moclobemide and clorgyline

moclobemide has been researched along with clorgyline in 57 studies

Research

Studies (57)

TimeframeStudies, this research(%)All Research%
pre-19909 (15.79)18.7374
1990's11 (19.30)18.2507
2000's12 (21.05)29.6817
2010's23 (40.35)24.3611
2020's2 (3.51)2.80

Authors

AuthorsStudies
Agostinelli, E; Artico, M; Befani, O; De Martino, G; La Regina, G; Palumbo, M; Silvestri, R; Turini, P1
Agostinelli, E; Artico, M; Befani, O; La Regina, G; Lavecchia, A; Novellino, E; Silvestri, R; Turini, P1
Alcaro, S; Bolasco, A; Carradori, S; Chimenti, F; Chimenti, P; Cirilli, R; Ferretti, R; Granese, A; La Torre, F; Maccioni, E; Orallo, F; Ortuso, F; Secci, D; Yáñez, M1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Agostinelli, E; Befani, O; Gatti, V; La Regina, G; Lavecchia, A; Novellino, E; Silvestri, R; Turini, P1
Ercan, A; Jayaprakash, V; Sinha, BN; Ucar, G1
Erol, K; Gökhan-Kelekçi, N; Kendi, E; Koyunoğlu, S; Ozgen, O; Uçar, G; Yabanoğlu, S; Yelekçi, K; Yeşilada, A1
Alcaro, S; Bizzarri, B; Bolasco, A; Carradori, S; Chimenti, F; Chimenti, P; Granese, A; Orallo, F; Ortuso, F; Secci, D; Yáñez, M1
Alcaro, S; Bolasco, A; Chimenti, F; Chimenti, P; Fioravanti, R; Orallo, F; Ortuso, F; Rossi, F; Secci, D; Yáñez, M1
Bizzarri, B; Bolasco, A; Carradori, S; Chimenti, F; Chimenti, P; Granese, A; Orallo, F; Secci, D; Yáñez, M1
Alcaro, S; Bolasco, A; Chimenti, F; Chimenti, P; Cirilli, R; Ferretti, R; Fioravanti, R; Orallo, F; Ortuso, F; Rossi, F; Sanna, ML; Secci, D; Yáñez, M1
Alcaro, S; Borges, F; Gaspar, A; Milhazes, N; Orallo, F; Ortuso, F; Uriarte, E; Yáñez, M1
Alcaro, S; Bolasco, A; Cardia, MC; Carradori, S; Chimenti, F; Chimenti, P; Cirilli, R; Distinto, S; Ferretti, R; Granese, A; Kirchmair, J; Langer, T; Maccioni, E; Orallo, F; Ortuso, F; Secci, D; Yáñez, M1
Alcaro, S; Bolasco, A; Carradori, S; Chimenti, F; Chimenti, P; Granese, A; Orallo, F; Ortuso, F; Secci, D; Yáñez, M1
Alcaro, S; Cardia, MC; Costa, G; Distinto, S; Maccioni, E; Meleddu, R; Orallo, F; Sanna, ML; Secci, D; Vigo, S; Yanez, M1
Bolasco, A; Carradori, S; Chimenti, F; Chimenti, P; Cirilli, R; Gallinella, B; Granese, A; Orallo, F; Sanna, ML; Secci, D; Yáñez, M1
Alcaro, S; Bolasco, A; Fioravanti, R; Manna, F; Orallo, F; Ortuso, F; Rossi, F; Vitali, A; Yáñez, M1
Alcaro, S; Bolasco, A; Desideri, N; Fioravanti, R; Monaco, LP; Orallo, F; Ortuso, F; Yáñez, M1
