miltefosine and pentamidine

miltefosine has been researched along with pentamidine in 51 studies

Research

Studies (51)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's11 (21.57)29.6817
2010's35 (68.63)24.3611
2020's5 (9.80)2.80

Authors

AuthorsStudies
Boykin, DW; Brun, R; Salem, MM; Stephens, CE; Tanious, F; Werbovetz, KA; Wilson, WD1
Goyal, N; Gupta, S; Pandey, S; Suryawanshi, SN1
Delfín, DA; Morgan, RE; Werbovetz, KA; Zhu, X1
Bisht, SS; Gupta, S; Kumar, A; Mishra, M; Mittal, M; Pandey, VP; Sane, SA; Siddiqi, MI; Tripathi, RP; Verma, A1
Boykin, DW; Hall, JE; Kyle, DE; Liu, Q; Madhubala, R; Mandal, S; Munde, M; Pandharkar, T; Parman, T; Riccio, E; Srivastava, A; Stephens, CE; Sweat, JM; Tidwell, RR; Wang, MZ; Werbovetz, KA; Wilson, WD; Zhu, X1
Baumann, K; Bischof, SK; Bringmann, G; Brun, R; Dreher, J; Gulder, T; Kaiser, M; Moll, H; Müller, S; Stich, A; Winter, C1
Carvalho, L; Castanys, S; Gamarro, F; Manzano, JI; Pérez-Victoria, JM1
Alami, M; Audisio, D; Bories, C; Brion, JD; Cojean, S; Huteau, F; Loiseau, PM; Messaoudi, S; Peyrat, JF1
Azas, N; Casanova, M; Castera-Ducros, C; Dumètre, A; Hutter, S; Kraiem-M'rabet, M; Laget, M; Mbatchi, L; Paloque, L; Rathelot, P; Rault, S; Remusat, V; Vanelle, P; Verhaeghe, P1
Chan, KF; Chan, TH; Chow, LM; Wong, IL1
Chauhan, PM; Gupta, S; Khan, S; Kidwai, S; Puri, SK; Shivahare, R; Srivastava, K; Tyagi, V1
Buisson, D; Fromentin, Y; Gaboriaud-Kolar, N; Grellier, P; Lallemand, MC; Lenta, BN; Loiseau, PM; Michel, S; Mouray, E; Wansi, JD1
Arafa, RK; Boykin, DW; Brun, R; Ismail, MA; Jones, SK; Pandharkar, T; Patrick, DA; Tidwell, RR; Wenzler, T; Werbovetz, KA; Zhu, X1
Abada, Z; Akagah, B; Cojean, S; Ferrié, L; Figadère, B; Loiseau, PM; Lormier, AT; Pomel, S1
Brun, R; Harel, D; Prinz, H; Schepmann, D; Schmidt, TJ; Wünsch, B1
Azas, N; Cantelli, C; Casanova, M; Castera-Ducros, C; Cohen, A; Crozet, MD; Hutter, S; Laget, M; Paloque, L; Rathelot, P; Remusat, V; Tanguy, F; Vanelle, P; Verhaeghe, P1
Chauhan, K; Chauhan, PM; Debnath, U; Gupta, S; Prabhakar, YS; Sharma, M; Shivahare, R1
Avery, VM; Baell, JB; Bergström, CA; Charman, SA; Ferrins, L; Gazdik, M; Jones, AJ; Kaiser, M; Rahmani, R; Ryan, E; Sykes, ML; Varghese, S; White, KL1
Blonski, C; Djilali, R; Jagu, E; Labruère, R; Loiseau, PM; Pethe, S; Pomel, S; Ramiandrasoa, F1
Azas, N; Castera-Ducros, C; Cohen, A; Hutter, S; Kieffer, C; Laget, M; M'Rabet, MK; Rathelot, P; Rault, S; Remusat, V; Vanelle, P; Verhaeghe, P1
Azas, N; Castera-Ducros, C; Cohen, A; Hutter, S; Kieffer, C; Laget, M; Paloque, L; Rathelot, P; Rault, S; Valentin, A; Vanelle, P; Verhaeghe, P1
Alexandre-Moreira, MS; da Matta, CB; DaCosta, JB; de Queiroz, AC; Del Cistia, Cde N; Gonçalves, VT; Sant'Anna, CM; Santos, MS1
Bosc, D; Cojean, S; Dubois, J; Franco, CH; Freitas-Junior, LH; Grellier, P; Loiseau, PM; Moraes, CB; Mouray, E1
Alunda, JM; Baptista, C; Behrens, B; Bifeld, E; Borsari, C; Clos, J; Cordeiro-da-Silva, A; Corral, MJ; Costantino, L; Costi, MP; Dello Iacono, L; Di Pisa, F; Eick, J; Ellinger, B; Ferrari, S; Gribbon, P; Gul, S; Henrich, S; Jiménez-Antón, MD; Keminer, O; Kohler, M; Kuzikov, M; Landi, G; Luciani, R; Mangani, S; Pellati, F; Poehner, I; Pozzi, C; Reinshagen, J; Santarem, N; Tait, A; Tejera Nevado, P; Torrado, J; Trande, M; Wade, RC; Witt, G; Wolf, M1
