Page last updated: 2024-09-05

muraglitazar and troglitazone

muraglitazar has been researched along with troglitazone in 3 studies

Compound Research Comparison

Studies
(muraglitazar)
Trials
(muraglitazar)
Recent Studies (post-2010)
(muraglitazar)
Studies
(troglitazone)
Trials
(troglitazone)
Recent Studies (post-2010) (troglitazone)
8510251,857146287

Protein Interaction Comparison

ProteinTaxonomymuraglitazar (IC50)troglitazone (IC50)
Bile salt export pumpRattus norvegicus (Norway rat)3.9
Bile salt export pumpHomo sapiens (human)5.05
Carbonic anhydrase 2Homo sapiens (human)0.97
Adenosine receptor A3Homo sapiens (human)5.208
Cytochrome P450 2C9 Homo sapiens (human)4
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)5.208
Thromboxane-A synthase Homo sapiens (human)2.966
Amine oxidase [flavin-containing] BHomo sapiens (human)2.07
Mitogen-activated protein kinase 1Homo sapiens (human)1.238
Peroxisome proliferator-activated receptor gammaHomo sapiens (human)1.03
5-hydroxytryptamine receptor 2BHomo sapiens (human)1.312
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)5.208
ATP-binding cassette sub-family C member 8Homo sapiens (human)1.285
ATP-sensitive inward rectifier potassium channel 11Homo sapiens (human)1.285
Indoleamine 2,3-dioxygenase 2Mus musculus (house mouse)4.5

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adams, WJ; Artman, GD; Colca, JR; Gadwood, RC; Kletzien, RF; Larsen, SD; Lee, PH; McDonald, WG; Parker, TT; Tanis, SP; Zeller, JB1
Claude, N; Guillouzo, A; Renaud, MP; Rogue, A; Spire, C1
Amacher, DE; Boucher, GG; Francone, O; Kerlin, RL; Morton, D; Pettersen, JC; Pruimboom-Brees, IM; Will, Y1

Other Studies

3 other study(ies) available for muraglitazar and troglitazone

ArticleYear
PPARγ-sparing thiazolidinediones as insulin sensitizers. Design, synthesis and selection of compounds for clinical development.
    Bioorganic & medicinal chemistry, 2018, 12-01, Volume: 26, Issue:22

    Topics: Dose-Response Relationship, Drug; Drug Design; Humans; Insulin Resistance; Molecular Structure; PPAR gamma; Structure-Activity Relationship; Thiazolidinediones

2018
Comparative gene expression profiles induced by PPARγ and PPARα/γ agonists in rat hepatocytes.
    Toxicology and applied pharmacology, 2011, Jul-01, Volume: 254, Issue:1

    Topics: Alkanesulfonates; Animals; Chromans; Gene Expression Profiling; Genes; Glycine; Hepatocytes; Humans; Male; Oligonucleotide Array Sequence Analysis; Oxazoles; Phenylpropionates; PPAR alpha; PPAR gamma; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Rosiglitazone; Thiazolidinediones; Troglitazone

2011
The development of subcutaneous sarcomas in rodents exposed to peroxisome proliferators agonists: hypothetical mechanisms of action and de-risking attitude.
    Toxicologic pathology, 2012, Volume: 40, Issue:5

    Topics: Adipogenesis; Adipose Tissue, Brown; Adipose Tissue, White; Animals; Cell Differentiation; Chromans; Diabetes Mellitus, Type 2; DNA Damage; Glycine; Hypoglycemic Agents; Ion Channels; Mice; Mitochondria; Mitochondrial Proteins; Oxazoles; Oxidative Stress; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Pioglitazone; PPAR alpha; PPAR gamma; Rats; RNA-Binding Proteins; Rodentia; Rosiglitazone; Sarcoma; Thermogenesis; Thiazolidinediones; Transcription Factors; Troglitazone; Uncoupling Protein 1

2012