Page last updated: 2024-08-21

muscarine and pirenzepine

muscarine has been researched along with pirenzepine in 76 studies

Research

Studies (76)

TimeframeStudies, this research(%)All Research%
pre-199029 (38.16)18.7374
1990's42 (55.26)18.2507
2000's4 (5.26)29.6817
2010's1 (1.32)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kimura, T; Satoh, S; Shimamura, T1
Dohi, T; Minami, N; Morita, K; Ohtsuki, H; Suemitsu, T; Tsujimoto, A1
Aguilar, JS; Ballesta, JJ; Criado, M; Palmero, M; Reig, JA; Viniegra, S1
Bungardt, E; Feifel, R; Lambrecht, G; Moser, U; Mutschler, E; Surprenant, A; Tacke, R; Vockert, E1
Akerman, KE; Heikkilä, J; Jansson, C1
Jiang, ZG; North, RA; Sugita, S; Uchimura, N1
North, RA; Uchimura, N1
Ringdahl, B; Vargas, HM1
Inoue, M; Kuriyama, H1
Nishimura, S; Sorimachi, M; Yamagami, K1
Barker, JL; Fiszman, ML; Jones, SV1
Black, JW; Durant, PA; Shankley, NP; Welsh, NJ1
Doods, HN1
Beume, R; Eltze, M; Häfner, D; Hanauer, G; Kilian, U; Schudt, C1
Fujimoto, K; Hayakawa, T; Kashima, Y; Kawashima, K; Oohata, H; Suzuki, T1
Aceves, J; Brassart, JL; Góngora-Alfaro, JL; Hernández-López, S; Martínez-Fong, D1
Felix, W; Schneider, E1
Angeli, P; Brasili, L; Cantalamessa, F; Marucci, G; Wess, J1
Angelici, O; Cereda, E; Donetti, A; Duranti, P; Giudici, L; Micheletti, R; Schiavone, A1
Burgard, EC; Sarvey, JM1
de Pont, JJ; Rodrigues de Miranda, JF; van Ginneken, CA; van Zwam, AJ; Willems, PH1
Allen, TG; Burnstock, G1
Black, JW; Shankley, NP2
Kahn, R; Malhotra, RK; Wakade, AR; Wakade, CG; Wakade, TD1
Kobayashi, H; Mochida, S1
Galvan, M1
Horwitz, J1
Rojas, E; Santos, RM1
Mihara, S; Nishi, S1
Kaneko, E; Ooi, S1
Connolly, GP; Newberry, NR1
Gilbert, MJ; Newberry, NR1
Ellerbrock, BR; Hoss, W; Messer, WS; Smith, DA1
Boer, R; Galvan, M; Schudt, C1
Boselli, C; Kenakin, T1
Giachetti, A; Micheletti, R; Montagna, E1
Angeli, P; Lambrecht, G; Melchiorre, C; Moser, U; Mutschler, E; Wess, J1
Broekkamp, CL; Hagan, JJ; van der Heijden, B1
Gallagher, JP; Hasuo, H; Shinnick-Gallagher, P1
Chung, FZ; Lai, J; Mei, L; Roeske, WR; Venter, JC; Yamamura, HI1
Falch, E; Krogsgaard-Larsen, P; Lembøl, HL; Meier, E; Sauerberg, P1
Ferkany, JW; Kinnier, WJ; Kirkien-Rzeszotarski, A; McPherson, DW; Noronha-Blob, L; Rzeszotarski, WJ1
Akiba, I; Bujo, H; Kubo, T; Maeda, A; Mishina, M; Nakai, J; Numa, S1
Newberry, NR; Priestley, T1
Brown, DA; Gähwiler, BH1
Kilbinger, H; Nafziger, M1
Beld, AJ; Klaassen, AB; Kuijpers, W; Rodrigues de Miranda, JF; Salden, HJ; Scheres, HM1
Newberry, NR; Priestley, T; Woodruff, GN1
Beld, AJ; Hermanussen, MW; Lammers, JW; Rodrigues de Miranda, JF; van Ginneken, CA; van Koppen, CJ1
Christophe, J; Dehaye, JP; Hermans, L; Poloczek, P; Winand, J1
Hackmiller, RC; Jumblatt, JE1
Duranti, P; Giudici, L; Sagrada, A; Schiavone, A1
Akasu, T; Gallagher, JP; Hasuo, H2
Burgard, EC; Cote, TE; Sarvey, JM1
Changeux, JP; Vidal, C1
Akaike, N; Furukawa, K; Nabekura, J1
Iwamoto, ET; Marion, L1
Chen, FF; Hsu, HF; Sung, TC; Wu, D; Yang, CM1
Wills-Karp, M1
Desrues, L; Garnier, M; Lamacz, M; Louiset, E; Tonon, MC; Vaudry, H1
Eglen, RM; Sharif, NA; To, ZP1
Asano, T; Ito, S; Nakazato, Y; Ohta, T; Otsuguro, K1
Alvarez, R; Diez, N; Gil, MJ; Lizcano, F; Llorente, I; Salvador, J; Sopena, M1
Travagli, RA1
Bargas, J; Galarraga, E; Hernández-Echeagaray, E1
Hu, HZ; Li, ZW; Shao, M1
Bargas, J; Bermudez-Rattoni, F; Galarraga, E; Hernández-López, S; Miranda, I; Reyes, A; Vilchis, C1
Bernardi, G; Bonci, A; Grillner, P; Mercuri, NB; Svensson, TH1
Acs, Z; Makara, GB; Némethy, Z1
Kato, T; Ogasawara, M; Sato, K; Shimoda, N; Sugaya, K1
Arredondo, J; Chernyavsky, AI; Grando, SA; Ndoye, A; Nguyen, VT; Wess, J; Zia, S1
Chen, SR; Pan, HL1
Dudel, J1
Aceves, JJ; Bargas, J; Galarraga, E; Hernández-Flores, T; Hernández-González, O; Hernández-Martínez, R; Rueda-Orozco, PE; Tapia, D1

