Page last updated: 2024-08-16

moxonidine and rilmenidine

moxonidine has been researched along with rilmenidine in 56 studies

Research

Studies (56)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's34 (60.71)18.2507
2000's17 (30.36)29.6817
2010's5 (8.93)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arrault, A; Guillaumet, G; Mérour, JY; Pfeiffer, B; Renard, P; Rettori, MC; Scalbert, E; Touzeau, F1
Agbaba, D; Filipic, S; Nikolic, K1
Bousquet, P; Ehrhardt, JD; Feldman, J; Fellmann, L; Gasparik, V; Greney, H; Schann, S1
Agbaba, D; Azzali, E; Costantino, G; Glisic, S; Laurila, JM; Nikolic, K; Perovic, V; Pieroni, M; Radi, M; Scheinin, M; Srdic-Rajic, T; Tassini, S; Veljkovic, N; Vucicevic, J1
Christen, O; Göthert, M; Michel, MC; Molderings, GJ; Schäfer, SG1
Gregoire, JR; Sheps, SG1
Starke, K; Szabo, B; Urban, R1
Jacob, R; Rupp, H1
Szabo, B; Urban, R2
Elliott, HL; MacPhee, G; Panfilov, V; Reid, JL1
Li, P; Penner, SB; Smyth, DD1
Christen, MO; Collins, LA; Dreshaj, I; Ernsberger, P; Graff, LM; Graves, ME; Grove, DL; Haxhiu, MA; Schäfer, SG1
Christen, O; Göthert, M; Molderings, GJ; Schäfer, SG1
Chan, CK; Head, GA; Sannajust, F1
Chudek, J; Nowicki, M; Wiecek, A1
Chan, CK; Head, GA1
Frishman, WH; Yu, A1
van Zwieten, PA3
Lada, W1
Piletz, JE; Reis, DJ1
Kunduzova, OR; Medvedev, OS; Medvedeva, NA; Murashev, AN3
Godwin, SJ; Head, GA; Parkin, ML; Tortelli, CF1
Blue, DR; Dillon, MP; Eglen, RM; Jasper, JR; Lesnick, JD; MacLennan, SJ; Zhu, QM2
Bock, C; Niederhoffer, N; Szabo, B1
Drzewoski, J; Wiśniewska-Jarosińska, M1
Bock, C; Niederhoffer, N; Nordheim, U; Szabo, B1
Head, GA1
Peters, SL; Van Zwieten, PA1
Masek, K; Sevcík, J1
Bousquet, P; Feldman, J1
Robles, NR1
Bönisch, H; Brüss, M; Göthert, M; Likungu, J; Molderings, GJ1
Spinar, J; Vítovec, J1
Schachter, M1
Fritz, T; Szabo, B; Wedzony, K1
Nurminen, ML1
Godwin, SJ; Head, GA; Parkin, ML1
Camilleri, G; Clerson, P; Portal, B; Quiniou, G1
Ernsberger, P; Koletsky, RJ; Velliquette, RA1
Burgdorf, C; Engelhardt, A; Kurz, T; Raasch, W; Richardt, G; Schäfer, U1
Forzley, B; Penner, SB; Pirnat, D; Smyth, DD1
de Arruda Camargo, LA; Guarda, IF; Guarda, RS; Saad, WA; Simões, S1
Kotanko, P1
Ernsberger, P; Kossover, R; Previs, SF; Velliquette, RA1
Cong, B; Li, F; Li, J; Lu, XQ; Su, RB; Wu, N; Xu, B; Zheng, JQ1
Sica, DA1
Li, F; Li, J; Liu, Y; Lu, XQ; Su, RB; Wu, N1
Bousquet, P; Lessa, MA; Nascimento, AR; Sabino, B; Tibiriçá, E1
Agbaba, D; Gemovic, B; Nikolic, K; Srdic-Rajic, T; Veljkovic, N1

Reviews

19 review(s) available for moxonidine and rilmenidine

ArticleYear
[Imidazole receptors: site of action of a new generation of antihypertensive drugs. Current status and future prospects].
    Deutsche medizinische Wochenschrift (1946), 1992, Jan-10, Volume: 117, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Binding Sites; Cattle; Humans; Imidazoles; Oxazoles; Rats; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1992
Newer antihypertensive drugs.
    Current opinion in cardiology, 1995, Volume: 10, Issue:5

    Topics: Antihypertensive Agents; Dibenzothiepins; Humans; Imidazoles; Methionine; Oxazoles; Piperazines; Protease Inhibitors; Rilmenidine

