Page last updated: 2024-09-04

mrz 2549 and fentanyl

mrz 2549 has been researched along with fentanyl in 1 studies

*Fentanyl: A potent narcotic analgesic, abuse of which leads to habituation or addiction. It is primarily a mu-opioid agonist. Fentanyl is also used as an adjunct to general anesthetics, and as an anesthetic for induction and maintenance. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1078) [MeSH]

*Fentanyl: A potent narcotic analgesic, abuse of which leads to habituation or addiction. It is primarily a mu-opioid agonist. Fentanyl is also used as an adjunct to general anesthetics, and as an anesthetic for induction and maintenance. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1078) [MeSH]

Compound Research Comparison

Studies
(mrz 2549)
Trials
(mrz 2549)
Recent Studies (post-2010)
(mrz 2549)
Studies
(fentanyl)
Trials
(fentanyl)
Recent Studies (post-2010) (fentanyl)
60015,2884,3104,483

Protein Interaction Comparison

ProteinTaxonomymrz 2549 (IC50)fentanyl (IC50)
ATP-dependent translocase ABCB1Homo sapiens (human)6.5
Delta-type opioid receptorMus musculus (house mouse)0.6342
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0122
Mu-type opioid receptorRattus norvegicus (Norway rat)0.1888
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0122
Mu-type opioid receptorHomo sapiens (human)0.0058
Delta-type opioid receptorHomo sapiens (human)0.3092
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)5.893
Kappa-type opioid receptorHomo sapiens (human)1.58
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0031
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.8197
Sigma non-opioid intracellular receptor 1Cavia porcellus (domestic guinea pig)4.973
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.354

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19901 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Rubini, P; Schulz, R; Wüster, M1

Other Studies

1 other study(ies) available for mrz 2549 and fentanyl

ArticleYear
The preference of putative pro-enkephalins for different types of opiate receptors.
    Life sciences, 1981, Sep-21, Volume: 29, Issue:12

    Topics: Animals; Benzomorphans; Brain; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Fentanyl; Guinea Pigs; Ileum; Male; Mice; Morphine; Protein Precursors; Rats; Receptors, Opioid; Vas Deferens

1981