Alcaro, S; Bolasco, A; Carradori, S; Chimenti, P; Ortuso, F; Secci, D; Yáñez, M1
Escobar, M; García-Mera, X; González-Díaz, H; Prado-Prado, F; Riera-Fernandez, P; Sobarzo-Sánchez, E; Yañez, M1
Alcaro, S; Bolasco, A; Cardia, MC; Distinto, S; Gaspari, M; Kirchmair, J; Maccioni, E; Markt, P; Meleddu, R; Ortuso, F; Sanna, ML; Secci, D; Wolber, G; Yáñez, M1
Abdalla, MM; Abdelhafez, OM; Ali, HI; Amin, KM; Batran, RZ1
Bolasco, A; Carradori, S; D'Ascenzio, M; Nescatelli, R; Secci, D; Yáñez, M1
Alcaro, S; Biava, M; Desideri, N; Fioravanti, R; Ortuso, F; Proietti Monaco, L; Yáñez, M2
Biava, M; Desideri, N; Fioravanti, R; Grammatica, L; Proietti Monaco, L; Yáñez, M1
Alcaro, S; Carradori, S; Cirilli, R; D'Ascenzio, M; De Monte, C; Mannina, L; Ortuso, F; Secci, D; Sobolev, AP; Yáñez, M1
Abdel Moneim, SA; Ali Ahmed, HE; Amer, A; Bekhit, AA; El Massry, AM; El-Faham, A; Hassan, SY; Khattab, SN1
Alam, MM; Alex, AT; Bansal, S; Chaudhary, A; Jaiswal, V; Joseph, A; Suthar, SK; Tiwari, A1
Alcaro, S; Arridu, A; Bianco, G; Cirilli, R; Cossu, P; Cottiglia, F; Distinto, S; Faggi, C; Maccioni, E; Meleddu, R; Ortuso, F; Sanna, ML; Yanez, M1
Borges, F; Delogu, GL; Fontenla, JA; Hripcsak, G; Matos, MJ; Mayán, L; Munín, J; Pintus, F; Vilar, S; Viña, D1
Acar Çevik, U; Kaplancıklı, ZA; Kaya Çavuşoğlu, B; Levent, S; Osmaniye, D; Özkay, Y; Sağlık, BN1
Bai, R; Jiang, X; Wu, K; Zhang, P; Zhang, Y1
Antonin, KH; Bieck, PR; Gleiter, CH; Mühlbauer, B; Nilsson, E1
Iwata, N; Kumagae, Y; Matsui, Y1
Stöcklin, K; Waldmeier, PC1
Fletcher, PJ; Yu, PH1
Rényi, L1
Bizière, K; Kan, JP; Roncucci, R; Wermuth, CG; Worms, P1
Bizière, K; Kan, JP; Mouget-Goniot, C; Steinberg, R; Worms, P1
Cesura, AM; Da Prada, M; Kettler, R; Richards, JG1
Finberg, JP; Youdim, MB1
Dowson, JH1
Demurov, EA; Gol'dina, OA; Koloskov, IuB; Tepliakov, VG; Zagorevskiĭ, VA1
Waldmeier, PC1
McIntyre, IM; Oxenkrug, GF; Requintina, PJ; White, K1
Youdim, MB1
Finberg, JP1
Alemany, R; García-Sevilla, JA; Olmos, G1
Gerardy, J1
Finberg, JP; Lavian, G; Youdim, MB1
Ametamey, SM; Antonini, A; Beer, HF; Guenther, I; Leenders, KL; Schubiger, PA; Waldmeier, PC1
Hibell, A; Hudson, AL; Lalies, MD; Nutt, DJ1
Bonnet, U; Leniger, T; Wiemann, M1
Culver, KE; Rosenfeld, JM; Szechtman, H1
Bejar, C; Drigues, N; Poltyrev, T; Weinstock, M; Youdim, MB1
Fisar, Z; Hroudová, J; Raboch, J1

