Page last updated: 2024-09-04

ml 1035 and cisapride

ml 1035 has been researched along with cisapride in 1 studies

*Cisapride: A substituted benzamide used for its prokinetic properties. It is used in the management of gastroesophageal reflux disease, functional dyspepsia, and other disorders associated with impaired gastrointestinal motility. (Martindale The Extra Pharmacopoeia, 31st ed) [MeSH]

*Cisapride: A substituted benzamide used for its prokinetic properties. It is used in the management of gastroesophageal reflux disease, functional dyspepsia, and other disorders associated with impaired gastrointestinal motility. (Martindale The Extra Pharmacopoeia, 31st ed) [MeSH]

Compound Research Comparison

Studies
(ml 1035)
Trials
(ml 1035)
Recent Studies (post-2010)
(ml 1035)
Studies
(cisapride)
Trials
(cisapride)
Recent Studies (post-2010) (cisapride)
10001,554390110

Protein Interaction Comparison

ProteinTaxonomyml 1035 (IC50)cisapride (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.767
3-hydroxy-3-methylglutaryl-coenzyme A reductaseHomo sapiens (human)3.37
Cytochrome P450 3A4Homo sapiens (human)0.3
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0098
Alpha-2A adrenergic receptorHomo sapiens (human)3.5923
Cytochrome P450 2D6Homo sapiens (human)0.07
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)0.1701
D(2) dopamine receptorHomo sapiens (human)0.35
Dipeptidyl peptidase 4Rattus norvegicus (Norway rat)2.69
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0098
Insulin receptor Rattus norvegicus (Norway rat)3.37
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)2.29
Alpha-2B adrenergic receptorHomo sapiens (human)3.3827
Alpha-2C adrenergic receptorHomo sapiens (human)3.26
DRattus norvegicus (Norway rat)0.0065
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)3.6495
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0065
D(1A) dopamine receptorHomo sapiens (human)1.7
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0065
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0065
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)2.29
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.0065
Alpha-1D adrenergic receptorHomo sapiens (human)0.083
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0054
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.2597
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)3.6495
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)4.47
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)4.47
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0098
Sodium-dependent serotonin transporterHomo sapiens (human)0.384
Alpha-1A adrenergic receptorHomo sapiens (human)0.03
Prostaglandin G/H synthase 2Homo sapiens (human)3.37
Alpha-1B adrenergic receptorHomo sapiens (human)0.03
D(3) dopamine receptorHomo sapiens (human)0.144
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.9
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0407
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)2.29
D(2) dopamine receptorRattus norvegicus (Norway rat)0.535
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.2536
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)0.1701
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.994
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.9

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ahmed, NK; Butler, BT; Gaddis, RR; Linnik, MD1

Other Studies

1 other study(ies) available for ml 1035 and cisapride

ArticleYear
Analysis of serotonergic mechanisms underlying benzamide-induced gastroprokinesis.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:2

    Topics: Animals; Benzamides; Cisapride; Electric Stimulation; Female; Gastric Emptying; Gastrointestinal Transit; Guinea Pigs; Ileum; In Vitro Techniques; Male; Metoclopramide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin Antagonists

1991