Reviews

2 review(s) available for muscarine and pirenzepine

ArticleYear
Selective muscarinic antagonists as bronchodilators.
    Agents and actions. Supplements, 1991, Volume: 34

    Topics: Animals; Bronchodilator Agents; Humans; Muscarine; Pirenzepine; Receptors, Muscarinic; Respiratory System; Salivation

1991
Telenzepine and its enantiomers, M1-selective antimuscarinics, in guinea pig lung function tests.
    Agents and actions. Supplements, 1991, Volume: 34

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Muscarine; Parasympatholytics; Pirenzepine; Respiratory Function Tests; Stereoisomerism; Trachea

1991

Other Studies

74 other study(ies) available for muscarine and pirenzepine

ArticleYear
Effects of pirenzepine and hexamethonium on adrenal catecholamine release in responses to endogenous and exogenous acetylcholine in anesthetized dogs.
    Journal of cardiovascular pharmacology, 1992, Volume: 20, Issue:6

    Topics: Acetylcholine; Adrenal Glands; Anesthesia; Animals; Catecholamines; Dogs; Epinephrine; Female; Hexamethonium Compounds; Male; Muscarine; Norepinephrine; Pirenzepine; Splanchnic Nerves

1992
Involvement of Ca2+ entry and inositol trisphosphate-induced internal Ca2+ mobilization in muscarinic receptor-mediated catecholamine release in dog adrenal chromaffin cells.
    Neurochemistry international, 1992, Volume: 21, Issue:2

    Topics: Acetylcholine; Adrenal Medulla; Animals; Atropine; Bethanechol; Bethanechol Compounds; Biological Transport; Calcium; Calcium Channel Blockers; Catecholamines; Cells, Cultured; Dogs; Female; Gallic Acid; Inositol 1,4,5-Trisphosphate; Kinetics; Male; Muscarine; Neomycin; Nicotine; Oxotremorine; Pirenzepine; Polymyxin B; Potassium Chloride; Receptors, Muscarinic; Retinaldehyde; Tetradecanoylphorbol Acetate

1992
Muscarinic receptor subtypes in bovine adrenal medulla.
    Neurochemical research, 1992, Volume: 17, Issue:12

    Topics: Adrenal Medulla; Animals; Atropine; Binding Sites; Binding, Competitive; Cattle; Cell Membrane; Dicyclomine; Muscarine; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic

1992
Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Arterioles; Benzodiazepinones; Carbachol; Guinea Pigs; Ileum; Methacholine Chloride; Muscarine; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandin Endoperoxides, Synthetic; Receptors, Muscarinic; Vasodilation

1992
Differential coupling of muscarinic receptors to Ca2+ mobilization and cyclic AMP in SH-SY5Y and IMR 32 neuroblastoma cells.
    European journal of pharmacology, 1991, Sep-12, Volume: 208, Issue:1

    Topics: Acetylcholine; Alprostadil; Atropine; Calcium; Carbachol; Cyclic AMP; Humans; Methacholine Chloride; Muscarine; Neuroblastoma; Pertussis Toxin; Pirenzepine; Receptors, Muscarinic; Tumor Cells, Cultured; Virulence Factors, Bordetella

1991
Distinct muscarinic receptors inhibit release of gamma-aminobutyric acid and excitatory amino acids in mammalian brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1991, Mar-15, Volume: 88, Issue:6

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Brain; Corpus Striatum; Diamines; gamma-Aminobutyric Acid; Glutamates; In Vitro Techniques; Kinetics; Muscarine; Neurons; Nucleus Accumbens; Organ Specificity; Parasympatholytics; Pirenzepine; Quinoxalines; Rats; Receptors, Muscarinic; Synapses