Reviews

4 review(s) available for moclobemide and clorgyline

ArticleYear
Functionalized quinoxalinones as privileged structures with broad-ranging pharmacological activities.
    European journal of medicinal chemistry, 2022, Feb-05, Volume: 229

    Topics: Animals; Anti-Allergic Agents; Anti-Bacterial Agents; Anti-Infective Agents; Anti-Inflammatory Agents; Antineoplastic Agents; Antioxidants; Antiviral Agents; Drug Development; Heterocyclic Compounds; Humans; Hypoglycemic Agents; Mice; Neuroprotective Agents; Photochemotherapy; Quinoxalines; Structure-Activity Relationship; Tubulin Modulators

2022
MAO inhibitors in mental disease: their current status.
    Journal of neural transmission. Supplementum, 1987, Volume: 23

    Topics: Benzamides; Clorgyline; Depressive Disorder; Drug Therapy, Combination; Humans; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenelzine; Tranylcypromine

1987
The advent of selective monoamine oxidase A inhibitor antidepressants devoid of the cheese reaction.
    Acta psychiatrica Scandinavica. Supplementum, 1995, Volume: 386

    Topics: Benzamides; Cheese; Clorgyline; Depressive Disorder; Humans; Hypertension; Moclobemide; Monoamine Oxidase Inhibitors; Selegiline; Tyramine

1995
Pharmacology of reversible and selective inhibitors of monoamine oxidase type A.
    Acta psychiatrica Scandinavica. Supplementum, 1995, Volume: 386

    Topics: Animals; Benzamides; Clorgyline; Dopamine; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Norepinephrine; Piperidines; Rats; Serotonin; Sympathetic Nervous System; Tyramine

1995

Other Studies

53 other study(ies) available for moclobemide and clorgyline

ArticleYear
Simple, potent, and selective pyrrole inhibitors of monoamine oxidase types A and B.
    Journal of medicinal chemistry, 2003, Mar-13, Volume: 46, Issue:6

    Topics: Alkynes; Amides; Amines; Animals; Brain; Cattle; Isoenzymes; Mitochondria; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pyrroles; Structure-Activity Relationship

2003
New pyrrole inhibitors of monoamine oxidase: synthesis, biological evaluation, and structural determinants of MAO-A and MAO-B selectivity.
    Journal of medicinal chemistry, 2007, Mar-08, Volume: 50, Issue:5

    Topics: Animals; Benzylamines; Binding Sites; Brain; Cattle; In Vitro Techniques; Isoenzymes; Mitochondria; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pyrroles; Stereoisomerism; Structure-Activity Relationship

2007
Synthesis, stereochemical identification, and selective inhibitory activity against human monoamine oxidase-B of 2-methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones.
    Journal of medicinal chemistry, 2008, Aug-28, Volume: 51, Issue:16

    Topics: Chromatography, High Pressure Liquid; Cyclohexanones; Humans; Hydrazones; Inhibitory Concentration 50; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Stereoisomerism; Thermodynamics; Thiazoles; Thiosemicarbazones

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Synthesis, structure-activity relationships and molecular modeling studies of new indole inhibitors of monoamine oxidases A and B.
    Bioorganic & medicinal chemistry, 2008, Nov-15, Volume: 16, Issue:22

    Topics: Binding Sites; Indoles; Kinetics; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Stereoisomerism; Structure-Activity Relationship

2008
Pyrazoline-based mycobactin analogues as MAO-inhibitors.
    Bioorganic & medicinal chemistry letters, 2008, Dec-15, Volume: 18, Issue:24

    Topics: Acetamides; Animals; Binding Sites; Catalytic Domain; Drug Design; Humans; Inhibitory Concentration 50; Linezolid; Liver; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Oxazolidinones; Pyrazoles; Rats; Siderophores

2008
New pyrazoline bearing 4(3H)-quinazolinone inhibitors of monoamine oxidase: synthesis, biological evaluation, and structural determinants of MAO-A and MAO-B selectivity.
    Bioorganic & medicinal chemistry, 2009, Jan-15, Volume: 17, Issue:2

    Topics: Binding Sites; Flavin-Adenine Dinucleotide; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pyrazoles; Quinazolinones

2009
Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins.
    Journal of medicinal chemistry, 2009, Apr-09, Volume: 52, Issue:7

    Topics: Coumarins; Crystallography, X-Ray; Humans; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2009
Chalcones: a valid scaffold for monoamine oxidases inhibitors.
    Journal of medicinal chemistry, 2009, May-14, Volume: 52, Issue:9

    Topics: Chalcones; Crystallography, X-Ray; Databases, Protein; Drug Design; Humans; Inhibitory Concentration 50; Isoenzymes; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors

2009
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:2

    Topics: Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pyrazoles

2010
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors.
    Bioorganic & medicinal chemistry, 2010, Volume: 18, Issue:3

