Page last updated: 2024-09-04

mk 767 and thiazoles

mk 767 has been researched along with thiazoles in 12 studies

Compound Research Comparison

Studies
(mk 767)
Trials
(mk 767)
Recent Studies (post-2010)
(mk 767)
Studies
(thiazoles)
Trials
(thiazoles)
Recent Studies (post-2010) (thiazoles)
3201033,1792,10012,330

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (33.33)18.2507
2000's8 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Akanuma, Y; Ide, T; Kadowaki, T; Mochizuki, T; Murakami, K; Ohashi, M; Tobe, K; Yazaki, Y1
Awano, K; Kinoshita, S; Maeda, T; Miyachi, H; Murakami, K; Nomura, M; Satoh, H; Tsunoda, M1
Ide, T; Kadowaki, T; Mochizuki, T; Murakami, K; Suzuki, M1
Ide, T; Mochizuki, T; Murakami, K; Ohashi, M; Tsunoda, M1
Ide, T; Mochizuki, T; Murakami, K; Nakazawa, T1
Chaput, E; Edgar, AD; Saladin, R; Silvestre, M1
Ide, T; Kadowaki, T; Mochizuki, T; Murakami, K; Nakazawa, T; Okazaki, T1
Yamanouchi, T1
Fujita, H; Hirose, H; Kawai, T; Miyashita, K; Ogawa, T; Saruta, T; Seto, Y; Ukeda, K; Yajima, K; Yamada, T; Yamamoto, Y1
Calkin, AC; Cooper, ME; Thomas, MC1
Narce, M; Poisson, JP1
Miyachi, H1

Reviews

3 review(s) available for mk 767 and thiazoles

ArticleYear
[KRP-297, MCC-555].
    Nihon rinsho. Japanese journal of clinical medicine, 2001, Volume: 59, Issue:11

    Topics: Animals; Clinical Trials, Phase II as Topic; Diabetes Mellitus; Glucose; Humans; Hypoglycemic Agents; Lipid Metabolism; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Thiazolidines; Transcription Factors

2001
MK-767. Kyorin/Banyu/Merck.
    Current opinion in investigational drugs (London, England : 2000), 2003, Volume: 4, Issue:4

    Topics: Animals; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Contraindications; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Thiazoles; Thiazolidines

2003
[Design and synthesis of subtype- and species-selective peroxisome proliferator-activated receptor (PPAR) alpha ligands].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 2004, Volume: 124, Issue:11

    Topics: Animals; Drug Design; Humans; Phenylpropionates; PPAR alpha; Species Specificity; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Thiazolidines

2004

Other Studies

9 other study(ies) available for mk 767 and thiazoles

ArticleYear
A novel insulin sensitizer acts as a coligand for peroxisome proliferator-activated receptor-alpha (PPAR-alpha) and PPAR-gamma: effect of PPAR-alpha activation on abnormal lipid metabolism in liver of Zucker fatty rats.
    Diabetes, 1998, Volume: 47, Issue:12

    Topics: Acyl-CoA Oxidase; Adipose Tissue; Animals; Blood Glucose; Body Weight; Carrier Proteins; Fatty Acid-Binding Protein 7; Fatty Acid-Binding Proteins; Fatty Acids; Gene Expression; Hypoglycemic Agents; Insulin; Ligands; Lipid Metabolism; Liver; Male; Myelin P2 Protein; Neoplasm Proteins; Nerve Tissue Proteins; Obesity; Organ Size; Oxidoreductases; Radioligand Assay; Rats; Rats, Wistar; Rats, Zucker; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Rosiglitazone; Thiazoles; Thiazolidinediones; Thiazolidines; Transcription Factors; Transcriptional Activation; Triglycerides

1998
(3-substituted benzyl)thiazolidine-2,4-diones as structurally new antihyperglycemic agents.
    Bioorganic & medicinal chemistry letters, 1999, Feb-22, Volume: 9, Issue:4

    Topics: Animals; Blood Glucose; Hypoglycemic Agents; Insulin; Mice; Mice, Obese; Pioglitazone; Structure-Activity Relationship; Thiazoles; Thiazolidinediones; Thiazolidines; Triglycerides

