Page last updated: 2024-09-03

mr 2034 and cyclazocine

mr 2034 has been researched along with cyclazocine in 12 studies

Compound Research Comparison

Studies
(mr 2034)
Trials
(mr 2034)
Recent Studies (post-2010)
(mr 2034)
Studies
(cyclazocine)
Trials
(cyclazocine)
Recent Studies (post-2010) (cyclazocine)
4800855307

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-199012 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chahl, LA1
Geppert, M; Illes, P; Jackisch, R1
Brenner, AS; Geppert, M; Illes, P; Jackisch, R1
Ensinger, HA2
Abbott, FV; Franklin, KB; Libman, RB1
Hart, JC; Leander, JD; Zerbe, RL1
Dykstra, LA; Gmerek, DE; Woods, JH1
Fitzjarrell, AT; Heath, RG; Walker, CF1
Johnson, N; Pasternak, GW1
Hayes, AG; Tyers, MB1
Altura, BM; Altura, BT; Quirion, R1

Other Studies

12 other study(ies) available for mr 2034 and cyclazocine

ArticleYear
Withdrawal responses of guinea-pig isolated ileum following brief exposure to opiates and opioid peptides.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:4

    Topics: Animals; Benzomorphans; Buprenorphine; Cyclazocine; Endorphins; Ethylketocyclazocine; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Naloxone; Narcotics; Substance P; Substance Withdrawal Syndrome

1986
Characterization of opioid receptors modulating noradrenaline release in the hippocampus of the rabbit.
    Journal of neurochemistry, 1986, Volume: 46, Issue:6

    Topics: Animals; Benzomorphans; Clonidine; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hippocampus; Morphine; Norepinephrine; Rabbits; Receptors, Opioid

1986
Presynaptic opioid receptors modulating acetylcholine release in the hippocampus of the rabbit.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2

    Topics: Acetylcholine; Animals; Benzomorphans; Choline; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hippocampus; Naloxone; Peptide Fragments; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Synapses

1986
Differentiating aspects of opioid receptor binding by [3H](-) (1R,5R,9R,2''S)-5,9-dimethyl-2-tetrahydrofurfuryl-2'-hydroxy-6,7- benzomorphan hydrochloride ([3H]Mr 2034), a drug preferentially acting on kappa-receptors.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Animals; Benzomorphans; Binding, Competitive; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1985
A dose-ratio comparison of mu and kappa agonists in formalin and thermal pain.
    Life sciences, 1986, Nov-24, Volume: 39, Issue:21

    Topics: Analgesia; Animals; Benzomorphans; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Fentanyl; Formaldehyde; Hot Temperature; Male; Naloxone; Pain; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sufentanil

1986
Kappa agonist-induced diuresis: evidence for stereoselectivity, strain differences, independence of hydration variables and a result of decreased plasma vasopressin levels.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Butorphanol; Cyclazocine; Diuresis; Drinking; Ethylketocyclazocine; Female; Male; Nalorphine; Pyrrolidines; Rats; Rats, Inbred Strains; Rats, Zucker; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Vasopressins; Water Deprivation

1987
Kappa opioids in rhesus monkeys. III. Dependence associated with chronic administration.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Cyclazocine; Drug Tolerance; Endorphins; Ethylketocyclazocine; Macaca mulatta; Morphinans; Morphine; Narcotic Antagonists; Pentobarbital; Pyrrolidines; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1987
Kappa opiate receptor agonists: effects on behavior and on brain function and structure in rhesus monkeys.
    Biological psychiatry, 1984, Volume: 19, Issue:7

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Behavior, Animal; Benzomorphans; Brain; Computers; Cyclazocine; Dose-Response Relationship, Drug; Electroencephalography; Ethylketocyclazocine; Evoked Potentials; Macaca mulatta; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa

1984
[3H]Mr 2034 labels a high affinity opioid kappa-receptor not accessible to naloxazone.
    European journal of pharmacology, 1983, Apr-22, Volume: 89, Issue:1-2

    Topics: Animals; Benzomorphans; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1983
The binding to rat brain homogenates of Mr2034, a universal opiate.
    Life sciences, 1983, Sep-05, Volume: 33, Issue:10

    Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid

1983
Determination of receptors that mediate opiate side effects in the mouse.
    British journal of pharmacology, 1983, Volume: 79, Issue:3

    Topics: Analgesics; Animals; Benzamides; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Female; Gastrointestinal Motility; Male; Mice; Narcotic Antagonists; Narcotics; Pentazocine; Pupil; Receptors, Opioid; Respiration; Rotation; Tail

1983
Identification of benzomorphan-kappa opiate receptors in cerebral arteries which subserve relaxation.
    British journal of pharmacology, 1984, Volume: 82, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Cerebral Arteries; Cyclazocine; Dinoprost; Dogs; Drug Interactions; Ethylketocyclazocine; Female; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Phencyclidine; Prostaglandins F; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa

1984