Blonski, C; Diez-Martinez, A; Jagu, E; Krauth-Siegel, RL; Labruère, R; Loiseau, PM; Pethe, S; Pomel, S; Ramiandrasoa, F1
Alcântara, LM; Alunda, JM; Baptista, C; Bertolacini, CD; Borsari, C; Bruno Dos Santos, P; Clos, J; Cordeiro-da-Silva, A; Corral, MJ; Costantino, L; Costi, MP; Ellinger, B; Ferrari, S; Fontana, V; Franco, CH; Freitas-Junior, LH; Gribbon, P; Gul, S; Kuzikov, M; Linciano, P; Moraes, CB; Olías, AI; Reinshagen, J; Santarem, N; Tait, A; Tejera Nevado, P; Torrado, J; Witt, G; Wolf, M1
Argüello-Garcia, R; Barbosa-Cabrera, E; Chan-Bacab, MJ; Colín-Lozano, B; Hernández-Núñez, E; León-Rivera, I; López-Guerrero, V; Moo-Puc, R; Navarrete-Vázquez, G; Ortega-Morales, BO; Scior, T1
Alcantara, LM; Cordeiro-da-Silva, A; Costantino, L; Costi, MP; Ellinger, B; Ferrari, S; Franco, CH; Freitas-Junior, LH; Gul, S; Kuzikov, M; Linciano, P; Luciani, R; Macedo, S; Moraes, CB; Pascoalino, B; Quotadamo, A; Santarem, N; Witt, G1
Ashok, P; Chander, S; Sankaranarayanan, M; Smith, TK1
Cantizani, J; Cogo, J; Corrêa, AG; Cotillo, I; Filho, BPD; Martín, JJ; Nakamura, CV; Sangi, DP; Ueda-Nakamura, T1
Azas, N; Basmaciyan, L; Belle Mbou, V; Boudot, C; Bourgeade-Delmas, S; Boutet-Robinet, É; Casanova, M; Castera-Ducros, C; Cohen, A; Courtioux, B; Fairlamb, AH; Fersing, C; Hutter, S; Laget, M; Milne, R; Pedron, J; Piednoel, M; Primas, N; Rathelot, P; Since, M; Sournia-Saquet, A; Valentin, A; Vanelle, P; Verhaeghe, P; Wyllie, S1
Baptista, C; Bonucci, A; Cordeiro-da-Silva, A; Costantino, L; Costi, MP; di Pisa, F; Ellinger, B; Ferrari, S; Franco, C; Gul, S; Iacono, LD; Kuzikov, M; Landi, G; Linciano, P; Luciani, R; Mangani, S; Moraes, CB; Müller, W; Pöhner, I; Pozzi, C; Quotadamo, A; Santarem, N; Sesenna, A; Witt, G; Wittig, U1
Bhatia, R; Gupta, O; Monga, V; Pradhan, T1
Carvalho, C; Cordeiro da Silva, A; Duarte, D; Kijjoa, A; Long, S; Moreira, R; Nogueira, F; Oliveira, R; Palmeira, A; Pinto, MMM; Resende, DISP; Santarém, N; Silva, AMS; Sousa, E1
Carvalho, MA; Cordeiro-da-Silva, A; Lopes, A; Santarém, N1
Sundar, S1
Berman, J1
Singh, S; Sivakumar, R1
Kumar, A; Sundar, S1
Bandyopadhyay, S; Chatterjee, M; Ganguly, S; Sarkar, A1
Minodier, P; Parola, P1
Acquaviva, V; Antinori, S; Bestetti, G; Corbellino, M; Foschi, A; Longhi, E; Meroni, L; Parravicini, C; Piolini, R; Trovati, S1
Chatterjee, M; Mandal, G; Sarkar, A; Singh, N; Sundar, S1
Click, J; Gee, SN; Hsu, MY; Rothschild, B; Saavedra, A; Sheth, V1
Kumar, M; Singh, N; Singh, RK1
Chirouze, C; Faucher, JF; Hoen, B; Le Moing, V; Morquin, D; Reynes, J1
de Paula, E; Giorgio, S; Ortega, V1
Calderón-Gomezcaseres, Á; Rodriguez-Morales, AJ; Villamil-Gómez, WE1
Alexandre-Moreira, MS; Alves, MA; Barreiro, EJ; Cavalcanti de Queiroz, A; Lima, LM1
Bano, S; Bibi, M; Choudhary, MI; Farooq, S; Khoso, BK; Shaikh, M; Yousuf, S; Zafar, H1
Kazemirad, E; Latifi, A; Mohebali, M; Rezaian, M; Soleimani, M; Yasami, S1

