metoclopramide and thioridazine

metoclopramide has been researched along with thioridazine in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-199014 (56.00)18.7374
1990's1 (4.00)18.2507
2000's5 (20.00)29.6817
2010's5 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Ahman, M; Holmén, AG; Wan, H1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Boriss, H; Braggio, S; Corbioli, S; Fontana, S; Helmdach, L; Longhi, R; Schiller, J; Vinco, F1
Artursson, P; Mateus, A; Matsson, P1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Costall, B; Naylor, RJ2
Budygin, EA; Gaĭnetdinov, RR; Kovalev, GI; Kudrin, VS; Raevskiĭ, KS1
Blackburn, JR; Phillips, AG1
Blackburn, JR; Fibiger, HC; Phillips, AG1
Jepsen, SA; Nielsen, EB1
Ekker, M; Sourkes, TL1
Hand, TH; Kasser, RJ; Wang, RY1
Blaha, CD; Lane, RF1
Cools, AR; Ellenbroek, BA; Honig, WM; Peeters, BW1
Greenberg, WM1
Marco, L; Stanford, GK; Velek, M1
Durko, A; Głuszcz-Zielińska, A; Kozubski, W; Prusiński, A; Rózniecki, J; Swatko, A1
Stanley, M; Wazer, D1
Kim, HS; Liebman, J; Welch, JJ1
Davidson, A; Hunter, C; Jankovic, J; Kenney, C1

Reviews

1 review(s) available for metoclopramide and thioridazine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

24 other study(ies) available for metoclopramide and thioridazine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
    Journal of medicinal chemistry, 2001, Jul-19, Volume: 44, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water

2001
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Relationship between brain tissue partitioning and microemulsion retention factors of CNS drugs.
    Journal of medicinal chemistry, 2009, Mar-26, Volume: 52, Issue:6

    Topics: Brain; Central Nervous System; Chromatography, Liquid; Emulsions; Mass Spectrometry

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Brain tissue binding of drugs: evaluation and validation of solid supported porcine brain membrane vesicles (TRANSIL) as a novel high-throughput method.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:2

    Topics: Absorption; Albumins; Animals; Brain; Brain Chemistry; Cell Membrane; Chromatography, High Pressure Liquid; Drug Evaluation, Preclinical; In Vitro Techniques; Lipids; Male; Microdialysis; Pharmaceutical Preparations; Protein Binding; Rats; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Swine; Tissue Distribution

2011
A high-throughput cell-based method to predict the unbound drug fraction in the brain.
    Journal of medicinal chemistry, 2014, Apr-10, Volume: 57, Issue:7

    Topics: Animals; Brain; Dialysis; HEK293 Cells; High-Throughput Screening Assays; Humans; Pharmaceutical Preparations; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2014
A comparison of the abilities of typical neuroleptic agents and of thioridazine, clozapine, sulpiride and metoclopramide to antagonise the hyperactivity induced by dopamine applied intracerebrally to areas of the extrapyramidal and mesolimbic systems.
    European journal of pharmacology, 1976, Volume: 40, Issue:1

    Topics: Animals; Brain; Clozapine; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Fluphenazine; Haloperidol; Limbic System; Male; Metoclopramide; Pimozide; Rats; Stereotaxic Techniques; Sulpiride; Thioridazine; Tranquilizing Agents

1976
[Different effects of typical and atypical neuroleptics on K+-stimulated dopamine release from isolated rat striatum].
    Biulleten' eksperimental'noi biologii i meditsiny, 1992, Volume: 114, Issue:7

    Topics: Animals; Antipsychotic Agents; Carbolines; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; In Vitro Techniques; Male; Metoclopramide; Potassium; Raclopride; Rats; Rats, Wistar; Remoxipride; Salicylamides; Stimulation, Chemical; Sulpiride; Thioridazine; Tiapamil Hydrochloride; Trifluoperazine

1992
Blockade of acquisition of one-way conditioned avoidance responding by haloperidol and metoclopramide but not by thioridazine or clozapine: implications for screening new antipsychotic drugs.
    Psychopharmacology, 1989, Volume: 98, Issue:4

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Clozapine; Dibenzazepines; Drug Evaluation, Preclinical; Haloperidol; Male; Metoclopramide; Rats; Thioridazine

1989
Dopamine and preparatory behavior: III. Effects of metoclopramide and thioridazine.
    Behavioral neuroscience, 1989, Volume: 103, Issue:4

    Topics: Animals; Arousal; Brain; Conditioning, Classical; Dopamine; Dose-Response Relationship, Drug; Feeding Behavior; Male; Metoclopramide; Motivation; Rats; Receptors, Dopamine; Thioridazine

