Page last updated: 2024-08-24

mibefradil and nicardipine

mibefradil has been researched along with nicardipine in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (15.38)18.2507
2000's6 (46.15)29.6817
2010's4 (30.77)24.3611
2020's1 (7.69)2.80

Authors

AuthorsStudies
Coassolo, P; Lavé, T; Schneider, G1
Topliss, JG; Yoshida, F1
Fischer, H; Huwyler, J; Poli, S; Schwab, D; Tabatabaei, A1
Lombardo, F; Obach, RS; Waters, NJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Fijorek, K; Glinka, A; Mendyk, A; Polak, S; Wiśniowska, B1
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ1
Capponi, AM; Ertel, EA; Rossier, MF; Vallotton, MB1
Kenyon, JL; Koh, SD; Mason, HS; Monaghan, K; Ro, S; Sanders, KM1
Angus, JA; Evans, RJ; Roberts, JA; Xi, Q; Ziogas, J1
Bayguinov, O; Kenyon, JL; Sanders, KM; Ward, SM1
Bieger, D; Ford, CA; Tabrizchi, R1
Goto, T; Tohkin, M; Yamazoe, Y1

Other Studies

13 other study(ies) available for mibefradil and nicardipine

ArticleYear
Combining in vitro and in vivo pharmacokinetic data for prediction of hepatic drug clearance in humans by artificial neural networks and multivariate statistical techniques.
    Journal of medicinal chemistry, 1999, Dec-16, Volume: 42, Issue:25

    Topics: Animals; Biological Availability; Dogs; Humans; Least-Squares Analysis; Liver; Multivariate Analysis; Neural Networks, Computer; Pharmacokinetics; Rats

1999
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Comparison of in vitro P-glycoprotein screening assays: recommendations for their use in drug discovery.
    Journal of medicinal chemistry, 2003, Apr-24, Volume: 46, Issue:9

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cells, Cultured; Drug Evaluation, Preclinical; Fluoresceins; Fluorescent Dyes; Humans; Indicators and Reagents; Mice; Models, Molecular; Rhodamines; Species Specificity; Swine

2003
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Predictive model for L-type channel inhibition: multichannel block in QT prolongation risk assessment.
    Journal of applied toxicology : JAT, 2012, Volume: 32, Issue:10

    Topics: Artificial Intelligence; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Computational Biology; Computer Simulation; Drugs, Investigational; Ether-A-Go-Go Potassium Channels; Expert Systems; Heart Rate; Humans; Models, Biological; Myocytes, Cardiac; NAV1.5 Voltage-Gated Sodium Channel; Potassium Channel Blockers; Quantitative Structure-Activity Relationship; Risk Assessment; Shaker Superfamily of Potassium Channels; Torsades de Pointes; Voltage-Gated Sodium Channel Blockers

2012
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:1

    Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity

2013
Inhibitory action of mibefradil on calcium signaling and aldosterone synthesis in bovine adrenal glomerulosa cells.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:3

    Topics: Aldosterone; Animals; Benzimidazoles; Calcium; Calcium Channel Blockers; Cattle; Cells, Cultured; Cytosol; Mibefradil; Nicardipine; Patch-Clamp Techniques; Pimozide; Potassium Chloride; Signal Transduction; Tetrahydronaphthalenes; Zona Glomerulosa

1998
Novel voltage-dependent non-selective cation conductance in murine colonic myocytes.
    The Journal of physiology, 2001, Jun-01, Volume: 533, Issue:Pt 2

    Topics: Action Potentials; Animals; Barium; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, T-Type; Cesium; Colon; Gadolinium; Gene Expression; Ion Channel Gating; Mibefradil; Mice; Mice, Inbred BALB C; Muscle, Smooth; Neural Inhibition; Nicardipine; Nickel; Patch-Clamp Techniques; Sodium; Temperature

2001
Involvement of T-type calcium channels in excitatory junction potentials in rat resistance mesenteric arteries.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: Adenosine Triphosphate; Animals; Calcium Channel Blockers; Calcium Channels, T-Type; Electric Stimulation; In Vitro Techniques; Male; Mesenteric Arteries; Mibefradil; Muscle Contraction; Neuromuscular Junction; Nicardipine; Nickel; omega-Conotoxin GVIA; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Vas Deferens; Vascular Resistance; Vasoconstriction

2002
Voltage-gated Ca2+ currents are necessary for slow-wave propagation in the canine gastric antrum.
    American journal of physiology. Cell physiology, 2007, Volume: 293, Issue:5

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Calcium-Transporting ATPases; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Indoles; Mibefradil; Muscle, Smooth; Myoelectric Complex, Migrating; Nicardipine; Nickel; Peristalsis; Pinacidil; Potassium; Potassium Channels; Pyloric Antrum; Stromal Cells; Time Factors

2007
Potassium-induced intermittent vasomotion in rat isolated pulmonary artery.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2011, Volume: 47, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Animals; Barium; Indoles; Male; Mibefradil; Nicardipine; Niflumic Acid; Potassium; Potassium Channels; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Verapamil

2011
Versatile applicability of a grid-based CYP3A4 Template to understand the interacting mechanisms with the small-size ligands; part 3 of CYP3A4 Template study.
    Drug metabolism and pharmacokinetics, 2020, Volume: 35, Issue:3

    Topics: Coumarins; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Humans; Ketoconazole; Ligands; Mibefradil; Molecular Structure; Nicardipine

2020