Page last updated: 2024-09-03

mr 2034 and morphinans

mr 2034 has been researched along with morphinans in 16 studies

Compound Research Comparison

Studies
(mr 2034)
Trials
(mr 2034)
Recent Studies (post-2010)
(mr 2034)
Studies
(morphinans)
Trials
(morphinans)
Recent Studies (post-2010) (morphinans)
48003,251307648

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-199016 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Iyengar, S; Kim, HS; Wood, PL1
Herz, A; Nikolarakis, K; Pfeiffer, A; Stalla, GK1
Männistö, PT; Rauhala, P; Tuominen, RK1
Coupar, JM; Quinn, MJ1
Ensinger, HA2
Wood, PL1
Brantl, V; Emrich, HM; Herz, A; Pfeiffer, A1
Brantl, V; Braun, S; Knepel, W; Lohmann, H; Meyer, HD; Pfeiffer, A1
Brantl, V; Braun, S; Mann, K; Meyer, HD; Pfeiffer, A1
Lanthier, D; Leibowitz, SF; Stanley, BG1
Dykstra, LA; Gmerek, DE; Woods, JH1
Gmerek, DE; Woods, JH1
Ensinger, HA; Gaida, W; Jennewein, HM; Merz, H; Stockhaus, K1
Faden, AI; Feuerstein, G; Kopin, IJ; Pfeiffer, A1
Johnson, N; Pasternak, GW1

Other Studies

16 other study(ies) available for mr 2034 and morphinans

ArticleYear
Reversal of the actions of morphine on mesocortical dopamine metabolism in the rat by the kappa agonist MR-2034: tentative mu-2 opioid control of mesocortical dopaminergic projections.
    Life sciences, 1987, Oct-05, Volume: 41, Issue:14

    Topics: Animals; Benzomorphans; Brain; Cerebral Cortex; Corpus Striatum; Dopamine; Frontal Lobe; Gyrus Cinguli; Male; Morphinans; Morphine; Olfactory Bulb; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu

1987
The role of CRF in the release of ACTH by opiate agonists and antagonists in rats.
    Brain research, 1987, Sep-22, Volume: 421, Issue:1-2

    Topics: Adrenocorticotropic Hormone; Animals; Benzomorphans; Corticotropin-Releasing Hormone; Immune Sera; Male; Morphinans; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid

1987
Opiate receptor subtypes in the regulation of thyrotropin and prolactin secretion in the rat.
    Hormone research, 1988, Volume: 29, Issue:5-6

    Topics: Animals; Benzomorphans; Cerebral Ventricles; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Injections, Intraventricular; Kinetics; Male; Morphinans; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reference Values; Thyrotropin

1988
The effects of the selective kappa-opioid agonist MR 2034 on the guinea-pig ileum.
    The Journal of pharmacy and pharmacology, 1988, Volume: 40, Issue:5

    Topics: Animals; Benzomorphans; Female; Guinea Pigs; Ileum; Male; Morphinans; Receptors, Opioid; Receptors, Opioid, kappa

1988
Differentiating aspects of opioid receptor binding by [3H](-) (1R,5R,9R,2''S)-5,9-dimethyl-2-tetrahydrofurfuryl-2'-hydroxy-6,7- benzomorphan hydrochloride ([3H]Mr 2034), a drug preferentially acting on kappa-receptors.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Animals; Benzomorphans; Binding, Competitive; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1985
N-tetrahydrofurfuryl benzomorphans: comparison of a kappa and an agonist/antagonist analgesic.
    Neuropeptides, 1985, Volume: 5, Issue:4-6

    Topics: 3,4-Dihydroxyphenylacetic Acid; Analgesics; Animals; Benzomorphans; Corpus Striatum; Dopamine; Homovanillic Acid; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Structure-Activity Relationship

1985
Psychotomimesis mediated by kappa opiate receptors.
    Science (New York, N.Y.), 1986, Aug-15, Volume: 233, Issue:4765

    Topics: Adult; Anxiety; Benzomorphans; Humans; Male; Middle Aged; Morphinans; Naloxone; Personality Tests; Phencyclidine; Receptors, Opioid; Receptors, Opioid, kappa

1986
Effects of a kappa-opioid agonist on adrenocorticotropic and diuretic function in man.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1986, Volume: 18, Issue:12

    Topics: Adrenocorticotropic Hormone; Adult; Benzomorphans; Diuresis; Humans; Hydrocortisone; Male; Morphinans; Naloxone; Pituitary Hormones; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Vasopressins

1986
Anterior pituitary hormone responses to a kappa-opioid agonist in man.
    The Journal of clinical endocrinology and metabolism, 1986, Volume: 62, Issue:1

    Topics: Adult; Benzomorphans; Follicle Stimulating Hormone; Growth Hormone; Humans; Kinetics; Luteinizing Hormone; Male; Morphinans; Naloxone; Pituitary Hormones, Anterior; Prolactin; Reference Values; Thyrotropin

1986
Multiple brain sites sensitive to feeding stimulation by opioid agonists: a cannula-mapping study.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:4

    Topics: Animals; Benzomorphans; Brain; Brain Mapping; Dose-Response Relationship, Drug; Enkephalin, Methionine; Feeding Behavior; Male; Morphinans; Morphine; Rats; Rats, Inbred Strains; Time Factors

1988
Kappa opioids in rhesus monkeys. III. Dependence associated with chronic administration.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Cyclazocine; Drug Tolerance; Endorphins; Ethylketocyclazocine; Macaca mulatta; Morphinans; Morphine; Narcotic Antagonists; Pentobarbital; Pyrrolidines; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1987
Substitution and primary dependence studies in animals.
    Drug and alcohol dependence, 1985, Volume: 14, Issue:3-4

    Topics: Animals; Behavior, Animal; Benzomorphans; Buprenorphine; Butorphanol; Codeine; Discrimination, Psychological; Humans; Macaca mulatta; Morphinans; Morphine; Morphine Dependence; Nalbuphine; Narcotic Antagonists; Pentazocine; Piperidines; Substance Withdrawal Syndrome

1985
Mr 2033 CL--a novel non-morphine-like opioid analgesic.
    NIDA research monograph, 1983, Volume: 43

    Topics: Analgesics, Opioid; Animals; Benzomorphans; Humans; Mice; Morphinans; Morphine; Naloxone; Rabbits; Rats; Reaction Time; Receptors, Opioid; Receptors, Opioid, kappa; Stereotyped Behavior

1983
[3H]Mr 2034 labels a high affinity opioid kappa-receptor not accessible to naloxazone.
    European journal of pharmacology, 1983, Apr-22, Volume: 89, Issue:1-2

    Topics: Animals; Benzomorphans; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1983
Cardiovascular and respiratory effects of mu-, delta- and kappa-opiate agonists microinjected into the anterior hypothalamic brain area of awake rats.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:3

    Topics: Animals; Anterior Hypothalamic Nucleus; Benzomorphans; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Heart Rate; Male; Microinjections; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Respiration; Wakefulness

1983
The binding to rat brain homogenates of Mr2034, a universal opiate.
    Life sciences, 1983, Sep-05, Volume: 33, Issue:10

    Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid

1983