mr 2034 has been researched along with enkephalin, leucine-2-alanine in 9 studies
| Studies (mr 2034) | Trials (mr 2034) | Recent Studies (post-2010) (mr 2034) | Studies (enkephalin, leucine-2-alanine) | Trials (enkephalin, leucine-2-alanine) | Recent Studies (post-2010) (enkephalin, leucine-2-alanine) |
|---|---|---|---|---|---|
| 48 | 0 | 0 | 1,581 | 23 | 74 |
| Protein | Taxonomy | mr 2034 (IC50) | enkephalin, leucine-2-alanine (IC50) |
|---|---|---|---|
| Delta-type opioid receptor | Mus musculus (house mouse) | 0.0915 | |
| Delta-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0017 | |
| Kappa-type opioid receptor | Mus musculus (house mouse) | 0.009 | |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0419 | |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | 1.4691 | |
| Mu-type opioid receptor | Mus musculus (house mouse) | 0.009 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 9 (100.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Smith, CB | 1 |
| Geppert, M; Illes, P; Jackisch, R | 1 |
| Brenner, AS; Geppert, M; Illes, P; Jackisch, R | 1 |
| Ensinger, HA | 1 |
| Havemann, U; Kuschinsky, K | 1 |
| Bradley, PB; Brookes, A | 1 |
| Rubini, P; Schulz, R; Wüster, M | 1 |
| Faden, AI; Feuerstein, G; Kopin, IJ; Pfeiffer, A | 1 |
| Johnson, N; Pasternak, GW | 1 |
9 other study(ies) available for mr 2034 and enkephalin, leucine-2-alanine
| Article | Year |
|---|---|
New approaches to the evaluation of opioid agonists and antagonists upon the isolated, electrically stimulated mouse vas deferens preparation.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Oligopeptides; Pyrrolidines; Receptors, Opioid; Vas Deferens | 1987 |
Characterization of opioid receptors modulating noradrenaline release in the hippocampus of the rabbit.
Topics: Animals; Benzomorphans; Clonidine; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hippocampus; Morphine; Norepinephrine; Rabbits; Receptors, Opioid | 1986 |
Presynaptic opioid receptors modulating acetylcholine release in the hippocampus of the rabbit.
Topics: Acetylcholine; Animals; Benzomorphans; Choline; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hippocampus; Naloxone; Peptide Fragments; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Synapses | 1986 |
Differentiating aspects of opioid receptor binding by [3H](-) (1R,5R,9R,2''S)-5,9-dimethyl-2-tetrahydrofurfuryl-2'-hydroxy-6,7- benzomorphan hydrochloride ([3H]Mr 2034), a drug preferentially acting on kappa-receptors.
Topics: Animals; Benzomorphans; Binding, Competitive; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa | 1985 |
Locomotor activity of rats after injection of various opioids into the nucleus accumbens and the septum mediale.
Topics: Animals; Benzomorphans; Drug Synergism; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Injections; Male; Morphine; Motor Activity; Naloxone; Narcotics; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Septum Pellucidum | 1985 |
The effects of kappa opioid agonists in the rat hippocampal slice.
Topics: Animals; Benzodiazepines; Benzomorphans; Electrophysiology; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Hippocampus; In Vitro Techniques; Male; Narcotics; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa | 1984 |
The preference of putative pro-enkephalins for different types of opiate receptors.
Topics: Animals; Benzomorphans; Brain; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Fentanyl; Guinea Pigs; Ileum; Male; Mice; Morphine; Protein Precursors; Rats; Receptors, Opioid; Vas Deferens | 1981 |
Cardiovascular and respiratory effects of mu-, delta- and kappa-opiate agonists microinjected into the anterior hypothalamic brain area of awake rats.
Topics: Animals; Anterior Hypothalamic Nucleus; Benzomorphans; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Heart Rate; Male; Microinjections; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Respiration; Wakefulness | 1983 |
The binding to rat brain homogenates of Mr2034, a universal opiate.
Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid | 1983 |