metoclopramide and bemesetron

metoclopramide has been researched along with bemesetron in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19905 (29.41)18.7374
1990's11 (64.71)18.2507
2000's1 (5.88)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Airey, JE; Campbell, HF; Golec, S; Klein, S; Powers, M; Rodriguez, W; Schnapper, M; Studt, W; Woodward, R; Youssefyeh, RD1
Bloomquist, W; Cohen, ML; Reid, LR; Robertson, DW; Schenck, K; Wong, DT1
Carr, AA; Hibert, MF; Hoffmann, R; Miller, RC1
Bourguignon, JJ; Didier, B; Hoffmann, R; Rival, Y; Rybaltchenko, V; Wermuth, CG1
Fukui, H; Sato, S; Yamamoto, M1
Gandara, DR; Hesketh, PJ1
Adler-Graschinsky, E; Butta, NV; Elgoyhen, AB1
Buchheit, KH; Costall, B; Engel, G; Gunning, SJ; Naylor, RJ; Richardson, BP1
Bradbury, AJ; Costall, B; Gunning, SJ; Naylor, RJ1
Kilbinger, H; Pfeuffer-Friederich, I1
Round, A; Wallis, DI1
Buchheit, KH; Buhl, T1
Pilot, MA; Qin, XY; Scott, M; Thompson, H1
Barrett, RJ; Hahne, WF; Heck, K; Homesley, HD; Lentz, SS; Lovelace, JV; McLees, B; Woodlief, L1
Janvier, JJ; Peyraud-Waïtzenegger, M; Soulier, P1
Deschaux, P; Ferrière, F; Khan, NA; Meyniel, JP1
Andrews, PL; Cheng, FH; Moreaux, B; Ngan, MP; Rudd, JA; Sam, TS; Wai, MK; Wan, C1

Trials

1 trial(s) available for metoclopramide and bemesetron

ArticleYear
Randomized comparison of the antiemetic efficacy of a serotonin type 3 receptor antagonist (MDL 72,222) with a high-dose metoclopramide regimen.
    American journal of clinical oncology, 1993, Volume: 16, Issue:2

    Topics: Adult; Aged; Antiemetics; Cisplatin; Diphenhydramine; Drug Therapy, Combination; Female; Genital Neoplasms, Female; Humans; Lorazepam; Metoclopramide; Middle Aged; Nausea; Pilot Projects; Serotonin Antagonists; Tropanes; Vomiting

1993

Other Studies

16 other study(ies) available for metoclopramide and bemesetron

ArticleYear
Development of high-affinity 5-HT3 receptor antagonists. 2. Two novel tricyclic benzamides.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Amides; Animals; Antiemetics; Benzamides; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Dogs; Ferrets; Guinea Pigs; Ileum; Molecular Structure; Muscle Contraction; Rats; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting; X-Ray Diffraction

1992
Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:12

    Topics: Animals; Cell Membrane; Cerebral Cortex; Guinea Pigs; Heart Rate; Ileum; Indazoles; Male; Methylation; Myocardium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tritium; Tropanes

1990
Conformation-activity relationship study of 5-HT3 receptor antagonists and a definition of a model for this receptor site.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Animals; Binding Sites; Guinea Pigs; Mice; Protein Conformation; Rabbits; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1990
5-HT3 antagonists derived from aminopyridazine-type muscarinic M1 agonists.
    Journal of medicinal chemistry, 1998, Jan-29, Volume: 41, Issue:3

    Topics: Animals; Brain Stem; Hippocampus; In Vitro Techniques; Models, Molecular; Muscarinic Agonists; Myocardium; Protein Conformation; Pyridazines; Rats; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists

1998
Vagal afferent fibers and peripheral 5-HT3 receptors mediate cisplatin-induced emesis in dogs.
    Japanese journal of pharmacology, 1992, Volume: 59, Issue:2

    Topics: Afferent Pathways; Animals; Cisplatin; Dogs; Female; Indoles; Male; Metoclopramide; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vagus Nerve; Vomiting

1992
Serotonin antagonists: a new class of antiemetic agents.
    Journal of the National Cancer Institute, 1991, May-01, Volume: 83, Issue:9

    Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting

1991
Different receptor subtypes mediate the dual presynaptic effects of 5-hydroxytryptamine on peripheral sympathetic neurones.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cats; Cyproheptadine; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Ketanserin; Male; Membranes; Metoclopramide; Neurons; Norepinephrine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes; Tropanes

1989
5-Hydroxytryptamine receptor antagonism by metoclopramide and ICS 205-930 in the guinea-pig leads to enhancement of contractions of stomach muscle strips induced by electrical field stimulation and facilitation of gastric emptying in-vivo.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:9

    Topics: Animals; Electric Stimulation; Gastric Emptying; Guinea Pigs; In Vitro Techniques; Indoles; Male; Metoclopramide; Muscle Contraction; Muscle, Smooth; Serotonin Antagonists; Stomach; Tropanes; Tropisetron

1985
Evidence that 5-hydroxytryptamine may exert both facilitatory and inhibitory control of electrical field stimulation-evoked contractions in longitudinal muscle taken from the body of guinea-pig stomach.
    The Journal of pharmacy and pharmacology, 1986, Volume: 38, Issue:3

    Topics: 5-Hydroxytryptophan; Animals; Electric Stimulation; Fenclonine; Guinea Pigs; In Vitro Techniques; Male; Methyldopa; Metoclopramide; Muscle Contraction; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Tropanes

1986
Two types of receptors for 5-hydroxytryptamine on the cholinergic nerves of the guinea-pig myenteric plexus.
    British journal of pharmacology, 1985, Volume: 85, Issue:2

    Topics: Acetylcholine; Animals; Binding, Competitive; Cocaine; Electric Stimulation; Female; Guinea Pigs; Ketanserin; Male; Methiothepin; Methysergide; Metoclopramide; Muscle Contraction; Myenteric Plexus; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes

1985
Further studies on the blockade of 5-HT depolarizations of rabbit vagal afferent and sympathetic ganglion cells by MDL 72222 and other antagonists.
    Neuropharmacology, 1987, Volume: 26, Issue:1

    Topics: Action Potentials; Animals; Female; Ganglia, Sympathetic; In Vitro Techniques; Male; Metoclopramide; Nodose Ganglion; Piperazines; Quipazine; Rabbits; Serotonin; Serotonin Antagonists; Tropanes; Vagus Nerve

1987
Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: 4-Aminobenzoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ligands; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Tetrodotoxin; Tropanes; Tropisetron

1994
Effects of cholinoceptor and 5-hydroxytryptamine3 receptor antagonism on erythromycin-induced canine intestinal motility disruption and emesis.
    British journal of pharmacology, 1993, Volume: 108, Issue:1

    Topics: Animals; Atropine; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cholinergic Antagonists; Dogs; Electromyography; Erythromycin; Female; Gastrointestinal Motility; Hexamethonium; Hexamethonium Compounds; Injections, Intravenous; Intestine, Small; Male; Metoclopramide; Muscle Contraction; Muscle, Smooth; Serotonin Antagonists; Tropanes; Vomiting

1993
Mediation of serotonin-induced hyperventilation via 5-HT3-receptor in European eel Anguilla anguilla.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 1996, Volume: 165, Issue:8

    Topics: Anguilla; Animals; Benzimidazoles; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Hyperventilation; Injections, Intravenous; Methysergide; Metoclopramide; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Respiration; Serotonin; Serotonin Antagonists; Tropanes

1996
Identification of lymphocyte 5-HT3 receptor subtype and its implication in fish T-cell proliferation.
    Immunology letters, 1997, Volume: 55, Issue:3

    Topics: Animals; Cell Cycle; Indoles; Lymphocyte Activation; Lymphocytes; Metoclopramide; Oncorhynchus mykiss; Phytohemagglutinins; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Sodium; Time Factors; Tritium; Tropanes; Tropisetron

1997
Evaluation of the anti-emetic potential of anti-migraine drugs to prevent resiniferatoxin-induced emesis in Suncus murinus (house musk shrew).
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Antiemetics; Butanols; Capsaicin; Cyclooxygenase Inhibitors; Dihydroergotamine; Diphenhydramine; Diterpenes; Domperidone; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Indomethacin; Malates; Methysergide; Metoclopramide; Migraine Disorders; Ondansetron; Piperidines; Ruthenium Red; Scopolamine; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Sumatriptan; Time Factors; Tropanes; Vomiting

2005