1995
Clinical pharmacology of drugs acting on imidazoline and adrenergic receptors. Studies with clonidine, moxonidine, rilmenidine, and atenolol.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Antihypertensive Agents; Atenolol; Clinical Trials as Topic; Clonidine; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Placebos; Receptors, Adrenergic; Receptors, Drug; Reference Values; Rilmenidine

1995
[Imidazole receptors and blood pressure regulation. High receptor selectivity of moxonidine].
    Deutsche medizinische Wochenschrift (1946), 1993, Jun-25, Volume: 118, Issue:25

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Cats; Clonidine; Humans; Hypertension; Imidazoles; Oxazoles; Rabbits; Rats; Receptors, Drug; Rilmenidine

1993
[Imidazol receptor agonists--new possibilities for treating hypertension].
    Postepy higieny i medycyny doswiadczalnej, 1995, Volume: 49, Issue:5

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Hemodynamics; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1995
Imidazoline receptor agonist drugs: a new approach to the treatment of systemic hypertension.
    Journal of clinical pharmacology, 1996, Volume: 36, Issue:2

    Topics: Animals; Antihypertensive Agents; Clinical Trials as Topic; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1996
From alpha and beta to I1: an overview of sympathetic receptors involved in blood pressure control targets for drug treatment.
    Journal of cardiovascular pharmacology, 1996, Volume: 27 Suppl 3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Drug; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Rilmenidine

1996
[Imidazoline receptors and use of drug blocking receptors I1].
    Polski merkuriusz lekarski : organ Polskiego Towarzystwa Lekarskiego, 1996, Volume: 1, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Antihypertensive Agents; Arrhythmias, Cardiac; Cimetidine; Histamine H2 Antagonists; Humans; Hypertension; Imidazoles; Myocardial Infarction; Oxazoles; Rilmenidine

1996
The imidazoline receptor in control of blood pressure by clonidine and allied drugs.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Humans; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Neurons; Oxazoles; Receptors, Drug; Rilmenidine

1997
Central imidazoline (I1) receptors as targets of centrally acting antihypertensives: moxonidine and rilmenidine.
    Journal of hypertension, 1997, Volume: 15, Issue:2

    Topics: Animals; Antihypertensive Agents; Brain; Humans; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1997
[Clinical pharmacology of hypotensive drugs acting on central imidazoline receptors].
    Polskie Archiwum Medycyny Wewnetrznej, 1998, Volume: 100, Issue:6

    Topics: Antihypertensive Agents; Clonidine; Drug Interactions; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1998
Central I1-imidazoline receptors as targets of centrally acting antihypertensive drugs. Clinical pharmacology of moxonidine and rilmenidine.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Brain; Clinical Trials as Topic; Clonidine; Hemodynamics; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1999
[New, modern, centrally active antihypertensive agents in the treatment of essential hypertension].
    Casopis lekaru ceskych, 1999, Jun-07, Volume: 138, Issue:12

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Imidazoles; Medulla Oblongata; Oxazoles; Rilmenidine

1999
Drugs acting on imidazoline receptors: a review of their pharmacology, their use in blood pressure control and their potential interest in cardioprotection.
    Drugs, 1999, Volume: 58, Issue:5

    Topics: Animals; Antihypertensive Agents; Arrhythmias, Cardiac; Clinical Trials as Topic; Heart Failure; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1999
Metabolic effects of moxonidine and other centrally acting antihypertensives.
    Diabetes, obesity & metabolism, 1999, Volume: 1, Issue:6

    Topics: Animals; Antihypertensive Agents; Diabetes Complications; Humans; Hypertension; Imidazoles; Insulin Resistance; Metabolism; Oxazoles; Rilmenidine; Sympathetic Nervous System; Sympatholytics; Syndrome

1999
[Central nervous system as a target for the new antihypertensive agents].
    Duodecim; laaketieteellinen aikakauskirja, 1999, Volume: 115, Issue:20

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Autonomic Fibers, Preganglionic; Brain; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Oxazoles; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Sympatholytics

1999
Centrally acting imidazoline I1-receptor agonists: do they have a place in the management of hypertension?
    American journal of cardiovascular drugs : drugs, devices, and other interventions, 2001, Volume: 1, Issue:5

    Topics: Animals; Antihypertensive Agents; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

2001
Cause and consequences of sympathetic hyperactivity in chronic kidney disease.
    Blood purification, 2006, Volume: 24, Issue:1

    Topics: Adrenergic alpha-Agonists; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Arginine; Brain Stem; Humans; Hyperkinesis; Hypertension, Renal; Imidazoles; Kidney Failure, Chronic; Nitric Oxide Synthase; Oxazoles; Receptor, Angiotensin, Type 1; Renal Dialysis; Rilmenidine; Sympathetic Nervous System; Sympatholytics