Reviews

7 review(s) available for miltefosine and pentamidine

ArticleYear
Recent advancements in anti-leishmanial research: Synthetic strategies and structural activity relationships.
    European journal of medicinal chemistry, 2021, Nov-05, Volume: 223

    Topics: Animals; Cell Line, Tumor; Heterocyclic Compounds; Humans; Leishmania; Leishmaniasis; Molecular Structure; Small Molecule Libraries; Structure-Activity Relationship; Trypanocidal Agents

2021
Current treatment approaches to leishmaniasis.
    Current opinion in infectious diseases, 2003, Volume: 16, Issue:5

    Topics: Amphotericin B; Antimony Sodium Gluconate; Antiprotozoal Agents; Clinical Trials as Topic; Fluconazole; Humans; Leishmaniasis; Paromomycin; Pentamidine; Phosphorylcholine

2003
Challenges and new discoveries in the treatment of leishmaniasis.
    Journal of infection and chemotherapy : official journal of the Japan Society of Chemotherapy, 2004, Volume: 10, Issue:6

    Topics: Amphotericin B; Animals; Antiprotozoal Agents; Drug Therapy, Combination; Humans; Leishmania; Leishmaniasis; Pentamidine; Phosphorylcholine; Psychodidae

2004
Cutaneous leishmaniasis treatment.
    Travel medicine and infectious disease, 2007, Volume: 5, Issue:3

    Topics: Administration, Cutaneous; Administration, Oral; Aminoquinolines; Amphotericin B; Animals; Antimony; Antiprotozoal Agents; Humans; Imiquimod; Injections, Intralesional; Injections, Intramuscular; Leishmaniasis, Cutaneous; Paromomycin; Pentamidine; Phosphorylcholine

2007
Post-kala-azar dermal leishmaniasis as an immune reconstitution inflammatory syndrome in a patient with acquired immune deficiency syndrome.
    The British journal of dermatology, 2007, Volume: 157, Issue:5

    Topics: Acquired Immunodeficiency Syndrome; Americas; Antiprotozoal Agents; Antiretroviral Therapy, Highly Active; Asia; Humans; Italy; Leishmaniasis, Cutaneous; Leishmaniasis, Visceral; Male; Middle Aged; Pentamidine; Phosphorylcholine; Travel

