metronidazole and diazepam

metronidazole has been researched along with diazepam in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-19906 (20.00)18.7374
1990's1 (3.33)18.2507
2000's11 (36.67)29.6817
2010's11 (36.67)24.3611
2020's1 (3.33)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Abraham, MH; Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY2
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Brown, AM; Bruening-Wright, A; Kramer, J; Kuryshev, YA; Myatt, G; Obejero-Paz, CA; Verducci, JS1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Chandrasekaran, B; Cherukupalli, S; Hampannavar, GA; Karpoormath, R; Palakollu, VN; Thapliyal, N1
Bajusz, D; Balogh, GT; Dargó, G; Müller, J; Simon, K1
Achumba, JI; Essien, EE; Ette, EI; Thomas, WO1
Gugler, R; Jensen, JC1
O'Neil, JT; Pogge, RC1
Marshall, RJ; McIndewar, IC1
Hill, LM; Kleinberg, F1
Bociaga-Jasik, M; Caban, J; Garlicki, A; Kluba-Wojewoda, U; Krukowiecki, J1
Georgiadis, G; Kazakos, G; Koutinas, AF; Koutinas, Ch; Polizopoulou, ZS; Soubasis, N1
Hanley, MR; O'Regan, W; Squires, S; Tate, C1
Cavanagh, S; Fleming, C; Muldoon, EG1
Carter, C; Viveash, S1
Coboeken, K; Dallmann, A; Eissing, T; Hempel, G; Ince, I1

Reviews

3 review(s) available for metronidazole and diazepam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
An insight on synthetic and medicinal aspects of pyrazolo[1,5-a]pyrimidine scaffold.
    European journal of medicinal chemistry, 2017, Jan-27, Volume: 126

    Topics: Animals; Chemistry Techniques, Synthetic; Humans; Pyrazoles; Pyrimidines

2017
Effects of drugs and chemicals on the fetus and newborn (2).
    Mayo Clinic proceedings, 1984, Volume: 59, Issue:11

    Topics: Abnormalities, Drug-Induced; Anticoagulants; Anticonvulsants; Diazepam; Drug-Related Side Effects and Adverse Reactions; Environmental Pollutants; Female; Fetal Alcohol Spectrum Disorders; Fetus; Hexachlorophene; Humans; Infant, Newborn; Metronidazole; Povidone-Iodine; Pregnancy; Smoking

1984

Other Studies

27 other study(ies) available for metronidazole and diazepam

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
ElogPoct: a tool for lipophilicity determination in drug discovery.
    Journal of medicinal chemistry, 2000, Jul-27, Volume: 43, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Solvents

2000
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
    Journal of medicinal chemistry, 2001, Jul-19, Volume: 44, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water

2001
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
    Journal of medicinal chemistry, 2002, Jun-20, Volume: 45, Issue:13

    Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding

2002
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
MICE models: superior to the HERG model in predicting Torsade de Pointes.
    Scientific reports, 2013, Volume: 3

    Topics: ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Models, Theoretical; Patch-Clamp Techniques; Predictive Value of Tests; Torsades de Pointes

2013
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Human Serum Albumin Binding in a Vial: A Novel UV-pH Titration Method To Assist Drug Design.
    Journal of medicinal chemistry, 2020, 02-27, Volume: 63, Issue:4

    Topics: Binding Sites; Chemistry, Pharmaceutical; Drug Design; Humans; Hydrogen-Ion Concentration; Molecular Docking Simulation; Pharmaceutical Preparations; Protein Binding; Serum Albumin, Human; Spectrophotometry, Ultraviolet; Titrimetry

2020
IARC monographs on the evaluation of the carcinogenic risk of chemicals to man: some miscellaneous pharmaceutical substances.
    IARC monographs on the evaluation of the carcinogenic risk of chemicals to man, 1977, Volume: 13

    Topics: Acriflavine; Animals; Anthralin; Aurothioglucose; Carcinogens; Chloroquine; Diazepam; Ethanolamines; Ethionamide; Female; Humans; Hycanthone; Male; Metronidazole; Neoplasms; Neoplasms, Experimental; Oxazepam; Oxymetholone; Oxyphenbutazone; Oxyquinoline; Phenacetin; Phenobarbital; Phenylbutazone; Phenytoin; Pregnancy; Pyrimethamine; Risk

1977
Chloroquine-induced acute dystonic reactions in the presence of metronidazole.
    Drug intelligence & clinical pharmacy, 1988, Volume: 22, Issue:4

    Topics: Adult; Basal Ganglia Diseases; Chloroquine; Diazepam; Drug Interactions; Dystonia; Female; Humans; Metronidazole

1988
Interaction between metronidazole and drugs eliminated by oxidative metabolism.
    Clinical pharmacology and therapeutics, 1985, Volume: 37, Issue:4

    Topics: Administration, Oral; Adult; Antipyrine; Chromatography, Gas; Diazepam; Drug Interactions; Female; Half-Life; Humans; Infusions, Parenteral; Kinetics; Male; Metronidazole; Phenytoin

1985
Relative safety of self inflicted overdose with relatively newer medications.
    Arizona medicine, 1973, Volume: 30, Issue:7

    Topics: Adult; Depression; Diazepam; Female; Humans; Lethal Dose 50; Metronidazole; Penicillin V; Substance-Related Disorders

1973
Interactions between the neuromuscular blocking drug Org NC 45 and some anaesthetic, analgesic and antimicrobial agents.
    British journal of anaesthesia, 1981, Volume: 53, Issue:8

    Topics: Analgesics; Anesthesia, Inhalation; Anesthesia, Intravenous; Anesthetics; Animals; Cats; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Female; Male; Metronidazole; Neuromuscular Blocking Agents; Pancuronium; Vecuronium Bromide

1981
[Modifications in treatment of tetanus and prognosis--observations from the Cracow Department of Infectious Diseases].
    Przeglad lekarski, 1999, Volume: 56, Issue:9

    Topics: Aged; Aged, 80 and over; Diazepam; Drug Therapy, Combination; Female; Humans; Length of Stay; Male; Mental Disorders; Metronidazole; Midazolam; Middle Aged; Penicillins; Survival Rate; Tetanus

1999
Presumed localized tetanus in two cats.
    Journal of feline medicine and surgery, 2002, Volume: 4, Issue:4

    Topics: Animals; Cat Diseases; Cats; Diagnosis, Differential; Diazepam; Electromyography; Forelimb; Male; Metronidazole; Physical Therapy Modalities; Tetanus

2002
Tetanus, pneumonia, and malaria in a tsunami victim in Banda Aceh, Indonesia.
    Military medicine, 2006, Volume: 171, Issue:12

    Topics: Adult; Ceftriaxone; Diazepam; Disasters; Female; Humans; Indonesia; Malaria; Metronidazole; Pneumonia; Prognosis; Tetanus

2006
Generalised tetanus in an unvaccinated adult.
    Irish journal of medical science, 2010, Volume: 179, Issue:1

    Topics: Aged; Anti-Bacterial Agents; Anti-Infective Agents; Clostridium tetani; Diazepam; Humans; Magnesium Sulfate; Male; Metronidazole; Muscle Relaxants, Central; Muscle Spasticity; Penicillin G; Tetanus; Tetanus Antitoxin; Tetanus Toxoid; Trismus

2010
Nursing a critically ill tetanus patient in an intensive care unit in Zambia.
    British journal of nursing (Mark Allen Publishing), 2017, May-11, Volume: 26, Issue:9

    Topics: Analgesics, Opioid; Anti-Infective Agents; Anticonvulsants; Back Pain; Critical Care Nursing; Critical Illness; Developing Countries; Diazepam; Fever; Humans; Immunoglobulins; Immunologic Factors; Magnesium; Male; Meperidine; Metronidazole; Muscle Weakness; Pain; Seizures; Tetanus; Trismus; Young Adult; Zambia

2017
A Physiologically Based Pharmacokinetic Model for Pregnant Women to Predict the Pharmacokinetics of Drugs Metabolized Via Several Enzymatic Pathways.
    Clinical pharmacokinetics, 2018, Volume: 57, Issue:6

    Topics: Caffeine; Cytochrome P-450 Enzyme System; Diazepam; Female; Granisetron; Humans; Metoprolol; Metronidazole; Midazolam; Models, Biological; Nifedipine; Ondansetron; Pharmaceutical Preparations; Pregnancy

2018