Page last updated: 2024-09-04

moxifloxacin and gs 4071

moxifloxacin has been researched along with gs 4071 in 3 studies

Compound Research Comparison

Studies
(moxifloxacin)
Trials
(moxifloxacin)
Recent Studies (post-2010)
(moxifloxacin)
Studies
(gs 4071)
Trials
(gs 4071)
Recent Studies (post-2010) (gs 4071)
3,1575521,69019016140

Protein Interaction Comparison

ProteinTaxonomymoxifloxacin (IC50)gs 4071 (IC50)
Neuraminidase Influenza A virus (A/Turkey/651242/2006(H5N1))1.4208
Neuraminidase Influenza A virus (A/Wilson-Smith/1933(H1N1))0.4952
Neuraminidase Influenza A virus (A/duck/Laos/25/2006(H5N1))1.63
NeuraminidaseInfluenza A virus (A/Puerto Rico/8/1934(H1N1))0.0175
NeuraminidaseInfluenza A virus (A/USSR/90/1977(H1N1))0.0079
NeuraminidaseInfluenza A virus (A/Wilson-Smith/1933(H1N1))0.1851
NeuraminidaseInfluenza A virus (A/Memphis/1/1971(H3N2))0.0039
NeuraminidaseInfluenza B virus (B/Lee/1940)0.0085
NeuraminidaseInfluenza A virus (A/udorn/1972(H3N2))0.5813
SialidaseClostridium perfringens0.001
Substance-P receptorCavia porcellus (domestic guinea pig)0.015
Histamine H1 receptorCavia porcellus (domestic guinea pig)2.8247
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0089
NeuraminidaseInfluenza A virus (A/duck/Ukraine/1/1963(H3N8))0.0089
Neuraminidase Influenza A virus (A/udorn/1972(H3N2))0.0029
Substance-K receptorCavia porcellus (domestic guinea pig)0.015
NeuraminidaseInfluenza A virus (A/swine/Hong Kong/127/1982(H3N2))0.17
Neuraminidase Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1))0.0007
NeuraminidaseInfluenza A virus (A/budgerigar/Hokkaido/1/1977(H4N6))0.0153
Integrase Human immunodeficiency virus 11.785

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1

Other Studies

3 other study(ies) available for moxifloxacin and gs 4071

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010