Page last updated: 2024-09-03

morphiceptin and u-50488

morphiceptin has been researched along with u-50488 in 6 studies

Compound Research Comparison

Studies
(morphiceptin)
Trials
(morphiceptin)
Recent Studies (post-2010)
(morphiceptin)
Studies
(u-50488)
Trials
(u-50488)
Recent Studies (post-2010) (u-50488)
1390121,6643209

Protein Interaction Comparison

ProteinTaxonomymorphiceptin (IC50)u-50488 (IC50)
Delta-type opioid receptorRattus norvegicus (Norway rat)2.15
Kappa-type opioid receptorMus musculus (house mouse)0.0027
Mu-type opioid receptorRattus norvegicus (Norway rat)2.15
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.7171
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.0958
Kappa-type opioid receptorHomo sapiens (human)0.0537

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19901 (16.67)18.7374
1990's4 (66.67)18.2507
2000's1 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Levine, JD; Miaskowski, C1
Członkowski, A; Widy-Tyszkiewicz, E1
Bero, LA; Kuhn, CM; Lurie, SN1
de Andrés, I; Reinoso-Barbero, F1
Joshi, S; Lee, JW; Wong, YH1
Barr, GA; Cheng, J; Limon, E; Luthmann, RA; Wang, S1

Other Studies

6 other study(ies) available for morphiceptin and u-50488

ArticleYear
Antinociception produced by receptor selective opioids: modulation of spinal antinociceptive effects by supraspinal opioids.
    Brain research, 1992, Nov-06, Volume: 595, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dose-Response Relationship, Drug; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Intraventricular; Injections, Spinal; Male; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Spinal Cord

1992
Normotensive Wistar rats differ from spontaneously hypertensive and renal hypertensive rats in their cardiovascular responses to opioid agonists.
    Clinical and experimental pharmacology & physiology, 1991, Volume: 18, Issue:12

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Amino Acid Sequence; Analgesics; Animals; Blood Pressure; Endorphins; Heart Rate; Hemodynamics; Hypertension, Renal; Injections, Intraventricular; Male; Molecular Sequence Data; Naloxone; Oligopeptides; Pyrrolidines; Rats; Rats, Inbred SHR; Rats, Inbred Strains

1991
Early ontogeny of kappa-opioid receptor regulation of prolactin secretion in the rat.
    Brain research, 1987, Dec-15, Volume: 465, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Dynorphins; Endorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Hydrazines; Morphine; Peptide Fragments; Prolactin; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serotonin

1987
Effects of opioid microinjections in the nucleus of the solitary tract on the sleep-wakefulness cycle states in cats.
    Anesthesiology, 1995, Volume: 82, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Cats; Drug Interactions; Electroencephalography; Endorphins; Microinjections; Morphine; Naloxone; Pyrrolidines; Receptors, Opioid; Sleep Stages; Sodium Chloride; Solitary Nucleus

1995
Stimulation of phospholipase C by the cloned mu, delta and kappa opioid receptors via chimeric G alpha(q) mutants.
    The European journal of neuroscience, 1999, Volume: 11, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclases; Analgesics; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Cloning, Molecular; COS Cells; DNA, Complementary; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Enzyme Activation; GTP-Binding Proteins; Mice; Naloxone; Narcotic Antagonists; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Recombinant Fusion Proteins; Type C Phospholipases

1999
Analgesia induced by local plantar injections of opiates in the formalin test in infant rats.
    Developmental psychobiology, 2003, Volume: 42, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Age Factors; Analgesics, Opioid; Animals; Animals, Newborn; Endorphins; Enkephalin, D-Penicillamine (2,5)-; Female; Formaldehyde; Hindlimb; Injections, Subcutaneous; Male; Pain Threshold; Rats; Rats, Sprague-Dawley

2003