Page last updated: 2024-08-24

mibefradil and nimodipine

mibefradil has been researched along with nimodipine in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (5.88)18.2507
2000's9 (52.94)29.6817
2010's7 (41.18)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Ekins, S; Williams, AJ; Xu, JJ1
Fijorek, K; Glinka, A; Mendyk, A; Polak, S; Wiśniowska, B1
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ1
Brust, PF; Hans, M; Harpold, MM; Prodanovich, P; Stauderman, KA; Urrutia, A; Washburn, MS; Williams, ME1
Andrade, R; Hu, HJ; Pan, ZH; Perring, P1
Connolly, TM; Figueroa, DJ; Lawlor, AM; Liang, HA; Liu, Y; Salata, JJ; Xia, M1
Kahlert, S; Martínez-Sánchez, M; Reiser, G; Reymann, KG; Schröder, UH; Striggow, F1
Berggren, PO; Billestrup, N; Kapelioukh, IL; Karlsen, AE; Mandrup-Poulsen, T; Størling, J; Zaitsev, SV1
Badawi, JK; Bross, S; Kamp, S; Kwon, ST; Langbein, S; Li, H1
Hata, R; Kato, Y; Kubota, E; Miyazaki, K; Ozawa, S; St-Pierre, Y; Tsukuda, M1
Fei, H; Wang, Q; Zhao, B; Zhao, S1
Du, X; Huang, D; Huang, S; Li, L; Yan, Y; Zhang, H; Zhou, N1
Braszko, JJ1

Other Studies

17 other study(ies) available for mibefradil and nimodipine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Predictive model for L-type channel inhibition: multichannel block in QT prolongation risk assessment.
    Journal of applied toxicology : JAT, 2012, Volume: 32, Issue:10

    Topics: Artificial Intelligence; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Computational Biology; Computer Simulation; Drugs, Investigational; Ether-A-Go-Go Potassium Channels; Expert Systems; Heart Rate; Humans; Models, Biological; Myocytes, Cardiac; NAV1.5 Voltage-Gated Sodium Channel; Potassium Channel Blockers; Quantitative Structure-Activity Relationship; Risk Assessment; Shaker Superfamily of Potassium Channels; Torsades de Pointes; Voltage-Gated Sodium Channel Blockers

2012
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:1

    Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity

2013
Structure and functional characterization of a novel human low-voltage activated calcium channel.
    Journal of neurochemistry, 1999, Volume: 72, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amiloride; Animals; Barium; Benzimidazoles; Blotting, Northern; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, T-Type; Cells, Cultured; Cloning, Molecular; Diuretics; DNA, Complementary; Electric Stimulation; Electrophysiology; Humans; Ion Channel Gating; Kidney; Kinetics; Membrane Potentials; Mibefradil; Molecular Sequence Data; Nickel; Nimodipine; Oocytes; Recombinant Proteins; RNA, Messenger; Sequence Homology, Amino Acid; Tetrahydronaphthalenes; Transcription, Genetic; Verapamil; Xenopus

1999
T-type Ca(2+) channels mediate neurotransmitter release in retinal bipolar cells.
    Neuron, 2001, Oct-11, Volume: 32, Issue:1

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels, T-Type; Chelating Agents; Cobalt; Egtazic Acid; Electric Capacitance; Exocytosis; Membrane Potentials; Mibefradil; Neurotransmitter Agents; Nimodipine; Patch-Clamp Techniques; Presynaptic Terminals; Rats; Rats, Long-Evans; Retina; RNA, Messenger; Synaptic Transmission

2001
Functional expression of L- and T-type Ca2+ channels in murine HL-1 cells.
    Journal of molecular and cellular cardiology, 2004, Volume: 36, Issue:1

    Topics: Animals; Calcium; Calcium Channels, L-Type; Calcium Channels, T-Type; Cell Line; Electric Conductivity; Heart Atria; Ion Transport; Mibefradil; Mice; Myocytes, Cardiac; Nimodipine; Patch-Clamp Techniques; Pimozide; Potassium; Verapamil