1991
Muscarine reduces inwardly rectifying potassium conductance in rat nucleus accumbens neurones.
    The Journal of physiology, 1990, Volume: 422

    Topics: Action Potentials; Animals; Calcium; Cobalt; In Vitro Techniques; Ion Channels; Magnesium; Male; Muscarine; Neurons; Nucleus Accumbens; Phorbol Esters; Pirenzepine; Potassium; Rats; Receptors, Muscarinic; Septal Nuclei; Serotonin

1990
Antimuscarinic potency and functional selectivity of oxotremorine analogs at muscarinic receptor subtypes in the rat.
    Life sciences, 1990, Volume: 47, Issue:22

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Blood Pressure; Heart Rate; Male; Muscarine; Oxotremorine; Parasympathomimetics; Physostigmine; Pirenzepine; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1990
Muscarinic receptor is coupled with a cation channel through a GTP-binding protein in guinea-pig chromaffin cells.
    The Journal of physiology, 1991, Volume: 436

    Topics: Adrenal Medulla; Animals; Barium; Calcium; Dose-Response Relationship, Drug; Female; GTP-Binding Proteins; Guinea Pigs; Ion Channels; Male; Membrane Potentials; Muscarine; Oxotremorine; Pirenzepine; Receptors, Muscarinic; Tetraethylammonium; Tetraethylammonium Compounds

1991
Internal Ca2+ mobilization by muscarinic stimulation increases secretion from adrenal chromaffin cells only in the presence of Ca2+ influx.
    Journal of neurochemistry, 1991, Volume: 57, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Atropine; Calcium; Catecholamines; Cats; Cattle; Cytosol; Gallopamil; Kinetics; Methacholine Chloride; Muscarine; Nicotine; Parasympatholytics; Pilocarpine; Pirenzepine; Receptors, Muscarinic

1991
Electrophysiological responses to muscarinic receptor stimulation in cultured hippocampal neurons.
    Brain research, 1991, Aug-23, Volume: 557, Issue:1-2

    Topics: Action Potentials; Animals; Atropine; Carbachol; Cells, Cultured; Electrophysiology; Female; Hippocampus; Kinetics; Membrane Potentials; Muscarine; Muscarinic Antagonists; Neurons; Parasympathomimetics; Pirenzepine; Pregnancy; Rats; Receptors, Muscarinic; Stimulation, Chemical

1991
Pharmacological analysis of agonist-antagonist interactions at acetylcholine muscarinic receptors in a new urinary bladder assay.
    British journal of pharmacology, 1991, Volume: 104, Issue:1

    Topics: Animals; Atropine; Atropine Derivatives; Guinea Pigs; Hemicholinium 3; In Vitro Techniques; Male; Mice; Muscarine; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Pirenzepine; Receptors, Muscarinic; Trachea; Urinary Bladder

1991
Determination of acetylcholine release in the striatum of anesthetized rats using in vivo microdialysis and a radioimmunoassay.
    Journal of neurochemistry, 1991, Volume: 57, Issue:3

    Topics: Acetylcholine; Administration, Topical; Animals; Atropine; Corpus Striatum; Dialysis; Male; Muscarine; Parasympatholytics; Physostigmine; Pirenzepine; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
Activation of nigral M1 and M2 muscarinic receptors produces opposing effects on striatal 3,4-dihydroxyphenylacetic acid measured by in vivo voltammetry.
    Brain research, 1991, Jul-19, Volume: 554, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Corpus Striatum; Electrochemistry; Functional Laterality; Male; Muscarine; Parasympatholytics; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereotaxic Techniques; Substantia Nigra

1991
Effects of acetylcholine on different muscarinic receptors in the perfused porcine ear vein.
    Cardiovascular research, 1991, Volume: 25, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Ear; Feedback; Gallamine Triethiodide; Indomethacin; Muscarine; Muscle, Smooth, Vascular; Organ Culture Techniques; Perfusion; Pirenzepine; Receptors, Muscarinic; Swine; Vasomotor System

1991
Determination of muscarinic agonist potencies at M1 and M2 muscarinic receptors in a modified pithed rat preparation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:6

    Topics: Animals; Bradycardia; Diamines; Dimethylamines; Dose-Response Relationship, Drug; Heart Rate; Heterocyclic Compounds; Male; Muscarine; Muscarinic Antagonists; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic; Stereoisomerism; Thiophenes

1990
Affinity profile of the novel muscarinic antagonist, guanylpirenzepine.
    Life sciences, 1990, Volume: 47, Issue:15

    Topics: Animals; Atrial Function; Duodenum; Guanine; Guinea Pigs; Ileum; Male; Muscarine; Muscarinic Antagonists; Muscle Relaxation; Pirenzepine; Rabbits; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Vas Deferens

