Page last updated: 2024-09-03

morphiceptin, n-me-phe(3)- and u 69593

morphiceptin, n-me-phe(3)- has been researched along with u 69593 in 3 studies

Compound Research Comparison

Studies
(morphiceptin, n-me-phe(3)-)
Trials
(morphiceptin, n-me-phe(3)-)
Recent Studies (post-2010)
(morphiceptin, n-me-phe(3)-)
Studies
(u 69593)
Trials
(u 69593)
Recent Studies (post-2010) (u 69593)
9511524075

Protein Interaction Comparison

ProteinTaxonomymorphiceptin, n-me-phe(3)- (IC50)u 69593 (IC50)
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0006
Mu-type opioid receptorHomo sapiens (human)0.194
Delta-type opioid receptorHomo sapiens (human)3.6437
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.0021
Kappa-type opioid receptorHomo sapiens (human)0.058
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.588

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A1
Ananthan, S; Bartlett, JL; Bilsky, EJ; Davis, P; Dersch, CM; Khare, NK; Porreca, F; Rothman, RB; Saini, SK; Seitz, LE1
Macdonald, RL; Moises, HC; Rusin, KI1

Other Studies

3 other study(ies) available for morphiceptin, n-me-phe(3)- and u 69593

ArticleYear
Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
    NIDA research monograph, 1998, Volume: 178

    Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders

1998
Identification of opioid ligands possessing mixed micro agonist/delta antagonist activity among pyridomorphinans derived from naloxone, oxymorphone, and hydromorphone [correction of hydropmorphone].
    Journal of medicinal chemistry, 2004, Mar-11, Volume: 47, Issue:6

    Topics: Analgesics; Animals; Binding Sites; Brain; Drug Tolerance; Electric Stimulation; Guinea Pigs; Hydromorphone; Ileum; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Morphinans; Muscle Contraction; Muscle, Smooth; Naloxone; Oxymorphone; Pyridines; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Vas Deferens

2004
Mu- and kappa-opioid receptors selectively reduce the same transient components of high-threshold calcium current in rat dorsal root ganglion sensory neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:10

    Topics: Analgesics; Animals; Benzeneacetamides; Calcium; Calcium Channels; Dynorphins; Endorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Evoked Potentials; Ganglia, Spinal; In Vitro Techniques; Naloxone; Naltrexone; Narcotic Antagonists; Neurons, Afferent; Pyrrolidines; Rats; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reference Values; Sensitivity and Specificity

1994