2006
Centrally acting antihypertensive agents: an update.
    Journal of clinical hypertension (Greenwich, Conn.), 2007, Volume: 9, Issue:5

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Clonidine; Contraindications; Guanabenz; Guanfacine; Humans; Hypertension; Imidazoles; Methyldopa; Oxazoles; Rilmenidine

2007

Trials

1 trial(s) available for moxonidine and rilmenidine

ArticleYear
[Comparison of the antihypertensive efficacy of and tolerance to 2 imidazoline receptor agonists: moxonidine and rilmenidine in monotherapy].
    Annales de cardiologie et d'angeiologie, 2001, Volume: 50, Issue:3

    Topics: Antihypertensive Agents; Female; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Male; Middle Aged; Oxazoles; Receptors, Drug; Rilmenidine; Severity of Illness Index

2001

Other Studies

36 other study(ies) available for moxonidine and rilmenidine

ArticleYear
Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.
    Journal of medicinal chemistry, 2003, May-08, Volume: 46, Issue:10

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Cattle; Frontal Lobe; Heart Rate; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Oxazines; Rabbits; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship

2003
QSAR study of imidazoline antihypertensive drugs.
    Bioorganic & medicinal chemistry, 2008, Aug-01, Volume: 16, Issue:15

    Topics: Antihypertensive Agents; Binding Sites; Imidazoline Receptors; Imidazolines; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship

2008
Synthesis and biological evaluation of 2-aryliminopyrrolidines as selective ligands for I1 imidazoline receptors: discovery of new sympatho-inhibitory hypotensive agents with potential beneficial effects in metabolic syndrome.
    Journal of medicinal chemistry, 2015, Jan-22, Volume: 58, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Blood-Brain Barrier; Drug Discovery; Heart Rate; Imidazoline Receptors; Ligands; Metabolic Syndrome; Pyrrolidines; Rats; Rats, Wistar; Structure-Activity Relationship; Sympatholytics

2015
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin.
    Bioorganic & medicinal chemistry, 2016, 07-15, Volume: 24, Issue:14

    Topics: Adrenergic alpha-Agonists; Antibiotics, Antineoplastic; Apoptosis; Doxorubicin; Drug Synergism; Humans; K562 Cells; Ligands; Molecular Structure; Oxazoles; Receptors, Adrenergic, alpha-2; Rilmenidine

2016
Involvement of peripheral presynaptic inhibition in the reduction of sympathetic tone by moxonidine, rilmenidine and UK 14304.
    European journal of pharmacology, 1995, Aug-25, Volume: 282, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Female; Imidazoles; Male; Neural Inhibition; Oxazoles; Peripheral Nervous System; Presynaptic Terminals; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Vasoconstrictor Agents

1995
Excess catecholamines and the metabolic syndrome: should central imidazoline receptors be a therapeutic target?
    Medical hypotheses, 1995, Volume: 44, Issue:3

    Topics: Animals; Antihypertensive Agents; Cardiovascular Diseases; Catecholamines; Energy Intake; Energy Metabolism; Humans; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Models, Biological; Neurons; Obesity; Oxazoles; Receptors, Drug; Rilmenidine; Social Conditions; Stress, Psychological; Sympathetic Nervous System

1995
Mechanism of sympathoinhibition by imidazolines.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzazepines; Brimonidine Tartrate; Dioxanes; Hemodynamics; Idazoxan; Imidazoles; Oxazoles; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1995
Attenuated renal response to moxonidine and rilmenidine in one kidney-one clip hypertensive rats.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Hemodynamics; Hypertension, Renovascular; Imidazoles; Infusions, Intra-Arterial; Kidney; Male; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Renal Circulation; Rilmenidine; Sodium; Urodynamics

1994
A novel mechanism of action for hypertension control: moxonidine as a selective I1-imidazoline agonist.
    Cardiovascular drugs and therapy, 1994, Volume: 8 Suppl 1

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Autoradiography; Binding Sites; Blood Pressure; Cattle; Cells, Cultured; Clonidine; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1994
Role of imidazoline receptors in the cardiovascular actions of moxonidine, rilmenidine and clonidine in conscious rabbits.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1996
Relative importance of central imidazoline receptors for the antihypertensive effects of moxonidine and rilmenidine.
    Journal of hypertension, 1996, Volume: 14, Issue:7

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiac Catheterization; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intravenous; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Time Factors

1996
Role of I1 imidazoline receptors in the sympathoinhibition produced by intracisternally administered rilmenidine and moxonidine.
    Arzneimittel-Forschung, 1997, Volume: 47, Issue:9