    Topics: Flavanones; Flavones; Humans; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Stereoisomerism; Sulfhydryl Compounds

2010
Chromone-2- and -3-carboxylic acids inhibit differently monoamine oxidases A and B.
    Bioorganic & medicinal chemistry letters, 2010, May-01, Volume: 20, Issue:9

    Topics: Binding Sites; Chromones; Computer Simulation; Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Protein Isoforms

2010
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors.
    Bioorganic & medicinal chemistry, 2010, Jul-15, Volume: 18, Issue:14

    Topics: Chromatography, High Pressure Liquid; Humans; Hydrazones; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship; Thiazoles

2010
Investigations on the 2-thiazolylhydrazyne scaffold: synthesis and molecular modeling of selective human monoamine oxidase inhibitors.
    Bioorganic & medicinal chemistry, 2010, Aug-01, Volume: 18, Issue:15

    Topics: Humans; Hydrazines; Hydrogen Peroxide; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2010
Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:10

    Topics: Animals; Cell Line; Humans; Insecta; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Protein Binding; Pyrazoles; Recombinant Proteins; Structure-Activity Relationship; Thioamides

2010
Synthesis, stereochemical separation, and biological evaluation of selective inhibitors of human MAO-B: 1-(4-arylthiazol-2-yl)-2-(3-methylcyclohexylidene)hydrazines.
    Journal of medicinal chemistry, 2010, Sep-09, Volume: 53, Issue:17

    Topics: Chromatography, High Pressure Liquid; Cyclohexanes; Humans; Hydrazines; Isoenzymes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Stereoisomerism; Structure-Activity Relationship; Triazoles

2010
Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors.
    Bioorganic & medicinal chemistry letters, 2010, Nov-15, Volume: 20, Issue:22

    Topics: Humans; Inhibitory Concentration 50; Models, Molecular; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Prenylation; Pyrazoles; Structure-Activity Relationship

2010
Homoisoflavonoids: natural scaffolds with potent and selective monoamine oxidase-B inhibition properties.
    Journal of medicinal chemistry, 2011, Apr-14, Volume: 54, Issue:7

    Topics: Drug Discovery; Flavonoids; Humans; Inhibitory Concentration 50; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Protein Conformation; Substrate Specificity

2011
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:10

    Topics: Coumarins; Humans; Inhibitory Concentration 50; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2011
2D MI-DRAGON: a new predictor for protein-ligands interactions and theoretic-experimental studies of US FDA drug-target network, oxoisoaporphine inhibitors for MAO-A and human parasite proteins.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:12

    Topics: Antiprotozoal Agents; Aporphines; Databases, Factual; Humans; Ligands; Malaria, Falciparum; Markov Chains; Models, Biological; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Plasmodium falciparum; Protozoan Proteins; Quantitative Structure-Activity Relationship; Software; United States

2011
Synthesis and biological assessment of novel 2-thiazolylhydrazones and computational analysis of their recognition by monoamine oxidase B.
    European journal of medicinal chemistry, 2012, Volume: 48

    Topics: Binding Sites; Humans; Hydrazones; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Dynamics Simulation; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Parkinson Disease; Protein Conformation; Structure-Activity Relationship; Tandem Mass Spectrometry; Thiazoles

2012
Synthesis of new 7-oxycoumarin derivatives as potent and selective monoamine oxidase A inhibitors.
    Journal of medicinal chemistry, 2012, Dec-13, Volume: 55, Issue:23

    Topics: Coumarins; Hydrogen Bonding; Magnetic Resonance Spectroscopy; Mass Spectrometry; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Spectrophotometry, Infrared

2012
Recent advances in the development of selective human MAO-B inhibitors: (hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines.
    European journal of medicinal chemistry, 2012, Volume: 58

    Topics: Dose-Response Relationship, Drug; Humans; Hydrazines; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2012
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors.
    European journal of medicinal chemistry, 2013, Volume: 59

    Topics: Cells, Cultured; Curcumin; Enzyme Activation; Humans; Inhibitory Concentration 50; Models, Molecular; Monoamine Oxidase Inhibitors; Quantum Theory; Structure-Activity Relationship