1990
Muscarinic receptor activation facilitates the induction of long-term potentiation (LTP) in the rat dentate gyrus.
    Neuroscience letters, 1990, Aug-14, Volume: 116, Issue:1-2

    Topics: Animals; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Kinetics; Muscarine; Pirenzepine; Rats; Receptors, Muscarinic

1990
Binding characteristics of the muscarinic receptor subtype in rabbit pancreas.
    Journal of receptor research, 1990, Volume: 10, Issue:1-2

    Topics: Animals; Binding, Competitive; Carbachol; Kinetics; Muscarine; Oxotremorine; Pancreas; Parasympathomimetics; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Time Factors; Tritium

1990
M1 and M2 muscarinic receptors mediate excitation and inhibition of guinea-pig intracardiac neurones in culture.
    The Journal of physiology, 1990, Volume: 422

    Topics: Action Potentials; Animals; Cells, Cultured; Ganglia; Guinea Pigs; Heart; Membrane Potentials; Muscarine; Neural Inhibition; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic

1990
Pharmacological analysis of the muscarinic receptors involved when McN-A 343 stimulates acid secretion in the mouse isolated stomach.
    British journal of pharmacology, 1985, Volume: 86, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Benzodiazepinones; Cimetidine; Drug Interactions; Gastric Acid; Histamine H2 Antagonists; In Vitro Techniques; Mice; Muscarine; Parietal Cells, Gastric; Pirenzepine; Quaternary Ammonium Compounds; Receptors, Muscarinic; Tetrodotoxin

1985
McN-A-343, a specific agonist of M1-muscarinic receptors, exerts antinicotinic and antimuscarinic effects in the rat adrenal medulla.
    Life sciences, 1986, Dec-01, Volume: 39, Issue:22

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adrenal Medulla; Animals; Catecholamines; Male; Muscarine; Nicotine; Oxotremorine; Parasympatholytics; Pirenzepine; Quaternary Ammonium Compounds; Rats

1986
Activation of M2 muscarinic receptors causes an alteration of action potentials by modulation of Ca entry in isolated sympathetic neurons of rabbits.
    Neuroscience letters, 1986, Dec-12, Volume: 72, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Action Potentials; Animals; Calcium; Cells, Cultured; Ganglia, Sympathetic; Male; Muscarine; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic

1986
Modulation of synaptic transmission in autonomic ganglia mediated via the activation of postganglionic muscarinic M1 receptors.
    Pharmacology, 1988, Volume: 37 Suppl 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Action Potentials; Animals; Ganglia, Autonomic; Ganglia, Sympathetic; In Vitro Techniques; Muscarine; Pirenzepine; Rabbits; Rats; Receptors, Muscarinic; Synapses; Synaptic Transmission

1988
Muscarinic receptor stimulation increases inositol-phospholipid metabolism and inhibits cyclic AMP accumulation in PC12 cells.
    Journal of neurochemistry, 1989, Volume: 53, Issue:1

    Topics: Animals; Cyclic AMP; Muscarine; N-Methylscopolamine; Pheochromocytoma; Phorbol Esters; Phosphatidylinositols; Phosphodiesterase Inhibitors; Pirenzepine; Protein Kinase C; Receptors, Muscarinic; Scopolamine Derivatives; Stimulation, Chemical; Tumor Cells, Cultured

1989
Muscarinic receptor modulation of glucose-induced electrical activity in mouse pancreatic B-cells.
    FEBS letters, 1989, Jun-05, Volume: 249, Issue:2

    Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Cells, Cultured; Glucose; In Vitro Techniques; Membrane Potentials; Mice; Muscarine; Pancreas; Pirenzepine; Receptors, Muscarinic

1989
Muscarinic excitation and inhibition of neurons in the submucous plexus of the guinea-pig caecum.
    Neuroscience, 1989, Volume: 31, Issue:1

    Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Electric Stimulation; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscarine; Parasympathomimetics; Pirenzepine; Potassium; Receptors, Muscarinic; Submucous Plexus; Thionucleotides

1989
Gastric acid secretion stimulated by modified sham-feeding, and the effects of histamine H2-antagonist and anti-muscarinic agent in patients with duodenal ulcer.
    Gastroenterologia Japonica, 1989, Volume: 24, Issue:5

    Topics: Adult; Cimetidine; Duodenal Ulcer; Gastric Acid; Histamine H2 Antagonists; Humans; Middle Aged; Muscarine; Pirenzepine; Reference Values

1989
Muscarinic pharmacology of the spinal cord of the neonatal rat in vitro.
    Neuropharmacology, 1989, Volume: 28, Issue:2

    Topics: Action Potentials; Animals; Animals, Newborn; Atropine; In Vitro Techniques; Muscarine; Pirenzepine; Rats; Rats, Inbred Strains; Spinal Cord

