Page last updated: 2024-09-04

moxifloxacin and amsacrine

moxifloxacin has been researched along with amsacrine in 4 studies

Compound Research Comparison

Studies
(moxifloxacin)
Trials
(moxifloxacin)
Recent Studies (post-2010)
(moxifloxacin)
Studies
(amsacrine)
Trials
(amsacrine)
Recent Studies (post-2010) (amsacrine)
3,1575521,6901,293127120

Protein Interaction Comparison

ProteinTaxonomymoxifloxacin (IC50)amsacrine (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)5
Multidrug resistance-associated protein 4Homo sapiens (human)7.43
DNA topoisomerase 2-alphaHomo sapiens (human)5.47
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)5
DNA topoisomerase 2-betaHomo sapiens (human)1.88
Aldehyde oxidaseHomo sapiens (human)3.2
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.2095
Aldehyde oxidase 1 Rattus norvegicus (Norway rat)6.4

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Sen, S; Sinha, N1
Kulkarni, P; Meda, N; Medapi, B; Sriram, D; Yogeeswari, P1

Other Studies

4 other study(ies) available for moxifloxacin and amsacrine

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
Development of acridine derivatives as selective Mycobacterium tuberculosis DNA gyrase inhibitors.
    Bioorganic & medicinal chemistry, 2016, Feb-15, Volume: 24, Issue:4

    Topics: Acridines; Animals; Antitubercular Agents; Bacterial Proteins; Cell Line; Cell Survival; Chlorobenzoates; DNA Gyrase; Dose-Response Relationship, Drug; Embryo, Nonmammalian; Ether-A-Go-Go Potassium Channels; Gene Expression; Heart Rate; Macrophages; Mice; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Piperidines; Quinolines; Structure-Activity Relationship; Topoisomerase II Inhibitors; Zebrafish; Zebrafish Proteins

2016