2013
Design, synthesis, and in vitro hMAO-B inhibitory evaluation of some 1-methyl-3,5-diphenyl-4,5-dihydro-1H-pyrazoles.
    Bioorganic & medicinal chemistry letters, 2013, Sep-15, Volume: 23, Issue:18

    Topics: Dose-Response Relationship, Drug; Drug Design; Enzyme Inhibitors; Humans; Molecular Structure; Monoamine Oxidase; Pyrazoles; Structure-Activity Relationship

2013
Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors.
    Bioorganic & medicinal chemistry, 2014, May-15, Volume: 22, Issue:10

    Topics: Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Design; Humans; Isoenzymes; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Stereoisomerism; Structure-Activity Relationship; Thiazoles

2014
Exploring new selective 3-benzylquinoxaline-based MAO-A inhibitors: design, synthesis, biological evaluation and docking studies.
    European journal of medicinal chemistry, 2015, Mar-26, Volume: 93

    Topics: Animals; Catalytic Domain; Cattle; Chemistry Techniques, Synthetic; Drug Design; Humans; Male; Mice; Molecular Docking Simulation; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quinoxalines; Stereoisomerism; Structure-Activity Relationship

2015
Design, synthesis, and biological evaluation of oxindole derivatives as antidepressive agents.
    Bioorganic & medicinal chemistry letters, 2015, Nov-15, Volume: 25, Issue:22

    Topics: Animals; Antidepressive Agents; Benzylidene Compounds; Clorgyline; Imipramine; Indoles; Lactams; Mice; Moclobemide; Molecular Docking Simulation; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2015
Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold.
    European journal of medicinal chemistry, 2016, Jan-27, Volume: 108

    Topics: Computer Simulation; Dose-Response Relationship, Drug; Drug Design; Humans; Molecular Dynamics Simulation; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxadiazoles; Structure-Activity Relationship

2016
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors.
    European journal of medicinal chemistry, 2016, Jul-19, Volume: 117

    Topics: Chromans; Humans; Hydrogen Bonding; Inhibitory Concentration 50; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Sensitivity and Specificity; Solvents; Structure-Activity Relationship

2016
MAO inhibitory activity of bromo-2-phenylbenzofurans: synthesis,
    MedChemComm, 2017, Sep-01, Volume: 8, Issue:9

    Topics:

2017
Novel 1,3,4-thiadiazole compounds as potential MAO-A inhibitors - design, synthesis, biological evaluation and molecular modelling.
    RSC medicinal chemistry, 2020, Sep-01, Volume: 11, Issue:9

    Topics:

2020
Effect of the selective MAO-A inhibitors brofaromine, clorgyline and moclobemide on human platelet MAO-B activity.
    Journal of neural transmission. General section, 1992, Volume: 89, Issue:1-2

    Topics: Adult; Benzamides; Blood Platelets; Clorgyline; Female; Humans; Male; Moclobemide; Monoamine Oxidase Inhibitors; Piperidines

1992
Deamination of norepinephrine, dopamine, and serotonin by type A monoamine oxidase in discrete regions of the rat brain and inhibition by RS-8359.
    Japanese journal of pharmacology, 1991, Volume: 55, Issue:1

    Topics: Animals; Benzamides; Biogenic Monoamines; Brain; Cerebral Cortex; Clorgyline; Corpus Striatum; Deamination; Dopamine; Dose-Response Relationship, Drug; Hippocampus; Male; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nitriles; Norepinephrine; Pyrimidines; Rats; Rats, Inbred Strains; Selegiline; Serotonin

1991
Binding of [3H]brofaromine to monoamine oxidase A in vivo: displacement by clorgyline and moclobemide.
    European journal of pharmacology, 1990, May-16, Volume: 180, Issue:2-3

    Topics: Animals; Benzamides; Binding, Competitive; Biogenic Monoamines; Clorgyline; In Vitro Techniques; Male; Microsomes, Liver; Moclobemide; Monoamine Oxidase; Piperidines; Proadifen; Propylamines; Rats; Rats, Inbred Strains; Tissue Distribution

1990
Enhancement of 5-HT-induced anorexia: a test of the reversibility of monoamine oxidase inhibitors.
    Psychopharmacology, 1989, Volume: 98, Issue:2

