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moxonidine and oxazoles

moxonidine has been researched along with oxazoles in 51 studies

Research

Studies (51)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's34 (66.67)18.2507
2000's15 (29.41)29.6817
2010's2 (3.92)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Christen, O; Göthert, M; Michel, MC; Molderings, GJ; Schäfer, SG1
Gregoire, JR; Sheps, SG1
Starke, K; Szabo, B; Urban, R1
Jacob, R; Rupp, H1
Szabo, B; Urban, R2
Elliott, HL; MacPhee, G; Panfilov, V; Reid, JL1
Li, P; Penner, SB; Smyth, DD1
Christen, MO; Collins, LA; Dreshaj, I; Ernsberger, P; Graff, LM; Graves, ME; Grove, DL; Haxhiu, MA; Schäfer, SG1
Christen, O; Göthert, M; Molderings, GJ; Schäfer, SG1
Chan, CK; Head, GA; Sannajust, F1
Chudek, J; Nowicki, M; Wiecek, A1
Chan, CK; Head, GA1
Frishman, WH; Yu, A1
van Zwieten, PA3
Lada, W1
Piletz, JE; Reis, DJ1
Kunduzova, OR; Medvedev, OS; Medvedeva, NA; Murashev, AN3
Godwin, SJ; Head, GA; Parkin, ML; Tortelli, CF1
Blue, DR; Dillon, MP; Eglen, RM; Jasper, JR; Lesnick, JD; MacLennan, SJ; Zhu, QM2
Bock, C; Niederhoffer, N; Szabo, B1
Drzewoski, J; Wiśniewska-Jarosińska, M1
Bock, C; Niederhoffer, N; Nordheim, U; Szabo, B1
Head, GA1
Peters, SL; Van Zwieten, PA1
Masek, K; Sevcík, J1
Bousquet, P; Feldman, J1
Robles, NR1
Bönisch, H; Brüss, M; Göthert, M; Likungu, J; Molderings, GJ1
Spinar, J; Vítovec, J1
Schachter, M1
Fritz, T; Szabo, B; Wedzony, K1
Nurminen, ML1
Godwin, SJ; Head, GA; Parkin, ML1
Camilleri, G; Clerson, P; Portal, B; Quiniou, G1
Ernsberger, P; Koletsky, RJ; Velliquette, RA1
Burgdorf, C; Engelhardt, A; Kurz, T; Raasch, W; Richardt, G; Schäfer, U1
Forzley, B; Penner, SB; Pirnat, D; Smyth, DD1
de Arruda Camargo, LA; Guarda, IF; Guarda, RS; Saad, WA; Simões, S1
Kotanko, P1
Ernsberger, P; Kossover, R; Previs, SF; Velliquette, RA1
Cong, B; Li, F; Li, J; Lu, XQ; Su, RB; Wu, N; Xu, B; Zheng, JQ1
Sica, DA1
Li, F; Li, J; Liu, Y; Lu, XQ; Su, RB; Wu, N1
Bousquet, P; Lessa, MA; Nascimento, AR; Sabino, B; Tibiriçá, E1
Agbaba, D; Gemovic, B; Nikolic, K; Srdic-Rajic, T; Veljkovic, N1

Reviews

19 review(s) available for moxonidine and oxazoles

ArticleYear
[Imidazole receptors: site of action of a new generation of antihypertensive drugs. Current status and future prospects].
    Deutsche medizinische Wochenschrift (1946), 1992, Jan-10, Volume: 117, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Binding Sites; Cattle; Humans; Imidazoles; Oxazoles; Rats; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1992
Newer antihypertensive drugs.
    Current opinion in cardiology, 1995, Volume: 10, Issue:5

    Topics: Antihypertensive Agents; Dibenzothiepins; Humans; Imidazoles; Methionine; Oxazoles; Piperazines; Protease Inhibitors; Rilmenidine

1995
Clinical pharmacology of drugs acting on imidazoline and adrenergic receptors. Studies with clonidine, moxonidine, rilmenidine, and atenolol.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Antihypertensive Agents; Atenolol; Clinical Trials as Topic; Clonidine; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Placebos; Receptors, Adrenergic; Receptors, Drug; Reference Values; Rilmenidine

