mr 2034 has been researched along with morphinans in 16 studies
Studies (mr 2034) | Trials (mr 2034) | Recent Studies (post-2010) (mr 2034) | Studies (morphinans) | Trials (morphinans) | Recent Studies (post-2010) (morphinans) |
---|---|---|---|---|---|
48 | 0 | 0 | 3,251 | 307 | 648 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 16 (100.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Iyengar, S; Kim, HS; Wood, PL | 1 |
Herz, A; Nikolarakis, K; Pfeiffer, A; Stalla, GK | 1 |
Männistö, PT; Rauhala, P; Tuominen, RK | 1 |
Coupar, JM; Quinn, MJ | 1 |
Ensinger, HA | 2 |
Wood, PL | 1 |
Brantl, V; Emrich, HM; Herz, A; Pfeiffer, A | 1 |
Brantl, V; Braun, S; Knepel, W; Lohmann, H; Meyer, HD; Pfeiffer, A | 1 |
Brantl, V; Braun, S; Mann, K; Meyer, HD; Pfeiffer, A | 1 |
Lanthier, D; Leibowitz, SF; Stanley, BG | 1 |
Dykstra, LA; Gmerek, DE; Woods, JH | 1 |
Gmerek, DE; Woods, JH | 1 |
Ensinger, HA; Gaida, W; Jennewein, HM; Merz, H; Stockhaus, K | 1 |
Faden, AI; Feuerstein, G; Kopin, IJ; Pfeiffer, A | 1 |
Johnson, N; Pasternak, GW | 1 |
16 other study(ies) available for mr 2034 and morphinans
Article | Year |
---|---|
Reversal of the actions of morphine on mesocortical dopamine metabolism in the rat by the kappa agonist MR-2034: tentative mu-2 opioid control of mesocortical dopaminergic projections.
Topics: Animals; Benzomorphans; Brain; Cerebral Cortex; Corpus Striatum; Dopamine; Frontal Lobe; Gyrus Cinguli; Male; Morphinans; Morphine; Olfactory Bulb; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu | 1987 |
The role of CRF in the release of ACTH by opiate agonists and antagonists in rats.
Topics: Adrenocorticotropic Hormone; Animals; Benzomorphans; Corticotropin-Releasing Hormone; Immune Sera; Male; Morphinans; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid | 1987 |
Opiate receptor subtypes in the regulation of thyrotropin and prolactin secretion in the rat.
Topics: Animals; Benzomorphans; Cerebral Ventricles; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Injections, Intraventricular; Kinetics; Male; Morphinans; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reference Values; Thyrotropin | 1988 |
The effects of the selective kappa-opioid agonist MR 2034 on the guinea-pig ileum.
Topics: Animals; Benzomorphans; Female; Guinea Pigs; Ileum; Male; Morphinans; Receptors, Opioid; Receptors, Opioid, kappa | 1988 |
Differentiating aspects of opioid receptor binding by [3H](-) (1R,5R,9R,2''S)-5,9-dimethyl-2-tetrahydrofurfuryl-2'-hydroxy-6,7- benzomorphan hydrochloride ([3H]Mr 2034), a drug preferentially acting on kappa-receptors.
Topics: Animals; Benzomorphans; Binding, Competitive; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa | 1985 |
N-tetrahydrofurfuryl benzomorphans: comparison of a kappa and an agonist/antagonist analgesic.
Topics: 3,4-Dihydroxyphenylacetic Acid; Analgesics; Animals; Benzomorphans; Corpus Striatum; Dopamine; Homovanillic Acid; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Structure-Activity Relationship | 1985 |
Psychotomimesis mediated by kappa opiate receptors.
Topics: Adult; Anxiety; Benzomorphans; Humans; Male; Middle Aged; Morphinans; Naloxone; Personality Tests; Phencyclidine; Receptors, Opioid; Receptors, Opioid, kappa | 1986 |
Effects of a kappa-opioid agonist on adrenocorticotropic and diuretic function in man.
Topics: Adrenocorticotropic Hormone; Adult; Benzomorphans; Diuresis; Humans; Hydrocortisone; Male; Morphinans; Naloxone; Pituitary Hormones; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Vasopressins | 1986 |
Anterior pituitary hormone responses to a kappa-opioid agonist in man.
Topics: Adult; Benzomorphans; Follicle Stimulating Hormone; Growth Hormone; Humans; Kinetics; Luteinizing Hormone; Male; Morphinans; Naloxone; Pituitary Hormones, Anterior; Prolactin; Reference Values; Thyrotropin | 1986 |
Multiple brain sites sensitive to feeding stimulation by opioid agonists: a cannula-mapping study.
Topics: Animals; Benzomorphans; Brain; Brain Mapping; Dose-Response Relationship, Drug; Enkephalin, Methionine; Feeding Behavior; Male; Morphinans; Morphine; Rats; Rats, Inbred Strains; Time Factors | 1988 |
Kappa opioids in rhesus monkeys. III. Dependence associated with chronic administration.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Cyclazocine; Drug Tolerance; Endorphins; Ethylketocyclazocine; Macaca mulatta; Morphinans; Morphine; Narcotic Antagonists; Pentobarbital; Pyrrolidines; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors | 1987 |
Substitution and primary dependence studies in animals.
Topics: Animals; Behavior, Animal; Benzomorphans; Buprenorphine; Butorphanol; Codeine; Discrimination, Psychological; Humans; Macaca mulatta; Morphinans; Morphine; Morphine Dependence; Nalbuphine; Narcotic Antagonists; Pentazocine; Piperidines; Substance Withdrawal Syndrome | 1985 |
Mr 2033 CL--a novel non-morphine-like opioid analgesic.
Topics: Analgesics, Opioid; Animals; Benzomorphans; Humans; Mice; Morphinans; Morphine; Naloxone; Rabbits; Rats; Reaction Time; Receptors, Opioid; Receptors, Opioid, kappa; Stereotyped Behavior | 1983 |
[3H]Mr 2034 labels a high affinity opioid kappa-receptor not accessible to naloxazone.
Topics: Animals; Benzomorphans; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa | 1983 |
Cardiovascular and respiratory effects of mu-, delta- and kappa-opiate agonists microinjected into the anterior hypothalamic brain area of awake rats.
Topics: Animals; Anterior Hypothalamic Nucleus; Benzomorphans; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Heart Rate; Male; Microinjections; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Respiration; Wakefulness | 1983 |
The binding to rat brain homogenates of Mr2034, a universal opiate.
Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |