mibefradil has been researched along with nicardipine in 13 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (15.38) | 18.2507 |
2000's | 6 (46.15) | 29.6817 |
2010's | 4 (30.77) | 24.3611 |
2020's | 1 (7.69) | 2.80 |
Authors | Studies |
---|---|
Coassolo, P; Lavé, T; Schneider, G | 1 |
Topliss, JG; Yoshida, F | 1 |
Fischer, H; Huwyler, J; Poli, S; Schwab, D; Tabatabaei, A | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ | 1 |
Fijorek, K; Glinka, A; Mendyk, A; Polak, S; Wiśniowska, B | 1 |
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ | 1 |
Capponi, AM; Ertel, EA; Rossier, MF; Vallotton, MB | 1 |
Kenyon, JL; Koh, SD; Mason, HS; Monaghan, K; Ro, S; Sanders, KM | 1 |
Angus, JA; Evans, RJ; Roberts, JA; Xi, Q; Ziogas, J | 1 |
Bayguinov, O; Kenyon, JL; Sanders, KM; Ward, SM | 1 |
Bieger, D; Ford, CA; Tabrizchi, R | 1 |
Goto, T; Tohkin, M; Yamazoe, Y | 1 |
13 other study(ies) available for mibefradil and nicardipine
Article | Year |
---|---|
Combining in vitro and in vivo pharmacokinetic data for prediction of hepatic drug clearance in humans by artificial neural networks and multivariate statistical techniques.
Topics: Animals; Biological Availability; Dogs; Humans; Least-Squares Analysis; Liver; Multivariate Analysis; Neural Networks, Computer; Pharmacokinetics; Rats | 1999 |
QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Comparison of in vitro P-glycoprotein screening assays: recommendations for their use in drug discovery.
Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cells, Cultured; Drug Evaluation, Preclinical; Fluoresceins; Fluorescent Dyes; Humans; Indicators and Reagents; Mice; Models, Molecular; Rhodamines; Species Specificity; Swine | 2003 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics | 2010 |
Predictive model for L-type channel inhibition: multichannel block in QT prolongation risk assessment.
Topics: Artificial Intelligence; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Computational Biology; Computer Simulation; Drugs, Investigational; Ether-A-Go-Go Potassium Channels; Expert Systems; Heart Rate; Humans; Models, Biological; Myocytes, Cardiac; NAV1.5 Voltage-Gated Sodium Channel; Potassium Channel Blockers; Quantitative Structure-Activity Relationship; Risk Assessment; Shaker Superfamily of Potassium Channels; Torsades de Pointes; Voltage-Gated Sodium Channel Blockers | 2012 |
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity | 2013 |
Inhibitory action of mibefradil on calcium signaling and aldosterone synthesis in bovine adrenal glomerulosa cells.
Topics: Aldosterone; Animals; Benzimidazoles; Calcium; Calcium Channel Blockers; Cattle; Cells, Cultured; Cytosol; Mibefradil; Nicardipine; Patch-Clamp Techniques; Pimozide; Potassium Chloride; Signal Transduction; Tetrahydronaphthalenes; Zona Glomerulosa | 1998 |
Novel voltage-dependent non-selective cation conductance in murine colonic myocytes.
Topics: Action Potentials; Animals; Barium; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, T-Type; Cesium; Colon; Gadolinium; Gene Expression; Ion Channel Gating; Mibefradil; Mice; Mice, Inbred BALB C; Muscle, Smooth; Neural Inhibition; Nicardipine; Nickel; Patch-Clamp Techniques; Sodium; Temperature | 2001 |
Involvement of T-type calcium channels in excitatory junction potentials in rat resistance mesenteric arteries.
Topics: Adenosine Triphosphate; Animals; Calcium Channel Blockers; Calcium Channels, T-Type; Electric Stimulation; In Vitro Techniques; Male; Mesenteric Arteries; Mibefradil; Muscle Contraction; Neuromuscular Junction; Nicardipine; Nickel; omega-Conotoxin GVIA; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Vas Deferens; Vascular Resistance; Vasoconstriction | 2002 |
Voltage-gated Ca2+ currents are necessary for slow-wave propagation in the canine gastric antrum.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Calcium-Transporting ATPases; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Indoles; Mibefradil; Muscle, Smooth; Myoelectric Complex, Migrating; Nicardipine; Nickel; Peristalsis; Pinacidil; Potassium; Potassium Channels; Pyloric Antrum; Stromal Cells; Time Factors | 2007 |
Potassium-induced intermittent vasomotion in rat isolated pulmonary artery.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Animals; Barium; Indoles; Male; Mibefradil; Nicardipine; Niflumic Acid; Potassium; Potassium Channels; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Verapamil | 2011 |
Versatile applicability of a grid-based CYP3A4 Template to understand the interacting mechanisms with the small-size ligands; part 3 of CYP3A4 Template study.
Topics: Coumarins; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Humans; Ketoconazole; Ligands; Mibefradil; Molecular Structure; Nicardipine | 2020 |