    Topics: Animals; Benzamides; Clorgyline; Drug Synergism; Feeding Behavior; Male; Moclobemide; Monoamine Oxidase Inhibitors; Oxazoles; Oxazolidinones; Piperidines; Rats; Rats, Inbred Strains; Serotonin

1989
The effects of monoamine oxidase inhibitors on the ejaculatory response induced by 5-methoxy-N,N-dimethyltryptamine in the rat.
    British journal of pharmacology, 1986, Volume: 88, Issue:4

    Topics: Animals; Benzamides; Clorgyline; Dose-Response Relationship, Drug; Ejaculation; Male; Methoxydimethyltryptamines; Moclobemide; Monoamine Oxidase Inhibitors; Nialamide; p-Chloroamphetamine; Pargyline; Rats; Receptors, Serotonin; Selegiline; Serotonin; Time Factors

1986
SR 95191, a selective inhibitor of type A monoamine oxidase with dopaminergic properties. I. Psychopharmacological profile in rodents.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: 5-Hydroxytryptophan; Amphetamines; Animals; Antidepressive Agents; Behavior, Animal; Benzamides; Body Temperature; Catalepsy; Clorgyline; Drug Interactions; Female; Haloperidol; Imipramine; Levodopa; Male; Mice; Moclobemide; Monoamine Oxidase Inhibitors; Motor Activity; Nomifensine; Oxotremorine; Pargyline; Piperidines; Pyridazines; Rats; Rats, Inbred Strains; Reserpine; Selegiline; Stereotyped Behavior

1987
SR 95191, a selective inhibitor of type A monoamine oxidase with dopaminergic properties. II. Biochemical characterization of monoamine oxidase inhibition.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: Animals; Benzamides; Biogenic Amines; Brain; Clorgyline; Dopamine; Duodenum; Harmaline; Isoenzymes; Liver; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Oxazolidinones; Pyridazines; Rats; Selegiline; Synaptosomes

1987
Reversible, enzyme-activated monoamine oxidase inhibitors: new advances.
    Pharmacological research communications, 1988, Volume: 20 Suppl 4

    Topics: Animals; Benzamides; Brain; Clorgyline; Humans; In Vitro Techniques; Male; Moclobemide; Monoamine Oxidase Inhibitors; Phenelzine; Picolinic Acids; Piperidines; Rats; Selegiline

1988
Potentiation of tyramine pressor responses in conscious rats by reversible inhibitors of monoamine oxidase.
    Journal of neural transmission. Supplementum, 1988, Volume: 26

    Topics: Animals; Benzamides; Blood Pressure; Clorgyline; Drug Synergism; Male; Moclobemide; Monoamine Oxidase Inhibitors; Oxazoles; Oxazolidinones; Phenethylamines; Piperidines; Rats; Rats, Inbred Strains; Tyramine

1988
[Effect of benzamide derivatives on convulsions induced by the toxic action of oxygen in rats].
    Biulleten' eksperimental'noi biologii i meditsiny, 1987, Volume: 104, Issue:10

    Topics: Animals; Anticonvulsants; Benzamides; Brain; Clorgyline; Drug Evaluation, Preclinical; Heart; Male; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Myocardium; Oxygen; Rats; Seizures

1987
On the reversibility of reversible MAO inhibitors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzamides; Brain; Clorgyline; Dopamine; Female; Homovanillic Acid; Kinetics; Liver; Moclobemide; Monoamine Oxidase Inhibitors; Oxazoles; Oxazolidinones; Phenethylamines; Piperidines; Rats; Rats, Inbred Strains; Serotonin

1985
Chronic effect of the irreversible and reversible selective MAO-A inhibitors on rat pineal melatonin biosynthesis.
    Journal of neural transmission. Supplementum, 1994, Volume: 41

    Topics: Animals; Benzamides; Clorgyline; Female; Hydroxyindoleacetic Acid; Melatonin; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pineal Gland; Rats; Rats, Inbred F344; Serotonin; Time Factors