2007
Leishmaniasis: current status of available drugs and new potential drug targets.
    Asian Pacific journal of tropical medicine, 2012, Volume: 5, Issue:6

    Topics: Aminoquinolines; Amphotericin B; Antigens, Protozoan; Antimony Sodium Gluconate; Antiprotozoal Agents; Caspase Inhibitors; Cyclin-Dependent Kinases; Drug Discovery; Enzyme Inhibitors; Folic Acid Antagonists; Humans; Leishmaniasis; Macrophages; Microbodies; Mitogen-Activated Protein Kinase Kinases; Paromomycin; Pentamidine; Phosphorylcholine; Polyamines; Protease Inhibitors; Sterols; Sulfhydryl Compounds; Topoisomerase Inhibitors

2012
Liposomal formulations in the pharmacological treatment of leishmaniasis: a review.
    Journal of liposome research, 2017, Volume: 27, Issue:3

    Topics: Amphotericin B; Animals; Antiprotozoal Agents; Drug Compounding; Drug Delivery Systems; Drug Liberation; Humans; Leishmaniasis; Liposomes; Nanoparticles; Paromomycin; Particle Size; Pentamidine; Phosphorylcholine; Surface Properties

2017

Other Studies

44 other study(ies) available for miltefosine and pentamidine

ArticleYear
The activity of diguanidino and 'reversed' diamidino 2,5-diarylfurans versus Trypanosoma cruzi and Leishmania donovani.
    Bioorganic & medicinal chemistry letters, 2003, Jun-16, Volume: 13, Issue:12

    Topics: Amidines; Animals; DNA; Furans; Guanidine; Inhibitory Concentration 50; Leishmania donovani; Macrophages; Nucleic Acid Denaturation; Oligodeoxyribonucleotides; Poly dA-dT; Protozoan Proteins; Structure-Activity Relationship; Temperature; Trypanocidal Agents; Trypanosoma cruzi

2003
Chemotherapy of leishmaniasis. Part V: Synthesis and in vitro bioevaluation of novel pyridinone derivatives.
    European journal of medicinal chemistry, 2007, Volume: 42, Issue:5

    Topics: Antiprotozoal Agents; Drug Evaluation, Preclinical; Humans; Leishmaniasis; Pyridones

2007
Redox-active dinitrodiphenylthioethers against Leishmania: synthesis, structure-activity relationships and mechanism of action studies.
    Bioorganic & medicinal chemistry, 2009, Jan-15, Volume: 17, Issue:2

    Topics: Animals; Antiprotozoal Agents; Chlorocebus aethiops; Leishmania donovani; Macrophages, Peritoneal; Membrane Potential, Mitochondrial; Mice; Mice, Inbred Strains; Oxidation-Reduction; Quantitative Structure-Activity Relationship; Reactive Oxygen Species; Sulfides; Vero Cells

2009
Synthesis and molecular docking studies of 1-phenyl-4-glycosyl-dihydropyridines as potent antileishmanial agents.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:6

    Topics: Animals; Antiprotozoal Agents; Cell Line; Leishmania donovani; Life Cycle Stages; Mice; Models, Molecular; Molecular Conformation; Oxidoreductases; Pyridines

2010
Novel arylimidamides for treatment of visceral leishmaniasis.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:6

    Topics: Amidines; Animals; Antiprotozoal Agents; Biological Availability; Cricetinae; Disease Models, Animal; Drug Discovery; Female; Furans; Humans; In Vitro Techniques; Leishmania donovani; Leishmania major; Leishmania mexicana; Leishmaniasis, Visceral; Liver; Mesocricetus; Mice; Mice, Inbred BALB C; Microsomes, Liver; Mutagenicity Tests; Parasitemia; Parasitic Sensitivity Tests; Spleen; Tissue Distribution

2010
QSAR guided synthesis of simplified antiplasmodial analogs of naphthylisoquinoline alkaloids.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:11

