Page last updated: 2024-09-03

mk 912 and rx 821002

mk 912 has been researched along with rx 821002 in 9 studies

Compound Research Comparison

Studies
(mk 912)
Trials
(mk 912)
Recent Studies (post-2010)
(mk 912)
Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010) (rx 821002)
6032317045

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (77.78)18.2507
2000's2 (22.22)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bouloumié, A; Devedjian, JC; Lafontan, M; Planat, V; Record, M; Saulnier-Blache, JS; Valet, P1
Uhlén, S; Wikberg, JE; Wikberg-Matsson, A1
Starke, K; Trendelenburg, AU; Wahl, CA1
Castan, I; Devedjian, JC; Lafontan, M; Paris, H; Valet, P1
Akerman, KE; Cockcroft, V; Huifang, G; Jansson, CC; Kukkonen, JP; Savola, JM; Wurster, S1
Dambrova, M; Gu, Y; Näsman, J; Schiöth, HB; Uhlén, S; Wikberg, JE; Wikberg-Matsson, A1
Cayla, C; Gales, C; Paris, H; Quinchon, F; Roquelaine, C; Schaak, S1
Bylund, DB; Gerety, ME; Happe, HK; Murrin, LC1
Cussac, D; Denis, C; Flordellis, C; Gales, C; Paris, H; Schaak, S1

Other Studies

9 other study(ies) available for mk 912 and rx 821002

ArticleYear
Alpha 2-adrenergic stimulation promotes preadipocyte proliferation. Involvement of mitogen-activated protein kinases.
    The Journal of biological chemistry, 1994, Dec-02, Volume: 269, Issue:48

    Topics: 3T3 Cells; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adipocytes; Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Bucladesine; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; Cells, Cultured; Clone Cells; Clonidine; Cyclic AMP; Dioxanes; Humans; Idazoxan; Kinetics; Male; Mice; Pertussis Toxin; Quinolizines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Transfection; Virulence Factors, Bordetella

1994
Identification of drugs subtype-selective for alpha 2A-, alpha 2B-, and alpha 2C-adrenoceptors in the pig cerebellum and kidney cortex.
    European journal of pharmacology, 1995, Sep-25, Volume: 284, Issue:3

    Topics: Animals; Binding, Competitive; Cerebellum; Dibenzazepines; Dioxanes; Idazoxan; Imidazoles; Kidney Cortex; Quinolizines; Receptors, Adrenergic, alpha-2; Swine

1995
Antagonists that differentiate between alpha 2A-and alpha 2D-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoreceptors; Benzofurans; Brimonidine Tartrate; Cerebral Cortex; Dioxanes; Electric Stimulation; Female; Guinea Pigs; Idazoxan; Imidazoles; Isotope Labeling; Male; Norepinephrine; Oxathiins; Quinolizines; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha-2; Structure-Activity Relationship; Tritium

1996
Human adipocytes express alpha 2-adrenergic receptor of the alpha 2A-subtype only: pharmacological and genetic evidence.
    Fundamental & clinical pharmacology, 1995, Volume: 9, Issue:6

    Topics: Adipocytes; Adrenergic alpha-Antagonists; Adult; Cell Line; Female; Humans; Idazoxan; In Vitro Techniques; Membranes; Middle Aged; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Ribonucleases; RNA; RNA Probes

1995
Different apparent modes of inhibition of alpha2A-adrenoceptor by alpha2-adrenoceptor antagonists.
    European journal of pharmacology, 1997, Sep-17, Volume: 335, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Humans; Idazoxan; Quinolizines; Receptors, Adrenergic, alpha-2; Tritium; Tumor Cells, Cultured; Yohimbine

1997
[3H]RS79948-197 binding to human, rat, guinea pig and pig alpha2A-, alpha2B- and alpha2C-adrenoceptors. Comparison with MK912, RX821002, rauwolscine and yohimbine.
    European journal of pharmacology, 1998, Feb-05, Volume: 343, Issue:1

    Topics: Adrenergic Agents; Animals; Guinea Pigs; Humans; Idazoxan; Isoquinolines; Naphthyridines; Quinolizines; Rats; Receptors, Adrenergic, alpha-2; Swine; Yohimbine

1998
Homologous regulation of the alpha2C-adrenoceptor subtype in human hepatocarcinoma, HepG2.
    British journal of pharmacology, 1999, Volume: 126, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Binding, Competitive; Brimonidine Tartrate; Carcinoma, Hepatocellular; Humans; Idazoxan; Quinolizines; Quinoxalines; Receptors, Adrenergic, alpha-2; RNA, Messenger; Tritium; Tumor Cells, Cultured

1999
Inverse agonism at alpha(2)-adrenoceptors in native tissue.
    European journal of pharmacology, 2000, Jun-16, Volume: 398, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Guanosine Triphosphate; Idazoxan; Kinetics; Protein Binding; Quinolizines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

2000
alpha(2B)-Adrenergic receptors activate MAPK and modulate proliferation of primary cultured proximal tubule cells.
    American journal of physiology. Renal physiology, 2002, Volume: 282, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Arachidonic Acid; Calcimycin; Cell Division; Cell Line; Cell Membrane; Cells, Cultured; Enzyme Activation; Epinephrine; Humans; Idazoxan; Ionophores; Kidney Tubules, Proximal; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Pertussis Toxin; Phosphorylation; Protein Kinase C; Quinolizines; Rats; Receptors, Adrenergic, alpha-2; Signal Transduction; Tritium; Virulence Factors, Bordetella

2002