Page last updated: 2024-09-03

mk 912 and phentolamine

mk 912 has been researched along with phentolamine in 2 studies

Compound Research Comparison

Studies
(mk 912)
Trials
(mk 912)
Recent Studies (post-2010)
(mk 912)
Studies
(phentolamine)
Trials
(phentolamine)
Recent Studies (post-2010) (phentolamine)
60329,141270265

Protein Interaction Comparison

ProteinTaxonomymk 912 (IC50)phentolamine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.396
Alpha-2A adrenergic receptorHomo sapiens (human)0.006
Cytochrome P450 2D6Homo sapiens (human)10
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0316
Alpha-2B adrenergic receptorHomo sapiens (human)0.018
Alpha-2C adrenergic receptorHomo sapiens (human)0.11
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0316
Alpha-1D adrenergic receptorHomo sapiens (human)0.0173
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.359
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.396
Alpha-1A adrenergic receptorHomo sapiens (human)0.0011
Alpha-1B adrenergic receptorHomo sapiens (human)0.0108
5-hydroxytryptamine receptor 2BHomo sapiens (human)3.807
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0316
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.5495

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dan, K; Hirose, H; Maruyama, H; Nakamura, K; Saruta, T; Seto, Y1
Goto, K; Ishikawa, T; Kashihara, T; Nakayama, K; Sahara, Y1

Other Studies

2 other study(ies) available for mk 912 and phentolamine

ArticleYear
Effects of alpha 2-adrenergic agonism, imidazolines, and G-protein on insulin secretion in beta cells.
    Metabolism: clinical and experimental, 1997, Volume: 46, Issue:10

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Cricetinae; Glucose; GTP-Binding Proteins; Humans; Imidazoles; Indoles; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Kinetics; Molecular Structure; Oxymetazoline; Pancreatic Neoplasms; Pertussis Toxin; Phentolamine; Pyrroles; Quinolizines; Receptors, Adrenergic, alpha-2; Tumor Cells, Cultured; Virulence Factors, Bordetella

1997
Differential involvement of alpha1-adrenoceptors in vasoconstrictor responses to cooling in mouse plantar arteries in vitro and in vivo.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2009, Volume: 45, Issue:2-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Brimonidine Tartrate; Cold Temperature; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle, Smooth, Vascular; Phentolamine; Phenylephrine; Quinolizines; Quinoxalines; Receptors, Adrenergic, alpha-1; Regional Blood Flow; Skin; Tetrodotoxin; Vasoconstriction

2009