1995
[Imidazole receptors and blood pressure regulation. High receptor selectivity of moxonidine].
    Deutsche medizinische Wochenschrift (1946), 1993, Jun-25, Volume: 118, Issue:25

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Cats; Clonidine; Humans; Hypertension; Imidazoles; Oxazoles; Rabbits; Rats; Receptors, Drug; Rilmenidine

1993
[Imidazol receptor agonists--new possibilities for treating hypertension].
    Postepy higieny i medycyny doswiadczalnej, 1995, Volume: 49, Issue:5

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Hemodynamics; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1995
Imidazoline receptor agonist drugs: a new approach to the treatment of systemic hypertension.
    Journal of clinical pharmacology, 1996, Volume: 36, Issue:2

    Topics: Animals; Antihypertensive Agents; Clinical Trials as Topic; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1996
From alpha and beta to I1: an overview of sympathetic receptors involved in blood pressure control targets for drug treatment.
    Journal of cardiovascular pharmacology, 1996, Volume: 27 Suppl 3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Drug; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Rilmenidine

1996
[Imidazoline receptors and use of drug blocking receptors I1].
    Polski merkuriusz lekarski : organ Polskiego Towarzystwa Lekarskiego, 1996, Volume: 1, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Antihypertensive Agents; Arrhythmias, Cardiac; Cimetidine; Histamine H2 Antagonists; Humans; Hypertension; Imidazoles; Myocardial Infarction; Oxazoles; Rilmenidine

1996
The imidazoline receptor in control of blood pressure by clonidine and allied drugs.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Humans; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Neurons; Oxazoles; Receptors, Drug; Rilmenidine

1997
Central imidazoline (I1) receptors as targets of centrally acting antihypertensives: moxonidine and rilmenidine.
    Journal of hypertension, 1997, Volume: 15, Issue:2

    Topics: Animals; Antihypertensive Agents; Brain; Humans; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1997
[Clinical pharmacology of hypotensive drugs acting on central imidazoline receptors].
    Polskie Archiwum Medycyny Wewnetrznej, 1998, Volume: 100, Issue:6

    Topics: Antihypertensive Agents; Clonidine; Drug Interactions; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1998
Central I1-imidazoline receptors as targets of centrally acting antihypertensive drugs. Clinical pharmacology of moxonidine and rilmenidine.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Brain; Clinical Trials as Topic; Clonidine; Hemodynamics; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1999
[New, modern, centrally active antihypertensive agents in the treatment of essential hypertension].
    Casopis lekaru ceskych, 1999, Jun-07, Volume: 138, Issue:12

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Imidazoles; Medulla Oblongata; Oxazoles; Rilmenidine

1999
Drugs acting on imidazoline receptors: a review of their pharmacology, their use in blood pressure control and their potential interest in cardioprotection.
    Drugs, 1999, Volume: 58, Issue:5

    Topics: Animals; Antihypertensive Agents; Arrhythmias, Cardiac; Clinical Trials as Topic; Heart Failure; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1999
Metabolic effects of moxonidine and other centrally acting antihypertensives.
    Diabetes, obesity & metabolism, 1999, Volume: 1, Issue:6

    Topics: Animals; Antihypertensive Agents; Diabetes Complications; Humans; Hypertension; Imidazoles; Insulin Resistance; Metabolism; Oxazoles; Rilmenidine; Sympathetic Nervous System; Sympatholytics; Syndrome

1999
[Central nervous system as a target for the new antihypertensive agents].
    Duodecim; laaketieteellinen aikakauskirja, 1999, Volume: 115, Issue:20

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Autonomic Fibers, Preganglionic; Brain; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Oxazoles; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Sympatholytics

1999
Centrally acting imidazoline I1-receptor agonists: do they have a place in the management of hypertension?
    American journal of cardiovascular drugs : drugs, devices, and other interventions, 2001, Volume: 1, Issue:5

    Topics: Animals; Antihypertensive Agents; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

2001
Cause and consequences of sympathetic hyperactivity in chronic kidney disease.
    Blood purification, 2006, Volume: 24, Issue:1