1999
Evidence for direct binding of fatty acids and eicosanoids to human peroxisome proliferators-activated receptor alpha.
    Biochemical and biophysical research communications, 1999, Jul-14, Volume: 260, Issue:3

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Eicosanoids; Fatty Acids; Fatty Acids, Unsaturated; Gene Expression Regulation; Genes, Reporter; Humans; Hydroxyeicosatetraenoic Acids; Inhibitory Concentration 50; Kinetics; Ligands; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidines; Transcription Factors; Transfection

1999
Amelioration by KRP-297, a new thiazolidinedione, of impaired glucose uptake in skeletal muscle from obese insulin-resistant animals.
    Metabolism: clinical and experimental, 1999, Volume: 48, Issue:11

    Topics: Animals; Blood Glucose; Glucose; Hypoglycemic Agents; Insulin Resistance; Male; Mice; Mice, Inbred C57BL; Muscle, Skeletal; Obesity; Thiazoles; Thiazolidines

1999
Tissue-specific actions of antidiabetic thiazolidinediones on the reduced fatty acid oxidation in skeletal muscle and liver of Zucker diabetic fatty rats.
    Metabolism: clinical and experimental, 2000, Volume: 49, Issue:4

    Topics: Administration, Oral; Animals; Chromans; Diabetes Mellitus; Fatty Acids; Hypoglycemic Agents; Liver; Male; Muscle, Skeletal; Obesity; Oxidation-Reduction; Palmitic Acid; Rats; Rats, Zucker; Reference Values; Substrate Specificity; Thiazoles; Thiazolidinediones; Thiazolidines; Triglycerides; Troglitazone

2000
Fenofibrate and rosiglitazone lower serum triglycerides with opposing effects on body weight.
    Biochemical and biophysical research communications, 2000, May-10, Volume: 271, Issue:2

    Topics: Acyl-CoA Oxidase; Animals; Apolipoprotein A-I; Apolipoprotein C-III; Apolipoproteins C; Body Weight; Carrier Proteins; Fatty Acid-Binding Protein 7; Fatty Acid-Binding Proteins; Fenofibrate; Hypolipidemic Agents; Male; Mice; Myelin P2 Protein; Neoplasm Proteins; Nerve Tissue Proteins; Oxidoreductases; Rats; Rats, Zucker; Receptors, Cytoplasmic and Nuclear; Rosiglitazone; Thiazoles; Thiazolidinediones; Thiazolidines; Time Factors; Transcription Factors; Triglycerides

2000
Fatty-acyl-CoA thioesters inhibit recruitment of steroid receptor co-activator 1 to alpha and gamma isoforms of peroxisome-proliferator-activated receptors by competing with agonists.
    The Biochemical journal, 2001, Jan-15, Volume: 353, Issue:Pt 2

    Topics: Acyl Coenzyme A; Animals; Binding, Competitive; Fatty Acids; Histone Acetyltransferases; Ligands; Liver; Male; Muscles; Nuclear Receptor Coactivator 1; Plasmids; Protein Isoforms; Rats; Rats, Zucker; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Thiazoles; Thiazolidines; Transcription Factors; Tritium

2001
Combination therapy with PPARgamma and PPARalpha agonists increases glucose-stimulated insulin secretion in db/db mice.
    American journal of physiology. Endocrinology and metabolism, 2003, Volume: 284, Issue:5

    Topics: Animals; Bezafibrate; Body Weight; Diabetes Mellitus; Drug Therapy, Combination; Glucose; Glucose Transporter Type 2; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Monosaccharide Transport Proteins; Pancreas; Pioglitazone; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Thiazolidines; Transcription Factors

2003
Novel PPARgamma-dependent and independent effects for thiazolidinediones.
    Current opinion in lipidology, 2003, Volume: 14, Issue:6

    Topics: Animals; Bezafibrate; Body Weight; Chromans; Diabetes Mellitus, Type 2; Gene Expression; Humans; Insulin-Like Growth Factor Binding Protein 1; Insulin-Like Growth Factor Binding Proteins; Mice; Monocytes; Pancreas; Pioglitazone; PPAR alpha; PPAR gamma; Pregnancy Proteins; Pregnane X Receptor; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Rosiglitazone; Thiazoles; Thiazolidinediones; Thiazolidines; Troglitazone; Tumor Necrosis Factor-alpha

2003