Page last updated: 2024-09-03

mk 0663 and gw406381x

mk 0663 has been researched along with gw406381x in 2 studies

Compound Research Comparison

Studies
(mk 0663)
Trials
(mk 0663)
Recent Studies (post-2010)
(mk 0663)
Studies
(gw406381x)
Trials
(gw406381x)
Recent Studies (post-2010) (gw406381x)
5491732651547

Protein Interaction Comparison

ProteinTaxonomymk 0663 (IC50)gw406381x (IC50)
Prostaglandin G/H synthase 2Homo sapiens (human)0.003

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beswick, P; Bingham, S; Bountra, C; Brown, T; Browning, K; Campbell, I; Chessell, I; Clayton, N; Collins, S; Corfield, J; Guntrip, S; Haslam, C; Lambeth, P; Lucas, F; Mathews, N; Murkit, G; Naylor, A; Pegg, N; Pickup, E; Player, H; Price, H; Stevens, A; Stratton, S; Wiseman, J1
Ramajayam, R1

Reviews

1 review(s) available for mk 0663 and gw406381x

ArticleYear
Medicinal chemistry of vicinal diaryl scaffold: A mini review.
    European journal of medicinal chemistry, 2019, Jan-15, Volume: 162

    Topics: Carbonic Anhydrase IV; Chemistry, Pharmaceutical; Cyclooxygenase 2 Inhibitors; Drug Discovery; Humans; Hydrocarbons, Aromatic; Structure-Activity Relationship

2019

Other Studies

1 other study(ies) available for mk 0663 and gw406381x

ArticleYear
Identification of 2,3-diaryl-pyrazolo[1,5-b]pyridazines as potent and selective cyclooxygenase-2 inhibitors.
    Bioorganic & medicinal chemistry letters, 2004, Nov-01, Volume: 14, Issue:21

    Topics: Administration, Oral; Animals; Arthritis, Experimental; Biological Availability; Brain; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Freund's Adjuvant; Humans; Infusions, Intravenous; Male; Membrane Proteins; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Pyridazines; Rats; Structure-Activity Relationship

2004