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Cisterna Magna; Dose-Response Relationship, Drug; Female; Guanabenz; Heart Rate; Imidazoles; Imidazoline Receptors; Injections; Male; Norepinephrine; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Yohimbine

1997
Chronopharmacological dependence of antihypertensive effects of the imidazoline-like drugs in stroke-prone spontaneously hypertensive rats.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cerebrovascular Disorders; Circadian Rhythm; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Imidazoles; Male; Motor Activity; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine

1998
Comparison of the baroreceptor-heart rate reflex effects of moxonidine, rilmenidine and clonidine in conscious rabbits.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Algorithms; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Clonidine; Female; Heart Rate; Imidazoles; Injections, Intraventricular; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Vagus Nerve

1998
Influence of sino-aortic barodenervation on the cardiovascular effects of imidazoline-like drugs.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Circadian Rhythm; Clonidine; Denervation; Heart Rate; Imidazoles; Injections, Intravenous; Male; Motor Activity; Oxazoles; Pressoreceptors; Rats; Rats, Wistar; Rilmenidine; Sinus of Valsalva; Telemetry

1998
Cardiovascular effects of rilmenidine, moxonidine and clonidine in conscious wild-type and D79N alpha2A-adrenoceptor transgenic mice.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Adrenergic alpha-Antagonists; Amino Acid Substitution; Animals; Binding, Competitive; Blood Pressure; Cardiovascular Agents; Cell Line; Clonidine; Consciousness; Dogs; Heart Rate; Humans; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Mice; Mice, Inbred Strains; Mice, Transgenic; Mutation; Naphthyridines; Oxazoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Rilmenidine; Saphenous Vein; Tritium

1999
Analysis of the receptor involved in the central hypotensive effect of rilmenidine and moxonidine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Benzofurans; Blood Pressure; Dose-Response Relationship, Drug; Drug Interactions; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Methyldopa; Norepinephrine; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Yohimbine

1999
Mechanism of the sympathoinhibition produced by the clonidine-like drugs rilmenidine and moxonidine.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Blood Pressure; Clonidine; Decerebrate State; Heart Rate; Imidazoles; Injections, Spinal; Medulla Oblongata; Microinjections; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1999
Central imidazoline- and alpha 2-receptors involved in the cardiovascular actions of centrally acting antihypertensive agents.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Microinjections; Models, Neurological; Norepinephrine; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Serotonin; Sympathetic Nervous System

1999
alpha 2A-adrenoceptors, not I1-imidazoline receptors, mediate the hypotensive effects of rilmenidine and moxonidine in conscious mice. In vivo and in vitro studies.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cell Line; Dogs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypotension; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Quinolizines; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Transfection

1999
Influence of sinoaortic barodenervation on the hypotensive effects of imidazoline-like drugs in stroke-prone spontaneously hypertensive rats.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cerebrovascular Disorders; Circadian Rhythm; Clonidine; Denervation; Heart Rate; Hypotension; Imidazoles; Male; Oxazoles; Pressoreceptors; Rats; Rats, Inbred SHR; Rilmenidine; Sinus of Valsalva; Time Factors

1999
[New central agents in the treatment of arterial hypertension].
    Anales de medicina interna (Madrid, Spain : 1984), 1999, Volume: 16, Issue:10

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Adult; Antihypertensive Agents; Atenolol; Calcium Channel Blockers; Clonidine; Diabetes Complications; Humans; Hypertension; Imidazoles; Nifedipine; Oxazoles; Renin-Angiotensin System; Reserpine; Rilmenidine; Risk Factors; Sympathetic Nervous System; Vasodilator Agents

1999
Species-specific pharmacological properties of human alpha(2A)-adrenoceptors.
    Hypertension (Dallas, Tex. : 1979), 2000, Volume: 36, Issue:3

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Amino Acid Sequence; Animals; Antihypertensive Agents; Female; Heart Atria; Humans; Imidazoles; Male; Middle Aged; Molecular Sequence Data; Norepinephrine; Oxazoles; Oxymetazoline; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha-2; Rilmenidine; Species Specificity; Tritium

2000
[Imidazole receptor agonists--a new advance in the treatment of hypertension?].
    Vnitrni lekarstvi, 2000, Volume: 46, Issue:2

    Topics: Antihypertensive Agents; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

2000
Effects of imidazoline antihypertensive drugs on sympathetic tone and noradrenaline release in the prefrontal cortex.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Guanabenz; Heart Rate; Imidazoles; Male; Microdialysis; Norepinephrine; Oxazoles; Prefrontal Cortex; Rats; Rats, Wistar; Rilmenidine; Sympathetic Nervous System