    Topics: Adrenergic alpha-Agonists; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Arginine; Brain Stem; Humans; Hyperkinesis; Hypertension, Renal; Imidazoles; Kidney Failure, Chronic; Nitric Oxide Synthase; Oxazoles; Receptor, Angiotensin, Type 1; Renal Dialysis; Rilmenidine; Sympathetic Nervous System; Sympatholytics

2006
Centrally acting antihypertensive agents: an update.
    Journal of clinical hypertension (Greenwich, Conn.), 2007, Volume: 9, Issue:5

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Clonidine; Contraindications; Guanabenz; Guanfacine; Humans; Hypertension; Imidazoles; Methyldopa; Oxazoles; Rilmenidine

2007

Trials

1 trial(s) available for moxonidine and oxazoles

ArticleYear
[Comparison of the antihypertensive efficacy of and tolerance to 2 imidazoline receptor agonists: moxonidine and rilmenidine in monotherapy].
    Annales de cardiologie et d'angeiologie, 2001, Volume: 50, Issue:3

    Topics: Antihypertensive Agents; Female; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Male; Middle Aged; Oxazoles; Receptors, Drug; Rilmenidine; Severity of Illness Index

2001

Other Studies

31 other study(ies) available for moxonidine and oxazoles

ArticleYear
Involvement of peripheral presynaptic inhibition in the reduction of sympathetic tone by moxonidine, rilmenidine and UK 14304.
    European journal of pharmacology, 1995, Aug-25, Volume: 282, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Female; Imidazoles; Male; Neural Inhibition; Oxazoles; Peripheral Nervous System; Presynaptic Terminals; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Vasoconstrictor Agents

1995
Excess catecholamines and the metabolic syndrome: should central imidazoline receptors be a therapeutic target?
    Medical hypotheses, 1995, Volume: 44, Issue:3

    Topics: Animals; Antihypertensive Agents; Cardiovascular Diseases; Catecholamines; Energy Intake; Energy Metabolism; Humans; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Models, Biological; Neurons; Obesity; Oxazoles; Receptors, Drug; Rilmenidine; Social Conditions; Stress, Psychological; Sympathetic Nervous System

1995
Mechanism of sympathoinhibition by imidazolines.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzazepines; Brimonidine Tartrate; Dioxanes; Hemodynamics; Idazoxan; Imidazoles; Oxazoles; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1995
Attenuated renal response to moxonidine and rilmenidine in one kidney-one clip hypertensive rats.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Hemodynamics; Hypertension, Renovascular; Imidazoles; Infusions, Intra-Arterial; Kidney; Male; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Renal Circulation; Rilmenidine; Sodium; Urodynamics

1994
A novel mechanism of action for hypertension control: moxonidine as a selective I1-imidazoline agonist.
    Cardiovascular drugs and therapy, 1994, Volume: 8 Suppl 1

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Autoradiography; Binding Sites; Blood Pressure; Cattle; Cells, Cultured; Clonidine; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1994
Role of imidazoline receptors in the cardiovascular actions of moxonidine, rilmenidine and clonidine in conscious rabbits.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1996
Relative importance of central imidazoline receptors for the antihypertensive effects of moxonidine and rilmenidine.
    Journal of hypertension, 1996, Volume: 14, Issue:7

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiac Catheterization; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intravenous; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Time Factors

1996
Role of I1 imidazoline receptors in the sympathoinhibition produced by intracisternally administered rilmenidine and moxonidine.
    Arzneimittel-Forschung, 1997, Volume: 47, Issue:9

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Cisterna Magna; Dose-Response Relationship, Drug; Female; Guanabenz; Heart Rate; Imidazoles; Imidazoline Receptors; Injections; Male; Norepinephrine; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Yohimbine

1997
Chronopharmacological dependence of antihypertensive effects of the imidazoline-like drugs in stroke-prone spontaneously hypertensive rats.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cerebrovascular Disorders; Circadian Rhythm; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Imidazoles; Male; Motor Activity; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine

1998
Comparison of the baroreceptor-heart rate reflex effects of moxonidine, rilmenidine and clonidine in conscious rabbits.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Algorithms; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Clonidine; Female; Heart Rate; Imidazoles; Injections, Intraventricular; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Vagus Nerve

1998
Influence of sino-aortic barodenervation on the cardiovascular effects of imidazoline-like drugs.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Circadian Rhythm; Clonidine; Denervation; Heart Rate; Imidazoles; Injections, Intravenous; Male; Motor Activity; Oxazoles; Pressoreceptors; Rats; Rats, Wistar; Rilmenidine; Sinus of Valsalva; Telemetry

1998
Cardiovascular effects of rilmenidine, moxonidine and clonidine in conscious wild-type and D79N alpha2A-adrenoceptor transgenic mice.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Adrenergic alpha-Antagonists; Amino Acid Substitution; Animals; Binding, Competitive; Blood Pressure; Cardiovascular Agents; Cell Line; Clonidine; Consciousness; Dogs; Heart Rate; Humans; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Mice; Mice, Inbred Strains; Mice, Transgenic; Mutation; Naphthyridines; Oxazoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Rilmenidine; Saphenous Vein; Tritium

1999
Analysis of the receptor involved in the central hypotensive effect of rilmenidine and moxonidine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Benzofurans; Blood Pressure; Dose-Response Relationship, Drug; Drug Interactions; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Methyldopa; Norepinephrine; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Yohimbine

1999
Mechanism of the sympathoinhibition produced by the clonidine-like drugs rilmenidine and moxonidine.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Blood Pressure; Clonidine; Decerebrate State; Heart Rate; Imidazoles; Injections, Spinal; Medulla Oblongata; Microinjections; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1999
Central imidazoline- and alpha 2-receptors involved in the cardiovascular actions of centrally acting antihypertensive agents.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Microinjections; Models, Neurological; Norepinephrine; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Serotonin; Sympathetic Nervous System

1999
alpha 2A-adrenoceptors, not I1-imidazoline receptors, mediate the hypotensive effects of rilmenidine and moxonidine in conscious mice. In vivo and in vitro studies.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cell Line; Dogs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypotension; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Quinolizines; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Transfection

1999
Influence of sinoaortic barodenervation on the hypotensive effects of imidazoline-like drugs in stroke-prone spontaneously hypertensive rats.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cerebrovascular Disorders; Circadian Rhythm; Clonidine; Denervation; Heart Rate; Hypotension; Imidazoles; Male; Oxazoles; Pressoreceptors; Rats; Rats, Inbred SHR; Rilmenidine; Sinus of Valsalva; Time Factors

1999
[New central agents in the treatment of arterial hypertension].
    Anales de medicina interna (Madrid, Spain : 1984), 1999, Volume: 16, Issue:10

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Adult; Antihypertensive Agents; Atenolol; Calcium Channel Blockers; Clonidine; Diabetes Complications; Humans; Hypertension; Imidazoles; Nifedipine; Oxazoles; Renin-Angiotensin System; Reserpine; Rilmenidine; Risk Factors; Sympathetic Nervous System; Vasodilator Agents

1999
Species-specific pharmacological properties of human alpha(2A)-adrenoceptors.
    Hypertension (Dallas, Tex. : 1979), 2000, Volume: 36, Issue:3

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Amino Acid Sequence; Animals; Antihypertensive Agents; Female; Heart Atria; Humans; Imidazoles; Male; Middle Aged; Molecular Sequence Data; Norepinephrine; Oxazoles; Oxymetazoline; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha-2; Rilmenidine; Species Specificity; Tritium

2000
[Imidazole receptor agonists--a new advance in the treatment of hypertension?].
    Vnitrni lekarstvi, 2000, Volume: 46, Issue:2

    Topics: Antihypertensive Agents; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

2000
Effects of imidazoline antihypertensive drugs on sympathetic tone and noradrenaline release in the prefrontal cortex.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Guanabenz; Heart Rate; Imidazoles; Male; Microdialysis; Norepinephrine; Oxazoles; Prefrontal Cortex; Rats; Rats, Wistar; Rilmenidine; Sympathetic Nervous System