2004
Na(+) and Ca(2+) homeostasis pathways, cell death and protection after oxygen-glucose-deprivation in organotypic hippocampal slice cultures.
    Neuroscience, 2004, Volume: 128, Issue:4

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Boron Compounds; Calcium; Calcium Channel Blockers; Cell Death; Clonazepam; Dantrolene; Dizocilpine Maleate; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Fura-2; Glucose; Hippocampus; Hypoxia; In Situ Nick-End Labeling; Indoles; Intracellular Space; Ion Exchange; Lidocaine; Mibefradil; Nimodipine; Organ Culture Techniques; Quinoxalines; Rats; Rats, Wistar; Sodium; Sodium Channel Blockers; Thiazepines; Thiourea; Time Factors

2004
Calcium has a permissive role in interleukin-1beta-induced c-jun N-terminal kinase activation in insulin-secreting cells.
    Endocrinology, 2005, Volume: 146, Issue:7

    Topics: Animals; Calcium; Calcium Channel Blockers; Cell Line; Drug Synergism; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Humans; Insulin; Insulin Secretion; Interleukin-1; Intracellular Membranes; Islets of Langerhans; JNK Mitogen-Activated Protein Kinases; Mibefradil; Mice; NF-kappa B; Nimodipine; p38 Mitogen-Activated Protein Kinases; Rats; Rats, Inbred WF; Signal Transduction

2005
Inhibitory effects of L- and T-type calcium antagonists on contractions of human detrusor muscle.
    European journal of clinical pharmacology, 2006, Volume: 62, Issue:5

    Topics: Adult; Aged; Analysis of Variance; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, T-Type; Carbachol; Diltiazem; Female; Humans; In Vitro Techniques; Male; Mibefradil; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Nimodipine; Potassium; Urinary Bladder; Verapamil

2006
Acidic extracellular pH increases calcium influx-triggered phospholipase D activity along with acidic sphingomyelinase activation to induce matrix metalloproteinase-9 expression in mouse metastatic melanoma.
    The FEBS journal, 2007, Volume: 274, Issue:12

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Line, Tumor; Chelating Agents; Desipramine; Egtazic Acid; Enzyme Activation; Extracellular Fluid; Hydrogen-Ion Concentration; Indolizines; MAP Kinase Signaling System; Matrix Metalloproteinase 9; Melanoma; Mibefradil; Mice; NF-kappa B; Nimodipine; Perhexiline; Phenethylamines; Phospholipase D; Phosphorylation; Promoter Regions, Genetic; Sphingomyelin Phosphodiesterase

2007
Requirements of calcium fluxes and ERK kinase activation for glucose- and interleukin-1beta-induced beta-cell apoptosis.
    Molecular and cellular biochemistry, 2008, Volume: 315, Issue:1-2

    Topics: Animals; Apoptosis; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Egtazic Acid; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Glucose; Humans; Insulin; Insulin Secretion; Insulin-Secreting Cells; Interleukin-1beta; Ion Channel Gating; Ionomycin; Mibefradil; Nimodipine; Rats; Sulfonamides; Thapsigargin

2008
Suppression of KV7/KCNQ potassium channel enhances neuronal differentiation of PC12 cells.
    Neuroscience, 2016, 10-01, Volume: 333

    Topics: Animals; Anthracenes; Calcium; Calcium Channels, T-Type; Central Nervous System Agents; Cerebral Cortex; KCNQ2 Potassium Channel; KCNQ3 Potassium Channel; Mibefradil; Nerve Growth Factor; Neurogenesis; Neurons; Nimodipine; PC12 Cells; Potassium; Rats; Rats, Sprague-Dawley; RNA, Messenger

2016
Indispensable role of the voltage-gated calcium channels in the procognitive effects of angiotensin IV.
    Brain research bulletin, 2017, Volume: 130

    Topics: Angiotensin II; Animals; Avoidance Learning; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, T-Type; Cognition; Exploratory Behavior; Male; Mental Recall; Mibefradil; Nimodipine; Nootropic Agents; Rats, Wistar; Recognition, Psychology

2017