Page last updated: 2024-08-21

metylperon and clozapine

metylperon has been researched along with clozapine in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19903 (21.43)18.7374
1990's3 (21.43)18.2507
2000's5 (35.71)29.6817
2010's3 (21.43)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Christensson, E; Egbe, P; Engel, J; Gustafsson, B1
Matsubara, S; Meltzer, HY1
Gudelsky, GA; Koenig, JI; Meltzer, HY; Nash, JF1
Gudelsky, GA; Meltzer, HY; Nash, JF1
Hippius, H; Klages, U; Müller-Spahn, F1
Evans, DL; Figur, LM; Lahti, RA; Stratman, NC1
Dai, J; Ichikawa, J; Li, Z; Meltzer, HY1
Baker, LE; Meltzer, HY; Prus, AJ1
Dahl, SG; Hjerde, E; Sylte, I1
Bobo, WV; Jayathilake, K; Lee, MA; Meltzer, HY2
Alam, R; Gadhia, S; Röhricht, F; Willis, M1

Reviews

1 review(s) available for metylperon and clozapine

ArticleYear
[Atypical neuroleptics, pharmacology and clinical importance].
    Fortschritte der Neurologie-Psychiatrie, 1993, Volume: 61, Issue:11

    Topics: Animals; Antipsychotic Agents; Brain; Butyrophenones; Clinical Trials as Topic; Clozapine; Humans; Psychotic Disorders; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin

1993

Trials

1 trial(s) available for metylperon and clozapine

ArticleYear
Melperone, an aytpical antipsychotic drug with clozapine-like effect on plasma prolactin: contrast with typical neuroleptics.
    Human psychopharmacology, 2009, Volume: 24, Issue:5

    Topics: Adult; Antipsychotic Agents; Butyrophenones; Clozapine; Female; Humans; Male; Mental Disorders; Prolactin; Sex Factors

2009

Other Studies

12 other study(ies) available for metylperon and clozapine

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Amperozide and conditioned behaviour in rats: potentiation by classical neuroleptics and alpha-methylparatyrosine.
    Pharmacology & toxicology, 1990, Volume: 66 Suppl 1

    Topics: alpha-Methyltyrosine; Animals; Antipsychotic Agents; Avoidance Learning; Behavior, Animal; Butyrophenones; Chlorpromazine; Clozapine; Conditioning, Operant; Drug Synergism; Female; Food; Haloperidol; Male; Methyltyrosines; Piperazines; Psychotropic Drugs; Rats; Rats, Inbred Strains; Reinforcement Schedule

1990
Effect of typical and atypical antipsychotic drugs on 5-HT2 receptor density in rat cerebral cortex.
    Life sciences, 1989, Volume: 45, Issue:15

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Butyrophenones; Cerebral Cortex; Chlorpromazine; Clozapine; Dibenzazepines; Dibenzothiazepines; Down-Regulation; Flupenthixol; Kinetics; Loxapine; Male; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiro Compounds; Time Factors

1989
Melperone and clozapine: neuroendocrine effects of atypical neuroleptic drugs.
    Acta psychiatrica Scandinavica. Supplementum, 1989, Volume: 352

    Topics: Animals; Antipsychotic Agents; Arcuate Nucleus of Hypothalamus; Butyrophenones; Clozapine; Corticosterone; Dibenzazepines; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Male; Median Eminence; Neurons; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine

1989
Antagonism of serotonin receptor mediated neuroendocrine and temperature responses by atypical neuroleptics in the rat.
    European journal of pharmacology, 1988, Jul-14, Volume: 151, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Body Temperature; Butyrophenones; Chlorpromazine; Clozapine; Corticosterone; Haloperidol; Male; Neurosecretory Systems; Pyrazines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1988
Dopamine D4 versus D2 receptor selectivity of dopamine receptor antagonists: possible therapeutic implications.
    European journal of pharmacology, 1993, Jun-04, Volume: 236, Issue:3

    Topics: Animals; Apomorphine; Butyrophenones; Cell Line; Chlorpromazine; Clozapine; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Raclopride; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Trifluoperazine

1993
Atypical antipsychotic drugs, quetiapine, iloperidone, and melperone, preferentially increase dopamine and acetylcholine release in rat medial prefrontal cortex: role of 5-HT1A receptor agonism.
    Brain research, 2002, Nov-29, Volume: 956, Issue:2

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Butyrophenones; Clozapine; Dibenzothiazepines; Dopamine; Haloperidol; Isoxazoles; Male; Microdialysis; Nucleus Accumbens; Piperidines; Prefrontal Cortex; Quetiapine Fumarate; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1

2002
Discriminative stimulus properties of 1.25 and 5.0 mg/kg doses of clozapine in rats: examination of the role of dopamine, serotonin, and muscarinic receptor mechanisms.
    Pharmacology, biochemistry, and behavior, 2004, Volume: 77, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Butyrophenones; Clozapine; Discrimination, Psychological; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Fluorobenzenes; Generalization, Stimulus; Haloperidol; Male; Muscarinic Antagonists; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Trihexyphenidyl

2004
Atypical and typical antipsychotic drug interactions with the dopamine D2 receptor.
    European journal of medicinal chemistry, 2005, Volume: 40, Issue:2

    Topics: Antipsychotic Agents; Binding Sites; Butyrophenones; Clozapine; Drug Interactions; Halogens; Humans; Ligands; Loxapine; Molecular Structure; Receptors, Dopamine D2

2005
Changes in weight and body mass index during treatment with melperone, clozapine and typical neuroleptics.
    Psychiatry research, 2010, Apr-30, Volume: 176, Issue:2-3

    Topics: Adult; Analysis of Variance; Antipsychotic Agents; Body Mass Index; Body Weight; Butyrophenones; Clozapine; Female; Humans; Male; Schizophrenia; Time Factors

2010
Auditing clinical outcomes after introducing off-licence prescribing of atypical antipsychotic melperone for patients with treatment refractory schizophrenia.
    TheScientificWorldJournal, 2012, Volume: 2012

    Topics: Adult; Antipsychotic Agents; Butyrophenones; Clozapine; Female; Follow-Up Studies; Humans; Male; Medical Audit; Middle Aged; Off-Label Use; Prospective Studies; Quality of Life; Schizophrenia; Severity of Illness Index; Treatment Outcome; Young Adult

2012