2001
Importance of imidazoline-preferring receptors in the cardiovascular actions of chronically administered moxonidine, rilmenidine and clonidine in conscious rabbits.
    Journal of hypertension, 2003, Volume: 21, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fourth Ventricle; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intraventricular; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

2003
The role of I(1)-imidazoline receptors and alpha(2)-adrenergic receptors in the modulation of glucose and lipid metabolism in the SHROB model of metabolic syndrome X.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Disease Models, Animal; Female; Glucagon; Glucose; Glucose Tolerance Test; Humans; Imidazoles; Imidazoline Receptors; Lipid Metabolism; Male; Metabolic Syndrome; Obesity; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Yohimbine

2003
Moxonidine displays a presynaptic alpha-2-adrenoceptor-dependent synergistic sympathoinhibitory action at imidazoline-1 receptors.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Bridged Bicyclo Compounds; Brimonidine Tartrate; Drug Synergism; Heart; Heptanes; Imidazoles; Imidazoline Receptors; Norepinephrine; Oxazoles; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Sympatholytics; Yohimbine

2003
Apparent absence of direct renal effect of imidazoline receptor agonists.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Diuretics; Furosemide; Imidazoles; Imidazoline Receptors; Kidney; Male; Natriuresis; Nephrectomy; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rilmenidine

2003
Moxonidine and rilmenidine injected into the medial septal area reduces the salivation induced by pilocarpine.
    Autonomic neuroscience : basic & clinical, 2004, May-31, Volume: 112, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Drug Interactions; Idazoxan; Imidazoles; Male; Muscarinic Agonists; Oxazoles; Pilocarpine; Rats; Rats, Sprague-Dawley; Rilmenidine; Salivation; Septum of Brain; Yohimbine

2004
Lipid-lowering actions of imidazoline antihypertensive agents in metabolic syndrome X.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 372, Issue:4

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Cell Membrane; Cholesterol; Clonidine; Disease Models, Animal; Female; Guanabenz; Hyperlipidemias; Imidazoles; Imidazoline Receptors; Liver; Male; Metabolic Syndrome; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine; Triglycerides

2006
Involvement of phosphatidylcholine-selective phospholipase C in activation of mitogen-activated protein kinase pathways in imidazoline receptor antisera-selected protein.
    Journal of cellular biochemistry, 2006, Aug-15, Volume: 98, Issue:6

    Topics: Animals; Cell Membrane; CHO Cells; Cricetinae; Diglycerides; Dose-Response Relationship, Drug; Extracellular Signal-Regulated MAP Kinases; Guanosine Triphosphate; Imidazoles; Imidazoline Receptors; Intracellular Signaling Peptides and Proteins; Ligands; MAP Kinase Signaling System; Oxazoles; Rilmenidine; Signal Transduction; Type C Phospholipases

2006
Comparison of agmatine with moxonidine and rilmenidine in morphine dependence in vitro: role of imidazoline I(1) receptors.
    European journal of pharmacology, 2009, Jun-10, Volume: 612, Issue:1-3

    Topics: Agmatine; Animals; Antihypertensive Agents; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Morphine Dependence; Oxazoles; Rilmenidine; RNA, Messenger; RNA, Small Interfering; Time Factors; Transfection

2009
Microvascular effects of centrally acting antihypertensive drugs in spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 2010, Volume: 55, Issue:3

    Topics: Administration, Oral; Animals; Antihypertensive Agents; Blood Pressure; Capillaries; Clonidine; Disease Models, Animal; Hypertension; Imidazoles; Male; Microcirculation; Microscopy, Video; Muscle, Skeletal; Oxazoles; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rilmenidine; Skin; Time Factors

2010
Imidazoline-1 receptor ligands as apoptotic agents: pharmacophore modeling and virtual docking study.
    Combinatorial chemistry & high throughput screening, 2013, Volume: 16, Issue:4

    Topics: Antineoplastic Agents; Apoptosis; Benzofurans; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Imidazoles; Imidazoline Receptors; K562 Cells; Ligands; Models, Molecular; Molecular Docking Simulation; Oxazoles; Quantitative Structure-Activity Relationship; Rilmenidine; Tumor Cells, Cultured

2013