    Topics: Alkaloids; Animals; Antimalarials; Isoquinolines; Magnetic Resonance Spectroscopy; Models, Molecular; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Spectrometry, Mass, Electrospray Ionization; Spectroscopy, Fourier Transform Infrared

2010
Increased glycolytic ATP synthesis is associated with tafenoquine resistance in Leishmania major.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:3

    Topics: Adenosine Triphosphate; Aminoquinolines; Antiprotozoal Agents; Drug Resistance; Glycolysis; Leishmania major; Pyruvate Kinase

2011
Synthesis and antikinetoplastid activities of 3-substituted quinolinones derivatives.
    European journal of medicinal chemistry, 2012, Volume: 52

    Topics: Animals; Antiprotozoal Agents; Cell Line, Tumor; Cell Proliferation; Drug Design; Leishmania donovani; Mice; Quinolones; Structure-Activity Relationship; Trypanosoma brucei brucei

2012
Discovery of a new antileishmanial hit in 8-nitroquinoline series.
    European journal of medicinal chemistry, 2012, Volume: 54

    Topics: Animals; Antiprotozoal Agents; Drug Discovery; Hep G2 Cells; Humans; Leishmania donovani; Life Cycle Stages; Mice; Nitroquinolines

2012
Flavonoid dimers as novel, potent antileishmanial agents.
    Journal of medicinal chemistry, 2012, Oct-25, Volume: 55, Issue:20

    Topics: Amines; Animals; Antiprotozoal Agents; Cell Line; Dimerization; Drug Resistance; Flavonoids; Leishmania; Macrophages, Peritoneal; Mice; Polyethylene Glycols; Structure-Activity Relationship

2012
A natural product inspired hybrid approach towards the synthesis of novel pentamidine based scaffolds as potential anti-parasitic agents.
    Bioorganic & medicinal chemistry letters, 2013, Jan-01, Volume: 23, Issue:1

    Topics: Antimalarials; Antiprotozoal Agents; Biological Products; Chalcone; Pentamidine; Plasmodium falciparum; Pyrimidines; Structure-Activity Relationship

2013
Synthesis of novel guttiferone A derivatives: in-vitro evaluation toward Plasmodium falciparum, Trypanosoma brucei and Leishmania donovani.
    European journal of medicinal chemistry, 2013, Volume: 65

    Topics: Antiprotozoal Agents; Benzophenones; Clusiaceae; Dose-Response Relationship, Drug; Leishmania donovani; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Seeds; Structure-Activity Relationship; Trypanosoma brucei brucei

2013
Synthesis and antiprotozoal activity of dicationic m-terphenyl and 1,3-dipyridylbenzene derivatives.
    Journal of medicinal chemistry, 2013, Jul-11, Volume: 56, Issue:13

    Topics: Animals; Antiprotozoal Agents; Benzene; Chagas Disease; Female; Leishmania donovani; Mice; Mice, Inbred Strains; Models, Chemical; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyridines; Structure-Activity Relationship; Terphenyl Compounds; Trypanosoma cruzi

2013
Synthesis and antiprotozoal activity of original porphyrin precursors and derivatives.
    European journal of medicinal chemistry, 2013, Volume: 67

    Topics: Antiprotozoal Agents; Dose-Response Relationship, Drug; Leishmania donovani; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium; Porphyrins; Structure-Activity Relationship; Trypanosoma brucei brucei

2013
Natural product derived antiprotozoal agents: synthesis, biological evaluation, and structure-activity relationships of novel chromene and chromane derivatives.
    Journal of medicinal chemistry, 2013, Sep-26, Volume: 56, Issue:18

    Topics: Antiprotozoal Agents; Biological Products; Chemistry Techniques, Synthetic; Chromans; Inhibitory Concentration 50; Structure-Activity Relationship

2013
Targeting the human parasite Leishmania donovani: discovery of a new promising anti-infectious pharmacophore in 3-nitroimidazo[1,2-a]pyridine series.
    Bioorganic & medicinal chemistry, 2013, Nov-15, Volume: 21, Issue:22

