mk 912 has been researched along with rx 821002 in 9 studies
Studies (mk 912) | Trials (mk 912) | Recent Studies (post-2010) (mk 912) | Studies (rx 821002) | Trials (rx 821002) | Recent Studies (post-2010) (rx 821002) |
---|---|---|---|---|---|
60 | 3 | 2 | 317 | 0 | 45 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 7 (77.78) | 18.2507 |
2000's | 2 (22.22) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bouloumié, A; Devedjian, JC; Lafontan, M; Planat, V; Record, M; Saulnier-Blache, JS; Valet, P | 1 |
Uhlén, S; Wikberg, JE; Wikberg-Matsson, A | 1 |
Starke, K; Trendelenburg, AU; Wahl, CA | 1 |
Castan, I; Devedjian, JC; Lafontan, M; Paris, H; Valet, P | 1 |
Akerman, KE; Cockcroft, V; Huifang, G; Jansson, CC; Kukkonen, JP; Savola, JM; Wurster, S | 1 |
Dambrova, M; Gu, Y; Näsman, J; Schiöth, HB; Uhlén, S; Wikberg, JE; Wikberg-Matsson, A | 1 |
Cayla, C; Gales, C; Paris, H; Quinchon, F; Roquelaine, C; Schaak, S | 1 |
Bylund, DB; Gerety, ME; Happe, HK; Murrin, LC | 1 |
Cussac, D; Denis, C; Flordellis, C; Gales, C; Paris, H; Schaak, S | 1 |
9 other study(ies) available for mk 912 and rx 821002
Article | Year |
---|---|
Alpha 2-adrenergic stimulation promotes preadipocyte proliferation. Involvement of mitogen-activated protein kinases.
Topics: 3T3 Cells; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adipocytes; Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Bucladesine; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; Cells, Cultured; Clone Cells; Clonidine; Cyclic AMP; Dioxanes; Humans; Idazoxan; Kinetics; Male; Mice; Pertussis Toxin; Quinolizines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Transfection; Virulence Factors, Bordetella | 1994 |
Identification of drugs subtype-selective for alpha 2A-, alpha 2B-, and alpha 2C-adrenoceptors in the pig cerebellum and kidney cortex.
Topics: Animals; Binding, Competitive; Cerebellum; Dibenzazepines; Dioxanes; Idazoxan; Imidazoles; Kidney Cortex; Quinolizines; Receptors, Adrenergic, alpha-2; Swine | 1995 |
Antagonists that differentiate between alpha 2A-and alpha 2D-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoreceptors; Benzofurans; Brimonidine Tartrate; Cerebral Cortex; Dioxanes; Electric Stimulation; Female; Guinea Pigs; Idazoxan; Imidazoles; Isotope Labeling; Male; Norepinephrine; Oxathiins; Quinolizines; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha-2; Structure-Activity Relationship; Tritium | 1996 |
Human adipocytes express alpha 2-adrenergic receptor of the alpha 2A-subtype only: pharmacological and genetic evidence.
Topics: Adipocytes; Adrenergic alpha-Antagonists; Adult; Cell Line; Female; Humans; Idazoxan; In Vitro Techniques; Membranes; Middle Aged; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Ribonucleases; RNA; RNA Probes | 1995 |
Different apparent modes of inhibition of alpha2A-adrenoceptor by alpha2-adrenoceptor antagonists.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Humans; Idazoxan; Quinolizines; Receptors, Adrenergic, alpha-2; Tritium; Tumor Cells, Cultured; Yohimbine | 1997 |
[3H]RS79948-197 binding to human, rat, guinea pig and pig alpha2A-, alpha2B- and alpha2C-adrenoceptors. Comparison with MK912, RX821002, rauwolscine and yohimbine.
Topics: Adrenergic Agents; Animals; Guinea Pigs; Humans; Idazoxan; Isoquinolines; Naphthyridines; Quinolizines; Rats; Receptors, Adrenergic, alpha-2; Swine; Yohimbine | 1998 |
Homologous regulation of the alpha2C-adrenoceptor subtype in human hepatocarcinoma, HepG2.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Binding, Competitive; Brimonidine Tartrate; Carcinoma, Hepatocellular; Humans; Idazoxan; Quinolizines; Quinoxalines; Receptors, Adrenergic, alpha-2; RNA, Messenger; Tritium; Tumor Cells, Cultured | 1999 |
Inverse agonism at alpha(2)-adrenoceptors in native tissue.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Guanosine Triphosphate; Idazoxan; Kinetics; Protein Binding; Quinolizines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine | 2000 |
alpha(2B)-Adrenergic receptors activate MAPK and modulate proliferation of primary cultured proximal tubule cells.
Topics: Adrenergic alpha-Antagonists; Animals; Arachidonic Acid; Calcimycin; Cell Division; Cell Line; Cell Membrane; Cells, Cultured; Enzyme Activation; Epinephrine; Humans; Idazoxan; Ionophores; Kidney Tubules, Proximal; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Pertussis Toxin; Phosphorylation; Protein Kinase C; Quinolizines; Rats; Receptors, Adrenergic, alpha-2; Signal Transduction; Tritium; Virulence Factors, Bordetella | 2002 |