Page last updated: 2024-09-03

mozavaptan and aldosterone

mozavaptan has been researched along with aldosterone in 5 studies

Compound Research Comparison

Studies
(mozavaptan)
Trials
(mozavaptan)
Recent Studies (post-2010)
(mozavaptan)
Studies
(aldosterone)
Trials
(aldosterone)
Recent Studies (post-2010) (aldosterone)
16582425,3331,5174,169

Protein Interaction Comparison

ProteinTaxonomymozavaptan (IC50)aldosterone (IC50)
Mineralocorticoid receptor Homo sapiens (human)0.0048
Mineralocorticoid receptorRattus norvegicus (Norway rat)0.043

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (60.00)18.2507
2000's2 (40.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Shimizu, K1
Fujihara, H; Inoue, T; Ohnishi, A; Okahara, R; Orita, Y; Tanaka, T; Yabuuchi, Y; Yamamura, Y1
Arroyo, V; Bordas, N; Bosch-Marcé, M; Jiménez, W; Leivas, A; Morales-Ruiz, M; Muñoz, RM; Pérez, M; Poo, JL; Rivera, F; Rodés, J1
Cadnapaphornchai, MA; Chen, YC; Falk, S; Li, C; Schrier, RW; Summer, SN; Wang, W1
Bie, P; Mølstrøm, S; Wamberg, S1

Trials

1 trial(s) available for mozavaptan and aldosterone

ArticleYear
Aquaretic effects of the nonpeptide V2 antagonist OPC-31260 in hydropenic humans.
    Kidney international, 1995, Volume: 48, Issue:1

    Topics: 6-Ketoprostaglandin F1 alpha; Adult; Aldosterone; Angiotensin II; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Atrial Natriuretic Factor; Benzazepines; Blood Pressure; Calcium; Creatinine; Dinoprostone; Epinephrine; Heart Rate; Humans; Male; Norepinephrine; Osmolar Concentration; Phosphates; Potassium; Sodium; Thromboxane B2; Uric Acid; Urine; Water; Water Deprivation

1995

Other Studies

4 other study(ies) available for mozavaptan and aldosterone

ArticleYear
Potent aquaretic agent. A novel nonpeptide selective vasopressin 2 antagonist (OPC-31260) in men.
    The Journal of clinical investigation, 1993, Volume: 92, Issue:6

    Topics: Adult; Aldosterone; Analysis of Variance; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Blood Pressure; Chlorides; Diuresis; Diuretics; Dose-Response Relationship, Drug; Furosemide; Heart Rate; Humans; Male; Osmolar Concentration; Potassium; Renin; Sodium; Time Factors; Urine

1993
Comparison of two aquaretic drugs (niravoline and OPC-31260) in cirrhotic rats with ascites and water retention.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:1

    Topics: Aldosterone; Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Benzeneacetamides; Body Water; Body Weight; Carbon Tetrachloride Poisoning; Diuretics; Hemodynamics; Hormones; Hypothalamus; Kidney; Liver Cirrhosis, Experimental; Male; Osmolar Concentration; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa; RNA, Messenger; Urodynamics; Vasopressins

1999
Molecular analysis of impaired urinary diluting capacity in glucocorticoid deficiency.
    American journal of physiology. Renal physiology, 2006, Volume: 290, Issue:5

    Topics: Aldosterone; Animals; Anti-Inflammatory Agents; Aquaporins; Benzazepines; Dexamethasone; Glucocorticoids; Male; Osmolar Concentration; Rats; Rats, Wistar; Sodium; Sodium Channels; Up-Regulation; Urine; Water-Electrolyte Balance

2006
Normotensive sodium loading in conscious dogs: regulation of renin secretion during beta-receptor blockade.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2009, Volume: 296, Issue:2

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Aldosterone; Angiotensin II; Animals; Antidiuretic Hormone Receptor Antagonists; Atrial Natriuretic Factor; Benzazepines; Blood Pressure; Consciousness; Diet, Sodium-Restricted; Dogs; Female; Glomerular Filtration Rate; Heart Rate; Hormone Antagonists; Infusions, Intravenous; Juxtaglomerular Apparatus; Metoprolol; Natriuresis; Norepinephrine; Potassium; Receptors, Adrenergic, beta-1; Receptors, Vasopressin; Renin; Renin-Angiotensin System; Sodium; Sodium Chloride; Sympathetic Nervous System; Time Factors

2009