1994
The effects of phenelzine and other monoamine oxidase inhibitor antidepressants on brain and liver I2 imidazoline-preferring receptors.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Benzamides; Binding, Competitive; Brain; Chlorphenamidine; Clorgyline; Cytochrome P-450 Enzyme System; Dioxanes; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Injections, Intraperitoneal; Isocarboxazid; Liver; Male; Moclobemide; Monoamine Oxidase Inhibitors; Pargyline; Phenelzine; Propylamines; Rats; Rats, Sprague-Dawley; Receptors, Drug; Tranylcypromine

1995
Effect of moclobemide on rat brain monoamine oxidase A and B: comparison with harmaline and clorgyline.
    Progress in neuro-psychopharmacology & biological psychiatry, 1994, Volume: 18, Issue:4

    Topics: Animals; Benzamides; Brain; Clorgyline; Harmaline; Male; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Rats; Rats, Wistar

1994
The advent of a new generation of monoamine oxidase inhibitor antidepressants: pharmacologic studies with moclobemide and brofaromine.
    Clinical neuropharmacology, 1993, Volume: 16 Suppl 2

    Topics: Animals; Antidepressive Agents; Benzamides; Blood Pressure; Clorgyline; Desipramine; Heart Rate; Kidney; Moclobemide; Monoamine Oxidase Inhibitors; Piperidines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System

1993
Radiosynthesis of [11C]brofaromine, a potential tracer for imaging monoamine oxidase A.
    Nuclear medicine and biology, 1996, Volume: 23, Issue:3

    Topics: Animals; Benzamides; Brain; Carbon Radioisotopes; Clorgyline; Female; Hydrocarbons, Iodinated; Indicators and Reagents; Isoenzymes; Isotope Labeling; Macaca mulatta; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Piperidines; Tomography, Emission-Computed

1996
Inhibition of central monoamine oxidase by imidazoline2 site-selective ligands.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Benzamides; Binding Sites; Brain; Clorgyline; Imidazoles; Imidazoline Receptors; Isoenzymes; Kinetics; Ligands; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenethylamines; Rats; Receptors, Drug; Selegiline; Serotonin

1999
Moclobemide reduces intracellular pH and neuronal activity of CA3 neurones in guinea-pig hippocampal slices-implication for its neuroprotective properties.
    Neuropharmacology, 2000, Aug-23, Volume: 39, Issue:11

    Topics: Action Potentials; Animals; Clorgyline; Guinea Pigs; Hippocampus; Hydrogen-Ion Concentration; Moclobemide; Monoamine Oxidase Inhibitors; Neurons; Neuroprotective Agents

2000
A switch mechanism between locomotion and mouthing implicated in sensitization to quinpirole in rats.
    Psychopharmacology, 2000, Volume: 151, Issue:2-3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Brain Chemistry; Clorgyline; Dopamine; Dopamine Agonists; Male; Moclobemide; Monoamine Oxidase Inhibitors; Motor Activity; Neostriatum; Quinpirole; Rats; Rats, Long-Evans; Serotonin; Stereotyped Behavior

2000
cDNA gene expression profile of rat hippocampus after chronic treatment with antidepressant drugs.
    Journal of neural transmission (Vienna, Austria : 1996), 2003, Volume: 110, Issue:12

    Topics: Activating Transcription Factor 1; Amitriptyline; Animals; Antidepressive Agents; Behavior, Animal; Clorgyline; Cyclic AMP; DNA Primers; DNA-Binding Proteins; DNA, Complementary; Hippocampus; Male; Moclobemide; Oligonucleotide Array Sequence Analysis; Rats; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Transcription Factors

2003
Inhibition of monoamine oxidase activity by antidepressants and mood stabilizers.
    Neuro endocrinology letters, 2010, Volume: 31, Issue:5

    Topics: Affect; Amitriptyline; Animals; Antidepressive Agents; Antimanic Agents; Benzodiazepines; Cerebral Cortex; Citalopram; Clorgyline; Cocaine; Cyclohexanols; Desipramine; Fluoxetine; Imipramine; In Vitro Techniques; Iproniazid; Lithium; Mianserin; Mirtazapine; Mitochondria; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Morpholines; Olanzapine; Pargyline; Reboxetine; Swine; Thiazepines; Valproic Acid; Venlafaxine Hydrochloride

2010