2001
Importance of imidazoline-preferring receptors in the cardiovascular actions of chronically administered moxonidine, rilmenidine and clonidine in conscious rabbits.
    Journal of hypertension, 2003, Volume: 21, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fourth Ventricle; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intraventricular; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

2003
The role of I(1)-imidazoline receptors and alpha(2)-adrenergic receptors in the modulation of glucose and lipid metabolism in the SHROB model of metabolic syndrome X.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Disease Models, Animal; Female; Glucagon; Glucose; Glucose Tolerance Test; Humans; Imidazoles; Imidazoline Receptors; Lipid Metabolism; Male; Metabolic Syndrome; Obesity; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Yohimbine

2003
Moxonidine displays a presynaptic alpha-2-adrenoceptor-dependent synergistic sympathoinhibitory action at imidazoline-1 receptors.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Bridged Bicyclo Compounds; Brimonidine Tartrate; Drug Synergism; Heart; Heptanes; Imidazoles; Imidazoline Receptors; Norepinephrine; Oxazoles; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Sympatholytics; Yohimbine

2003
Apparent absence of direct renal effect of imidazoline receptor agonists.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Diuretics; Furosemide; Imidazoles; Imidazoline Receptors; Kidney; Male; Natriuresis; Nephrectomy; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rilmenidine

2003
Moxonidine and rilmenidine injected into the medial septal area reduces the salivation induced by pilocarpine.
    Autonomic neuroscience : basic & clinical, 2004, May-31, Volume: 112, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Drug Interactions; Idazoxan; Imidazoles; Male; Muscarinic Agonists; Oxazoles; Pilocarpine; Rats; Rats, Sprague-Dawley; Rilmenidine; Salivation; Septum of Brain; Yohimbine

2004
Lipid-lowering actions of imidazoline antihypertensive agents in metabolic syndrome X.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 372, Issue:4

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Cell Membrane; Cholesterol; Clonidine; Disease Models, Animal; Female; Guanabenz; Hyperlipidemias; Imidazoles; Imidazoline Receptors; Liver; Male; Metabolic Syndrome; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine; Triglycerides

2006
Involvement of phosphatidylcholine-selective phospholipase C in activation of mitogen-activated protein kinase pathways in imidazoline receptor antisera-selected protein.
    Journal of cellular biochemistry, 2006, Aug-15, Volume: 98, Issue:6

    Topics: Animals; Cell Membrane; CHO Cells; Cricetinae; Diglycerides; Dose-Response Relationship, Drug; Extracellular Signal-Regulated MAP Kinases; Guanosine Triphosphate; Imidazoles; Imidazoline Receptors; Intracellular Signaling Peptides and Proteins; Ligands; MAP Kinase Signaling System; Oxazoles; Rilmenidine; Signal Transduction; Type C Phospholipases

2006
Comparison of agmatine with moxonidine and rilmenidine in morphine dependence in vitro: role of imidazoline I(1) receptors.
    European journal of pharmacology, 2009, Jun-10, Volume: 612, Issue:1-3

    Topics: Agmatine; Animals; Antihypertensive Agents; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Morphine Dependence; Oxazoles; Rilmenidine; RNA, Messenger; RNA, Small Interfering; Time Factors; Transfection

2009
Microvascular effects of centrally acting antihypertensive drugs in spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 2010, Volume: 55, Issue:3

    Topics: Administration, Oral; Animals; Antihypertensive Agents; Blood Pressure; Capillaries; Clonidine; Disease Models, Animal; Hypertension; Imidazoles; Male; Microcirculation; Microscopy, Video; Muscle, Skeletal; Oxazoles; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rilmenidine; Skin; Time Factors

2010
Imidazoline-1 receptor ligands as apoptotic agents: pharmacophore modeling and virtual docking study.
    Combinatorial chemistry & high throughput screening, 2013, Volume: 16, Issue:4

    Topics: Antineoplastic Agents; Apoptosis; Benzofurans; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Imidazoles; Imidazoline Receptors; K562 Cells; Ligands; Models, Molecular; Molecular Docking Simulation; Oxazoles; Quantitative Structure-Activity Relationship; Rilmenidine; Tumor Cells, Cultured

2013
INN Common stem: -onidine.
    Prescrire international, 2017, Volume: 26, Issue:181

    Topics: Adrenergic alpha-2 Receptor Agonists; Antimalarials; Brimonidine Tartrate; Cinchona Alkaloids; Clonidine; Humans; Hypertension; Imidazoles; Ocular Hypertension; Rilmenidine; Rosacea; Terminology as Topic

2017