1989
Antagonism of the amphetamine cue by both classical and atypical antipsychotic drugs.
    European journal of pharmacology, 1985, May-08, Volume: 111, Issue:2

    Topics: Animals; Antipsychotic Agents; Cues; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Humans; Male; Metoclopramide; Pimozide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Thioridazine

1985
Differential effects of thioridazine, clozapine and metoclopramide on the induction of adrenomedullary enzymes by apomorphine.
    Neuropharmacology, 1985, Volume: 24, Issue:11

    Topics: Adrenal Medulla; Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Enzyme Induction; Male; Metoclopramide; Ornithine Decarboxylase; Rats; Rats, Inbred Strains; Substantia Nigra; Thioridazine; Tyrosine 3-Monooxygenase

1985
Effects of acute thioridazine, metoclopramide and SCH 23390 on the basal activity of A9 and A10 dopamine cells.
    European journal of pharmacology, 1987, Jun-04, Volume: 137, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Thioridazine

1987
Chronic treatment with classical and atypical antipsychotic drugs differentially decreases dopamine release in striatum and nucleus accumbens in vivo.
    Neuroscience letters, 1987, Jul-22, Volume: 78, Issue:2

    Topics: Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Haloperidol; Male; Metoclopramide; Nucleus Accumbens; Promethazine; Rats; Rats, Inbred Strains; Septal Nuclei; Thioridazine

1987
The paw test: a behavioural paradigm for differentiating between classical and atypical neuroleptic drugs.
    Psychopharmacology, 1987, Volume: 93, Issue:3

    Topics: Animals; Antipsychotic Agents; Chlorpromazine; Clozapine; Desipramine; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Forelimb; Haloperidol; Hindlimb; Male; Metoclopramide; Morphine; Motor Activity; Rats; Rats, Inbred Strains; Thioridazine

1987
Mechanism of neuroleptic-associated priapism.
    The American journal of psychiatry, 1988, Volume: 145, Issue:3

    Topics: Antipsychotic Agents; Dopamine Antagonists; Humans; Male; Metoclopramide; Priapism; Receptors, Adrenergic, alpha; Thioridazine

1988
Priapism associated with concurrent use of thioridazine and metoclopramide.
    The American journal of psychiatry, 1987, Volume: 144, Issue:6

    Topics: Adult; Drug Synergism; Drug Therapy, Combination; Gastroesophageal Reflux; Humans; Male; Metoclopramide; Priapism; Schizophrenia, Paranoid; Thioridazine

1987
[Acute dystonic reactions after administration of neuroleptics and other drugs].
    Wiadomosci lekarskie (Warsaw, Poland : 1960), 1985, Mar-01, Volume: 38, Issue:5

    Topics: Acute Disease; Adult; Child; Droperidol; Dystonia; Female; Humans; Male; Metoclopramide; Middle Aged; Thioridazine

1985
Is there a relationship between the involvement of extrapyramidal and mesolimbic brain areas with the cataleptic action of neuroleptic agents and their clinical antipsychotic effect?
    Psychopharmacologia, 1973, Volume: 32, Issue:2

    Topics: Animals; Aporphines; Benzoates; Butyrophenones; Catalepsy; Dioxoles; Extrapyramidal Tracts; Humans; Hypothalamus; Male; Metoclopramide; Perphenazine; Piperidines; Rats; Spiro Compounds; Thioridazine; Tranquilizing Agents

1973
High plasma concentrations of metoclopramide are not detected by radioreceptor assay.
    Neuropsychobiology, 1983, Volume: 10, Issue:2-3

    Topics: Animals; Corpus Striatum; Dose-Response Relationship, Drug; Humans; Male; Metoclopramide; Prolactin; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Schizophrenia; Thioridazine

1983
Amphetamine-induced increases in dopaminergic single cell firing rate after haloperidol pretreatment. Correlation with extrapyramidal side effects.
    Neuropharmacology, 1980, Volume: 19, Issue:4

    Topics: Animals; Apomorphine; Brain; Clozapine; Dextroamphetamine; Dopamine; Drug Interactions; Extrapyramidal Tracts; Haloperidol; Male; Metoclopramide; Neurons; Rats; Substantia Nigra; Thioridazine

1980
Metoclopramide, an increasingly recognized cause of tardive dyskinesia.
    Journal of clinical pharmacology, 2008, Volume: 48, Issue:3

    Topics: Adverse Drug Reaction Reporting Systems; Aged; Amitriptyline; Dyskinesia, Drug-Induced; Haloperidol; Humans; Metoclopramide; Middle Aged; Perphenazine; Retrospective Studies; Texas; Thioridazine; Time Factors

2008