Page last updated: 2024-09-03

mk 912 and moxonidine

mk 912 has been researched along with moxonidine in 3 studies

Compound Research Comparison

Studies
(mk 912)
Trials
(mk 912)
Recent Studies (post-2010)
(mk 912)
Studies
(moxonidine)
Trials
(moxonidine)
Recent Studies (post-2010) (moxonidine)
60325058689

Protein Interaction Comparison

ProteinTaxonomymk 912 (IC50)moxonidine (IC50)
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.7021
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.7021

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Campbell, WR; Potter, DE1
Blue, DR; Dillon, MP; Eglen, RM; Jasper, JR; Lesnick, JD; MacLennan, SJ; Zhu, QM2

Other Studies

3 other study(ies) available for mk 912 and moxonidine

ArticleYear
The central effects of moxonidine on intraocular pressure and its antagonism by L-659, 066 and L-657, 743 in the rabbit.
    Progress in neuro-psychopharmacology & biological psychiatry, 1994, Volume: 18, Issue:6

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Imidazoles; Injections, Intravenous; Injections, Intraventricular; Intraocular Pressure; Male; Pupil; Quinolizines; Rabbits

1994
Cardiovascular effects of rilmenidine, moxonidine and clonidine in conscious wild-type and D79N alpha2A-adrenoceptor transgenic mice.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Adrenergic alpha-Antagonists; Amino Acid Substitution; Animals; Binding, Competitive; Blood Pressure; Cardiovascular Agents; Cell Line; Clonidine; Consciousness; Dogs; Heart Rate; Humans; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Mice; Mice, Inbred Strains; Mice, Transgenic; Mutation; Naphthyridines; Oxazoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Rilmenidine; Saphenous Vein; Tritium

1999
alpha 2A-adrenoceptors, not I1-imidazoline receptors, mediate the hypotensive effects of rilmenidine and moxonidine in conscious mice. In vivo and in vitro studies.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cell Line; Dogs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypotension; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Quinolizines; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Transfection

1999