1989
Biphasic dose-response curve to muscarine on the rat superior cervical ganglion.
    European journal of pharmacology, 1989, Apr-25, Volume: 163, Issue:2-3

    Topics: Animals; Dose-Response Relationship, Drug; Gallamine Triethiodide; Ganglia, Spinal; In Vitro Techniques; Muscarine; Pertussis Toxin; Pirenzepine; Rats; Virulence Factors, Bordetella

1989
Regional differences in the binding of selective muscarinic receptor antagonists in rat brain: comparison with minimum-energy conformations.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:6

    Topics: Animals; Autoradiography; Brain; Computer Simulation; Diencephalon; Mesencephalon; Molecular Conformation; Molecular Structure; Muscarine; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Rhombencephalon; Structure-Activity Relationship; Telencephalon; Thermodynamics; Tissue Distribution

1989
Interaction of telenzepine with muscarinic receptors in mammalian sympathetic ganglia.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Ganglia, Sympathetic; Male; Membrane Potentials; Muscarine; Parasympatholytics; Pirenzepine; Rabbits; Rats; Receptors, Muscarinic; Time Factors

1989
Pharmacologic discrimination between receptor heterogeneity and allosteric interaction: resultant analysis of gallamine and pirenzepine antagonism of muscarinic responses in rat trachea.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3

    Topics: Allosteric Regulation; Animals; Atropine; Binding Sites; Carbachol; Dose-Response Relationship, Drug; Gallamine Triethiodide; In Vitro Techniques; Male; Muscarine; Oxotremorine; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine; Trachea

1989
Pharmacological analysis of muscarinic receptors coupled to oxyntic cell secretion in the mouse stomach.
    British journal of pharmacology, 1985, Volume: 86, Issue:3

    Topics: Animals; Atropine; Atropine Derivatives; Benzodiazepinones; Binding, Competitive; Cimetidine; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Mice; Muscarine; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Parietal Cells, Gastric; Pirenzepine; Receptors, Muscarinic; Trachea

1985
AF-DX 116, a cardioselective muscarinic antagonist.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: Animals; Atropine; Bethanechol; Bethanechol Compounds; Carbachol; Cats; Dimethylphenylpiperazinium Iodide; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gastric Acid; Gastric Emptying; Guinea Pigs; Heart; Heart Rate; Male; Muscarine; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Pirenzepine; Rats; Receptors, Muscarinic

1987
Methoctramine selectively blocks cardiac muscarinic M2 receptors in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:3

    Topics: Animals; Atropine; Blood Pressure; Diamines; Heart Rate; Male; Methacholine Chloride; Methacholine Compounds; Muscarine; Myocardium; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1988
The relative potencies of cholinomimetics and muscarinic antagonists on the rat iris in vivo: effects of pH on potency of pirenzepine and telenzepine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:5

    Topics: Animals; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Iris; Male; Muscarine; Ophthalmic Solutions; Parasympathomimetics; Pirenzepine; Pupil; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1988
Disinhibition in the rat septum mediated by M1 muscarinic receptors.
    Brain research, 1988, Jan-12, Volume: 438, Issue:1-2

    Topics: Action Potentials; Animals; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Muscarine; Neural Inhibition; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Septal Nuclei

1988
The cloned murine M1 muscarinic receptor is associated with the hydrolysis of phosphatidylinositols in transfected murine B82 cells.
    Life sciences, 1988, Volume: 42, Issue:24

    Topics: Animals; Atropine; Binding, Competitive; Carbachol; Cell Line; Cell Membrane; DNA, Recombinant; Fibroblasts; Guanylyl Imidodiphosphate; Hydrolysis; Mice; Muscarine; Nucleic Acid Hybridization; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Recombinant Proteins; Sequence Homology, Nucleic Acid; Transfection

1988
Heterocyclic muscarinic agonists. Synthesis and biological activity of some bicyclic sulfonium arecoline bioisosteres.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:7

    Topics: Animals; Arecoline; Brain; Chemical Phenomena; Chemistry; Guinea Pigs; Ileum; Muscarine; Myocardium; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1988
Affinity and selectivity of the optical isomers of 3-quinuclidinyl benzilate and related muscarinic antagonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:7

    Topics: Adenylyl Cyclase Inhibitors; Animals; Cattle; Chemical Phenomena; Chemistry; Corpus Striatum; Inositol Phosphates; Male; Muscarine; Myocardium; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship

1988
Primary structure of porcine muscarinic acetylcholine receptor III and antagonist binding studies.
    FEBS letters, 1988, Aug-01, Volume: 235, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Base Sequence; DNA, Recombinant; Glycosylation; Molecular Sequence Data; Muscarine; Oocytes; Piperidines; Pirenzepine; Protein Conformation; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; RNA, Messenger; Sequence Homology, Nucleic Acid; Swine; Xenopus laevis