    Topics: Animals; Antiprotozoal Agents; Cell Line; Cell Survival; Drug Evaluation, Preclinical; Hep G2 Cells; Humans; Imidazoles; Leishmania donovani; Mice; Pyridines; Structure-Activity Relationship

2013
Discovery of triazine mimetics as potent antileishmanial agents.
    ACS medicinal chemistry letters, 2013, Nov-14, Volume: 4, Issue:11

    Topics:

2013
Pyridyl benzamides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei.
    Journal of medicinal chemistry, 2014, Aug-14, Volume: 57, Issue:15

    Topics: Animals; Benzamides; Cell Line; HEK293 Cells; Humans; Microsomes, Liver; Myoblasts; Pyridines; Rats; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma brucei rhodesiense

2014
Design, synthesis and in vitro antikinetoplastid evaluation of N-acylated putrescine, spermidine and spermine derivatives.
    Bioorganic & medicinal chemistry letters, 2015, Jan-15, Volume: 25, Issue:2

    Topics: Acylation; Antiprotozoal Agents; Drug Design; Drug Evaluation, Preclinical; Kinetoplastida; Leishmania donovani; Putrescine; Spermidine; Spermine; Trypanosoma brucei brucei

2015
Looking for new antileishmanial derivatives in 8-nitroquinolin-2(1H)-one series.
    European journal of medicinal chemistry, 2015, Mar-06, Volume: 92

    Topics: Antiprotozoal Agents; Dose-Response Relationship, Drug; Leishmania donovani; Molecular Structure; Nitroquinolines; Parasitic Sensitivity Tests; Structure-Activity Relationship

2015
Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series.
    Bioorganic & medicinal chemistry, 2015, May-15, Volume: 23, Issue:10

    Topics: Antiprotozoal Agents; Drug Design; Hep G2 Cells; Humans; Leishmania donovani; Leishmania infantum; Life Cycle Stages; Macrophages; Nitroquinolines; Parasitic Sensitivity Tests; Pentamidine; Phosphorylcholine; Structure-Activity Relationship

2015
Novel dialkylphosphorylhydrazones: Synthesis, leishmanicidal evaluation and theoretical investigation of the proposed mechanism of action.
    European journal of medicinal chemistry, 2015, Aug-28, Volume: 101

    Topics: Animals; Dose-Response Relationship, Drug; Hexokinase; Hydrazones; Leishmania; Macrophages; Mice; Molecular Docking Simulation; Molecular Structure; Parasitic Sensitivity Tests; Structure-Activity Relationship; Trypanocidal Agents

2015
Highly improved antiparasitic activity after introduction of an N-benzylimidazole moiety on protein farnesyltransferase inhibitors.
    European journal of medicinal chemistry, 2016, Feb-15, Volume: 109

    Topics: Alkyl and Aryl Transferases; Animals; Antiparasitic Agents; Cell Line; Enzyme Inhibitors; Humans; Imidazoles; Leishmania donovani; Leishmaniasis, Visceral; Malaria, Falciparum; Mice; Parasitic Sensitivity Tests; Plasmodium falciparum; Trypanosoma; Trypanosoma brucei brucei; Trypanosoma cruzi; Trypanosomiasis

2016
Profiling of Flavonol Derivatives for the Development of Antitrypanosomatidic Drugs.
    Journal of medicinal chemistry, 2016, 08-25, Volume: 59, Issue:16

    Topics: Animals; Biological Products; Cell Line; Dose-Response Relationship, Drug; Flavonols; Humans; Macrophages; Mice; Mice, Inbred BALB C; Models, Molecular; Molecular Structure; Parasitic Sensitivity Tests; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei

2016
Synthesis and in vitro antikinetoplastid activity of polyamine-hydroxybenzotriazole conjugates.
    Bioorganic & medicinal chemistry, 2017, 01-01, Volume: 25, Issue:1

    Topics: Animals; Antiprotozoal Agents; Humans; Leishmania donovani; Leishmaniasis, Visceral; NADH, NADPH Oxidoreductases; Spermidine; Triazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2017
Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds.
    European journal of medicinal chemistry, 2017, Jan-27, Volume: 126

