Factors | 2007 |
Muscarinic presynaptic modulation in GABAergic pallidal synapses of the rat.
Topics: Animals; Atropine; Cholinergic Neurons; Globus Pallidus; Inhibitory Postsynaptic Potentials; Intercellular Signaling Peptides and Proteins; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Peptides; Pirenzepine; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Muscarinic M1; Synapses | 2015 |