1988
Pharmacological differences between two muscarinic responses of the rat superior cervical ganglion in vitro.
    British journal of pharmacology, 1987, Volume: 92, Issue:4

    Topics: Acetylcholine; Animals; Atropine Derivatives; Calcium Chloride; Carbachol; Evoked Potentials; Ganglia, Spinal; In Vitro Techniques; Male; Muscarine; Neuromuscular Depolarizing Agents; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic

1987
Muscarine affects calcium-currents in rat hippocampal pyramidal cells in vitro.
    Neuroscience letters, 1987, May-19, Volume: 76, Issue:3

    Topics: Animals; Atropine; Calcium; Electric Conductivity; Hippocampus; In Vitro Techniques; Membrane Potentials; Muscarine; Neurons; Pirenzepine; Rats; Tubocurarine

1987
Two types of neuronal muscarine receptors modulating acetylcholine release from guinea-pig myenteric plexus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 328, Issue:3

    Topics: Acetylcholine; Animals; Benzodiazepinones; Guinea Pigs; Ileum; In Vitro Techniques; Muscarine; Muscle Contraction; Myenteric Plexus; Oxotremorine; Pilocarpine; Pirenzepine; Receptors, Muscarinic; Scopolamine

1985
Muscarinic receptors in rat nasal mucosa are predominantly of the low affinity agonist type.
    European journal of pharmacology, 1985, Jul-31, Volume: 113, Issue:3

    Topics: Animals; Benzodiazepinones; Female; In Vitro Techniques; Kinetics; Male; Methacholine Compounds; Muscarine; Nasal Mucosa; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism

1985
Pharmacological distinction between two muscarinic responses on the isolated superior cervical ganglion of the rat.
    European journal of pharmacology, 1985, Oct-08, Volume: 116, Issue:1-2

    Topics: Animals; Atropine Derivatives; Benzodiazepinones; Calcium Chloride; Carbachol; Evoked Potentials; Gallamine Triethiodide; Ganglia, Spinal; In Vitro Techniques; Muscarine; Pirenzepine; Rats; Receptors, Muscarinic

1985
Characterization of the muscarinic receptor in human tracheal smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 331, Issue:2-3

    Topics: Adolescent; Adult; Aged; Airway Resistance; Benzodiazepinones; Binding, Competitive; Child; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Kinetics; Methacholine Chloride; Methacholine Compounds; Middle Aged; Muscarine; Muscle, Smooth; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Trachea

1985
Inhibitory effects of pirenzepine on muscarinic stimulation of rat pancreas.
    European journal of pharmacology, 1983, Sep-02, Volume: 92, Issue:3-4

    Topics: alpha-Amylases; Animals; Atropine; Benzodiazepinones; Calcium; Carbachol; Male; Muscarine; Pancreas; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1983
M2-type muscarinic receptors mediate prejunctional inhibition of norepinephrine release in the human iris-ciliary body.
    Experimental eye research, 1994, Volume: 58, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Carbachol; Child; Ciliary Body; Diamines; Dose-Response Relationship, Drug; Electric Stimulation; Humans; In Vitro Techniques; Iris; Middle Aged; Muscarine; Norepinephrine; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic

1994
Himbacine discriminates between putative muscarinic M1 receptor-mediated responses.
    Life sciences, 1994, Volume: 54, Issue:17

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Alkaloids; Animals; Binding, Competitive; Dogs; Female; Furans; Male; Muscarine; Naphthalenes; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Saphenous Vein; Superior Cervical Ganglion; Vas Deferens

1994
Muscarine increases a voltage-independent potassium conductance through an M4 receptor in rat dorsolateral septal nucleus neurons.
    Neuroscience letters, 1995, Apr-21, Volume: 189, Issue:3

    Topics: Animals; Electrophysiology; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Male; Membrane Potentials; Muscarine; Neurons; Patch-Clamp Techniques; Pertussis Toxin; Pirenzepine; Potassium Channels; Rats; Rats, Inbred WKY; Receptors, Muscarinic; Septal Nuclei; Virulence Factors, Bordetella

1995
Muscarinic depression of synaptic transmission and blockade of norepinephrine-induced long-lasting potentiation in the dentate gyrus.
    Neuroscience, 1993, Volume: 54, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Analysis of Variance; Animals; Cyclic AMP; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; Muscarine; Norepinephrine; Parasympatholytics; Pertussis Toxin; Piperidines; Pirenzepine; Pyramidal Tracts; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Synapses; Synaptic Transmission; Virulence Factors, Bordetella

1993
Nicotinic and muscarinic modulations of excitatory synaptic transmission in the rat prefrontal cortex in vitro.
    Neuroscience, 1993, Volume: 56, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Atropine; Bungarotoxins; Cerebral Cortex; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Evoked Potentials; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Male; Mecamylamine; Membrane Potentials; Muscarine; Neurons; Nicotine; Pirenzepine; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Scopolamine; Synaptic Transmission; Tubocurarine