    Topics: Animals; Antiparasitic Agents; Cell Line, Tumor; Chalcones; Cyclodextrins; Drug Carriers; Mice; Solubility; Trypanosomatina

2017
Synthesis, in vitro and in vivo giardicidal activity of nitrothiazole-NSAID chimeras displaying broad antiprotozoal spectrum.
    Bioorganic & medicinal chemistry letters, 2017, 08-01, Volume: 27, Issue:15

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antiprotozoal Agents; Drug Design; Female; Giardia lamblia; Giardiasis; Humans; Leishmania; Mice; Nitro Compounds; Protozoan Infections; Thiazoles; Trichomonas vaginalis; Trypanosoma cruzi

2017
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections.
    European journal of medicinal chemistry, 2018, Feb-25, Volume: 146

    Topics: Antiprotozoal Agents; Chagas Disease; Dose-Response Relationship, Drug; Humans; Macrophages; Molecular Structure; Parasitic Sensitivity Tests; Structure-Activity Relationship; Thiosemicarbazones; Trypanosoma

2018
Design, synthesis and biological evaluation of piperazinyl-β-carbolinederivatives as anti-leishmanial agents.
    European journal of medicinal chemistry, 2018, Apr-25, Volume: 150

    Topics: Antineoplastic Agents; Antiprotozoal Agents; Carbolines; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; HeLa Cells; Humans; Leishmania donovani; Leishmania infantum; Molecular Structure; Parasitic Sensitivity Tests; Piperazines; Structure-Activity Relationship

2018
Quinoxaline derivatives as potential antitrypanosomal and antileishmanial agents.
    Bioorganic & medicinal chemistry, 2018, 08-07, Volume: 26, Issue:14

    Topics: Antiprotozoal Agents; Dose-Response Relationship, Drug; Leishmania donovani; Molecular Structure; Parasitic Sensitivity Tests; Quinoxalines; Structure-Activity Relationship; Trypanosoma brucei brucei; Trypanosoma cruzi

2018
Nongenotoxic 3-Nitroimidazo[1,2-
    ACS medicinal chemistry letters, 2019, Jan-10, Volume: 10, Issue:1

    Topics:

2019
Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections.
    Journal of medicinal chemistry, 2019, 04-25, Volume: 62, Issue:8

    Topics: Animals; Antiprotozoal Agents; Benzothiazoles; Binding Sites; Catalytic Domain; Crystallography, X-Ray; Drug Design; Enzyme Inhibitors; Half-Life; Leishmania major; Mice; Mice, Inbred BALB C; Molecular Docking Simulation; Oxidoreductases; Protozoan Proteins; Structure-Activity Relationship; Trypanosoma brucei brucei; Trypanosomiasis

2019
Indole-Containing Pyrazino[2,1-
    ACS medicinal chemistry letters, 2022, Feb-10, Volume: 13, Issue:2

    Topics:

2022
Pyrimido[5,4-
    ACS medicinal chemistry letters, 2022, Sep-08, Volume: 13, Issue:9

    Topics:

2022
Drug resistance in Indian visceral leishmaniasis.
    Tropical medicine & international health : TM & IH, 2001, Volume: 6, Issue:11

    Topics: Aminoquinolines; Amphotericin B; Antimony; Antiprotozoal Agents; Dose-Response Relationship, Drug; Drug Resistance; Geography; History, 20th Century; History, 21st Century; Humans; India; Leishmaniasis, Visceral; Paromomycin; Pentamidine; Phosphorylcholine; Treatment Outcome

2001
Challenges in the management of visceral leishmaniasis.
    Indian pediatrics, 2005, Volume: 42, Issue:6

    Topics: Amebicides; Amphotericin B; Antimony Sodium Gluconate; Antiparasitic Agents; Antiprotozoal Agents; Enzyme-Linked Immunosorbent Assay; Fluorescent Antibody Technique, Indirect; Humans; Immunoglobulin G; Leishmaniasis, Visceral; Paromomycin; Pentamidine; Phosphorylcholine

