Page last updated: 2024-09-03

mr 2034 and bremazocine

mr 2034 has been researched along with bremazocine in 5 studies

Compound Research Comparison

Studies
(mr 2034)
Trials
(mr 2034)
Recent Studies (post-2010)
(mr 2034)
Studies
(bremazocine)
Trials
(bremazocine)
Recent Studies (post-2010) (bremazocine)
480032304

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19905 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bergman, J; Howell, LL; Morse, WH1
Ensinger, HA1
Hart, JC; Leander, JD; Zerbe, RL1
Hayes, AG; Tyers, MB1
Altura, BM; Altura, BT; Quirion, R1

Other Studies

5 other study(ies) available for mr 2034 and bremazocine

ArticleYear
Effects of levorphanol and several kappa-selective opioids on respiration and behavior in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Behavior, Animal; Benzodiazepines; Benzomorphans; Carbon Dioxide; Levorphanol; Macaca mulatta; Male; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Respiration

1988
Differentiating aspects of opioid receptor binding by [3H](-) (1R,5R,9R,2''S)-5,9-dimethyl-2-tetrahydrofurfuryl-2'-hydroxy-6,7- benzomorphan hydrochloride ([3H]Mr 2034), a drug preferentially acting on kappa-receptors.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Animals; Benzomorphans; Binding, Competitive; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1985
Kappa agonist-induced diuresis: evidence for stereoselectivity, strain differences, independence of hydration variables and a result of decreased plasma vasopressin levels.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Butorphanol; Cyclazocine; Diuresis; Drinking; Ethylketocyclazocine; Female; Male; Nalorphine; Pyrrolidines; Rats; Rats, Inbred Strains; Rats, Zucker; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Vasopressins; Water Deprivation

1987
Determination of receptors that mediate opiate side effects in the mouse.
    British journal of pharmacology, 1983, Volume: 79, Issue:3

    Topics: Analgesics; Animals; Benzamides; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Female; Gastrointestinal Motility; Male; Mice; Narcotic Antagonists; Narcotics; Pentazocine; Pupil; Receptors, Opioid; Respiration; Rotation; Tail

1983
Identification of benzomorphan-kappa opiate receptors in cerebral arteries which subserve relaxation.
    British journal of pharmacology, 1984, Volume: 82, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Cerebral Arteries; Cyclazocine; Dinoprost; Dogs; Drug Interactions; Ethylketocyclazocine; Female; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Phencyclidine; Prostaglandins F; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa

1984