1993
Nicotinic and muscarinic acetylcholine responses in differentiated PC12 cells.
    Brain research, 1994, Feb-28, Volume: 638, Issue:1-2

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Cell Differentiation; Cell Membrane Permeability; Egtazic Acid; Hexamethonium; Hexamethonium Compounds; Membrane Potentials; Muscarine; Nerve Growth Factors; Nicotine; Nystatin; Parasympatholytics; PC12 Cells; Pirenzepine; Potassium; Receptors, Muscarinic; Receptors, Nicotinic; Tubocurarine

1994
Characterization of the antinociception produced by intrathecally administered muscarinic agonists in rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: Adrenergic alpha-Antagonists; Analgesia; Animals; Carbachol; Diamines; Dioxolanes; Dose-Response Relationship, Drug; Drug Interactions; Injections, Spinal; Male; Mecamylamine; Muscarine; Narcotic Antagonists; Nociceptors; Pain Measurement; Parasympathomimetics; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Receptors, Serotonin; Spinal Cord; Time Factors; Tissue Distribution

1993
Pharmacological characterization of muscarinic receptors in neonatal rat cardiomyocytes.
    The American journal of physiology, 1993, Volume: 265, Issue:3 Pt 1

    Topics: Animals; Animals, Newborn; Cells, Cultured; Cyclic AMP; Inositol Phosphates; Kinetics; Muscarine; Muscarinic Antagonists; Myocardium; N-Methylscopolamine; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine Derivatives

1993
Age-related changes in pulmonary muscarinic receptor binding properties.
    The American journal of physiology, 1993, Volume: 265, Issue:2 Pt 1

    Topics: Aging; Animals; Binding, Competitive; Guinea Pigs; Lung; Male; Muscarine; Parasympathomimetics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic

1993
Nicotine-induced stimulation of alpha-MSH release in frog pituitary melanotrophs is mediated through a novel type of receptor.
    Annals of the New York Academy of Sciences, 1993, May-31, Volume: 680

    Topics: alpha-MSH; Animals; Atropine; Calcium; Gallamine Triethiodide; In Vitro Techniques; Muscarine; Nicotine; Nifedipine; Pirenzepine; Pituitary Gland, Posterior; Ranidae; Receptors, Muscarinic; Tetrodotoxin

1993
Muscarinic M3 receptors mediate total inositol phosphates accumulation in murine HSDM1C1 fibrosarcoma cells.
    European journal of pharmacology, 1993, Jan-04, Volume: 244, Issue:1

    Topics: Animals; Binding, Competitive; Carbachol; Dioxolanes; Fibrosarcoma; Inositol Phosphates; Mice; Muscarine; Muscarinic Antagonists; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pirenzepine; Radioligand Assay; Receptors, Muscarinic; Scopolamine Derivatives; Tumor Cells, Cultured

1993
Muscarinic receptor subtypes mediating catecholamine secretion and increase in intracellular Ca2+ concentration in adrenal chromaffin cells of the guinea pig.
    The Journal of veterinary medical science, 1995, Volume: 57, Issue:6

    Topics: Adrenal Medulla; Animals; Calcium; Cells, Cultured; Cholinergic Agents; Chromatography, High Pressure Liquid; Diamines; Dose-Response Relationship, Drug; Epinephrine; Female; Guinea Pigs; Kinetics; Male; Methacholine Chloride; Muscarine; Norepinephrine; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic

1995
Cholinergic modulation of spontaneous hypothalamic-pituitary-adrenal activity and its circadian variation in man.
    The Journal of clinical endocrinology and metabolism, 1996, Volume: 81, Issue:8

    Topics: Adrenocorticotropic Hormone; Adult; Cholinesterase Inhibitors; Circadian Rhythm; Drug Combinations; Growth Hormone; Humans; Hydrocortisone; Hypothalamo-Hypophyseal System; Male; Muscarine; Parasympathetic Nervous System; Pirenzepine; Pituitary-Adrenal System; Pyridostigmine Bromide

1996
Muscarine activates a nonselective cation current through a M3 muscarinic receptor subtype in rat dorsolateral septal nucleus neurons.
    Journal of neurophysiology, 1996, Volume: 76, Issue:4

    Topics: Animals; Cations; Diamines; Electric Conductivity; GTP-Binding Proteins; In Vitro Techniques; Ion Channels; Membrane Potentials; Microelectrodes; Muscarine; Muscarinic Agonists; Neurons; Patch-Clamp Techniques; Pirenzepine; Rats; Receptors, Muscarinic; Septal Nuclei

1996
Muscarine receptor activation in the substantia gelatinosa of the spinal trigeminal nucleus of the guinea pig.
    Journal of neurophysiology, 1996, Volume: 76, Issue:6