2005
Development of a semi-automated colorimetric assay for screening anti-leishmanial agents.
    Journal of microbiological methods, 2006, Volume: 66, Issue:1

    Topics: Amphotericin B; Animals; Antiprotozoal Agents; Colorimetry; Drug Evaluation, Preclinical; Humans; Indicators and Reagents; Inhibitory Concentration 50; Kinetics; Leishmania; Leishmania donovani; Leishmaniasis, Visceral; Pentamidine; Phosphorylcholine; Tetrazolium Salts; Thiazoles

2006
Flow cytometric determination of intracellular non-protein thiols in Leishmania promastigotes using 5-chloromethyl fluorescein diacetate.
    Experimental parasitology, 2009, Volume: 122, Issue:4

    Topics: Animals; Antimony Sodium Gluconate; Antiprotozoal Agents; Culture Media, Serum-Free; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Humans; Leishmania donovani; Pentamidine; Phosphorylcholine; Sensitivity and Specificity; Sulfhydryl Compounds

2009
Tender ulceronecrotic nodules in a patient with leukemia. Cutaneous acanthamebiasis.
    Archives of dermatology, 2011, Volume: 147, Issue:7

    Topics: Acanthamoeba; Amebiasis; Antiprotozoal Agents; Drug Therapy, Combination; Female; Fluconazole; Flucytosine; Humans; Leukemia, Lymphocytic, Chronic, B-Cell; Middle Aged; Necrosis; Pentamidine; Phosphorylcholine; Pyrimidines; Skin Diseases, Parasitic; Skin Ulcer; Sulfadoxine; Triazoles; Voriconazole

2011
Serial use of pentamidine and miltefosine for treating Leishmania infantum-HIV coinfection.
    Parasitology international, 2016, Volume: 65, Issue:5 Pt A

    Topics: Antiprotozoal Agents; Coinfection; HIV Infections; Humans; Immunocompromised Host; Leishmania infantum; Leishmaniasis, Visceral; Pentamidine; Phosphorylcholine

2016
Visceral leishmaniasis in a patient with systemic lupus erythematosus from Colombia, Latin America.
    Le infezioni in medicina, 2019, Mar-01, Volume: 27, Issue:1

    Topics: Adult; Antiprotozoal Agents; Colombia; Humans; Leishmaniasis, Visceral; Lupus Erythematosus, Systemic; Male; Pentamidine; Phosphorylcholine

2019
Semicarbazone derivatives as promising therapeutic alternatives in leishmaniasis.
    Experimental parasitology, 2019, Volume: 201

    Topics: Analysis of Variance; Animals; Antiprotozoal Agents; Caspases; Cell Cycle; Cell Line; Cell Membrane; Cell Membrane Permeability; Female; Flow Cytometry; Inhibitory Concentration 50; Leishmania mexicana; Leishmaniasis, Cutaneous; Macrophages; Membrane Potential, Mitochondrial; Mice; Mice, Inbred BALB C; Pentamidine; Phospholipids; Phosphorylcholine; Semicarbazones

2019
Anti-leishmanial physalins-Phytochemical investigation, in vitro evaluation against clinical and MIL-resistant L. tropica strains and in silico studies.
    PloS one, 2022, Volume: 17, Issue:11

    Topics: Antiprotozoal Agents; Humans; Leishmania major; Leishmaniasis, Cutaneous; Molecular Docking Simulation; Pentamidine; Phosphorylcholine; Phytochemicals

2022
Comparing cytotoxicity and efficacy of miltefosine and standard antimicrobial agents against Acanthamoeba trophozoites and cyst forms: An in vitro study.
    Acta tropica, 2023, Volume: 247

    Topics: Acanthamoeba; Acanthamoeba Keratitis; Animals; Anti-Infective Agents; Chlorhexidine; Chlorocebus aethiops; Cysts; Humans; Pentamidine; Trophozoites; Vero Cells

2023