midazolam and isoxazoles

midazolam has been researched along with isoxazoles in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19903 (25.00)18.7374
1990's1 (8.33)18.2507
2000's4 (33.33)29.6817
2010's4 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Graeff, FG; Milani, H1
Brunner, EA; Cheng, SC1
Jensen, MS; Lambert, JD1
Kristiansen, U; Lambert, JD1
Feldman, J; Ibrahim, A; Karim, A; Kharasch, E1
France, CP; McMahon, LR1
D'Arienzo, C; Ewing, WR; Gu, Z; Humphreys, WG; Li, W; Li, YX; Murugesan, N; Shyu, WC; Yao, M; Zhang, D; Zhang, H; Zhu, Y1
Darbra, S; Pallarès, M1
Ding, X; Fang, C; Jia, K; Zhang, P; Zhang, QY; Zhou, X1
France, CP; Gerak, LR1
Gerak, LR; Ibarra, MH; Pressly, JD; Smith, KR; Zanettini, C1
Bint, L; Czarniak, P; Landwehr, C; Parsons, R; Richardson, J; Sunderland, B1

Trials

1 trial(s) available for midazolam and isoxazoles

ArticleYear
The influence of parecoxib, a parenteral cyclooxygenase-2 specific inhibitor, on the pharmacokinetics and clinical effects of midazolam.
    Anesthesia and analgesia, 2002, Volume: 95, Issue:3

    Topics: Adult; Area Under Curve; Biotransformation; Cyclooxygenase Inhibitors; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Double-Blind Method; Drug Interactions; Electroencephalography; Female; Half-Life; Humans; Hypnotics and Sedatives; Injections, Intravenous; Isoxazoles; Male; Midazolam; Mixed Function Oxygenases; Nausea; Reflex; Vomiting

2002

Other Studies

11 other study(ies) available for midazolam and isoxazoles

ArticleYear
GABA-benzodiazepine modulation of aversion in the medial hypothalamus of the rat.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:1

    Topics: Animals; Avoidance Learning; Bicuculline; Dose-Response Relationship, Drug; Electric Stimulation; Electrodes, Implanted; Flumazenil; Hypothalamus, Middle; Isoxazoles; Male; Microinjections; Midazolam; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Inducing anesthesia with a GABA analog, THIP.
    Anesthesiology, 1985, Volume: 63, Issue:2

    Topics: Analgesics; Anesthesia, Intravenous; Anesthetics; Animals; Benzodiazepines; gamma-Aminobutyric Acid; Isoxazoles; Ketamine; Male; Mice; Midazolam; Oxazoles; Rats; Rats, Inbred Strains; Sodium Oxybate; Time Factors

1985
Modulation of the responses to the GABA-mimetics, THIP and piperidine-4-sulphonic acid, by agents which interact with benzodiazepine receptors. An electrophysiological study on cultured mouse neurones.
    Neuropharmacology, 1984, Volume: 23, Issue:12A

    Topics: Animals; Benzodiazepines; Carbolines; Cells, Cultured; Convulsants; Electrophysiology; Female; gamma-Aminobutyric Acid; Iontophoresis; Isoxazoles; Mice; Midazolam; Neurons; Oxazoles; Piperidines; Receptors, GABA-A

1984
Benzodiazepine and barbiturate ligands modulate responses of cultured hippocampal neurones to the GABAA receptor partial agonist, 4-PIOL.
    Neuropharmacology, 1996, Volume: 35, Issue:9-10

    Topics: Animals; Barbiturates; Benzodiazepines; Carbolines; Cells, Cultured; Convulsants; Electrophysiology; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; Hippocampus; Hypnotics and Sedatives; Isonicotinic Acids; Isoxazoles; Membrane Potentials; Midazolam; Neurons; Patch-Clamp Techniques; Pentobarbital; Piperidines; Rats

1996
Combined discriminative stimulus effects of midazolam with other positive GABAA modulators and GABAA receptor agonists in rhesus monkeys.
    Psychopharmacology, 2005, Volume: 178, Issue:4

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Discrimination Learning; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Ethanol; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Injections, Subcutaneous; Isoxazoles; Macaca mulatta; Male; Midazolam; Pentobarbital; Pregnanolone; Receptors, GABA-A; Time Factors; Triazolam; Women

2005
Reduction of site-specific CYP3A-mediated metabolism for dual angiotensin and endothelin receptor antagonists in various in vitro systems and in cynomolgus monkeys.
    Drug metabolism and disposition: the biological fate of chemicals, 2007, Volume: 35, Issue:5

    Topics: Amides; Angiotensin Receptor Antagonists; Animals; Area Under Curve; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Endothelin A Receptor Antagonists; GABA Modulators; Humans; Hydroxylation; Isoxazoles; Macaca fascicularis; Male; Microsomes, Liver; Midazolam; Molecular Structure; Sulfonamides; Tandem Mass Spectrometry

2007
Neonatal allopregnanolone increases novelty-directed locomotion and disrupts behavioural responses to GABA(A) receptor modulators in adulthood.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 2009, Volume: 27, Issue:6

    Topics: Animals; Animals, Newborn; Behavior, Animal; Brain; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Exploratory Behavior; Flumazenil; GABA Modulators; Isoxazoles; Lorazepam; Male; Maze Learning; Midazolam; Motor Activity; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A

2009
Dietary regulation of mouse intestinal P450 expression and drug metabolism.
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:2

    Topics: Animal Feed; Animals; Bile Acids and Salts; Biotransformation; Cytochrome P-450 Enzyme System; Diet; Female; Hydroxylation; Intestines; Isoenzymes; Isoxazoles; Liver; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Microsomes, Liver; Midazolam; NADPH-Ferrihemoprotein Reductase; Receptors, Cytoplasmic and Nuclear; Substrate Specificity

2013
Discriminative stimulus effects of pregnanolone in rhesus monkeys.
    Psychopharmacology, 2014, Volume: 231, Issue:1

    Topics: Animals; Conditioning, Operant; Data Interpretation, Statistical; Discrimination, Psychological; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Flumazenil; Flunitrazepam; GABA Modulators; Gonadal Steroid Hormones; Hypnotics and Sedatives; Isoxazoles; Macaca mulatta; Male; Midazolam; Pregnanolone; Receptors, GABA-A; Reinforcement Schedule

2014
Comparing the discriminative stimulus effects of modulators of GABAA receptors containing α4-δ subunits with those of gaboxadol in rats.
    Psychopharmacology, 2016, Volume: 233, Issue:10

    Topics: Animals; Dose-Response Relationship, Drug; Ethanol; Flumazenil; GABA Agonists; GABA Modulators; Isoxazoles; Male; Midazolam; Pregnanolone; Protein Subunits; Rats; Receptors, GABA-A

2016
Cross-sectional survey of off-label and unlicensed prescribing for inpatients at a paediatric teaching hospital in Western Australia.
    PloS one, 2019, Volume: 14, Issue:1

    Topics: Australia; Child; Child, Preschool; Clonidine; Drug Administration Routes; Drug Prescriptions; Female; Humans; Inpatients; Isoxazoles; Legislation, Drug; Male; Midazolam; Off-Label Use; Oxycodone; Pediatrics

2019