    Topics: Animals; Carbachol; Cricetinae; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Patch-Clamp Techniques; Pirenzepine; Receptors, Glutamate; Substantia Gelatinosa; Trigeminal Nucleus, Spinal

1996
3-Alpha-chloro-imperialine, a potent blocker of cholinergic presynaptic modulation of glutamatergic afferents in the rat neostriatum.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: 4-Aminopyridine; Afferent Pathways; Animals; Atropine; Bicuculline; Carbachol; Cevanes; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA-A Receptor Antagonists; Gallamine Triethiodide; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Neurons; Pirenzepine; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Muscarinic; Synapses

1998
Enhancement of GABA-activated current by muscarine in rat dorsal root ganglion neurons.
    Neuroscience, 1999, Volume: 89, Issue:3

    Topics: Acetylcholine; Action Potentials; Animals; Atropine; Bicuculline; Carbachol; Carbolines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Female; GABA Agonists; GABA Modulators; Gallamine Triethiodide; gamma-Aminobutyric Acid; Ganglia, Spinal; Ion Channel Gating; Ion Channels; Male; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nerve Tissue Proteins; Nicotinic Antagonists; Patch-Clamp Techniques; Pentobarbital; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Muscarinic

1999
Cholinergic modulation of neostriatal output: a functional antagonism between different types of muscarinic receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, May-01, Volume: 19, Issue:9

    Topics: Acetylcholine; Animals; Cadmium Chloride; Cesium; Chlorides; Electric Stimulation; In Vitro Techniques; Membrane Potentials; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Neurons; Physostigmine; Pirenzepine; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptor, Muscarinic M4; Receptors, Muscarinic; Tetrodotoxin

1999
Presynaptic muscarinic (M3) receptors reduce excitatory transmission in dopamine neurons of the rat mesencephalon.
    Neuroscience, 1999, Volume: 91, Issue:2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Atropine; Carbachol; Diamines; Dicyclomine; Dopamine; Electric Stimulation; Excitatory Postsynaptic Potentials; Mesencephalon; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Reaction Time; Receptor, Muscarinic M3; Receptors, Muscarinic; Synaptic Transmission; Tetrodotoxin

1999
Effect of cholinergic drugs on the concentration of intracellular free calcium of rat pituitary intermediate lobe cells.
    Brain research bulletin, 1999, Sep-01, Volume: 50, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Age Factors; Animals; Atropine; Calcium; Carbachol; Cells, Cultured; Cholinergic Agonists; Cytosol; Female; Male; Melanocytes; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nicotinic Agonists; Piperidines; Pirenzepine; Pituitary Gland; Rats; Rats, Wistar; Vasodilator Agents

1999
[The effects of the antagonists of muscarinic acetylcholine receptor subtypes in rat brain on urinary bladder contraction].
    Nihon Hinyokika Gakkai zasshi. The japanese journal of urology, 2002, Volume: 93, Issue:3

    Topics: Animals; Atropine; Brain; Female; Muscarine; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Urinary Bladder; Urination

2002
The M4 muscarinic receptor-selective effects on keratinocyte crawling locomotion.
    Life sciences, 2003, Mar-28, Volume: 72, Issue:18-19

    Topics: Animals; Atropine; Cell Movement; Humans; Infant, Newborn; Keratinocytes; Mice; Mice, Knockout; Muscarine; Muscarinic Agonists; Piperidines; Pirenzepine; Receptor, Muscarinic M4; Receptors, Muscarinic; Stimulation, Chemical

2003
Up-regulation of spinal muscarinic receptors and increased antinociceptive effect of intrathecal muscarine in diabetic rats.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 307, Issue:2

    Topics: Analgesics; Animals; Binding Sites; Diabetic Neuropathies; Guanosine 5'-O-(3-Thiotriphosphate); Injections, Spinal; Male; Muscarine; Muscarinic Agonists; Pain; Pain Measurement; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Spinal Cord; Sulfur Radioisotopes; Tritium; Up-Regulation

2003
The time course of transmitter release in mouse motor nerve terminals is differentially affected by activation of muscarinic M1 or M2 receptors.
    The European journal of neuroscience, 2007, Volume: 26, Issue:8

    Topics: Animals; Diamines; Diaphragm; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; In Vitro Techniques; Mice; Mice, Inbred BALB C; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neuromuscular Junction; Neurotransmitter Agents; Pirenzepine; Presynaptic Terminals; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Time Factors

2007
Muscarinic presynaptic modulation in GABAergic pallidal synapses of the rat.
    Journal of neurophysiology, 2015, Feb-01, Volume: 113, Issue:3

    Topics: Animals; Atropine; Cholinergic Neurons; Globus Pallidus; Inhibitory Postsynaptic Potentials; Intercellular Signaling Peptides and Proteins; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Peptides; Pirenzepine; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Muscarinic M1; Synapses

2015