Page last updated: 2024-08-24

mibefradil and amiloride

mibefradil has been researched along with amiloride in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (15.38)18.2507
2000's8 (61.54)29.6817
2010's2 (15.38)24.3611
2020's1 (7.69)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S1
Campillo, NE; Guerra, A; Páez, JA1
Bellera, CL; Bruno-Blanch, LE; Castro, EA; Duchowicz, PR; Goodarzi, M; Ortiz, EV; Pesce, G; Talevi, A1
Brust, PF; Hans, M; Harpold, MM; Prodanovich, P; Stauderman, KA; Urrutia, A; Washburn, MS; Williams, ME1
Derambure, P; Niespodziany, I; Poulain, P1
Bourinet, E; Chemin, J; Lory, P; Mennessier, G; Monteil, A; Nargeot, J1
Benquet, P; Frere, S; Pichon, Y; Tiaho, F1
Baldi, E; Bonaccorsi, L; Forti, G1
Lambert, S; Oberwinkler, J1
Coste, B; Crest, M; Delmas, P1
Chen, H; Chen, SR; Pan, HL; Yuan, WX1
Abbasloo, E; Abdollahi, F; Akhlaghinasab, F; Esmaeili-Mahani, S; Kaeidi, A; Kobeissy, FH; Oryan, S; Saberi, A; Sheibani, V; Thomas, TC1

Other Studies

13 other study(ies) available for mibefradil and amiloride

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship

2009
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Prediction of drug intestinal absorption by new linear and non-linear QSPR.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Humans; Intestinal Absorption; Linear Models; Molecular Conformation; Nonlinear Dynamics; Permeability; Pharmaceutical Preparations; Probability; Quantitative Structure-Activity Relationship; Thermodynamics

2011
Structure and functional characterization of a novel human low-voltage activated calcium channel.
    Journal of neurochemistry, 1999, Volume: 72, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Amiloride; Animals; Barium; Benzimidazoles; Blotting, Northern; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, T-Type; Cells, Cultured; Cloning, Molecular; Diuretics; DNA, Complementary; Electric Stimulation; Electrophysiology; Humans; Ion Channel Gating; Kidney; Kinetics; Membrane Potentials; Mibefradil; Molecular Sequence Data; Nickel; Nimodipine; Oocytes; Recombinant Proteins; RNA, Messenger; Sequence Homology, Amino Acid; Tetrahydronaphthalenes; Transcription, Genetic; Verapamil; Xenopus

1999
Properties of T-type calcium current in enkephalinergic neurones in guinea-pig hypothalamic slices.
    Pflugers Archiv : European journal of physiology, 1999, Volume: 437, Issue:6

    Topics: Amiloride; Animals; Barium; Benzimidazoles; Calcium; Calcium Channel Blockers; Calcium Channels; Electric Conductivity; Enkephalins; Female; Guinea Pigs; Hypothalamus; Mibefradil; Neurons; Octanols; Patch-Clamp Techniques; Tetrahydronaphthalenes; Tetrodotoxin

1999
Molecular and functional properties of the human alpha(1G) subunit that forms T-type calcium channels.
    The Journal of biological chemistry, 2000, Mar-03, Volume: 275, Issue:9

    Topics: Amiloride; Amino Acid Sequence; Calcium; Calcium Channels, T-Type; Cell Line; Cloning, Molecular; Electrophysiology; Gene Expression Regulation; Humans; Mibefradil; Molecular Sequence Data; Nickel; RNA, Messenger; Sequence Alignment

2000
Properties and development of calcium currents in embryonic cockroach neurons.
    Neuroscience letters, 2000, Nov-10, Volume: 294, Issue:1

    Topics: Amiloride; Animals; Barium; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, N-Type; Calcium Channels, P-Type; Calcium Channels, T-Type; Dose-Response Relationship, Drug; In Vitro Techniques; Isradipine; Membrane Potentials; Mibefradil; Neurons; omega-Agatoxin IVA; omega-Conotoxin GVIA; Patch-Clamp Techniques; Periplaneta; Verapamil

2000
Low-voltage-activated calcium channels are not involved in capacitation and biological response to progesterone in human sperm.
    International journal of andrology, 2001, Volume: 24, Issue:6

    Topics: Amiloride; Calcium Channel Blockers; Calcium Channels; Fluoresceins; Humans; Ion Channel Gating; Male; Mibefradil; Phosphorylation; Pimozide; Progesterone; Sperm Capacitation; Tyrosine

2001
Characterization of a proton-activated, outwardly rectifying anion channel.
    The Journal of physiology, 2005, Aug-15, Volume: 567, Issue:Pt 1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Anions; Astrocytes; Calcium; Calcium Channel Blockers; Cell Line; Chlorides; Diuretics; Hippocampus; Humans; Hydrogen-Ion Concentration; Hypotonic Solutions; Ion Channels; Kidney; Magnesium; Membrane Potentials; Mibefradil; Mice; Mice, Inbred C57BL; Protons

2005
Pharmacological dissection and distribution of NaN/Nav1.9, T-type Ca2+ currents, and mechanically activated cation currents in different populations of DRG neurons.
    The Journal of general physiology, 2007, Volume: 129, Issue:1

    Topics: Action Potentials; Amiloride; Animals; Cadmium; Calcium Channel Blockers; Calcium Channels, T-Type; Cations; Cells, Cultured; Electrophysiology; Ganglia, Spinal; Lanthanum; Male; Mechanoreceptors; Mibefradil; NAV1.9 Voltage-Gated Sodium Channel; Neuropeptides; Nickel; Nociceptors; Rats; Rats, Wistar; Sodium Channel Blockers; Sodium Channels

2007
Stimulation of alpha(1)-adrenoceptors reduces glutamatergic synaptic input from primary afferents through GABA(A) receptors and T-type Ca(2+) channels.
    Neuroscience, 2009, Feb-18, Volume: 158, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Afferent Pathways; Amiloride; Animals; Biophysical Phenomena; Calcium Channel Blockers; Calcium Channels, T-Type; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; Glutamic Acid; Male; Mibefradil; Muscimol; Patch-Clamp Techniques; Phenylephrine; Phosphinic Acids; Picrotoxin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, GABA-A; Sensory Receptor Cells; Spinal Cord; Synapses

2009
Involvement of T-type calcium channels in the mechanism of low dose morphine-induced hyperalgesia in adult male rats.
    Neuropeptides, 2021, Volume: 90

    Topics: Amiloride; Analgesics, Opioid; Animals; Calcium Channels, T-Type; Dose-Response Relationship, Drug; Hyperalgesia; Injections, Intraperitoneal; Male; Mibefradil; Morphine; Pain Measurement; Pain Threshold; Posterior Horn Cells; Rats; Rats, Wistar; Receptors, Opioid, mu

2021