metoclopramide and ketanserin

metoclopramide has been researched along with ketanserin in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19908 (42.11)18.7374
1990's4 (21.05)18.2507
2000's2 (10.53)29.6817
2010's5 (26.32)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Calderó, JM; del Río, J; García, E; Lasheras, B; Monge, A; Palop, JA; Peña, MC; Roca, J; Romero, G1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
al-Humayyd, MS; Mobarok Ali, AT1
Bianconi, L; Buonanno, G; Caiazza, A; Capretti, L; Cavazzini, U; Chiodera, P; Coiro, V; Marcato, A; Speroni, G; Volpi, R1
Adler-Graschinsky, E; Butta, NV; Elgoyhen, AB1
Andries, LJ; Brutsaert, DL; Meulemans, AL; Shah, AM1
Bianconi, L; Caiazza, A; Capretti, L; Chiodera, P; Coiro, V; Fagnoni, F; Schianchi, L; Speroni, G; Volpi, R1
Costall, B; Gunning, SJ; Naylor, RJ; Tattersall, FD1
Kilbinger, H; Pfeuffer-Friederich, I1
Ozaki, L; Stern, N; Tuck, ML1
Bianconi, M; Degli Uberti, EC; Margutti, AR; Pansini, P; Rotola, CA; Trasforini, G1
Creese, I; Hamblin, MW; Leff, SE1
Deschaux, P; Ferriere, F; Khan, NA; Meyniel, JP1

Trials

1 trial(s) available for metoclopramide and ketanserin

ArticleYear
5-HT1-, but not 5-HT2-serotonergic, M1-, M2-muscarinic cholinergic or dopaminergic receptors mediate the ACTH/cortisol response to metoclopramide in man.
    Hormone research, 1990, Volume: 33, Issue:6

    Topics: Adrenocorticotropic Hormone; Adult; Atropine; Bromocriptine; Dose-Response Relationship, Drug; Humans; Hydrocortisone; Ketanserin; Male; Metergoline; Metoclopramide; Pirenzepine; Receptors, Adrenergic; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Muscarinic; Receptors, Serotonin

1990

Other Studies

18 other study(ies) available for metoclopramide and ketanserin

ArticleYear
Synthesis of 2-piperazinylbenzothiazole and 2-piperazinylbenzoxazole derivatives with 5-HT3 antagonist and 5-HT4 agonist properties.
    Journal of medicinal chemistry, 1994, Apr-29, Volume: 37, Issue:9

    Topics: Animals; Benzothiazoles; Binding, Competitive; Cerebral Cortex; Female; Gastric Emptying; Granisetron; Guinea Pigs; Ileum; Male; Molecular Structure; Mucous Membrane; Ondansetron; Piperazines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles

1994
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Enhancement of antithrombotic effect of aspirin by metoclopramide in rats.
    Thrombosis research, 1991, Feb-15, Volume: 61, Issue:4

    Topics: 5-Hydroxytryptophan; Administration, Oral; Animals; Aspirin; Benzamides; Body Temperature; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Drug Combinations; Drug Interactions; Female; Fibrinolytic Agents; Injections, Intravenous; Ketanserin; Metoclopramide; Rats; Receptors, Cell Surface; Thrombosis

1991
Different receptor subtypes mediate the dual presynaptic effects of 5-hydroxytryptamine on peripheral sympathetic neurones.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cats; Cyproheptadine; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Ketanserin; Male; Membranes; Metoclopramide; Neurons; Norepinephrine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes; Tropanes

1989
Endocardium modulates myocardial inotropic response to 5-hydroxytryptamine.
    The American journal of physiology, 1989, Volume: 257, Issue:6 Pt 2

    Topics: Animals; Cats; Endocardium; Endothelium, Vascular; In Vitro Techniques; Ketanserin; Kinetics; Metoclopramide; Microscopy, Electron, Scanning; Myocardial Contraction; Papillary Muscles; Prazosin; Propranolol; Serotonin; Ventricular Function

1989
Muscarinic cholinergic, but not serotoninergic mediation of arginine vasopressin response to metoclopramide in man.
    Clinical endocrinology, 1989, Volume: 31, Issue:4

    Topics: Adult; Arginine Vasopressin; Atropine; Dose-Response Relationship, Drug; Humans; Ketanserin; Kinetics; Male; Metergoline; Metoclopramide; Pirenzepine; Receptors, Muscarinic; Receptors, Serotonin

1989
Modification of electrical field stimulation-induced contractions in the guinea-pig ileum by metoclopramide and ICS 205-930 depends on the integrity of the mucosa.
    The Journal of pharmacy and pharmacology, 1986, Volume: 38, Issue:11

    Topics: Animals; Drug Interactions; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Intestinal Mucosa; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Muscle, Smooth; Serotonin Antagonists; Tropisetron

1986
Two types of receptors for 5-hydroxytryptamine on the cholinergic nerves of the guinea-pig myenteric plexus.
    British journal of pharmacology, 1985, Volume: 85, Issue:2

    Topics: Acetylcholine; Animals; Binding, Competitive; Cocaine; Electric Stimulation; Female; Guinea Pigs; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Myenteric Plexus; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes

1985
Evidence for dopaminergic binding sites in the human adrenal cortex.
    Metabolism: clinical and experimental, 1986, Volume: 35, Issue:12

    Topics: Adrenal Cortex; Adult; Aged; Apomorphine; Binding, Competitive; Bromocriptine; Domperidone; Dopamine; Epinephrine; Female; Humans; Ketanserin; Male; Metoclopramide; Middle Aged; Receptors, Dopamine; Spiperone; Sulpiride; Time Factors

1986
Effect of ketanserin, an inhibitor of 5-HT2 receptors, on the aldosterone-stimulating action of metoclopramide.
    Hormone research, 1983, Volume: 17, Issue:3

    Topics: Adolescent; Adult; Aldosterone; Humans; Ketanserin; Kinetics; Male; Metoclopramide; Piperidines; Potassium; Prolactin; Receptors, Serotonin; Renin; Serotonin Antagonists

1983
Interactions of agonists with D-2 dopamine receptors: evidence for a single receptor population existing in multiple agonist affinity-states in rat striatal membranes.
    Biochemical pharmacology, 1984, Mar-15, Volume: 33, Issue:6

    Topics: Animals; Binding, Competitive; Butyrophenones; Corpus Striatum; Domperidone; Dopamine Antagonists; Guanine Nucleotides; Ketanserin; Metoclopramide; Piperidines; Radioligand Assay; Rats; Receptors, Dopamine; Sodium; Spiperone; Temperature

1984
5-Hydroxytryptamine-induced calcium-channel gating in rainbow trout (Oncorhynchus mykiss) peripheral blood lymphocytes.
    The Biochemical journal, 1997, Apr-01, Volume: 323 ( Pt 1)

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Calcium Channels; Dopamine Antagonists; Ion Channel Gating; Ionomycin; Ionophores; Ketanserin; Lymphocytes; Metoclopramide; Oncorhynchus mykiss; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulpiride

1997